Calcium Channel
Calcium channels are membrane proteins that regulate the flow of calcium ions into and out of cells, which is essential for various cellular functions, including muscle contraction, neurotransmitter release, and gene expression. Dysregulation of calcium channel activity is associated with conditions such as hypertension, cardiac arrhythmias, and neurological disorders. At CymitQuimica, we provide a wide selection of calcium channel modulators to support your research in cardiovascular health, neurobiology, and signal transduction.
Found 573 products of "Calcium Channel"
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ω-Conotoxin FVIA
ω-Conotoxin FVIA is an inhibitor of N-type Ca²⁺ channels (Caᵥ2.2), shown to alleviate mechanical and thermal pain abnormalities in a rat model of caudal nerveFormula:C98H164N36O33S6Purity:98%Color and Shape:SolidMolecular weight:2566.96PACAP-38 (31-38), human, mouse, rat TFA
PACAP-38 (31-38), human, mouse, rat (TFA) demonstrates potent, efficacious, and sustained stimulatory effects on sympathetic neuronal.Formula:C49H84F3N17O13Purity:98%Color and Shape:SolidMolecular weight:1176.29ω-Agatoxin TK
CAS:Selective blocker of CaV2.1 P/Q-type calcium channels.Formula:C215H337N65O70S10Purity:98%Color and Shape:SolidMolecular weight:5273.02Vesnarinone HCl
Vesnarinone HCl is an oral PDE3 inhibitor improving heart contractility, affecting calcium and potassium flux. Used in heart failure research.Formula:C22H26ClN3O4Purity:99.17%Color and Shape:SoildMolecular weight:431.91Calcium Channel Compound Library
A unique collection of 140 calcium channel blockers and agonists for high throughput and high content screening;Color and Shape:Odour SolidRef: TM-L7200
1mgTo inquire30μL*10mM (DMSO)To inquire50μL*10mM (DMSO)To inquire100μL*10mM (DMSO)To inquire250μL*10mM (DMSO)To inquireMyoregulin TFA
Myoregulin (MLN peptide) TFA, belonging to the regulin family, is a regulator of muscle performance through modulation of intracellular calcium dynamics.Formula:C239H391N53O67S3·xC2HF3O2Purity:98%Color and Shape:SolidMolecular weight:5175.17 (free base)Huwentoxin I
CAS:Huwentoxin I (HWTX-I) is a peptide toxin that targets and inhibits both voltage-gated sodium channels and N-type calcium channels.Formula:C161H246N48O44S6Purity:98%Color and Shape:SolidMolecular weight:3750.36Ser-Ala-alloresact acetate
Ser-Ala-alloresact acetate is a sperm-activating peptide (SAP) that is released by marine invertebrate eggs and plays an important role in fertilization.Formula:C44H75N13O16S2Purity:98.52%Color and Shape:SolidMolecular weight:1106.28(±)5(6)-DiHETE
CAS:Eicosapentaenoic acid is an ω-3 polyunsaturated fatty acid that is abundant in marine organisms and fish oils.Formula:C20H32O4Color and Shape:SolidMolecular weight:336.472Chlorocresol
CAS:Chlorocresol (4-Chloro-3-methylphenol) is an antiseptic medication.Formula:C7H7ClOColor and Shape:SolidMolecular weight:142.58Ethyl 4-chloro-2-oxo-1,2-dihydroquinoline-3-carboxylate
CAS:ethyl 4-chloro-2-oxo-1,2-dihydroquinoline-3-carboxylate inhibits NAD(P)H: quinone oxidoreductase 1.Formula:C12H10ClNO3Purity:99.17%Color and Shape:SolidMolecular weight:251.671-(aminomethyl)cyclopropanecarboxylic acid hydrochloride
CAS:1-(aminomethyl)cyclopropanecarboxylic acid hydrochloride inhibits L amino acid transporter proteins and the α2δ subunit of voltage-gated calcium channels.1-(
Formula:C5H10ClNO2Purity:>99.99%Color and Shape:SolidMolecular weight:151.59Caloxin 3A1
Caloxin 3A1, a biologically active peptide, is a member of the caloxins, which are inhibitors of the extracellular plasma membrane (PM) Ca2+ pumps.Formula:C83H126N22O30Purity:98%Color and Shape:SolidMolecular weight:1912.02PD 0299685
CAS:PD 0299685 is a potent α2δ ligand of the Ca2+ channel for the treatment of interstitial cystitis.Formula:C10H21NO2Purity:97.20%Color and Shape:SoildMolecular weight:187.28Cyclic ADP-ribose ammonium
cADPR ammonium is a second messenger that boosts cytosolic calcium via Ryanodine receptors and TRPM2 channels.Color and Shape:Liquidω-Conotoxin CVIF
ω-Conotoxin CVIF is a selective inhibitor of Ca v 2.2 channels, demonstrating an IC50 value of 34.3 nM in isolated rat DRG neurons.Formula:C101H170N40O33S6Purity:98%Color and Shape:SolidMolecular weight:2665.07Levamlodipine besylate Hemipentahydrate
CAS:Levamlodipine besylate hemipentahydrate is the besylate hemipentahydrate salt form of Levamlodipine. It is an orally effective calcium channel blocker with antioxidative and vasodilatory properties. This compound can reduce serum malondialdehyde (MDA) levels, enhance the activity of superoxide dismutase (SOD), and alleviate oxidative stress. Levamlodipine besylate hemipentahydrate is relevant for research in vascular dementia, hypertension, and cerebrovascular diseases.Formula:C20H25ClN2O5·C6H6O3SH2OColor and Shape:SolidMolecular weight:1224.18MCU-i11
CAS:MCU-i11 is a novel negative modulator of the MCU, binding MICU1 and impairing muscle cell growth.Formula:C28H28N4O5SPurity:98.3%Color and Shape:SolidMolecular weight:532.61Ref: TM-T9960
1mg160.00€5mg359.00€10mg512.00€25mg847.00€50mg1,159.00€100mg1,568.00€1mL*10mM (DMSO)437.00€KT-362 free base
CAS:KT-362 is a calcium channel blocker with antihypertensive properties that can be used in the study of cardiovascular disease.Formula:C22H28N2O3SPurity:99.91%Color and Shape:SoildMolecular weight:400.53MMK 1
CAS:Potent hFPR2 agonist; EC50: 1 nM (mFPR2), 2 nM (hFPR2), >10,000 nM (hFPR1). Induces monocyte/neutrophil migration, boosts IL-1β/IL-6, activates NADPH-oxidase.Formula:C75H123N19O18SPurity:98%Color and Shape:SolidMolecular weight:1610.97Candidalysin
CAS:Candidalysin is a cytolytic peptide toxin initially isolated from *Candida albicans*, exhibiting both toxic and non-toxic properties. It activates epithelial cell signaling pathways by interacting with the epithelial growth factor receptor (EGFR) on host cells, leading to the activation of matrix metalloproteinases (MMP) and calcium ion influx, which results in inflammatory responses and immune cell recruitment. Additionally, Candidalysin exhibits cytotoxicity by causing membrane damage to host cells.Formula:C153H266N38O38S2Color and Shape:SolidMolecular weight:3310.11Fasudil
CAS:Fasudil (HA-1077) is a potent inhibitor of ROCK1, PKA, PKC, and MLCK.Formula:C14H17N3O2SPurity:99.79% - 99.84%Color and Shape:SolidMolecular weight:291.37Lnd 796
CAS:Lnd 796 is an aminosteroid related to LND 623.Formula:C27H45NO7Color and Shape:SolidMolecular weight:495.65Maurocalcine TFA
Maurocalcine TFA acts as an agonist for ryanodine receptor (RyR) channels 1, 2, and 3, demonstrating cell-penetrating capabilities. It induces binding of [3H]ryanodine to RyR1 with an EC50 of 2558 nM and exhibits an apparent affinity of 14 nM for RyR2. This compound is applicable for in vivo cell tracking or other cellular imaging techniques.Formula:C156H270N56O46S6·xC2HF3O2Color and Shape:SolidMolecular weight:3858.55 (free base)Calcium Ionophore I
CAS:Calcium Ionophore I has a wide range of applications in life science related research.Formula:C38H72N2O8Color and Shape:SolidMolecular weight:685.0N-Palmitoyl Glycine
CAS:Acyl amides like AEA modulate pain/inflammation. PalGly, similar to N-acyl ethanolamines, inhibits nociception and induces calcium influx in cells.Formula:C18H35NO3Color and Shape:SolidMolecular weight:313.48Almorexant hydrochloride
CAS:Almorexant hydrochloride (ACT 078573 hydrochloride) is a dual orexin receptor antagonist that induces apoptosis and can be used to study sleep disorders.Formula:C29H32ClF3N2O3Purity:99.85%Color and Shape:SolidMolecular weight:549.02MRS1845
CAS:MRS1845 is a selective inhibitor of store-operated calcium (SOC) channel (IC50 of 1.7 μM).Formula:C21H22N2O6Purity:99.69%Color and Shape:SolidMolecular weight:398.41YM-244769
CAS:YM-244769 (3-Pyridinecarboxamide, N-[(3-aminophenyl)methyl]-6-[4-[(3-fluorophenyl)methoxy]phenoxy]-) is an effective inhibitor of Na+/Ca2+ exchange 3 (NCX3)Formula:C26H22FN3O3Purity:95.62%Color and Shape:SolidMolecular weight:443.47YM-244769 dihydrochloride
CAS:YM-244769 dihydrochloride is an effective inhibitor of Na+/Ca2+ exchange 3 (NCX3) with an IC50 of 18 nM.Formula:C26H24Cl2FN3O3Purity:98%Color and Shape:SolidMolecular weight:516.39(R)-(+)-Bay-K-8644
CAS:(R)-(+)-Bay-K-8644, a Ca2+ channel agonist, is a dihydropyridine agonist that induces central respiratory depression and inhibits platelet activation in cats.
Formula:C16H15F3N2O4Purity:96.51% - 96.51%Color and Shape:SolidMolecular weight:356.3Catharanthine
CAS:Catharanthine ((+)-3,4-Didehydrocoronaridine) suppresses nicotinic receptor-mediated diaphragm contractions (IC50=59.6 μM).Formula:C21H24N2O2Purity:99.11%Color and Shape:White PowderMolecular weight:336.43CCT129957
CAS:CCT129957 is a novel and potent phospholipase C-γ (PLC-γ) inhibitor with an IC50 of about 3 μM and a GC50 of 15 μM.CCT129957 exhibits anticancer activity andFormula:C17H15N3O3Purity:99.69%Color and Shape:SolidMolecular weight:309.32Ref: TM-T14903
1mg44.00€5mg93.00€10mg126.00€25mg220.00€50mg330.00€100mg497.00€500mg1,054.00€1mL*10mM (DMSO)92.00€TPC2-A1-N
CAS:TPC2-A1-N is a TPC2 small molecule agonist that can be used to detect different functions of TPC2 channels in intact cells.Formula:C17H9Cl2F3N2O2Purity:99.86%Color and Shape:SolidMolecular weight:401.17(S)-Lercanidipine D3 hydrochloride
CAS:(S)-Lercanidipine D3 hydrochloride is a deuterium labeled Lercanidipine D3 hydrochloride. (S)-Lercanidipine hydrochloride is an agent of antihypertensive.Formula:C36H42ClN3O6Purity:98%Color and Shape:SolidMolecular weight:651.21Norverapamil-d7 HCl
CAS:Norverapamil-d7 HCl (D591-d7 HCl) is a 2H-labeled Norverapamil HCl, a calcium channel blocker and P-gp inhibitor, also a coronary vasodilator.Formula:C26H37ClN2O4Color and Shape:SolidMolecular weight:484.08(R)-Nicardipine
CAS:(R)-Nicardipine is the less active R enantiomer of Nicardipine. Nicardipine is a blocker of calcium channel(IC50 of 1 μM for blocking cardiac calcium channels).Formula:C26H29N3O6Color and Shape:SolidMolecular weight:479.53β-Cyfluthrin
CAS:β-Cyfluthrin is a type II synthetic pyrethroid compound commonly utilized as an active ingredient in agricultural insecticide products.Formula:C22H18Cl2FNO3Color and Shape:SolidMolecular weight:434.29(R)-Lercanidipine-d3 hydrochloride
CAS:(R)-lercanidipine D3 hydrochloride is a deuterium labeled (R)-Lercanidipine hydrochloride. (R)-Lercanidipine D3 (hydrochloride) is a calcium channel blocker.Formula:C36H42ClN3O6Purity:98%Color and Shape:SolidMolecular weight:651.21Nicardipine-d3 hydrochloride
CAS:Nicardipine D3 hydrochloride is the deuterium labeled Nicardipine hydrochloride.Formula:C26H30ClN3O6Purity:98%Color and Shape:SolidMolecular weight:519HSK16149
CAS:HSK16149 is a novel ligand of voltage-gated calcium channel (VGCC) α 2 δ subunit with analgesic activity.Formula:C12H19NO2Color and Shape:SolidMolecular weight:209.28A 839977
CAS:A 839977 is a P2X7 receptor antagonist with analgesic activity that inhibits BzATP-induced calcium efflux from the P2X7 receptor for the study of renal fibrosisFormula:C19H14Cl2N6OPurity:98.01%Color and Shape:SolidMolecular weight:413.26(S)-Nicardipine
CAS:(S)-Nicardipine is the less active S enantiomer of Nicardipine. Nicardipine is a blocker of calcium channel(IC50 of 1 μM for blocking cardiac calcium channels).Formula:C26H29N3O6Color and Shape:SolidMolecular weight:479.53Norverapamil-d7
CAS:Norverapamil D7 is a deuterium labeled Norverapamil . Norverapamil is a blocker of L-type calcium channel and an inhibitor of P-glycoprotein (P-gp) function .Formula:C26H36N2O4Purity:98%Color and Shape:SolidMolecular weight:447.62Hexadecylphosphoserine TFA
Hexadecylphosphoserine is a type of phospholipid molecule that incorporates a long-chain alkyl group (hexadecyl) and a phosphatidylserine group, granting it high affinity for cell membranes. This compound exhibits antitumor activity by modulating [Ca++]i and related signaling pathways, making it useful for breast cancer research.Formula:C21H41F3NO8PColor and Shape:SolidMolecular weight:523.52Magnesium sulfate
CAS:Magnesium sulfate: anticonvulsant for eclampsia, tocolytic agent.Formula:MgSO4Purity:98%Color and Shape:SolidMolecular weight:120.37Etripamil
CAS:Etripamil is a fast-acting intranasal L-type calcium-channel blocker for Paroxysmal Supraventricular Tachycardia.Formula:C27H36N2O4Purity:99.47% - 99.83%Color and Shape:SolidMolecular weight:452.59Ref: TM-T15257
1mg52.00€2mg74.00€5mg110.00€10mg169.00€25mg295.00€50mg447.00€100mg670.00€200mg1,054.00€Dronedarone
CAS:Dronedarone (SR 33589) is an amiodarone analogue which has an effective and promising treatment for Atrial fibrillation.Formula:C31H44N2O5SPurity:98.85% - 99.99%Color and Shape:SolidMolecular weight:556.76L-Phenylalanine
CAS:L-Phenylalanine (3-Phenyl-L-alanine) is an essential amino acid and the precursor of the amino acid tyrosine, acts as an antagonist at α2δ calcium channels.Formula:C9H11NO2Purity:99.37% - 99.87%Color and Shape:Solid CrystallineMolecular weight:165.19JNJ-26990990
CAS:"JNJ-26990990: broad-spectrum anticonvulsant, less side effects than topiramate, potential for pain and depression treatment; Phase II in 2007."Formula:C9H10N2O2S2Purity:97.37%Color and Shape:SolidMolecular weight:242.32Ref: TM-T27673
1mg131.00€5mg286.00€10mg424.00€25mg702.00€50mg938.00€100mg1,311.00€1mL*10mM (DMSO)261.00€
