Inhibitor Enzymes
Inhibitor enzymes are molecules that decrease or block the activity of enzymes, preventing them from catalyzing their specific reactions. These inhibitors can be reversible or irreversible and are crucial tools in research and drug development for studying enzyme mechanisms, controlling metabolic pathways, and developing therapeutic agents. Inhibitor enzymes are widely used to modulate biological processes and to treat various diseases by targeting specific enzymes. At CymitQuimica, we offer a comprehensive range of high-quality enzyme inhibitors to support your research and pharmaceutical development needs.
Found 123 products of "Inhibitor Enzymes"
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Retorphan
CAS:Controlled Product<p>Applications Retorphan is a powerful and selective inhibitors of neprilysin and is being developed as a therapeutic agent. Retorphan behave as the prodrug of the enantiomers of Thiorphan (T369500).<br>References Monteil, T., et al.: Mini. Rev. Med. Chem., 2, 209 (2002); Roques, B.P., et al.: Nature, 288, 286 (1980); Tiraboschi, G., et al.: Protein Engineering, 12, 2, 141 (1999)<br></p>Formula:C21H23NO4SColor and Shape:NeatMolecular weight:385.48(1R,2R)-2-Fluorocyclopentanamine Hydrochloride
CAS:Controlled Product<p>Applications A cyclopentanamine used in the preparation of heterocyclic and aromatic ureas and amides as CEPT inhibitors.<br></p>Formula:C5H11ClFNColor and Shape:NeatMolecular weight:139.61-Deoxy-L-altronojirimycin Hydrochloride
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications α-Glycosidase inhibitor.<br>References Jefferies, I., et al.: Bioorg. Med. Chem. Lett., 7, 1171 (1997), Hassan, A., et al.: Carbohydr. Res., 339, 1565 (2004),<br></p>Formula:C6H13NO4·ClHPurity:>90%Color and Shape:NeatMolecular weight:199.634-Fluorobenzoic Acid-d4
CAS:Controlled Product<p>Applications 4-Fluorobenzoic Acid-d4 is used as a reagent in the synthesis of Flurofamide-d4 (F596687); the isotope labelled analog of Fluorofamide (F596685) which is a compound that acts as a urease inhibitor, useful in the treatment of gastritis and irregular urease activity in the urinary tract.<br>References Loes, A. et al.: Lett. App. Microbiol., 58, 31 (2014); Ohta, T.et al.: Biochem. Biophys, Res. Comm., 285, 728 (2001)<br></p>Formula:C7HD4FO2Color and Shape:NeatMolecular weight:144.14tert-Butyl (3-(4,4,5,5-Tetramethyl-1,3,2-dioxaborolan-2-yl)cyclohex-3-en-1-yl)carbamate
CAS:Controlled ProductFormula:C17H30BNO4Color and Shape:NeatMolecular weight:323.24n-Pentyl-d11 chloroformate
CAS:Controlled Product<p>Applications n-Pentyl-d11 chloroformate is labelled n-Pentyl chloroformate which can be used to synthesize 1,3-disubstituted ureas as potent inhibitors of the soluble epoxide hydrolase.<br>References Kim, I., et al.: J. Med. Chem., 47, 2110 (2004); Hammock, B., et al.: PCT Int. Appl. (2006), WO 2006045119 A2 20060427.<br></p>Formula:C6D11ClO2Color and Shape:NeatMolecular weight:161.674-Pyridin-2,3,5,6-d4-ol-d
CAS:Controlled Product<p>Applications 4-Pyridin-2,3,5,6-d4-ol-d is one of the azepanone derivatives studies as CGRP receptor antagonists.<br>References Liu, J.: PCT Int. Appl. (2010), WO 2010108103 A1 20100923.<br></p>Formula:C5D5NOColor and Shape:NeatMolecular weight:100.13n-Propyl-2,2,3,3,3-d5-amine Hydrochloride
CAS:Controlled Product<p>Applications n-Propyl-2,2,3,3,3-d5-amine Hydrochloride is the hydrochloride salt of 1-Propyl-d5-amine (P833702); the isotope labelled analog of 1-Propylamine (P833700) which is used in the synthesis of pyrimidine derivatives as novel and highly potent PDE4 inhibitors. It is also used in the preparation of fluorenone analogs with DNA topisomerase I inhibitors.<br>References Goto, T. et al.: Bioorg. Med. Chem., 21, 7025 (2013); Lee, C. et al.: Bioorg. Med. Chem. 21, 7125, (2013)<br></p>Formula:C3H5D5ClNColor and Shape:NeatMolecular weight:100.6tert-Butyl 4-Bromo-2-(1H-pyrrolo[2,3-b]pyridin-5-yloxy)benzoate
CAS:Controlled ProductFormula:C18H17BrN2O3Color and Shape:NeatMolecular weight:389.24GW4869 TFA Salt (~90%, ~10% inorganics)
CAS:Controlled Product<p>Applications GW4869 is a selective inhibitor of N-SMase.<br>References Lallemand, T., et al.: Arterioscler. Thromb. Vasc. Biol., 38, 1479 (2018); Figuera-Losada, M., et al.: PLoS One, 10, 0124481 (2015)<br></p>Formula:C30H28N6O2·xC2HF3O2Color and Shape:NeatMolecular weight:504.58 + x(114.02)N-Fmoc-glycine-d2
CAS:Controlled Product<p>Applications Isotope labelled N-Fmoc-glycine is an N-Fmoc-protected form of Glycine (G615990). Glycine is a nonessential amino acid that acts as an inhibitory neyrotransmitter in the vertebrate central nervous system. Glycine also posesses cytoprotective against oxidant damage in the kidney.<br>References Eulenberg, V., et al.: Trend. Biochem. Sci., 30, 325 (2005); Gundersen, R., et al.: Acta Anaesth. Scand., 49, 1108 (2005); Lockart, R. & Eagle, H.: Science, 129, 252 (1959); Sogabe, K., et al.: Kidn. Int., 50, 845 (1996)<br></p>Formula:C17H13D2NO4Color and Shape:NeatMolecular weight:299.32Ethyl Palmitate-d31
CAS:Controlled Product<p>Applications A labelled fatty acid found in Amaranth oil; it shows inhibitory activity.<br>References Fidler, N., et al.: J. Lipid Res., 41, 1376 (2000), Yang, T., et al.: Food Chem., 80, 473 (2003), Gamel, T., et al.: J. Food Lipids, 14, 323 (2007),<br></p>Formula:C18H5D31O2Color and Shape:NeatMolecular weight:315.671-Propyl-d5-amine
CAS:Controlled Product<p>Applications 1-Propyl-d5-amine is labelled 1-Propylamine (P833700) which is used in the synthesis of pyrimidine derivatives as novel and highly potent PDE4 inhibitors. It is also used in the preparation of fluorenone analogs with DNA topisomerase I inhibitors.<br> Not a dangerous good if item is equal to or less than 1g/ml and there is less than 100g/ml in the package<br></p>Formula:C3H4D5NColor and Shape:NeatMolecular weight:64.14(3R,5S,6E)-7-(2-Cyclopropyl-4-phenyl-3-quinolinyl)-3,5-dihydroxy-6-heptenoic Acid Sodium Salt
CAS:Controlled Product<p>Stability Hygroscopic<br>Applications (3R,5S,6E)-7-(2-cyclopropyl-4-phenyl-3-quinolinyl)-3,5-dihydroxy-6-heptenoic Acid Sodium Salt is an impurity of Pitavastatin (P531000), a HMG CoA reductase inhibitor and an antilipemic agent.<br>References Suzukim M., et al.: Bioorg. Med. Chem., 9, 2977 (1999); Yen, H., et al.: J. Clin. Invest., 98, 1253 (1996); Zou, Y., et al.: J. Biol. Chem., 274, 9760 (1999); Sun, X., et al.: Cancer Res., et al.: 61, 3382 (2001); Ladas, E.J., et al.: Clin. Oncol., 22, 517 (2004);<br></p>Formula:C25H24NNaO4Color and Shape:NeatMolecular weight:425.45rac-1,2-Dioctanoyl-3-Chloropropanediol
CAS:Controlled Product<p>Stability Moisture Sensitive<br>Applications rac-1,2-Dioctanoyl-3-Chloropropanediol was studied for its ability to act as an inhibitor of protein kinase C.<br>References Briggs, Josie C., et al.: Carbohydrate Res., 234, 23-35 (1992)<br></p>Formula:C19H35ClO4Color and Shape:NeatMolecular weight:362.93N-(n-Butyl)phosphoric Triamide
CAS:<p>Applications N-Alkyl phosphoric triamide useful as urease inhibitors.<br></p>Formula:C4H14N3OPColor and Shape:White SolidMolecular weight:151.153-Amino-N-(Tertbutylbenzenesulfonamide
CAS:Controlled Product<p>Applications 3-Amino-N-(Tert-Butyl)Benzenesulfonamide (cas# 608523-94-0) is a useful research chemical.<br></p>Formula:C10H16N2O2SColor and Shape:NeatMolecular weight:228.31(E)-a-Hydroxy Tamoxifen
CAS:Controlled Product<p>Applications A metabolite of the chemotherapeutic drug Tamoxifen (T006000). Exhibits a more potent estrogen agonist/antagonist activity than the parent drug. Also active as an intramembranous inhibitor of lipid peroxidation.<br>References Kupfer, D., et al.: Cancer Res., 54, 3140 (1994), Custodio, J.B.A., et al.: Biochem. Pharmacol., 47, 1989 (1994),<br></p>Formula:C26H29NO2Color and Shape:NeatMolecular weight:387.51Valtrate
CAS:Controlled Product<p>Applications Valtrate is a Rev-transport inhibitor with anti-HIV activity from Valerianae Radix.<br>References Murakami, N., et al.: Bioorg. Med. Chem. Lett., 12, 2807 (2002); Watanabe, K., et al.: Drug Discoveries Ther., 5, 26 92011)<br></p>Formula:C22H30O8Color and Shape:Light Brown To Dark YellowMolecular weight:422.47A 83-01
CAS:Controlled Product<p>Stability Moisture Sensitive<br>Applications A 83-01 is a selective inhibitor of TGF-β type I receptor. A 83-01 treatment increases tumor permeability.<br>References Minowa, T. et al.: British. J. Canc., 101, 1884 (2009)<br></p>Formula:C25H19N5SColor and Shape:Off-WhiteMolecular weight:421.52
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