
Somatostatin
Somatostatin is a peptide hormone that inhibits the release of several other hormones, including growth hormone, insulin, and glucagon. It acts by binding to somatostatin receptors, which are G protein-coupled receptors expressed in various tissues. Somatostatin analogs are used in the treatment of acromegaly, neuroendocrine tumors, and gastrointestinal disorders. These analogs are also valuable tools for studying hormone secretion and signaling. At CymitQuimica, we provide a comprehensive range of high-quality somatostatin analogs to support your research in endocrinology, hormone regulation, and therapeutic development.
Found 64 products for "Somatostatin".
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L-796778 acetate
CAS:L-796778 acetate is a selective sst3 receptor agonist. In CHO-K1 cells expressing hsst3 receptors, it acts as a partial agonist that inhibits Forskolin-induced cAMP production, with an IC50 value of 18 nM. Additionally, L-796778 acetate exhibits anticonvulsant properties.Formula:C31H44N6O9Color and Shape:SolidMolecular weight:644.716SST1 receptor antagonist-2
CAS:SST1 receptor antagonist-2 (Example 2) is a piperazine derivative and an antagonist of the somatostatin receptor 1 (SST1). It can be utilized in research on psychiatric disorders, neurodegenerative diseases, tumors, vascular disorders, and immune diseases.Formula:C29H31F2N3OMolecular weight:475.57SSTR5 antagonist 6
CAS:SSTR5 antagonist 6, an orally active antagonist specific to the somatostatin receptor subtype 5 (SSTR5), exhibits an IC50 value of 24 nM. This compound is utilized in researching type 2 diabetes [1].Formula:C22H28ClN3O4Color and Shape:SolidMolecular weight:433.93Tau conotoxin CnVA
CAS:Tau conotoxin CnVA, a small peptide found in the venom of Conus consors (cone snail), is a member of the T1 cone snail peptide superfamily. It demonstrates high selectivity for the somatostatin sst3 receptor with a Ki value of 1.5 µM. Tau conotoxin CnVA is unique as the only known toxin interacting with this subfamily of G protein-coupled receptors (GPCR). This compound is useful for research related to diseases associated with the sst3 receptor, such as pancreatic cancer or pituitary adenomas.Formula:C72H116N24O17S4Color and Shape:SolidMolecular weight:1718.1
