CAS 94-15-5

Dimethocaine

Description:

Dimethocaine, also known as ethyl 4-(dimethylamino)benzoate, is a local anesthetic compound that belongs to the ester class of anesthetics. It is structurally related to cocaine and exhibits similar pharmacological properties, primarily acting as a sodium channel blocker to inhibit nerve impulse transmission. Dimethocaine is characterized by its ability to provide localized pain relief, making it useful in various medical applications. The compound is typically a white crystalline powder and is soluble in organic solvents but has limited solubility in water. Its chemical formula is C11H15N O2, and it has a molecular weight that reflects its complex structure. While it has potential therapeutic uses, dimethocaine is also associated with recreational use and can pose risks of toxicity and dependence. As with many anesthetics, careful consideration of dosage and administration is crucial to minimize adverse effects. Due to its structural similarities to controlled substances, dimethocaine is subject to regulatory scrutiny in many jurisdictions.

Formula: C₁₆H₂₆N₂O₂

InChI: InChI=1S/C16H26N2O2/c1-5-18(6-2)11-16(3,4)12-20-15(19)13-7-9-14(17)10-8-13/h7-10H,5-6,11-12,17H2,1-4H3

InChI key: InChIKey=OWQIUQKMMPDHQQ-UHFFFAOYSA-N

SMILES: C(OCC(CN(CC)CC)(C)C)(=O)C1=CC=C(N)C=C1

Synonyms:

• (3-Diethylamino-2,2-dimethyl)propyl 4-aminobenzoat
• 1-Propanol, 2-[(diethylamino)methyl]-2-methyl-, 1-(4-aminobenzoate)
• 1-Propanol, 3-(diethylamino)-2,2-dimethyl-, 4-aminobenzoate (ester)
• 1-Propanol, 3-(diethylamino)-2,2-dimethyl-, p-amino benzoate
• 1-Propanol, 3-(diethylamino)-2,2-dimethyl-, p-aminobenzoate
• 1-Propanol, 3-(diethylamino)-2,2-dimethyl-, p-aminobenzoate (ester)
• 4-Aminobenzoesaeure-3-diethylamino-2,2-dimethylproplylester
• Brn 2215967
• Dimethocaine
• Larocaine
• Nsc 68927
• Unii-R3L4A6Gowz

Dimethocaine

CAS: 94-15-5

Dimethocaine (Larocaine) is a local anesthetic which also effects on the central nervous system acting as dopamine-reuptake-inhibitor.

Formula: C₁₆H₂₆N₂O₂

Purity: 99.52%

Color and Shape: Solid

Molecular weight: 278.39

Ref: TM-T7118

Dimethocaine

Controlled Product

CAS: 94-15-5

Applications Dimethocaine is a local anesthetic with stimulatory properties that is half the potency of cocaine.
References Meyer, M.R., et al.: Toxicol. Lett., 217, 137 (2013); Wilcox, K.M., et al.: Synapse., 58, 220 (2005); Rigon, A.R., et al.: Psychopharmacol., 127, 323 (1996);

Formula: C₁₆H₂₆N₂O₂

Color and Shape: Neat

Molecular weight: 278.39

Ref: TR-D479515

Dimethocaine

Controlled Product

CAS: 94-15-5

Dimethocaine is a local anesthetic that is used in ophthalmology and dentistry. It is also used as a topical anesthetic, especially in the treatment of mouth sores. Dimethocaine has been shown to inhibit angiogenesis by preventing the release of various angiogenic factors from endothelial cells. Dimethocaine binds to dopamine receptors, which causes its uptake into cells, including human liver cells. The binding affinity for dopamine receptors increases with increasing basicity of the structure of dimethocaine.

Formula: C₁₆H₂₆N₂O₂

Purity: Min. 95%

Color and Shape: Powder

Molecular weight: 278.39 g/mol

Ref: 3D-FD178421

Dimethocaine

CAS: 94-15-5

Formula: C₁₆H₂₆N₂O₂

Color and Shape: Solid

Molecular weight: 278.3898

Ref: IN-DA003PKH