EGFR
EGFR (epidermal growth factor receptor) inhibitors are compounds that block the signaling of EGFR, a receptor that is often overexpressed in various cancers and plays a critical role in angiogenesis. EGFR inhibitors are used to prevent tumor growth and metastasis by disrupting the pathways that promote blood vessel formation in tumors. These inhibitors are widely used in cancer research and therapy. At CymitQuimica, we offer a diverse selection of high-quality EGFR inhibitors to support your research in oncology and angiogenesis.
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PD-161570
CAS:192705-80-9
PD-161570 is a potent and ATP-competitive human FGF-1 receptor inhibitor with an IC50 of 39.9 …
Formula:
C26H35Cl2N7O
Purity:
99.23%
Color and Shape:
Solid
Molecular weight:
532.51
Ref: TM-T23127
| 1mg | 35.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 149.00 € | ||
| 25mg | 305.00 € | ||
| 50mg | 492.00 € | ||
| 100mg | 700.00 € | ||
| 200mg | 938.00 € | ||
| 1mL*10mM (DMSO) | 125.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Lazertinib
CAS:1903008-80-9
Lazertinib (GNS-1480) is a potent, selective, irreversible EGFR-TKI; IC50: 1.7-76 nM for various EGFR mutations.
Formula:
C30H34N8O3
Purity:
98.7% - 99.53%
Color and Shape:
Solid
Molecular weight:
554.64
Ref: TM-T4485
| 1mg | 48.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 150.00 € | ||
| 25mg | 240.00 € | ||
| 50mg | 325.00 € | ||
| 100mg | 472.00 € | ||
| 500mg | 1,093.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Tyrphostin A1
CAS:2826-26-8
Tyrphostin A1 (Tyrphostin 1) is an inhibitor of EGFR tyrosine kinase .
Formula:
C11H8N2O
Purity:
99.13%
Color and Shape:
Solid
Molecular weight:
184.19
Ref: TM-T7649
| 10mg | 35.00 € | ||
| 25mg | 58.00 € | ||
| 50mg | 84.00 € | ||
| 100mg | 97.00 € | ||
| 200mg | 140.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
WZ4002
CAS:1213269-23-8
WZ4002 is a mutant-selective EGFR inhibitor for EGFR(L858R) and EGFR(T790M) with IC50 of 2 nM/8 …
Formula:
C25H27ClN6O3
Purity:
98.12%
Color and Shape:
Solid
Molecular weight:
494.97
Ref: TM-T6238
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 73.00 € | ||
| 25mg | 117.00 € | ||
| 50mg | 187.00 € | ||
| 100mg | 329.00 € | ||
| 200mg | 490.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Brigatinib
CAS:1197953-54-0
Brigatinib (AP-26113) is a highly potent and selective ALK inhibitor.
Formula:
C29H39ClN7O2P
Purity:
100% - 99.93%
Color and Shape:
Solid
Molecular weight:
584.09
Ref: TM-T3621
| 2mg | 35.00 € | ||
| 5mg | 50.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 96.00 € | ||
| 50mg | 114.00 € | ||
| 100mg | 166.00 € | ||
| 200mg | 240.00 € | ||
| 500mg | 406.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
MAZ51
CAS:163655-37-6
MAZ51 is a VEGFR-3 (Flt-4) tyrosine kinase inhibitor.
Formula:
C21H18N2O
Purity:
98.53%
Color and Shape:
Solid
Molecular weight:
314.38
Ref: TM-T8496
| 1mg | 40.00 € | ||
| 2mg | 51.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 243.00 € | ||
| 50mg | 406.00 € | ||
| 100mg | 607.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Gefitinib-based PROTAC 3
CAS:2230821-27-7
Gefitinib-PROTAC 3 degrades EGFR in cancer cells; DC50s: 11.7 nM (HCC827) and 22.3 nM (H3255).
Formula:
C47H57ClFN7O8S
Purity:
97.29% - 98.25%
Color and Shape:
Solid
Molecular weight:
934.51
Ref: TM-T5437
| 2mg | 46.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 105.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 259.00 € | ||
| 100mg | 374.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Dacomitinib hydrate
CAS:1042385-75-0
Dacomitinib hydrate (PF 299804) is a highly selective and second-generation small-molecule inhibitor of the pan-epidermal …
Formula:
C24H27ClFN5O3
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
487.96
Ref: TM-T19965
| 5mg | 50.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 105.00 € | ||
| 50mg | 140.00 € | ||
| 100mg | 212.00 € | ||
| 200mg | 311.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Almonertinib
CAS:1899921-05-1
Almonertinib (HS-10296) is an inhibitor of EGFR activation mutation and tolerant mutation of EGFR T790M, …
Formula:
C30H35N7O2
Purity:
99.99%
Color and Shape:
Solid
Molecular weight:
525.64
Ref: TM-T5462
| 1mg | 89.00 € | ||
| 5mg | 197.00 € | ||
| 10mg | 311.00 € | ||
| 25mg | 525.00 € | ||
| 50mg | 757.00 € | ||
| 100mg | 1,035.00 € | ||
| 500mg | 2,110.00 € | ||
| 1mL*10mM (DMSO) | 249.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
G5-7
CAS:939681-36-4
G5-7 is an oral JAK2 inhibitor targeting EGFR/STAT3 phosphorylation with potential for glioma research.
Formula:
C22H19F2NO3
Purity:
97.30%
Color and Shape:
Solid
Molecular weight:
383.39
Ref: TM-T8742
| 1mg | 50.00 € | ||
| 5mg | 97.00 € | ||
| 10mg | 145.00 € | ||
| 25mg | 259.00 € | ||
| 50mg | 374.00 € | ||
| 100mg | 523.00 € | ||
| 200mg | 710.00 € | ||
| 1mL*10mM (DMSO) | 105.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
AG-494
CAS:133550-35-3
AG-494 (Tyrphostin B48) is an inhibitor of epidermal growth factor receptor kinase.
Formula:
C16H12N2O3
Purity:
98.69%
Color and Shape:
Solid
Molecular weight:
280.28
Ref: TM-T4205
| 10mg | 44.00 € | ||
| 25mg | 82.00 € | ||
| 50mg | 117.00 € | ||
| 100mg | 198.00 € | ||
| 200mg | 283.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Neratinib
CAS:698387-09-6
Neratinib (HKI-272) (HKI-272) is an orally available, irreversible tyrosine kinase inhibitor for HER2 and EGFR …
Formula:
C30H29ClN6O3
Purity:
100% - 98.55%
Color and Shape:
Solid
Molecular weight:
557.04
Ref: TM-T2325
| 5mg | 35.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 93.00 € | ||
| 100mg | 124.00 € | ||
| 200mg | 187.00 € | ||
| 500mg | 311.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Osimertinib mesylate
CAS:1421373-66-1
Osimertinib mesylate (AZD-9291 mesylate) is an EGFR third-generation inhibitor. Osimertinib mesylate has antitumor activity. Cost-effective …
Formula:
C29H37N7O5S
Purity:
100% - 99.88%
Color and Shape:
Solid
Molecular weight:
595.71
Ref: TM-T3634
| 1g | 153.00 € | ||
| 5mg | 49.00 € | ||
| 10mg | 60.00 € | ||
| 50mg | 88.00 € | ||
| 100mg | 96.00 € | ||
| 200mg | 113.00 € | ||
| 500mg | 131.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
RG13022
CAS:136831-48-6
RG13022 (Tyrphostin RG13022) is a tyrosine kinase inhibitor; inhibits the autophosphorylation reaction of the EGF …
Formula:
C16H14N2O2
Purity:
98.38%
Color and Shape:
Solid
Molecular weight:
266.29
Ref: TM-T3545
| 2mg | 47.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 88.00 € | ||
| 25mg | 180.00 € | ||
| 50mg | 304.00 € | ||
| 100mg | 480.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
RG14620
CAS:136831-49-7
RG14620 (Tyrphostin RG14620) is an epidermal growth factor receptor (EGFR) inhibitor.
Formula:
C14H8Cl2N2
Purity:
99.56% - 99.79%
Color and Shape:
Solid
Molecular weight:
275.13
Ref: TM-T3554
| 2mg | 35.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 77.00 € | ||
| 25mg | 137.00 € | ||
| 50mg | 259.00 € | ||
| 100mg | 432.00 € | ||
| 500mg | 938.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Allitinib tosylate
CAS:1050500-29-2
Allitinib tosylate (AST-1306) is a novel irreversible inhibitor of EGFR and ErbB2 with IC50 of …
Formula:
C31H26ClFN4O5S
Purity:
98.46% - 98.68%
Color and Shape:
Solid
Molecular weight:
621.08
Ref: TM-T6331
| 1mg | 52.00 € | ||
| 5mg | 111.00 € | ||
| 10mg | 175.00 € | ||
| 25mg | 329.00 € | ||
| 50mg | 494.00 € | ||
| 100mg | 700.00 € | ||
| 1mL*10mM (DMSO) | 155.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
(S)-Sunvozertinib
CAS:2370013-49-1
(S)-Sunvozertinib (DZD9008) is a rationally designed selective, irreversible EGFR/HER2 inhibitor.
Formula:
C29H35ClFN7O3
Purity:
99.64%
Color and Shape:
Solid
Molecular weight:
584.08
Ref: TM-T9304
| 1mg | 63.00 € | ||
| 5mg | 137.00 € | ||
| 10mg | 210.00 € | ||
| 25mg | 424.00 € | ||
| 50mg | 627.00 € | ||
| 100mg | 893.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
BI-4020
CAS:2664214-60-0
BI-4020 is a fourth-generation, orally active, and non-covalent inhibitor of EGFR tyrosine kinase.
Formula:
C30H38N8O2
Purity:
100.00% - 98.44%
Color and Shape:
Solid
Molecular weight:
542.68
Ref: TM-T10534
| 1mg | 170.00 € | ||
| 5mg | 398.00 € | ||
| 10mg | 568.00 € | ||
| 25mg | 848.00 € | ||
| 50mg | 1,130.00 € | ||
| 100mg | 1,510.00 € | ||
| 200mg | 2,062.00 € | ||
| 1mL*10mM (DMSO) | 472.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Avitinib
CAS:1557267-42-1
Avitinib (AC0010), also known as AC0010 or AC0010MA, is an orally available, irreversible, epidermal growth …
Formula:
C26H26FN7O2
Purity:
100%
Color and Shape:
Solid
Molecular weight:
487.53
Ref: TM-T3024
| 2mg | 48.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 216.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 522.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
Avitinib maleate
CAS:1557268-88-8
Avitinib maleate is a pyrrolopyrimidine-based irreversible epidermal growth factor receptor (EGFR) inhibitor.
Formula:
C30H30FN7O6
Purity:
98% - 99.74%
Color and Shape:
Solid
Molecular weight:
603.61
Ref: TM-T3721
| 5mg | 73.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 208.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 567.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Thursday 3 Apr 2025
