Chromatin/Epigenetics
Chromatin/epigenetics inhibitors are compounds that modulate the structure and function of chromatin or interfere with epigenetic modifications, such as DNA methylation and histone modification. These inhibitors are essential tools for studying gene expression regulation and the role of epigenetics in diseases like cancer, neurological disorders, and developmental abnormalities. By targeting epigenetic processes, these inhibitors can alter gene expression patterns and offer new therapeutic avenues. At CymitQuimica, we provide a wide selection of high-quality chromatin/epigenetics inhibitors to support your research in molecular biology, genetics, and epigenetics.
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Subcategories of "Chromatin/Epigenetics"
Products of "Chromatin/Epigenetics"
SP-96
CAS:2682114-54-9
SP-96: Aurora B inhibitor, IC50=0.316 nM, selectively hinders MDA-MD-468 growth, GI50=107 nM, for triple-negative breast …
Formula:
C25H20FN7O
Purity:
99.52%
Color and Shape:
Solid
Molecular weight:
453.47
Ref: TM-T41256
| 1mg | 47.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 151.00 € | ||
| 25mg | 285.00 € | ||
| 50mg | 414.00 € | ||
| 100mg | 582.00 € | ||
| 200mg | 784.00 € | ||
| 1mL*10mM (DMSO) | 103.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
BRM/BRG1 ATP Inhibitor-2
CAS:2368900-77-8
BRM/BRG1 ATP Inhibitor-2 is an inhibitor of BRG1/BRM ATPase and can be used in studies …
Formula:
C20H20N4O2S2
Purity:
99.88%
Color and Shape:
Solid
Molecular weight:
412.53
Ref: TM-T60032
| 1mg | 39.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 126.00 € | ||
| 25mg | 246.00 € | ||
| 50mg | 362.00 € | ||
| 100mg | 516.00 € | ||
| 200mg | 699.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
PROTAC BET Degrader-1
CAS:2093386-22-0
PROTAC BET Degrader-1 is a potent degrader of BET based on PROTAC.
Formula:
C44H45N11O9
Purity:
98%
Color and Shape:
Solid
Molecular weight:
871.9
Ref: TM-T13849
| 5mg | 431.00 € | ||
| 10mg | 658.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | To inquire | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 469.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
Tulmimetostat
CAS:2567686-02-4
Tulmimetostat (CPI-0209) is an orally active EZH1/EZH2 inhibitor.Tulmimetostat has antitumor activity and is used in …
Formula:
C28H36ClN3O5S
Purity:
98.04%
Color and Shape:
Solid
Molecular weight:
562.12
Ref: TM-T40199
| 1mg | 36.00 € | ||
| 5mg | 68.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 180.00 € | ||
| 50mg | 270.00 € | ||
| 100mg | 532.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
EZH2-IN-15
CAS:2098545-98-1
A compound inhibits EZH2, overexpressed in cancers, affecting Treg activity and innate immunity.
Formula:
C32H44N4O4
Purity:
98.85%
Color and Shape:
Liquid
Molecular weight:
548.72
Ref: TM-T67883
| 1mg | 154.00 € | ||
| 5mg | 339.00 € | ||
| 10mg | 515.00 € | ||
| 25mg | 816.00 € | ||
| 50mg | 1,103.00 € | ||
| 100mg | 1,476.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
KDM2B-IN-2
CAS:1965248-01-4
KDM2B-IN-2 is a potent histone demethylase (kdm2b) inhibitor.
Formula:
C21H26N4O2S2
Purity:
97.57%
Color and Shape:
Solid
Molecular weight:
430.59
Ref: TM-T39389
| 1mg | 65.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 398.00 € | ||
| 50mg | 597.00 € | ||
| 100mg | 829.00 € | ||
| 500mg | 1,698.00 € | ||
| 1mL*10mM (DMSO) | 158.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
DC-S239
CAS:303141-21-1
Ethyl 2-amino-4-methyl-5-thiophene carboxylate is a SETD7 inhibitor (IC50=4.59μM) with anticancer properties.
Formula:
C15H15N3O5S
Purity:
99.36%
Color and Shape:
Liquid
Molecular weight:
349.36
Ref: TM-T60002
| 1mg | 62.00 € | ||
| 5mg | 141.00 € | ||
| 10mg | 218.00 € | ||
| 25mg | 365.00 € | ||
| 50mg | 519.00 € | ||
| 100mg | 703.00 € | ||
| 200mg | 903.00 € | ||
| 1mL*10mM (DMSO) | 147.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
TCIP 1
TCIP 1 is a small molecule in the category of transcriptional/epigenetic covalent inhibitor probes (TCIPs) …
Formula:
C50H58Cl2N12O6S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1026.04
Ref: TM-T79801
| 25mg | 2,275.00 € | ||
| 50mg | 2,990.00 € | ||
| 100mg | 4,043.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
LSD1-IN-24
CAS:4734-59-2
LSD1-IN-24 is a selective and potent LSD1 inhibitor with an IC50 value of 0.247 μM.LSD1-IN-24 …
Formula:
C18H20N2OS
Purity:
99.53%
Color and Shape:
Soild
Molecular weight:
312.43
Ref: TM-T67871
| 1mg | 79.00 € | ||
| 5mg | 173.00 € | ||
| 10mg | 270.00 € | ||
| 25mg | 540.00 € | ||
| 50mg | 865.00 € | ||
| 100mg | 1,150.00 € | ||
| 500mg | 2,327.00 € | ||
| 1mL*10mM (DMSO) | 184.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
PROTAC BRD9 Degrader-1
CAS:2097971-01-0
PROTAC BRD9 Degrader-1 is a lead PROTAC BRD9 chemical degrader with IC50 of 13.5 nM.
Formula:
C42H45N7O12S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
903.98
Ref: TM-T12560
| 5mg | 692.00 € | ||
| 10mg | 1,151.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
JQAD1
CAS:2417097-18-6
JQAD1, a potent EP300 degrader (DC50≤31.6 nM), induces apoptosis, suppresses tumor growth, and selectively downregulates …
Formula:
C48H52F4N6O9
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
932.95
Ref: TM-T41180
| 1mg | 126.00 € | ||
| 5mg | 305.00 € | ||
| 10mg | 463.00 € | ||
| 25mg | 754.00 € | ||
| 50mg | 1,049.00 € | ||
| 100mg | 1,417.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
PROTAC BRD4 Degrader-3
CAS:2313234-00-1
PROTAC BRD4 Degrader-3 is an efficacious degrader of PROTAC BRD4.
Formula:
C55H65F2N9O9S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1098.3
Ref: TM-T13835
| 100mg | To inquire | ||
| 500mg | To inquire |
Estimated delivery in United States, on Wednesday 6 Nov 2024
UNC 0631
CAS:1320288-19-4
UNC 0631 is a effectvie histone methyltransferase G9a inhibitor (IC50=4 nM).
Formula:
C37H61N7O2
Purity:
98.76%
Color and Shape:
Solid
Molecular weight:
635.93
Ref: TM-T2354
| 1mg | 49.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 150.00 € | ||
| 25mg | 291.00 € | ||
| 50mg | 459.00 € | ||
| 100mg | 668.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
JAK2-IN-6
CAS:353512-04-6
JAK2-IN-6: A potent JAK2-specific inhibitor (IC50=22.86μg/mL), blocks JAK2 signaling, has anticancer properties, and is inactive …
Formula:
C14H10ClN3OS2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
335.83
Ref: TM-T40443
| 1mg | 46.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 204.00 € | ||
| 50mg | 305.00 € | ||
| 100mg | 454.00 € | ||
| 500mg | 985.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
LSD1-IN-30
CAS:1289575-45-6
LSD1-IN-30 is a lysine-specific demethylase 1 (LSD1) inhibitor with anticancer activity for the study of …
Formula:
C15H14N2O3
Purity:
98.42%
Color and Shape:
Soild
Molecular weight:
270.28
Ref: TM-T83966
| 1mg | 115.00 € | ||
| 5mg | 278.00 € | ||
| 10mg | 444.00 € | ||
| 25mg | 891.00 € | ||
| 50mg | 1,430.00 € | ||
| 100mg | 2,290.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
HIF-1α-IN-2 hydrochloride
HIF-1α-IN-2 hydrochloride is a potent HIF-1α inhibitor exhibiting anticancer activity, demonstrated by IC50 values of …
Formula:
C21H20ClN3OS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
397.92
Ref: TM-T78123
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 6 Nov 2024
PARP-1/2-IN-2
PARP-1/2-IN-2-IN-1 (Compound 12e) effectively inhibits PARP1/2 and CDK12 with IC 50 values of 34 nM, …
Formula:
C25H23IN8O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
610.41
Ref: TM-T78787
| 5mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Wednesday 6 Nov 2024
GNE-987
CAS:2417371-71-0
GNE-987 is a potent chimeric BET degrader, binding BRD4 BD1/BD2 at IC50: 4.7/4.4 nM & …
Formula:
C56H67F2N9O8S2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
1096.31
Ref: TM-T11441
| 1mg | 467.00 € | ||
| 5mg | 1,057.00 € | ||
| 10mg | 1,680.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
Dihydro-5-azacytidine
CAS:62488-57-7
Dihydro-5-azacytidine (DHAC) is a nucleoside analog that interrupts DNA methylation by integrating into DNA. It …
Formula:
C8H14N4O5
Purity:
100%
Color and Shape:
Solid
Molecular weight:
246.22
Ref: TM-T40713
| 25mg | 1,422.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
RBN-3143
CAS:2360853-16-1
RBN-3143: potent PARP14 inhibitor (IC50= 4 nM), blocks ADP-ribosylation, may treat lung inflammation.
Formula:
C22H28FN3O4S
Purity:
98.64%
Color and Shape:
Soild
Molecular weight:
449.54
Ref: TM-T67844
| 1mg | 94.00 € | ||
| 5mg | 199.00 € | ||
| 10mg | 291.00 € | ||
| 25mg | 495.00 € | ||
| 50mg | 713.00 € | ||
| 100mg | 1,003.00 € | ||
| 500mg | 2,014.00 € | ||
| 1mL*10mM (DMSO) | 221.00 € |
Estimated delivery in United States, on Wednesday 6 Nov 2024
