CAS 962-58-3

Diazoxon

Description:

Diazoxon, with the CAS number 962-58-3, is an organophosphate compound that serves as a potent inhibitor of the enzyme acetylcholinesterase. This inhibition leads to the accumulation of acetylcholine in the synaptic cleft, resulting in prolonged stimulation of the nervous system. Diazoxon is primarily recognized for its role as a metabolite of the pesticide diazinon, which is used in agricultural applications. The compound is characterized by its relatively high toxicity to both insects and mammals, making it a subject of concern in environmental and health contexts. Physically, diazoxon is typically a colorless to pale yellow liquid with a distinctive odor. It is soluble in organic solvents but has limited solubility in water. Due to its toxicological properties, exposure to diazoxon can lead to symptoms associated with cholinergic toxicity, including respiratory distress, muscle twitching, and neurological effects. Proper handling and safety measures are essential when working with this substance to mitigate risks associated with its toxicity.

Formula: C₁₂H₂₁N₂O₄P

InChI: InChI=1S/C12H21N2O4P/c1-6-16-19(15,17-7-2)18-11-8-10(5)13-12(14-11)9(3)4/h8-9H,6-7H2,1-5H3

InChI key: InChIKey=VBLJFQYCTRKKKF-UHFFFAOYSA-N

SMILES: O(P(OCC)(OCC)=O)C1=NC(C(C)C)=NC(C)=C1

Synonyms:

• 4-Pyrimidinol, 2-isopropyl-6-methyl-, diethyl phosphate
• Diazinon oxon
• Diazinon oxygen analog
• Diazoxon
• Diethyl 2-isopropyl-6-methyl-4-pyrimidinyl phosphate
• Diethyl 2-isopropyl-6-methylpyrimidin-4-yl phosphate
• Diethyl 6-Methyl-2-(1-Methylethyl)Pyrimidin-4-Yl Phosphate
• Diethyl 6-methyl-2-(1-methylethyl)-4-pyrimidinyl phosphate
• Diethyl-2-isopropyl-6-methyl-4-pyrimidinylphosphat
• O,O-Diethyl O-(2-isopropyl-6-methyl-4-pyrimidinyl) phosphate
• O,O-Diethyl-O-(2-isopropyl-4-methylpyrimidyl-6) phosphate
• Oxodiazinon
• Phosphoric acid, diethyl 2-isopropyl-6-methyl-4-pyrimidinyl ester

Diazinon Oxon (Diazoxon)

CAS: 962-58-3

Formula: C₁₂H₂₁N₂O₄P

Molecular weight: 288.28

Ref: 4Z-D-183003

Diazinon-oxon 100 µg/mL in Acetonitrile

CAS: 962-58-3

Formula: C₁₂H₂₁N₂O₄P

Color and Shape: Single Solution

Molecular weight: 288.28

Ref: 04-A12210200AL-100

Diazinon-oxon

Controlled Product

CAS: 962-58-3

Formula: C₁₂H₂₁N₂O₄P

Color and Shape: Neat

Molecular weight: 288.28

Ref: 04-CA12210200

Diazoxon

CAS: 962-58-3

Formula: C₁₂H₂₁N₂O₄P

Molecular weight: 288.28

Ref: 4Z-D-181001

Diazoxon

Controlled Product

CAS: 962-58-3

Applications Diazoxon, is the oxidized form of Diazinon (D416880), an organophosphate insecticide. Diazoxon, is shown to be a more potent acetylcholinesterase (AChE) inhibitor.
Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package
References Lazarevic-Pasti, T. D., et al.: J. Electroanal. Chem., 692 (2013); Pasti, T. L., J. Environ. Protect. Ecology, 12, 1168 (2011);

Formula: C₁₂H₂₁N₂O₄P

Color and Shape: Colourless

Molecular weight: 288.28

Ref: TR-D416890

Diazoxon-d10

Controlled Product

CAS: 962-58-3

Applications Isotope laballed Diazoxon, is the oxidized form of Diazinon (D416880), an organophosphate insecticide. Diazoxon, is shown to be a more potent acetylcholinesterase (AChE) inhibitor.
Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package
References Lazarevic-Pasti, T. D., et al.: J. Electroanal. Chem., 692 (2013); Pasti, T. L., J. Environ. Protect. Ecology, 12, 1168 (2011);

Formula: C₁₂H₁₁D₁₀N₂O₄P

Color and Shape: Neat

Molecular weight: 199.27

Ref: TR-D416893

Diazoxon

CAS: 962-58-3

Diazoxon is the oxidized form of Diazinon -- an organophosphate insecticide. Diazoxon is shown to be a more potent acetylcholinesterase (AChE) inhibitor.

Formula: C₁₂H₂₁N₂O₄P

Color and Shape: Solid

Molecular weight: 288.28

Ref: TM-T68217