Chromatin/Epigenetics
Chromatin/epigenetics inhibitors are compounds that modulate the structure and function of chromatin or interfere with epigenetic modifications, such as DNA methylation and histone modification. These inhibitors are essential tools for studying gene expression regulation and the role of epigenetics in diseases like cancer, neurological disorders, and developmental abnormalities. By targeting epigenetic processes, these inhibitors can alter gene expression patterns and offer new therapeutic avenues. At CymitQuimica, we provide a wide selection of high-quality chromatin/epigenetics inhibitors to support your research in molecular biology, genetics, and epigenetics.
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Subcategories of "Chromatin/Epigenetics"
Products of "Chromatin/Epigenetics"
A1874
CAS:2064292-12-0
A1874 is a nutlin-based and BRD4-degrading PROTAC which induces BRD4 degradation in cells. Effective in …
Formula:
C58H62Cl3F2N9O7S
Purity:
≥95%
Color and Shape:
Solid
Molecular weight:
1173.59
Ref: TM-T5442
| 1mg | 212.00 € | ||
| 2mg | 296.00 € | ||
| 5mg | 453.00 € | ||
| 10mg | 644.00 € | ||
| 25mg | 1,016.00 € | ||
| 50mg | 1,374.00 € | ||
| 100mg | 1,850.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
M1001
CAS:874590-32-6
M1001 is a HIF-2α agonist.
Formula:
C17H17N3O2S
Purity:
98.83%
Color and Shape:
Solid
Molecular weight:
327.4
Ref: TM-T7802
| 1mg | 38.00 € | ||
| 5mg | 82.00 € | ||
| 10mg | 122.00 € | ||
| 25mg | 219.00 € | ||
| 50mg | 326.00 € | ||
| 100mg | 451.00 € | ||
| 200mg | 627.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
Cucurbitacin I
CAS:2222-07-3
Cucurbitacin I (JSI-124), a natural compound, is a selective inhibitor of JAK2/STAT3 with anti-cancer activity.
Formula:
C30H42O7
Purity:
96.69% - 98.2%
Color and Shape:
Solid
Molecular weight:
514.65
Ref: TM-TQ0196
| 1mg | 83.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 222.00 € | ||
| 25mg | 367.00 € | ||
| 50mg | 546.00 € | ||
| 1mL*10mM (DMSO) | 184.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
BRD4 Inhibitor-24
CAS:309951-18-6
BRD4 Inhibitor-24 is a BRD4 small molecule inhibitor with antitumor activity.
Formula:
C13H14N2O4
Purity:
98.65%
Color and Shape:
Solid
Molecular weight:
262.26
Ref: TM-T9629
| 5mg | 44.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 113.00 € | ||
| 50mg | 181.00 € | ||
| 100mg | 297.00 € | ||
| 200mg | 423.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
CBP/EP300-IN-1
CAS:2443789-32-8
CBP/EP300-IN-1 is a CBP/EP300 bromodomain inhibitor.
Formula:
C23H23FN2O5
Purity:
99.05%
Color and Shape:
Solid
Molecular weight:
426.44
Ref: TM-T7264
| 1mg | 47.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 155.00 € | ||
| 25mg | 255.00 € | ||
| 50mg | 360.00 € | ||
| 100mg | 511.00 € | ||
| 200mg | 696.00 € | ||
| 1mL*10mM (DMSO) | 102.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
Ruxolitinib phosphate
CAS:1092939-17-7
Ruxolitinib phosphate (INCB18424 phosphate) is a JAK1/2 inhibitor with IC50 of 3.3 nM/2.8 nM. Cost-effective …
Formula:
C17H21N6O4P
Purity:
100% - 99.91%
Color and Shape:
Solid
Molecular weight:
404.36
Ref: TM-T3043
| 1g | 604.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 81.00 € | ||
| 50mg | 95.00 € | ||
| 100mg | 144.00 € | ||
| 200mg | 223.00 € | ||
| 500mg | 408.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
(+)-JQ-1
CAS:1268524-70-4
(+)-JQ-1 (JQ1) is a BET bromine domain inhibitor that inhibits BRD4 (1/2) (IC50=77/33 nM) with …
Formula:
C23H25ClN4O2S
Purity:
97.57% - ≥95%
Color and Shape:
Solid
Molecular weight:
456.99
Ref: TM-T2110
| 1mg | 36.00 € | ||
| 2mg | 44.00 € | ||
| 5mg | 59.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 94.00 € | ||
| 50mg | 142.00 € | ||
| 100mg | 185.00 € | ||
| 200mg | 282.00 € | ||
| 500mg | 504.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
AZD-2461
CAS:1174043-16-3
AZD2461 is a novel PARP inhibitor.
Formula:
C22H22FN3O3
Purity:
98% - 99.25%
Color and Shape:
Solid
Molecular weight:
395.43
Ref: TM-T2484
| 2mg | 38.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 97.00 € | ||
| 50mg | 122.00 € | ||
| 100mg | 193.00 € | ||
| 1mL*10mM (DMSO) | 58.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
Cycloastragenol
CAS:78574-94-4
Cycloastragenol, a saponin from Astragalus, could be a new depression treatment.
Formula:
C30H50O5
Purity:
99.92% - 99.98%
Color and Shape:
Solid
Molecular weight:
490.71
Ref: TM-T5575
| 5mg | 46.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 87.00 € | ||
| 50mg | 115.00 € | ||
| 100mg | 170.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
dBET6
CAS:1950634-92-0
dBET6 is a selective and cell-permeable degrader of BET based on PROTAC (IC50: 14 nM). …
Formula:
C42H45ClN8O7S
Purity:
97.57% - 99.12%
Color and Shape:
Solid
Molecular weight:
841.37
Ref: TM-T5130
| 1mg | 52.00 € | ||
| 5mg | 95.00 € | ||
| 10mg | 166.00 € | ||
| 25mg | 302.00 € | ||
| 50mg | 481.00 € | ||
| 100mg | 699.00 € | ||
| 200mg | 878.00 € | ||
| 500mg | 1,287.00 € | ||
| 1mL*10mM (DMSO) | 156.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
5-AIQ
CAS:93117-08-9
5-aminoisoquinolin-1(2H)-one is the inhibitor of calf thymus PARP1.
Formula:
C9H8N2O
Purity:
95.00%
Color and Shape:
Solid
Molecular weight:
160.17
Ref: TM-T50044
| 25mg | 35.00 € | ||
| 50mg | 49.00 € | ||
| 100mg | 79.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
GSK-LSD1 dihydrochloride
CAS:2102933-95-7
GSK-LSD1 dihydrochloride: potent LSD1 inhibitor, >1000x selective over MAO-A/B, LSD2, IC50: 16 nM.
Formula:
C14H22Cl2N2
Purity:
100% - 99.22%
Color and Shape:
Solid
Molecular weight:
289.24
Ref: TM-T2315
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 70.00 € | ||
| 10mg | 101.00 € | ||
| 25mg | 206.00 € | ||
| 50mg | 312.00 € | ||
| 100mg | 513.00 € | ||
| 500mg | 1,093.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
Deoxyshikonin
CAS:43043-74-9
1.
Formula:
C16H16O4
Purity:
99.36% - ≥95%
Color and Shape:
Solid
Molecular weight:
272.3
Ref: TM-T5S2347
| 10mg | 125.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
PFI-90
CAS:53995-62-3
PFI-90, a selective histone demethylase (KDM3B) inhibitor, targets PAX3-FOXO1 action and demonstrates potential antitumor activity.
Formula:
C11H10N4O
Purity:
99.5%
Color and Shape:
Solid
Molecular weight:
214.22
Ref: TM-T9243
| 25mg | 40.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
PF-CBP1 hydrochloride
CAS:2070014-93-4
PF-CBP1 HCl selectively inhibits CREBBP bromodomain (IC50: 125 nM) and p300 (IC50: 363 nM).
Formula:
C29H37ClN4O3
Purity:
95.87% - 99%
Color and Shape:
Solid
Molecular weight:
525.08
Ref: TM-T3217
| 5mg | 46.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 118.00 € | ||
| 50mg | 184.00 € | ||
| 100mg | 343.00 € | ||
| 200mg | 447.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
UMB298
CAS:2266569-73-5
UMB298 is a potent and selective CBP/P300 bromodomain inhibitor. UMB298 inhibits BRD4 with IC50 of …
Formula:
C27H31ClN4O2
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
479.01
Ref: TM-T9194
| 1mg | 62.00 € | ||
| 5mg | 136.00 € | ||
| 10mg | 211.00 € | ||
| 25mg | 364.00 € | ||
| 50mg | 511.00 € | ||
| 100mg | 698.00 € | ||
| 200mg | 904.00 € | ||
| 1mL*10mM (DMSO) | 144.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
(S)-CPI203
CAS:1446144-04-2
CPI-203 is an effective BET bromodomain inhibitor (IC50: 37 nM for BRD4).
Formula:
C19H18ClN5OS
Purity:
98.96% - 99.36%
Color and Shape:
Solid
Molecular weight:
399.9
Ref: TM-T6026
| 2mg | 35.00 € | ||
| 5mg | 57.00 € | ||
| 10mg | 91.00 € | ||
| 25mg | 173.00 € | ||
| 50mg | 274.00 € | ||
| 100mg | 433.00 € | ||
| 200mg | 605.00 € | ||
| 1mL*10mM (DMSO) | 60.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
RO8191
CAS:691868-88-9
RO8191 (CDM-3008) (CDM-3008) is an agonist of interferon (IFN) receptor.
Formula:
C14H5F6N5O
Purity:
98.85% - ≥98%
Color and Shape:
Solid
Molecular weight:
373.21
Ref: TM-T22142
| 1mg | 45.00 € | ||
| 2mg | 58.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 301.00 € | ||
| 50mg | 478.00 € | ||
| 100mg | 698.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
C646
CAS:328968-36-1
C646, a histone acetyltransferase inhibitor, inhibits p300 (Ki: 400 nM, in a cell-free assay).
Formula:
C24H19N3O6
Purity:
98% - 99.21%
Color and Shape:
Solid
Molecular weight:
445.42
Ref: TM-T2452
| 2mg | 53.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 100.00 € | ||
| 25mg | 197.00 € | ||
| 50mg | 377.00 € | ||
| 100mg | 557.00 € | ||
| 500mg | 1,179.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
Brevilin A
CAS:16503-32-5
Brevilin A, a sesquiterpene from Centipeda minima, hinders JAK and blocks STAT3 (IC50=10.6μM), inducing apoptosis …
Formula:
C20H26O5
Purity:
100% - 99.74%
Color and Shape:
Solid
Molecular weight:
346.42
Ref: TM-T4672
| 1mg | 94.00 € | ||
| 5mg | 212.00 € | ||
| 10mg | 362.00 € | ||
| 25mg | 601.00 € | ||
| 50mg | 822.00 € | ||
| 100mg | 1,112.00 € | ||
| 500mg | 2,265.00 € | ||
| 1mL*10mM (DMSO) | 235.00 € |
Estimated delivery in United States, on Wednesday 13 Nov 2024
