CAS 94651-09-9
:Cicloprolol
Description:
Cicloprolol is a beta-blocker medication primarily used for the treatment of hypertension and certain heart conditions. It is characterized by its selective action on beta-1 adrenergic receptors, which helps to reduce heart rate and myocardial contractility, ultimately lowering blood pressure. Cicloprolol also exhibits some intrinsic sympathomimetic activity, which means it can partially stimulate beta receptors while blocking them, potentially leading to fewer side effects compared to non-selective beta-blockers. The compound has a relatively short half-life, necessitating multiple doses throughout the day for sustained therapeutic effects. Additionally, Cicloprolol may possess vasodilatory properties, contributing to its antihypertensive effects. Its pharmacokinetics can be influenced by factors such as age, liver function, and concomitant medications. As with other beta-blockers, common side effects may include fatigue, dizziness, and bradycardia. Overall, Cicloprolol represents a valuable option in the management of cardiovascular conditions, particularly for patients who may benefit from its unique pharmacological profile.
Formula:C18H29NO4
InChI:InChI=1S/C18H29NO4/c1-14(2)19-11-16(20)13-23-18-7-5-17(6-8-18)22-10-9-21-12-15-3-4-15/h5-8,14-16,19-20H,3-4,9-13H2,1-2H3
InChI key:InChIKey=JNDJPKHYZWRRIS-UHFFFAOYSA-N
SMILES:O(CC(CNC(C)C)O)C1=CC=C(OCCOCC2CC2)C=C1
Synonyms:- 1-[4-[2-(Cyclopropylmethoxy)ethoxy]phenoxy]-3-[(1-methylethyl)amino]-2-propanol
- 2-Propanol,1-[4-[2-(cyclopropylmethoxy)ethoxy]phenoxy]-3-[(1-methylethyl)amino]-, (?à)-
- Cicloprolol
- 2-Propanol, 1-[4-[2-(cyclopropylmethoxy)ethoxy]phenoxy]-3-[(1-methylethyl)amino]-, (±)-
- 2-Propanol, 1-[4-[2-(cyclopropylmethoxy)ethoxy]phenoxy]-3-[(1-methylethyl)amino]-
- [Synonyms]
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Found 3 products.
Cicloprolol-d5
CAS:Cicloprolol-d5 is a protein inhibitor that belongs to the class of medicinal compounds known as cyclin-dependent kinase inhibitors. It works by blocking the activity of kinases, which are enzymes involved in cell cycle regulation and proliferation. Cicloprolol-d5 has been shown to induce apoptosis, or programmed cell death, in cancer cells. This compound has demonstrated anticancer activity in Chinese hamster ovary cells and human tumor cell lines. It is a potent inhibitor of cyclin-dependent kinases and may have potential as an anticancer agent.
Formula:C18H29NO4Purity:Min. 95%Molecular weight:323.4 g/mol
