Somatostatin
Somatostatin is a peptide hormone that inhibits the release of several other hormones, including growth hormone, insulin, and glucagon. It acts by binding to somatostatin receptors, which are G protein-coupled receptors expressed in various tissues. Somatostatin analogs are used in the treatment of acromegaly, neuroendocrine tumors, and gastrointestinal disorders. These analogs are also valuable tools for studying hormone secretion and signaling. At CymitQuimica, we provide a comprehensive range of high-quality somatostatin analogs to support your research in endocrinology, hormone regulation, and therapeutic development.
Found 57 products of "Somatostatin"
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Edotreotide
CAS:Edotreotide (SMT-487) is an Indicator and Reagent. It also is used in the Diagnosis and Staging of Tumors Expressing Somatostatin Receptors.Formula:C65H92N14O18S2Purity:96.95%Color and Shape:SolidMolecular weight:1421.64Octreotide Acetate
CAS:Octreotide Acetate (Sandostatin) is a potent, long-acting synthetic somatostatin octapeptide analog that inhibits secretion of growth hormone.Formula:C51H70N10O12S2Purity:99.03% - 99.87%Color and Shape:Less To Off-White Lyophilised Solid Colourless To Off-White Lyophilised SolidMolecular weight:1079.30L-803087
CAS:L-803087: potent sst4 receptor agonist, 0.7 nM Ki, 280x selectivity, boosts AMPA responses & seizures in mice.Formula:C25H29F2N5O3Purity:99.37%Color and Shape:SolidMolecular weight:485.53Ref: TM-T11800
1mg50.00€5mg112.00€10mg175.00€25mg366.00€50mg585.00€100mg928.00€200mg1,234.00€1mL*10mM (DMSO)126.00€SST1 receptor antagonist-1
CAS:SST1 receptor antagonist-1 (Compound 23) is a selective antagonist of the somatostatin receptor 1 (SST1), showing a pKd of 9.11 for rSST1 and 8.79 for hSST1. This compound is applicable in research related to retinal and endocrine dysfunction, cancer, and neuropsychiatric disorders.Formula:C29H31F2N3O2Color and Shape:SolidMolecular weight:491.57SSTR4 agonist 5
CAS:SSTR4 agonist5 (Compound 5) is an orally active agonist of the somatostatin receptor 4 (SSTR4) with an EC50 of 0.228 nM. It demonstrates good stability in human/rat liver microsomes and can inhibit mechanical hyperalgesia in rat models.Formula:C20H26N4OMolecular weight:338.447L-796778 acetate
CAS:L-796778 acetate is a selective sst3 receptor agonist. In CHO-K1 cells expressing hsst3 receptors, it acts as a partial agonist that inhibits Forskolin-induced cAMP production, with an IC50 value of 18 nM. Additionally, L-796778 acetate exhibits anticonvulsant properties.Formula:C31H44N6O9Color and Shape:SolidMolecular weight:644.716SSTR5 antagonist 6
CAS:SSTR5 antagonist 6, an orally active antagonist specific to the somatostatin receptor subtype 5 (SSTR5), exhibits an IC50 value of 24 nM. This compound is utilized in researching type 2 diabetes [1].Formula:C22H28ClN3O4Color and Shape:SolidMolecular weight:433.93
