Chromatin/Epigenetics
Chromatin/epigenetics inhibitors are compounds that modulate the structure and function of chromatin or interfere with epigenetic modifications, such as DNA methylation and histone modification. These inhibitors are essential tools for studying gene expression regulation and the role of epigenetics in diseases like cancer, neurological disorders, and developmental abnormalities. By targeting epigenetic processes, these inhibitors can alter gene expression patterns and offer new therapeutic avenues. At CymitQuimica, we provide a wide selection of high-quality chromatin/epigenetics inhibitors to support your research in molecular biology, genetics, and epigenetics.
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Subcategories of "Chromatin/Epigenetics"
Products of "Chromatin/Epigenetics"
EML741
CAS:2328074-38-8
EML741 also inhibits DNMT1 (IC50, 3.1 μM), with no effect on DNMT3a or DNMT3b.
Formula:
C31H49N5O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
523.75
Ref: TM-T11185
| 25mg | 1,406.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
CARM1-IN-1
CAS:1020399-49-8
CARM1-IN-1 (CARM1-IN-7G) is a selective inhibitor of CARM1 with IC50 of 8.6 μM. CARM1-IN-1 shows …
Formula:
C26H21Br2NO3
Purity:
97.35%
Color and Shape:
Solid
Molecular weight:
555.26
Ref: TM-T10682L
| 1mg | 41.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 123.00 € | ||
| 25mg | 241.00 € | ||
| 50mg | 392.00 € | ||
| 100mg | 610.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
CX-6258
CAS:1202916-90-2
CX-6258 is an orally valid Pim 1/2/3 kinase(IC50=5 nM/25 nM/16 nM) inhibitor. It has good …
Formula:
C26H24ClN3O3
Purity:
95.88%
Color and Shape:
Solid
Molecular weight:
461.94
Ref: TM-T1834
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 86.00 € | ||
| 10mg | 124.00 € | ||
| 25mg | 237.00 € | ||
| 50mg | 386.00 € | ||
| 100mg | 548.00 € | ||
| 200mg | 796.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
EZM 2302
CAS:1628830-21-6
EZM 2302 (GSK3359088) is a selective, and orally available arginine methyltransferase CARM1 inhibitor (IC50: 6 …
Formula:
C29H37ClN6O5
Purity:
97.47% - ≥98%
Color and Shape:
Solid
Molecular weight:
585.09
Ref: TM-T5605
| 1mg | 73.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 231.00 € | ||
| 25mg | 441.00 € | ||
| 50mg | 588.00 € | ||
| 100mg | 831.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
OXF BD 02
CAS:1429129-68-9
OXF BD 02 is a potent and selective BRD4(1) inhibitor (IC50: 382 nM) with anticancer …
Formula:
C18H17NO3
Purity:
98.25%
Color and Shape:
Solid
Molecular weight:
295.33
Ref: TM-T23115
| 1mg | 96.00 € | ||
| 5mg | 229.00 € | ||
| 10mg | 345.00 € | ||
| 25mg | 639.00 € | ||
| 50mg | 914.00 € | ||
| 100mg | 1,224.00 € | ||
| 500mg | 2,466.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
3-Deazaneplanocin A
CAS:102052-95-9
3-Deazaneplanocin A (DZNep) is an attractive epigenetic anticancer agent through the inhibition of the cellular …
Formula:
C12H14N4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
262.26
Ref: TM-T6292
| 1mg | 153.00 € | ||
| 5mg | 398.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
WDR5-0102
CAS:824960-50-1
WDR5-0102 inhibits WDR5-MLL1 (Kd=4 μM), blocks MLL1 HMT activity, but doesn't affect SETD7 and 6 …
Formula:
C18H19ClN4O3
Purity:
97.16%
Color and Shape:
Solid
Molecular weight:
374.82
Ref: TM-T67947
| 1mg | 75.00 € | ||
| 5mg | 167.00 € | ||
| 10mg | 270.00 € | ||
| 25mg | 540.00 € | ||
| 50mg | 779.00 € | ||
| 100mg | 1,067.00 € | ||
| 500mg | 2,125.00 € | ||
| 1mL*10mM (DMSO) | 213.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
PARP10-IN-2
CAS:1042780-52-8
PARP10-IN-2 is a potent inhibitor of PARP10, a mono-ADP-ribosyltransferase, with an IC50 value of 3.64 …
Formula:
C14H10N2O2
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
238.24
Ref: TM-T73007
| 5mg | 69.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 305.00 € | ||
| 100mg | 500.00 € | ||
| 500mg | 1,068.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
BAY1238097
CAS:1564268-08-1
BAY1238097 is a BET inhibitor with anticancer activity and antiproliferative activity for the study of …
Formula:
C25H33N5O3
Purity:
98.55%
Color and Shape:
Solid
Molecular weight:
451.56
Ref: TM-T12660L
| 1mg | 98.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Dot1L-IN-2
CAS:1940206-71-2
Dot1l-in-2 is an effective, selective and oral bioutilization inhibitor of histone methyltransferase Dot1L, with IC50 …
Formula:
C27H24N8O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
476.53
Ref: TM-T11082
| 25mg | 1,545.00 € | ||
| 50mg | 2,031.00 € | ||
| 100mg | 2,609.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Corin
CAS:1808113-09-8
Corin is an irreversible inhibitor of HDAC1(IC50 = 147 nM) and LSD1(Ki = 110 nM).
Formula:
C26H28N4O2
Purity:
98.22%
Color and Shape:
Solid
Molecular weight:
428.53
Ref: TM-T10864
| 1mg | 167.00 € | ||
| 5mg | 423.00 € | ||
| 10mg | 625.00 € | ||
| 25mg | 984.00 € | ||
| 50mg | 1,328.00 € | ||
| 100mg | 1,784.00 € | ||
| 1mL*10mM (DMSO) | 463.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Guadecitabine sodium
CAS:929904-85-8
Guadecitabine sodium is a inhibitor of second-generation DNA methyltransferases (DNMT) .
Formula:
C18H24N9NaO10P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
580.407
Ref: TM-T12790
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
DW14800
CAS:2243709-60-4
DW14800 is an inhibitor of PRMT5 (IC50 = 17 nM), enhances the transcription of HNF4α, …
Formula:
C31H36N4O3
Purity:
97.26% - 99.12%
Color and Shape:
Solid
Molecular weight:
512.64
Ref: TM-T11131
| 1mg | 56.00 € | ||
| 5mg | 130.00 € | ||
| 10mg | 218.00 € | ||
| 25mg | 415.00 € | ||
| 50mg | 548.00 € | ||
| 1mL*10mM (DMSO) | 147.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
PARP14 inhibitor H10
CAS:2084811-68-5
PARP14 inhibitor H10 is a selective inhibitor against PARP14 with IC50 of 490 nM
Formula:
C24H27N7O7S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
557.58
Ref: TM-T12366
| 1mg | 880.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
Trotabresib
CAS:1706738-98-8
Trotabresib (CC-90010) is an orally active inhibitor of BET and can be used in studies …
Formula:
C21H21NO4S
Purity:
99.03%
Color and Shape:
Solid
Molecular weight:
383.46
Ref: TM-T36395
| 1mg | 90.00 € | ||
| 5mg | 184.00 € | ||
| 10mg | 305.00 € | ||
| 25mg | 516.00 € | ||
| 50mg | 738.00 € | ||
| 100mg | 993.00 € | ||
| 1mL*10mM (DMSO) | 210.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
PARP/PI3K-IN-1
CAS:2337386-47-5
PARP/PI3K-IN-1 is a PARP and PI3K dual inhibitor with anticancer and antiproliferative activities for the …
Formula:
C33H28F4N8O3
Purity:
99.59%
Color and Shape:
Solid
Molecular weight:
660.62
Ref: TM-T12365
| 1mg | 95.00 € | ||
| 5mg | 237.00 € | ||
| 10mg | 368.00 € | ||
| 25mg | 640.00 € | ||
| 50mg | 993.00 € | ||
| 100mg | 1,345.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
DDP-38003 dihydrochloride
CAS:1831167-98-6
DDP-38003 dihydrochloride is an orally available histone lysine-specific demethylase 1A (KDM1A/LSD1) inhibitor (IC50: 84 nM).
Formula:
C21H28Cl2N4O
Purity:
99.5%
Color and Shape:
Solid
Molecular weight:
423.38
Ref: TM-T10983L
| 1mg | 79.00 € | ||
| 5mg | 135.00 € | ||
| 10mg | 224.00 € | ||
| 25mg | 498.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
JAK1-IN-4
CAS:2091134-35-7
JAK1-IN-4 selectively blocks JAK1 (IC50 = 85 nM) over JAK2/JAK3 and halts STAT3 phosphorylation in …
Formula:
C26H32FN9O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
521.59
Ref: TM-T15606
| 25mg | 1,549.00 € | ||
| 50mg | 2,038.00 € | ||
| 100mg | 2,617.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
IACS-9571
CAS:1800477-30-8
IACS-9571 is a selective and potent inhibitor of TRIM24 and BRPF1, (IC50: 8 nM for …
Formula:
C32H42N4O8S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
642.76
Ref: TM-T11597
| 25mg | 8,469.00 € | ||
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Friday 27 Dec 2024
MS0124
CAS:1197196-63-6
MS0124 is a potent and selective G9A-like protein (GLP) inhibitor with IC50 values of 13±4 …
Formula:
C20H29N5O3
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
387.48
Ref: TM-T28112
| 1mg | 306.00 € | ||
| 5mg | 741.00 € | ||
| 10mg | 1,013.00 € | ||
| 25mg | 1,532.00 € | ||
| 50mg | 2,083.00 € | ||
| 100mg | 2,719.00 € |
Estimated delivery in United States, on Friday 27 Dec 2024
