EGFR
EGFR (epidermal growth factor receptor) inhibitors are compounds that block the signaling of EGFR, a receptor that is often overexpressed in various cancers and plays a critical role in angiogenesis. EGFR inhibitors are used to prevent tumor growth and metastasis by disrupting the pathways that promote blood vessel formation in tumors. These inhibitors are widely used in cancer research and therapy. At CymitQuimica, we offer a diverse selection of high-quality EGFR inhibitors to support your research in oncology and angiogenesis.
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WZ8040
CAS:1214265-57-2
WZ8040 is a novel mutant-selective irreversible EGFRT790M inhibitor, does not inhibit ERBB2 phosphorylation (T798I).
Formula:
C24H25ClN6OS
Purity:
97.42%
Color and Shape:
Solid
Molecular weight:
481.01
Ref: TM-T6734
| 1mg | 48.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 150.00 € | ||
| 25mg | 246.00 € | ||
| 50mg | 365.00 € | ||
| 100mg | 538.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
ZM39923 hydrochloride
CAS:1021868-92-7
ZM39923 hydrochloride (JAK3 Inhibitor IV) is an JAK1/3 inhibitor, almost no activity to JAK2 and …
Formula:
C23H25NO·HCl
Purity:
98.05%
Color and Shape:
Solid
Molecular weight:
367.91
Ref: TM-T6145
| 5mg | 59.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 310.00 € | ||
| 100mg | 464.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
SU5214
CAS:186611-04-1
SU5214 is a modulator of tyrosine kinase signal transduction.
Formula:
C16H13NO2
Purity:
99.52% - 99.55%
Color and Shape:
Solid
Molecular weight:
251.28
Ref: TM-T3569
| 5mg | 39.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 111.00 € | ||
| 50mg | 170.00 € | ||
| 100mg | 279.00 € | ||
| 200mg | 405.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
Canertinib dihydrochloride
CAS:289499-45-2
Canertinib dihydrochloride (PD-183805 dihydrochloride) is the hydrochloride salt of an orally bio-available quinazoline with potential …
Formula:
C24H27Cl3FN5O3
Purity:
99.23%
Color and Shape:
Solid
Molecular weight:
558.86
Ref: TM-T2501
| 10mg | 35.00 € | ||
| 25mg | 42.00 € | ||
| 50mg | 49.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
Chrysophanol
CAS:481-74-3
Chrysophanol (Turkey Rhubarb) is an EGFR/mTOR pathway inhibitor, which can be found in rhubarb, and …
Formula:
C15H10O4
Purity:
97.91% - 99.7%
Color and Shape:
Physical Description Golden Yellow Plates Or Brown Powder Melting Point 196°C
Molecular weight:
254.24
Ref: TM-T2995
| 50mg | 38.00 € | ||
| 100mg | 52.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
AG490
CAS:133550-30-8
AG490 inhibits EGFR (0.1 μM IC50), 135x >selective than ErbB2, blocks JAK2, spares Lyn, Lck, …
Formula:
C17H14N2O3
Purity:
98.6% - 99.7%
Color and Shape:
Yellow Solid
Molecular weight:
294.3
Ref: TM-T2600
| 10mg | 50.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 87.00 € | ||
| 100mg | 97.00 € | ||
| 200mg | 160.00 € | ||
| 500mg | 283.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
SYR127063
CAS:871026-18-5
SYR127063 (BDBM-92454) (BDBM92454) is a potent and selective HER2 inhibitor, binds to HER2 in a …
Formula:
C23H20ClF3N4O3
Purity:
98.57%
Color and Shape:
Solid
Molecular weight:
492.88
Ref: TM-T34760
| 1mg | 131.00 € | ||
| 5mg | 286.00 € | ||
| 10mg | 430.00 € | ||
| 25mg | 710.00 € | ||
| 50mg | 998.00 € | ||
| 1mL*10mM (DMSO) | 354.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
AZD8931 diFuMaric acid
CAS:1196531-39-1
AZD8931 is a reversible and ATP competitive inhibitor of EGFR, ErbB2 and ErbB3 (IC50 of …
Formula:
C31H33ClFN5O11
Purity:
99%
Color and Shape:
Solid
Molecular weight:
706.1
Ref: TM-T8751
| 1mg | 88.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 259.00 € | ||
| 25mg | 425.00 € | ||
| 50mg | 598.00 € | ||
| 100mg | 810.00 € | ||
| 200mg | 1,074.00 € | ||
| 1mL*10mM (DMSO) | 255.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
CP-724714
CAS:383432-38-0
CP-724714 (CP724714) is an effective and selective HER2/ErbB2 inhibitor (IC50: 10 nM), >640-fold selectivity against …
Formula:
C27H27N5O3
Purity:
97.10% - 98.82%
Color and Shape:
Solid
Molecular weight:
469.54
Ref: TM-T4014
| 1mg | 44.00 € | ||
| 2mg | 58.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 273.00 € | ||
| 50mg | 454.00 € | ||
| 100mg | 660.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
PF-6274484
CAS:1035638-91-5
PF-6274484 is an EGFR inhibitor with Ki values of 0.14 and 0.18 nM for EGFR-L858R/T790M …
Formula:
C18H14ClFN4O2
Purity:
97.71%
Color and Shape:
Solid
Molecular weight:
372.78
Ref: TM-T22396
| 2mg | 40.00 € | ||
| 5mg | 60.00 € | ||
| 10mg | 92.00 € | ||
| 25mg | 187.00 € | ||
| 50mg | 350.00 € | ||
| 100mg | 522.00 € | ||
| 500mg | 1,130.00 € | ||
| 1mL*10mM (DMSO) | 66.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
WS3
CAS:1421227-52-2
WS3, a β cell proliferation inducer, regulates Erb3 binding protein-1 (EBP1) and the IκB kinase …
Formula:
C28H30F3N7O3
Purity:
97.93% - 98.81%
Color and Shape:
Solid
Molecular weight:
569.58
Ref: TM-T2055
| 5mg | 52.00 € | ||
| 10mg | 77.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 213.00 € | ||
| 100mg | 394.00 € | ||
| 1mL*10mM (DMSO) | 70.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
CL-387785
CAS:194423-06-8
CL-387785 is an irreversible EGFR inhibitor with IC50 of 370 pM; overcomes T790M mutation resistance.
Formula:
C18H13BrN4O
Purity:
96.68% - 98.09%
Color and Shape:
Solid
Molecular weight:
381.23
Ref: TM-T2245
| 5mg | 39.00 € | ||
| 10mg | 58.00 € | ||
| 25mg | 105.00 € | ||
| 50mg | 169.00 € | ||
| 100mg | 264.00 € | ||
| 200mg | 373.00 € | ||
| 1mL*10mM (DMSO) | 44.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
Tyrphostin B44, (+) enantiomer
CAS:133550-37-5
Tyrphostin B44, (+) enantiomer is an inhibitor of epidermal growth factor receptor (EGFR) kinase with …
Formula:
C18H16N2O3
Purity:
97.18%
Color and Shape:
Solid
Molecular weight:
308.33
Ref: TM-T22450
| 1mg | 51.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 105.00 € | ||
| 10mg | 164.00 € | ||
| 25mg | 275.00 € | ||
| 50mg | 378.00 € | ||
| 100mg | 543.00 € | ||
| 200mg | 738.00 € | ||
| 1mL*10mM (DMSO) | 117.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
lavendustin C
CAS:125697-93-0
lavendustin C (NSC 666251) is a potent inhibitor of epidermal growth factor (EGF) receptor-associated tyrosine …
Formula:
C14H13NO5
Purity:
97.77%
Color and Shape:
Yellow To Tan Powder
Molecular weight:
275.26
Ref: TM-T4185
| 1mg | 44.00 € | ||
| 2mg | 58.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 160.00 € | ||
| 25mg | 349.00 € | ||
| 50mg | 518.00 € | ||
| 100mg | 747.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
Canertinib
CAS:267243-28-7
Canertinib (CI-1033), a pan-erbB inhibitor, effectively targets esophageal cancer in vitro/vivo, altering metabolism and reducing …
Formula:
C24H25ClFN5O3
Purity:
100% - 99.18%
Color and Shape:
White Or Similar To White Crystalline Powder
Molecular weight:
485.94
Ref: TM-T6136
| 5mg | 37.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 70.00 € | ||
| 50mg | 87.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
AG-1557 hydrochloride (189290-58-2(free base))
AG-1557 hydrochloride is an inhibitor of the epidermal growth factor receptor (EGFR) tyrosine kinase (pIC50: …
Formula:
C16H15ClIN3O2
Purity:
98.95%
Color and Shape:
Solid
Molecular weight:
443.66
Ref: TM-T4694
| 5mg | 35.00 € | ||
| 10mg | 50.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 155.00 € | ||
| 100mg | 269.00 € | ||
| 200mg | 394.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
Tyrphostin AG 879
CAS:148741-30-4
Tyrphostin AG 879 (AG 879) effectively inhibits HER2/ErbB2 (IC50: 1 μM), 100- and 500-fold higher …
Formula:
C18H24N2OS
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
316.46
Ref: TM-T6712
| 5mg | 50.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 156.00 € | ||
| 50mg | 250.00 € | ||
| 100mg | 427.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
Daphnetin
CAS:486-35-1
Daphnetin (7,8-Dihydroxycoumarin), a natural coumarin derivative, is a protein kinase inhibitor with inhibitory for EGFR …
Formula:
C9H6O4
Purity:
98.33% - 99.82%
Color and Shape:
Solid
Molecular weight:
178.14
Ref: TM-T2851
| 10mg | 50.00 € | ||
| 25mg | 95.00 € | ||
| 50mg | 166.00 € | ||
| 100mg | 244.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
NS309
CAS:18711-16-5
NS309 activates SK/KCa2, IK/KCa3.1 (0.12-1.2 μM EC50, 10-90 nM EC50), and Kv11.1 channels; doesn't affect …
Formula:
C8H4Cl2N2O2
Purity:
95.87%
Color and Shape:
Solid
Molecular weight:
231.04
Ref: TM-T4612
| 5mg | 57.00 € | ||
| 10mg | 69.00 € | ||
| 25mg | 119.00 € | ||
| 50mg | 216.00 € | ||
| 100mg | 323.00 € | ||
| 200mg | 470.00 € | ||
| 500mg | 752.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
Cetuximab
CAS:205923-56-4
Cetuximab (C225) is a monoclonal antibody that is an inhibitor of human epidermal growth factor …
Formula:
C107H179N35O36S7
Purity:
100.00% - SDS-PAGE:98.4%；SEC-HPLC: 99.7%
Color and Shape:
Liquid
Molecular weight:
152 kDa
Ref: TM-T9905
| 1mg | 187.00 € | ||
| 2mg | 274.00 € | ||
| 5mg | 457.00 € | ||
| 10mg | 662.00 € | ||
| 25mg | 1,035.00 € | ||
| 50mg | 1,396.00 € | ||
| 100mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 11 Mar 2025
