Androgen Receptor
The androgen receptor (AR) is a nuclear hormone receptor that is activated by binding to androgens, such as testosterone and dihydrotestosterone. This receptor plays a crucial role in the development and maintenance of male characteristics, as well as in the regulation of several physiological processes, including muscle growth, libido, and bone density. Androgen receptor inhibitors are widely studied in the context of prostate cancer, where AR signaling is often upregulated. At CymitQuimica, we offer a range of high-quality androgen receptor modulators to support your research in endocrinology, cancer biology, and hormone regulation.
Found 229 products of "Androgen Receptor"
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LG-121071
CAS:LG-121071: oral SARM, high-affinity AR full agonist, Ki=17 nM.Formula:C15H15F3N2OPurity:98%Color and Shape:SolidMolecular weight:296.29AR antagonist 5
CAS:Compound 30a, known as AR Antagonist 5, is a selective androgen receptor (AR) antagonist that demonstrates an IC 50 value of 134.8 nM. It exhibits favorable pharmacokinetic properties, characterized by high skin exposure and low plasma exposure [1].Formula:C23H21F3N6O2Color and Shape:SolidMolecular weight:470.45(R)-Bicalutamide
CAS:(R)-Bicalutamide, an AR antagonist with antitumor properties, is crucial in prostate cancer research.Formula:C18H14F4N2O4SColor and Shape:SolidMolecular weight:430.37AR antagonist 2
CAS:AR antagonist 2 (compound 58) is a potent inhibitor of the androgen receptor (AR) (IC50: 0.95 μM).Formula:C22H17ClFN5O2SColor and Shape:SolidMolecular weight:469.92Bromopropylate
CAS:Bromopropylate is an insecticide. Bromopropylate is the active substance in fumigant strips for mites.Formula:C17H16Br2O3Purity:98%Color and Shape:White Crystalline Solid Yellowish CrystalsMolecular weight:428.11S-40503
CAS:S-40503 is an investigational selective androgen receptor modulator (SARM).Formula:C15H23N3O3Color and Shape:SolidMolecular weight:293.36Ralaniten
CAS:Ralaniten (EPI-002), a potent AR-NTD antagonist, inhibits AR with IC50 of 7.4 μM, for CRPC study.Formula:C21H27ClO5Purity:99.96%Color and Shape:SolidMolecular weight:394.89Ref: TM-T28502
1mg40.00€5mg88.00€10mg126.00€25mg250.00€50mg393.00€100mg628.00€200mg879.00€1mL*10mM (DMSO)87.00€Androgen receptor antagonist 1
CAS:Androgen receptor antagonist 1, an oral full AR antagonist (IC50 59 nM), for PROTAC synthesis, reducing AR protein by 24–47% in LNCaP cells at 1–10 μM.Formula:C21H25ClN4O3Purity:99.054%Color and Shape:SolidMolecular weight:416.9RU 58642
CAS:RU 58642 is an effective systemic antiandrogen for androgen-dependent disorders.Formula:C15H11F3N4O2Purity:98%Color and Shape:SolidMolecular weight:336.27Cyprodinil
CAS:Cyprodinil is a fungicide blocking methionine synthesis in fungi and hinders B. cinerea, P. herpotrichoides, H. oryzae growth; it's also an AR agonist.Formula:C14H15N3Color and Shape:SolidMolecular weight:225.29VPC-14449
CAS:VPC-14449 is a selective androgen receptor DNA-binding domain (AR-DBD) inhibitor, useful in prostate cancer research.Formula:C10H10Br2N4OSPurity:99.56%Color and Shape:SolidMolecular weight:394.09BMS-564929
CAS:BMS-564929 is an AR agonist that upregulates the expression and activity of fat-producing enzymes, reducing VAT content and lipid levels.Formula:C14H12ClN3O3Purity:98.17%Color and Shape:SolidMolecular weight:305.72VPC-13789
CAS:VPC-13789: potent, selective oral antiandrogen for CRPC with 0.19 μM IC50 in LNCaP cells.Formula:C21H16F3N3OColor and Shape:SolidMolecular weight:383.37Androgen receptor antagonist 3
CAS:Androgen receptor antagonist 3 (Compound C18) has anticancer activities that is an antagonist of androgen receptor (AR) (IC 50 = 2.4 μM) [1].Formula:C22H18ClNColor and Shape:SolidMolecular weight:331.84(R)-UT-155
CAS:(R)-UT-155 is a selective androgen receptor degrader (SARD) ligand.Formula:C20H15F4N3O2Color and Shape:SolidMolecular weight:405.35Lubabegron fumarate
CAS:Lubabegron (LY591281, LY488756 fumarate) is a beta-agonist approved in 2018 to lower ammonia in cattle waste, aiding environment and health.Formula:C29H29N3O3SC4H4O4Color and Shape:SolidMolecular weight:557.66MK-4541
CAS:MK-4541: oral, selective AR modulator, blocks 5α-reductase, curbs AR+ prostate cancer growth, effective in mouse model.Formula:C22H31F3N2O3Color and Shape:SolidMolecular weight:428.49HG122
CAS:HG122 promotes AR degradation via proteasome, inhibiting castration-resistant prostate cancer.Formula:C15H13N5O5Color and Shape:SolidMolecular weight:343.29LGD-2226
CAS:LGD-2226: selective oral androgen receptor modulator, EC50: 0.2nM, Ki: 1.5nM. Treats muscle loss, osteoporosis, sexual issues.Formula:C14H9F9N2OPurity:98%Color and Shape:SolidMolecular weight:392.22Dimethomorph
CAS:Dimethomorph is a fungicide and sterol biosynthesis inhibitor that inhibits fungal cell wall formation,. inhibits androgen receptor (AR) .Formula:C21H22ClNO4Purity:99.20%Color and Shape:Solid CrystallineMolecular weight:387.86CSRM617
CAS:CSRM617: selective ONECUT2 inhibitor, Kd 7.43 uM, binds OC2-HOX, induces apoptosis, tolerable in mouse prostate cancer model.Formula:C10H13N3O5Purity:98%Color and Shape:SolidMolecular weight:255.23MK-3984
CAS:MK-3984 is a selective androgen receptor modulator, used in the study of conditions caused by androgen deficiency.Formula:C17H12F7NO2Purity:99.91%Color and Shape:SolidMolecular weight:395.27TFM-4AS-1
CAS:androgen receptor modulatorFormula:C27H33F3N2O2Purity:98%Color and Shape:SolidMolecular weight:474.56VPC-3033
CAS:VPC-3033 is an antagonist of the androgen receptor. It acts by inhibiting the LNCaP cell line as well as cell lines with the wild-type androgen receptor.Formula:C21H14O2Purity:98%Color and Shape:SolidMolecular weight:298.33Topterone
CAS:Topterone (Win 17,665) is a potent topical antiandrogen that inhibits the stimulation of lumbar organ development by testosterone and dihydrotestosterone inFormula:C22H34O2Purity:>99.99%Color and Shape:SolidMolecular weight:330.5Ar-V7-IN-1
CAS:Ar-V7-IN-1 (compound 47) is a potent inhibitor of Ar-V7,associated with resistance to AR-targeted therapy with desmoplasia-resistant prostate cancer (mCRPC).Formula:C10H10Br2N4OSColor and Shape:SolidMolecular weight:394.09Carbazole derivative 1
CAS:Carbazole derivative 1 is used to reduce androgen or oestrogen levels in mammals.Formula:C18H13FN2Purity:98%Color and Shape:SolidMolecular weight:276.31Seviteronel
CAS:Seviteronel (VT-464) is a novel CYP17 cleavage enzyme inhibitor and androgen receptor antagonist for the study of breast and prostate cancer.Formula:C18H17F4N3O3Purity:99.67% - 99.98%Color and Shape:SolidMolecular weight:399.34BMS-641988
CAS:BMS-641988 is a novel nonsteroidal androgen receptor antagonist for the treatment of prostate cancer.Formula:C20H20F3N3O5SPurity:99.3% - 99.92%Color and Shape:SoildMolecular weight:471.45Rosolutamide
CAS:Rosolutamide (ALZ-003) is a curcumin analog, an Nrf1 and Nrf2 activator.Formula:C28H32O6Purity:95.48% - 99.15%Color and Shape:SolidMolecular weight:464.55Ralaniten triacetate
CAS:Ralaniten triacetate (EPI-506) is a precursor of Ralaniten, an AR-NTD inhibitor, which can be used in the study of prostate and breast cancer.Formula:C27H33ClO8Purity:98.69%Color and Shape:SolidMolecular weight:521.00Ref: TM-T36375
1mg154.00€5mg371.00€10mg620.00€25mg1,341.00€50mg1,783.00€100mg2,250.00€1mL*10mM (DMSO)425.00€ONC1-13B
CAS:ONC1-13B, an androgen receptor antagonist, is used potentially for the treatment of prostate cancer.Formula:C22H16F4N4O3SPurity:99.36% - 99.85%Color and Shape:SolidMolecular weight:492.45GLPG0492
CAS:GLPG0492 is a novel selective androgen receptor modulator.Formula:C19H14F3N3O3Purity:99.58%Color and Shape:SolidMolecular weight:389.33Ref: TM-T11410L
1mg71.00€5mg156.00€10mg224.00€25mg358.00€50mg515.00€100mg692.00€200mg888.00€1mL*10mM (DMSO)166.00€Androgen receptor antagonist 5
CAS:AR antagonist 5 blocks AR (IC50: 6.17 μM), hinders LNCaP cell growth, and has anti-tumor effects in mouse models.Formula:C21H15F4N5O3SColor and Shape:SolidMolecular weight:493.43Celiprolol hydrochloride
CAS:Celiprolol hydrochloride (Selectrol) is a cardioselective beta-1 adrenergic antagonist that has intrinsic sympathomimetic activity.Formula:C20H33N3O4·HClColor and Shape:White Crystalline SolidMolecular weight:415.96VPC-14228
CAS:VPC-14228 is a specific AR-DBD inhibitor that acts by inhibiting both Y594A and Q592A mutants.Formula:C13H14N2OSPurity:99.96%Color and Shape:SolidMolecular weight:246.33N-Nitrosodicyclohexylamine
CAS:N-Nitrosodicyclohexylamine (NDCHA), an N-nitrosocompound, exhibits anti-androgenic activity by competitively binding to the androgen receptor (AR) in oppositionFormula:C12H22N2OPurity:98%Color and Shape:SolidMolecular weight:210.32Androgen receptor degrader-2
CAS:Androgen Receptor Degrader-2 (Compound 9) is a potent degrader of androgen receptors, with potential application in cancer research [1].Formula:C16H16ClN3O4Purity:98%Color and Shape:SolidMolecular weight:349.77(rel)-BMS-641988
CAS:(rel)-BMS-641988, a relative configuration of the potent nonsteroidal androgen receptor antagonist BMS-641988, holds potential for prostate cancer research.Formula:C20H20F3N3O5SPurity:98%Color and Shape:SolidMolecular weight:471.45JNJ-26146900
CAS:JNJ-26146900 is a nonsteroidal androgen receptor (AR) ligand with tissue-selective activity in rats. JNJ-26146900 binds to the rat AR with a K(i) of 400nM.Formula:C15H15F3N2O3SPurity:98%Color and Shape:SolidMolecular weight:360.35Trimegestone
CAS:Trimegestone, a highly effective oral progestogen, is used for endometrial protection, all doses inducing secretory endometrial transformation.Formula:C22H30O3Purity:98%Color and Shape:SolidMolecular weight:342.47YXG-158
CAS:YXG-158 (Compound 23-h), an orally active androgen receptor (AR) degrader and cytochrome P450 17A1 (CYP17A1) inhibitor, exhibits AR degradation with a DC50 of 1Formula:C30H36FN3OPurity:98%Color and Shape:SolidMolecular weight:473.62Androgen receptor degrader-3
CAS:Androgen Receptor Degrader-3 (ARD-3) is a compound that inhibits androgen receptor signaling and promotes the degradation of the receptor, with potentialFormula:C45H51ClN8O5Purity:98%Color and Shape:SolidMolecular weight:819.39PLK1/BRD4-IN-1
CAS:PLK1/BRD4-IN-1 (9b) is an orally active dual inhibitor of PLK1 (IC50: 22 nM) and BRD4 (IC50: 109 nM).Formula:C31H43N9O2Color and Shape:SolidMolecular weight:573.73Androgen receptor-IN-5
CAS:Androgen receptor-IN-5 is a potent inhibitor of the androgen receptor with anticancer properties.Formula:C22H10Cl2F4N4OSPurity:98%Color and Shape:SolidMolecular weight:525.31Androgen receptor degrader-1
CAS:Androgen Receptor Degrader-1 (Compound 18) is a potent agent for androgen receptor degradation, applicable in cancer research [1].Formula:C15H14ClN3O4Purity:98%Color and Shape:SolidMolecular weight:335.74JJH260
CAS:JJH260, a N-hydroxy hydantoin carbamate, inhibits AIG1 and ADTRP with IC50 values of 0.57 μM and 8.5 μM, respectively, and targets ABHD6, LYPLA1/2.Formula:C29H34ClN5O5Color and Shape:SolidMolecular weight:568.06EPI-7170
CAS:EPI-7170: Ralaniten analogue, blocks androgen receptor, inhibits transcription in AR & variants, fights enzalutamide-resistant prostate cancer.Formula:C22H28Cl3NO6SColor and Shape:SolidMolecular weight:540.88LGD-2941
CAS:LGD-2941 is an androgen receptor modulator. LGD-2941 is used for the treatment of hypogonadism, female sexual dysfunction and menopausal syndrome.Formula:C17H16F6N2O2Color and Shape:SolidMolecular weight:394.31RU 59063
CAS:RU 59063 is a prototype of a new class of high-affinity nonsteroidal androgen receptor (AR) ligands.Formula:C17H18F3N3O2SPurity:99.09%Color and Shape:SolidMolecular weight:385.4Ref: TM-T20761
1mg93.00€5mg182.00€10mg269.00€25mg429.00€50mg610.00€100mg820.00€200mg1,071.00€1mL*10mM (DMSO)197.00€
