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GABA Receptor

GABA Receptor

GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.

Found 336 products of "GABA Receptor"

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  • CP-409092 hydrochloride

    CAS:
    <p>CP-409092 hydrochloride is a partial agonist of the GABAA receptor with anti-anxiety activity.</p>
    Formula:C17H20ClN3O2
    Color and Shape:Solid
    Molecular weight:333.81
  • CGP 46381

    CAS:
    <p>CGP 46381 is a GABAB receptor antagonist.</p>
    Formula:C10H22NO2P
    Purity:98%
    Color and Shape:White Solid
    Molecular weight:219.26
  • GABAA receptor agent 5

    CAS:
    <p>Compound 018 is a potent γ-GABAAR antagonist, Ki of 0.020 μM, with low membrane permeability.</p>
    Formula:C21H25N3O2S
    Color and Shape:Solid
    Molecular weight:383.51
  • BGT1-IN-9

    CAS:
    <p>BGT1-IN-9 is an M1 muscarinic agonist.</p>
    Formula:C5H10ClN3O2
    Color and Shape:Solid
    Molecular weight:179.605
  • CCD-3693

    CAS:
    <p>CCD-3693 is a gamma-aminobutyric acid (GABA) receptor agonist.</p>
    Formula:C21H31F3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:372.46
  • GABA-AT-IN-1

    CAS:
    <p>GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.</p>
    Formula:C23H18N2O6
    Color and Shape:Solid
    Molecular weight:418.4
  • GABAA receptor agent 8

    CAS:
    <p>Compound 5e, a GABAA receptor modulator, shows potent anticonvulsant effects with low neurotoxicity for epilepsy research.</p>
    Formula:C19H16N4O
    Color and Shape:Solid
    Molecular weight:316.36
  • ZAPA sulfate

    CAS:
    <p>GABAA receptors agonist</p>
    Formula:C4H8N2O6S2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:244.25
  • TPMPA

    CAS:
    <p>GABAA-ρ antagonist</p>
    Formula:C6H12NO2P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:161.14
  • TG41

    CAS:
    <p>TG41 is a GABAA receptors positive modulator.</p>
    Formula:C18H13BrCl2N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:440.12
  • FG8119

    CAS:
    <p>FG8119 is a novel benzodiazepine agonist with potential anticonvulsant and antiepileptic activity for the study of neurological disorders.</p>
    Formula:C17H15N5O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:321.33
  • GABAA receptor agent 6

    CAS:
    <p>GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with low cellular membrane permeability (Ki = 0.56 μM) [1].</p>
    Formula:C18H25N3O2
    Color and Shape:Solid
    Molecular weight:315.41
  • TB 21007

    CAS:
    <p>GABAA receptor inverse agonist</p>
    Formula:C15H17NO2S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:339.5
  • SL-651498

    CAS:
    <p>SL-651498, a GABAA receptor agonist, is used potentially for the treatment of anxiety.</p>
    Formula:C23H20FN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:389.42
  • Bamaluzole

    CAS:
    <p>Bamaluzole is an agonist of GABA receptor.</p>
    Formula:C14H12ClN3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:273.72
  • NAP-1

    CAS:
    <p>NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).</p>
    Formula:C20H18ClNO2
    Color and Shape:Solid
    Molecular weight:339.82
  • GABAA receptor agent 7

    CAS:
    <p>Compound 5c, a GABAA receptor modulator with anticonvulsant properties and low neurotoxicity, is promising for epilepsy research.</p>
    Formula:C18H13ClN4O
    Color and Shape:Solid
    Molecular weight:336.77
  • MRK-623

    CAS:
    <p>MRK-623 (14k) is an oral GABA A agonist with high affinity for α1/α2/α3/α5 subunits and anxiolytic properties.</p>
    Formula:C20H17FN4O
    Color and Shape:Solid
    Molecular weight:348.37
  • Etbicyphat

    CAS:
    <p>Etbicyphat: potent GABA(A) antagonist, induces epileptiform activity, binds to GABA/benzodiazepine receptors.</p>
    Formula:C6H11O4P
    Color and Shape:Solid
    Molecular weight:178.12
  • TCS 1105

    CAS:
    <p>TCS 1105 is a GABAA BZR ligand, blocking Sema3A and altering mouse anxiety, aggression, and social dominance.</p>
    Formula:C17H13FN2O2
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:296.3
  • Pipazethate

    CAS:
    <p>Pipipyrazine is a nonnarcotic oral cough suppressant, cough suppressant.</p>
    Formula:C21H25N3O3S
    Color and Shape:Solid
    Molecular weight:399.51
  • NNC052090

    CAS:
    <p>NNC052090 inhibits GABA uptake, favoring hBGT-1 (Ki=1.4μM), affects α1/D2 receptors (IC50=266/1632nM).</p>
    Formula:C27H30N2O2
    Color and Shape:Solid
    Molecular weight:414.54
  • RU 33965

    CAS:
    <p>RU 33965, a 3-cyclopropyl carbonyl imidazobenzodiazepine, act as a low-efficacy benzodiazepine receptor inverse agonist.</p>
    Formula:C16H15N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:281.31
  • ZK93423

    CAS:
    <p>ZK93423: potent benzodiazepine agonist, IC50=1nM, non-selective, Ki=4.1-6nM for α1-α5 GABAA subunits.</p>
    Formula:C23H22N2O4
    Color and Shape:Solid
    Molecular weight:390.43
  • GABAA receptor modulator-2

    CAS:
    <p>Compound 20: Selective, oral α5-GABAAR inhibitor, Ki: 4.1 nM. High stability, CNS safe.</p>
    Formula:C22H22FN3O5S
    Color and Shape:Solid
    Molecular weight:459.49
  • Carburazepam

    CAS:
    <p>Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.</p>
    Formula:C17H16ClN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.78
  • UMB68 sodium

    CAS:
    <p>UMB-68 is a GHB receptor ligand with no affinity (IC(50) &gt;100 microM) at GABA(A) or GABA(B) receptors.</p>
    Formula:C6H12NaO3
    Color and Shape:Solid
    Molecular weight:155.149
  • (+)-Nipecotic acid

    CAS:
    <p>(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.</p>
    Formula:C6H11NO2
    Purity:99.38%
    Color and Shape:Solid
    Molecular weight:129.16
  • (S)-SNAP5114

    CAS:
    <p>(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.</p>
    Formula:C30H35NO6
    Purity:97%
    Color and Shape:Solid
    Molecular weight:505.6
  • Radequinil

    CAS:
    <p>Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).</p>
    Formula:C18H14N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:334.33
  • 3α,21-Dihydroxy-5α-pregnan-20-one

    CAS:
    <p>3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.</p>
    Formula:C21H34O3
    Purity:98.00%
    Color and Shape:Solid
    Molecular weight:334.49
  • Chlormethiazole edisylate

    CAS:
    <p>Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic.</p>
    Formula:C8H14ClNO6S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:351.85
  • COR628

    CAS:
    <p>COR628 is the GABA(B) receptor positive allosteric modulator.</p>
    Formula:C16H23NO3S
    Color and Shape:Solid
    Molecular weight:309.42
  • trans-4-Hydroxycrotonic acid

    CAS:
    <p>ligand of γ-hydroxybutyric acid (GHB) receptor</p>
    Formula:C4H6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:102.09
  • LY 81067

    CAS:
    <p>LY 81067, a new anticonvulsant, prevents PTZ- and picrotoxin-induced seizures in mice via picrotoxin site interaction.</p>
    Formula:C22H24N4O
    Color and Shape:Solid
    Molecular weight:360.45
  • U 90042

    CAS:
    <p>GABAA receptor ligand</p>
    Formula:C17H13ClN6O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.78
  • COR627

    CAS:
    <p>COR627 is the GABA receptor positive allosteric modulator.</p>
    Formula:C20H27NO3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:361.5
  • CPP-115

    CAS:
    <p>CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.</p>
    Formula:C7H9F2NO2
    Color and Shape:Solid
    Molecular weight:177.15
  • JY-XHe-053

    CAS:
    <p>JY-XHe-053 is a selective modulator of GABAA receptors.</p>
    Formula:C22H16FN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:373.38
  • HIE-124

    CAS:
    <p>HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.</p>
    Formula:C10H12N2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:240.28
  • Suclofenide

    CAS:
    <p>Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.</p>
    Formula:C16H13ClN2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:364.8
  • (S)-Baclofen

    CAS:
    <p>(S)-Baclofen may treat hyperacusis and tinnitus by reducing auditory pathway excitation.</p>
    Formula:C10H12ClNO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:213.66
  • ABP-700

    CAS:
    <p>ABP-700 is a positive allosteric modulator of the GABAA receptor.</p>
    Formula:C17H18N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:314.34
  • DAA-1097

    CAS:
    <p>DAA-1097 is a novel ligand of peripheral benzodiazepine receptor.</p>
    Formula:C24H24ClNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:409.91
  • (S)-3-Carboxy-4-hydroxyphenylglycine

    CAS:
    <p>group I metabotropic glutamate receptor antagonist and group II mGlu agonist</p>
    Formula:C9H9NO5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:211.17
  • PNU-107484A

    CAS:
    <p>PNU-107484A is a unique GABA(A) receptor ligand.</p>
    Formula:C18H23ClN6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:358.87
  • GS 39783

    CAS:
    <p>GS 39783 is a positive allosteric modulator (PAM) of GABABR, which reduces the motivational properties of alcohol and the conditioned reinforcement and</p>
    Formula:C15H23N5O2S
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:337.44
  • SCH 50911

    CAS:
    <p>SCH 50911 is a selective GABA(B) receptor antagonist with IC50: 1.1 μM, boosting 3H overflow at IC50: 3 μM.</p>
    Formula:C8H15NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:173.21
  • Anxiolytic/nonsedative agent-1

    CAS:
    <p>TCS 1205: Selective GABAA agonist, BzR affinity in bovine brain (Kis: 14-239 nM), α2 efficacy in vitro, anxioselective in vivo.</p>
    Formula:C18H15N3O4
    Purity:98.61%
    Color and Shape:Solid
    Molecular weight:337.33
  • SCH 50911 hydrochloride

    CAS:
    <p>SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).</p>
    Formula:C8H16ClNO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:209.67
  • Bifenazate

    CAS:
    <p>Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.</p>
    Formula:C17H20N2O3
    Purity:99.62%
    Color and Shape:Solid Crystalline
    Molecular weight:300.35
  • E2730

    CAS:
    <p>E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.</p>
    Formula:C9H8F4N2O2S
    Purity:98.22% - 98.54%
    Color and Shape:Solid
    Molecular weight:284.23
  • U-89843A

    CAS:
    <p>U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].</p>
    Formula:C16H24ClN5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:321.85
  • (R)-Baclofen hydrochloride

    CAS:
    <p>Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.</p>
    Formula:C10H13Cl2NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:250.12
  • Lesogaberan

    CAS:
    <p>Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity (Ki 1.4 μM).</p>
    Formula:C3H9FNO2P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:141.08
  • Tracazolate hydrochloride

    CAS:
    <p>Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.</p>
    Formula:C16H25ClN4O2
    Purity:99.52%
    Color and Shape:Solid
    Molecular weight:340.85
  • RO 4938581

    CAS:
    <p>RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).</p>
    Formula:C13H8BrF2N5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.14
  • AZD 3043

    CAS:
    <p>AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.</p>
    Formula:C19H29NO5
    Purity:98.19% - 99.55%
    Color and Shape:Solid
    Molecular weight:351.44
  • Phaclofen

    CAS:
    <p>GABAB antagonist</p>
    Formula:C9H13ClNO3P
    Purity:99.32%
    Color and Shape:White Solid
    Molecular weight:249.63
  • Panadiplon

    CAS:
    <p>Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment of</p>
    Formula:C18H17N5O2
    Purity:98.30% - 98.94%
    Color and Shape:Solid
    Molecular weight:335.36
  • Cirsimaritin

    CAS:
    <p>Cirsimaritin has anti-bacterial, anti-inflammatory, anti-tumor, antioxidant effects, and protects kidneys; it weakly targets GABAA receptors.</p>
    Formula:C17H14O6
    Purity:99.9%
    Color and Shape:Solid
    Molecular weight:314.29
  • Progabide

    CAS:
    <p>Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.</p>
    Formula:C17H16ClFN2O2
    Purity:99.68%
    Color and Shape:Solid
    Molecular weight:334.77
  • Saripidem

    CAS:
    <p>Saripidem (SL-85.0274) is a compound with anxiolytic activity.</p>
    Formula:C19H20ClN3O
    Purity:99.45%
    Color and Shape:Solid
    Molecular weight:341.83
  • NS-2710

    CAS:
    <p>NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.</p>
    Formula:C22H20N4O
    Purity:99.7% - 99.82%
    Color and Shape:Solid
    Molecular weight:356.42
  • ELB-139

    CAS:
    <p>ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.</p>
    Formula:C14H16ClN3O
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:277.75
  • Ru-32514

    CAS:
    <p>Ru-32514 is a benzodiazepine receptor agonist.</p>
    Formula:C18H17N3O2
    Purity:99.21%
    Color and Shape:Solid
    Molecular weight:307.35
  • Fengabine

    CAS:
    <p>Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.</p>
    Formula:C17H17Cl2NO
    Purity:99%
    Color and Shape:Solid
    Molecular weight:322.23
  • Nerisopam

    CAS:
    <p>Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.</p>
    Formula:C18H19N3O2
    Purity:97.07%
    Color and Shape:Solid
    Molecular weight:309.36
  • DMCM hydrochloride

    CAS:
    <p>DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.</p>
    Formula:C17H19ClN2O4
    Purity:99.56%
    Color and Shape:Solid
    Molecular weight:350.8
  • Suriclone

    CAS:
    <p>Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.</p>
    Formula:C20H20ClN5O3S2
    Purity:99.21% - 99.73%
    Color and Shape:Solid
    Molecular weight:477.99
  • NNC 05-711

    CAS:
    <p>NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.</p>
    Formula:C21H23ClN2O3
    Purity:99.92%
    Color and Shape:Solid
    Molecular weight:386.87
  • Riluzole hydrochloride

    CAS:
    <p>Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).</p>
    Formula:C8H6ClF3N2OS
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:270.66
  • BPDBA

    CAS:
    <p>BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and</p>
    Formula:C19H20Cl2N2O
    Purity:99.37% - 99.95%
    Color and Shape:Solid
    Molecular weight:363.28
  • RWJ-51204

    CAS:
    <p>RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.</p>
    Formula:C21H19F2N3O3
    Purity:99.57% - 99.95%
    Color and Shape:Solid
    Molecular weight:399.39
  • Lirequinil

    CAS:
    <p>Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.</p>
    Formula:C26H25ClN2O3
    Purity:98.54%
    Color and Shape:Solid
    Molecular weight:448.94
  • L-838417

    CAS:
    <p>L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disorders</p>
    Formula:C19H19F2N7O
    Purity:98.12% - 99.70%
    Color and Shape:Solid
    Molecular weight:399.4
  • Divaplon

    CAS:
    <p>Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.</p>
    Formula:C17H17N3O2
    Purity:97.44% - 98.25%
    Color and Shape:Solid
    Molecular weight:295.34
  • Alpidem

    CAS:
    <p>Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.</p>
    Formula:C21H23Cl2N3O
    Purity:99.56% - 99.97%
    Color and Shape:White To Off-White Solid
    Molecular weight:404.33
  • Sarmazenil

    CAS:
    <p>Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.</p>
    Formula:C15H14ClN3O3
    Purity:99.46%
    Color and Shape:Solid
    Molecular weight:319.74
  • Golexanolone

    CAS:
    <p>Golexanolone can be used to study neurological diseases.</p>
    Formula:C21H31NO2
    Purity:99.90% - 99.99%
    Color and Shape:Solid
    Molecular weight:329.48
  • Muscimol HBr

    CAS:
    <p>Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.</p>
    Formula:C4H7BrN2O2
    Purity:98.13%
    Color and Shape:Off-White Powder
    Molecular weight:195.01
  • DSP-0565

    CAS:
    <p>DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.</p>
    Formula:C14H12FNO
    Purity:99.51% - 99.56%
    Color and Shape:Solid
    Molecular weight:229.25
  • CGP 55845 hydrochloride

    CAS:
    <p>CGP55845 hydrochloride is a potent and selective GABAB receptor antagonist with an IC 50 of 6 nM which can be used in neurological research [1] [2].</p>
    Formula:C18H23Cl3NO3P
    Color and Shape:Solid
    Molecular weight:438.71
  • FGIN-1-27

    CAS:
    <p>FGIN-1-27 is a high-affinity agonist of the translocator protein and a specific peripheral benzodiazepine receptor (PBR) ligand(Ki = 5.0 nM).</p>
    Formula:C28H37FN2O
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:436.6
  • GMA-839

    CAS:
    <p>GMA-839 is a selective modulator of gamma-aminobutyric acid(A) receptors.</p>
    Formula:C21H31F3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:388.46
  • NO-711ME

    CAS:
    <p>NO-711ME (N-O711 Methyl ester) is a prodrug of NO-711. It also is a potent and selective GABA uptake inhibitor.</p>
    Formula:C22H24N2O3
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:364.44
  • U 89843A

    CAS:
    <p>U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.</p>
    Formula:C16H23N5
    Purity:99.62%
    Color and Shape:Solid
    Molecular weight:285.39
  • (+)-Bicuculline methiodide

    CAS:
    <p>(+)-Bicuculline methiodide is a GABAA receptor blocker that blocks epileptogens and may be used in the study of neurological disorders.</p>
    Formula:C21H20INO6
    Purity:99.24%
    Color and Shape:Solid
    Molecular weight:509.29
  • CP-409092

    CAS:
    <p>CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.</p>
    Formula:C17H19N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:297.35
  • mGAT3/4-IN-2

    CAS:
    <p>mGAT3/4-IN-2 are potent inhibitors of mGAT3/mGAT4 with their pIC50 values of 5.44 and 5.25, respectively.</p>
    Formula:C26H32ClN3OS2
    Color and Shape:Solid
    Molecular weight:502.13
  • COR659

    CAS:
    <p>COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.</p>
    Formula:C16H16ClNO3S
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:337.82
  • Diproqualone

    CAS:
    <p>Diproqualone, analogous to methaqualone, exhibits sedative, anxiolytic, anti-inflammatory, and analgesic properties [1].</p>
    Formula:C12H14N2O3
    Color and Shape:Solid
    Molecular weight:234.255
  • ADX71441

    CAS:
    <p>ADX71441, a GABAB PAM, lengthens urinary latencies, lessens events &amp; volume, and may aid in alcoholism and bladder pain.</p>
    Formula:C19H15ClF2N4O4
    Color and Shape:Solid
    Molecular weight:436.8
  • Adipiplon

    CAS:
    <p>Adipiplon(NG2-73, NG273) is a novel selective gamma-aminobutyric acid (GABA) partial agonist.</p>
    Formula:C18H18FN7
    Color and Shape:Solid
    Molecular weight:351.38
  • PZ-II-029

    CAS:
    <p>PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.</p>
    Formula:C18H15N3O3
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:321.33
  • CGP 64213

    CAS:
    <p>CGP 64213 is a GABAb receptor agonist.</p>
    Formula:C26H36IN2O7P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:646.45
  • (-)-Bicuculline methochloride

    CAS:
    <p>(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.</p>
    Formula:C21H20ClNO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:417.84
  • GABAA receptor agent 2 TFA

    CAS:
    <p>Potent GABAA antagonist; IC50: 24 nM (α1β2γ2), Ki: 28 nM (rat); inactive on human GABA transporters.</p>
    Formula:C22H22F3N3O3
    Color and Shape:Solid
    Molecular weight:433.42
  • JM-1232

    CAS:
    <p>JM-1232 is a sedative and hypnotic drug being researched as a potential anesthetic.</p>
    Formula:C24H27N3O2
    Color and Shape:Solid
    Molecular weight:389.49
  • CGP-54626 free base

    CAS:
    <p>CGP-54626 is a selective antagonist of the GABAB receptor (IC50 = 4 nM ).</p>
    Formula:C18H28Cl2NO3P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:408.3