GPR
G protein-coupled receptors (GPRs) are a large family of cell surface receptors that play a crucial role in transmitting signals from hormones, neurotransmitters, and other extracellular ligands into the cell. GPRs are involved in a wide range of physiological processes, including hormone regulation, immune response, and sensory perception. Modulating GPR activity is a key strategy in the development of therapeutics for various diseases, including endocrine disorders, cardiovascular diseases, and neurological conditions. At CymitQuimica, we offer a selection of high-quality GPR modulators to support your research in cell signaling, endocrinology, and drug discovery.
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Vincamine
CAS:1617-90-9
Vincamine, from Vinca minor, is an alkaloid used as a vasodilator and antihypertensive for brain …
Formula:
C21H26N2O3
Purity:
99.52%
Color and Shape:
White To Almost White Fine Crystalline Powder
Molecular weight:
354.44
Ref: TM-T1286
| 1g | 66.00 € | ||
| 500mg | 53.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Fezagepras
CAS:1002101-19-0
Fezagepras (Setogepram) is an orally active GPR40 agonist and is an antagonist or inverse agonist …
Formula:
C13H18O2
Purity:
96.73% - 99.38%
Color and Shape:
Solid
Molecular weight:
206.28
Ref: TM-T12883
| 1mg | 52.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 138.00 € | ||
| 25mg | 240.00 € | ||
| 50mg | 343.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
BI-671800
CAS:1093108-50-9
BI-671800 (AP-761) is a DP2/CRTH2 antagonist with IC50 values of 4.5 nM and 3.7 nM, …
Formula:
C25H26F3N5O3
Purity:
99.19%
Color and Shape:
Solid
Molecular weight:
501.5
Ref: TM-T14565
| 1mg | 57.00 € | ||
| 5mg | 127.00 € | ||
| 10mg | 200.00 € | ||
| 25mg | 360.00 € | ||
| 50mg | 511.00 € | ||
| 100mg | 694.00 € | ||
| 200mg | 906.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
FTBMT
CAS:1358575-02-6
FTBMT is a selective GPR52 agonist (EC50: 75 nM) and it also has antipsychotic and …
Formula:
C19H16F4N4O
Purity:
99.12%
Color and Shape:
Solid
Molecular weight:
392.35
Ref: TM-T15352
| 1mg | 38.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 125.00 € | ||
| 25mg | 279.00 € | ||
| 50mg | 496.00 € | ||
| 100mg | 771.00 € | ||
| 200mg | 1,021.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
NE 52-QQ57
CAS:1401728-56-0
NE 52-QQ57 is a selective, and orally available antagonist of GPR4(IC50 : 70 nM),with anti-inflammatory …
Formula:
C24H28N6O
Purity:
98.63%
Color and Shape:
Solid
Molecular weight:
416.52
Ref: TM-T11461
| 1mg | 73.00 € | ||
| 5mg | 158.00 € | ||
| 10mg | 231.00 € | ||
| 25mg | 386.00 € | ||
| 50mg | 573.00 € | ||
| 100mg | 821.00 € | ||
| 1mL*10mM (DMSO) | 168.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
Ramatroban
CAS:116649-85-5
Ramatroban (BAY u3405) (BAY u3405) is a thromboxane A(2) (TxA(2)) antagonist marketed for allergic rhinitis.
Formula:
C21H21FN2O4S
Purity:
98.12% - 99.96%
Color and Shape:
Crystalline Solid
Molecular weight:
416.47
Ref: TM-T2396
| 5mg | 38.00 € | ||
| 10mg | 56.00 € | ||
| 25mg | 93.00 € | ||
| 50mg | 167.00 € | ||
| 100mg | 268.00 € | ||
| 200mg | 347.00 € | ||
| 500mg | 587.00 € | ||
| 1mL*10mM (DMSO) | 63.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
GSK256073
CAS:862892-90-8
GSK256073 is an orally active GPR109A agonist.
Formula:
C10H13ClN4O2
Purity:
98.03%
Color and Shape:
Solid
Molecular weight:
256.69
Ref: TM-T15432
| 1mg | 72.00 € | ||
| 2mg | 95.00 € | ||
| 5mg | 157.00 € | ||
| 10mg | 245.00 € | ||
| 25mg | 430.00 € | ||
| 50mg | 633.00 € | ||
| 100mg | 900.00 € | ||
| 1mL*10mM (DMSO) | 168.00 € |
Estimated delivery in United States, on Wednesday 4 Dec 2024
7-FluorotryptaMine HCl
CAS:159730-09-3
7-FluorotryptaMine HCl is a potent aromatic monoamine GPRC5A agonist that induces GPRC5A-mediated β-arrestin recruitment.7-FluorotryptaMine HCl …
Formula:
C10H12ClFN2
Purity:
98.06%
Color and Shape:
Liquid
Molecular weight:
214.67
Ref: TM-T77673
| 1mg | 36.00 € | ||
| 5mg | 69.00 € | ||
| 10mg | 101.00 € | ||
| 25mg | 207.00 € | ||
| 50mg | 312.00 € | ||
| 100mg | 463.00 € | ||
| 500mg | 1,050.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
TUG-499
CAS:1206629-08-4
TUG-499 is a selective free fatty acid receptor 1 (FFAR1 or GPR40) agonist (EC50: 7.39).TUG-499 …
Formula:
C16H11Cl2NO2
Purity:
99.59%
Color and Shape:
Soild
Molecular weight:
320.17
Ref: TM-T60184
| 1mg | 52.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 157.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 346.00 € | ||
| 100mg | 453.00 € | ||
| 500mg | 984.00 € | ||
| 1mL*10mM (DMSO) | 114.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Latanoprost acid
CAS:41639-83-2
Latanoprost acid is a prostanoid receptor agonist that blocks RANKL and can be used to …
Formula:
C23H34O5
Purity:
96.97%
Color and Shape:
Pale Yellow Oil
Molecular weight:
390.51
Ref: TM-T15718
| 1mg | 56.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 220.00 € | ||
| 25mg | 440.00 € | ||
| 50mg | 653.00 € | ||
| 100mg | 897.00 € | ||
| 200mg | 1,190.00 € | ||
| 1mL*10mM (DMSO) | 156.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
NOX-6-18
CAS:898211-21-7
NOX-6-18 (GPR132-B-160) is a GPR132 antagonist with insulin-promoting activity and reduced weight gain.
Formula:
C18H17NO5S
Purity:
99.29%
Color and Shape:
Soild
Molecular weight:
359.4
Ref: TM-T83972
| 1mg | 75.00 € | ||
| 5mg | 160.00 € | ||
| 10mg | 250.00 € | ||
| 25mg | 502.00 € | ||
| 50mg | 809.00 € | ||
| 100mg | 1,290.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
(1S,2R)-2-PCCA
(1S,2R)-2-PCCA is a novel and potent small molecule GPR88 receptor agonist with an EC50 value …
Formula:
C30H39Cl2N3O
Purity:
99.34%
Color and Shape:
Soild
Molecular weight:
528.56
Ref: TM-T13423L
| 1mg | 183.00 € | ||
| 5mg | 435.00 € | ||
| 10mg | 635.00 € | ||
| 25mg | 1,000.00 € | ||
| 50mg | 1,336.00 € | ||
| 100mg | 1,803.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
WAY-298630
CAS:303134-93-2
Fluorophenoxy benzimidazole, a CRTH2 blocker, IC50 < 10 μM for rhinitis, COPD, arthritis, eczema, conjunctivitis.
Formula:
C17H15FN2O3S
Purity:
97.13%
Color and Shape:
Liquid
Molecular weight:
346.38
Ref: TM-T77601
| 1mg | 181.00 € | ||
| 5mg | 400.00 € | ||
| 10mg | 595.00 € | ||
| 25mg | 917.00 € | ||
| 50mg | 1,263.00 € | ||
| 100mg | 1,710.00 € | ||
| 500mg | 3,428.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
PU-WS13 hydrobromide
PU-WS13 hydrobromide is a GRP94 inhibitor with anti-inflammatory activity and inhibits the proliferation of M2-like …
Formula:
C17H21BrCl2N6S
Purity:
98%
Color and Shape:
Soild
Molecular weight:
492.26
Ref: TM-T5351L
| 1mg | 42.00 € | ||
| 5mg | 85.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 217.00 € | ||
| 50mg | 420.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
BMS-903452
CAS:1339944-47-6
BMS-903452: potent GPR119 agonist, EC50 = 14 nM, treats rodent diabetes, no P450 inhibition, safe …
Formula:
C21H19Cl2FN4O4S
Purity:
100% - 100%
Color and Shape:
Liquid
Molecular weight:
513.37
Ref: TM-T67791
| 1mg | 149.00 € | ||
| 5mg | 359.00 € | ||
| 10mg | 510.00 € | ||
| 25mg | 766.00 € | ||
| 50mg | 1,035.00 € | ||
| 100mg | 1,398.00 € | ||
| 500mg | 2,739.00 € | ||
| 1mL*10mM (DMSO) | 426.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
2-Oleoylglycerol
CAS:3443-84-3
2-Oleoylglycerol is a lipid found in palm kernels that acts as a GPR119 agonist with …
Formula:
C21H40O4
Purity:
98%
Color and Shape:
Liquid
Molecular weight:
356.54
Ref: TM-T37526
| 1mg (28mM*100μL in Ethanol) | 92.00 € | ||
| 25mg (28mM*2.5mL in Ethanol) | To inquire |
Estimated delivery in United States, on Thursday 5 Dec 2024
GPCR agonist-2
CAS:291528-35-3
GPCR agonist-2 (4-(Cyclopropylamino)-3-nitrobenzoic acid) is an agonist of the orphan human GPCR GPR109B.
Formula:
C10H10N2O4
Purity:
99.94%
Color and Shape:
Solid
Molecular weight:
222.2
Ref: TM-T60074
| 10mg | 35.00 € | ||
| 25mg | 47.00 € | ||
| 50mg | 60.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
15(R)-15-methyl Prostaglandin D2
CAS:210978-26-0
15(R)-15-methyl Prostaglandin D2 (15(R)15methyl PGD2) is a synthetic analog of PGD2 and a CRTH2/DP2 receptor …
Formula:
C21H34O5
Color and Shape:
Liquid
Molecular weight:
366.49
Ref: TM-T37264
| 1mg | 313.00 € | ||
| 500µg | 185.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
NCRW0005-F05
CAS:342779-66-2
NCRW0005-F05 is a potent agonist of orphan G-protein coupled receptor GPR139 with an IC 50 …
Formula:
C16H13F2NO2
Purity:
99.48%
Color and Shape:
Solid
Molecular weight:
289.28
Ref: TM-T60199
| 5mg | 46.00 € | ||
| 10mg | 77.00 € | ||
| 25mg | 144.00 € | ||
| 50mg | 222.00 € | ||
| 100mg | To inquire | ||
| 1mL*10mM (DMSO) | 50.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Kynurenic acid
CAS:492-27-3
Kynurenic acid (Quinurenic acid) is an NMDA, glutamate, α7 nicotinic acetylcholine receptor triple antagonist and …
Formula:
C10H7NO3
Purity:
99.69%
Color and Shape:
Liquid
Molecular weight:
189.17
Ref: TM-T65135
| 50mg | 36.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
