GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
Found 371 products of "GABA Receptor"
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U-7524
CAS:U-7524 (AOAA), an inhibitor of GABA-T and other PLP-dependent enzymes, disrupts the Schiff base linkage, forming oxime complexes.Formula:C2H5NO3Color and Shape:SolidMolecular weight:91.07Alfadolone
CAS:Alfadolone is an anesthetic derivative of pregnanedione.Formula:C21H32O4Color and Shape:SolidMolecular weight:348.48Y 23684
CAS:Y-23684 is an anxiolytic drug with a novel chemical structure. It has similar effects to benzodiazepine drugs and is classed as a nonbenzodiazepine anxiolytic.Formula:C18H13ClN2O2SPurity:98%Color and Shape:SolidMolecular weight:356.83Ro 22-8515
CAS:Ro 22-8515 is the ligand of benzodiazepine receptor.Formula:C18H12Cl2N2OColor and Shape:SolidMolecular weight:343.21Cyprodenate
CAS:Cyprodenate (Actebral) is a potent orally active brain-activating agent with appetite-suppressing properties, useful in studying metabolic.Formula:C13H25NO2Color and Shape:SolidMolecular weight:227.34Ref: TM-T72977
1mg37.00€5mg72.00€10mg99.00€25mg169.00€50mg229.00€100mg320.00€200mg479.00€1mL*10mM (DMSO)79.00€ZK-91296
CAS:ZK-91296: GABA agonist, lowers anxiety without sedation, may target specific BZ receptor subtype.Formula:C23H22N2O4Purity:98%Color and Shape:SolidMolecular weight:390.43DS1
CAS:DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse.Formula:C18H10Br2ClN3OSColor and Shape:SolidMolecular weight:511.62SCH-50910 free base
CAS:SCH-50910 is an antagonist of GABAB receptor.Formula:C8H15NO3Color and Shape:SolidMolecular weight:173.21Profadol hydrochloride
CAS:Profadol hydrochloride acts as a mixed agonist-antagonist of the μ-opioid receptor with analgesic activity.Formula:C14H22ClNOPurity:98%Color and Shape:SolidMolecular weight:255.783-Methyl-GABA
CAS:3-Methyl-GABA activates GABA aminotransferase, fits GABAaR, stimulates GAD, and acts as an anticonvulsant.Formula:C20H30N2O10S2Purity:98%Color and Shape:SolidMolecular weight:522.59Ro15-4513
CAS:Ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. Ro15-4513 is an effective ethanol antagonist.Formula:C15H14N6O3Purity:98%Color and Shape:SolidMolecular weight:326.31Ro 14-7437
CAS:Ro 14-7437 is an antagonist of GABA-benzodiazepine receptor.Formula:C15H15N3O3Color and Shape:SolidMolecular weight:285.3Adinazolam Mesylate
CAS:Adinazolam Mesylate is an anxiolytic and antidepressant agent. Adinazolam Mesylate binds to peripheral-type benzodiazepine receptors that interact allosterically with GABA receptors as an agonist to produce inhibitory effects.Formula:C20H22ClN5O3SPurity:98%Color and Shape:SolidMolecular weight:447.94Ro 15-1310
CAS:Ro 15-3505, a benzodiazepine receptor partial inverse agonist, has shown the ability to improve impaired recent memory of aged mice.Formula:C15H14ClN3O3Color and Shape:SolidMolecular weight:319.74CP-457920
CAS:CP-457920 is a selective α5 GABAA receptor inverse agonist that is suitable for investigating dementia in Alzheimer's disease.Formula:C18H17N3O3Purity:99.06% - 99.74%Color and Shape:SolidMolecular weight:323.352-Hydroxysaclofen
CAS:2-Hydroxysaclofen is a GABAB receptor antagonist.Formula:C9H12ClNO4SPurity:98%Color and Shape:White SolidMolecular weight:265.71CGS 20625
CAS:partial agonist for the benzodiazepine binding site of the GABAA receptorFormula:C18H19N3O2Purity:99.61%Color and Shape:SolidMolecular weight:309.36SX-3228
CAS:SX-3228 is a selective agonist of benzodiazepine1 (BZ1) receptor(IC50 of 17 nM).Formula:C18H18N4O3Purity:98%Color and Shape:SolidMolecular weight:338.36Org 20599
CAS:GABAA receptor agonistFormula:C25H40ClNO3Purity:98%Color and Shape:SolidMolecular weight:438.04U-101017
CAS:U-101017 is a partial benzodiazepine receptor and GABAA receptor agonist.Formula:C23H27ClN4O3Purity:98%Color and Shape:SolidMolecular weight:442.94TPA-023B
CAS:TPA-023B: oral GABAA α2/α3 agonist (Kis: 0.73/2 nM), α1 antagonist (Ki: 1.8 nM), non-sedating anxiolytic.Formula:C21H15F2N5OPurity:98%Color and Shape:SolidMolecular weight:391.37CGP 7930
CAS:Positive allosteric modulator of GABAB receptorsFormula:C19H32O2Purity:98%Color and Shape:SolidMolecular weight:292.46SCH 50911 hydrochloride
CAS:SCH 50911 hydrochloride is a selective, orally-active and competitive antagonist of γ-Aminobutyric acid B GABA(B) receptor(IC50 : 1.1 μM).Formula:C8H16ClNO3Purity:98%Color and Shape:SolidMolecular weight:209.67BHF-177
CAS:BHF-177 is a positive allosteric modulator of the GABAB receptor. BHF-177 reduces self-administration of nicotine in animal studies.Formula:C19H20F3N3Color and Shape:SolidMolecular weight:347.38CGS8216
CAS:CGS8216 shows analgesic activity at high doses, has anxiolytic activity, and can be used to study immune system disorders.Formula:C16H11N3OPurity:98.53%Color and Shape:SolidMolecular weight:261.28DS2
CAS:Positive allosteric modulator of δ-subunit containing GABAA receptorsFormula:C18H12ClN3OSPurity:98%Color and Shape:SolidMolecular weight:353.83(±)-Homoproline Hydrochloride
CAS:(±)-Homoproline Hydrochloride. Affordable Excellence: Reliable Quality You Can TrustFormula:C6H12ClNO2Purity:99.69%Color and Shape:SolidMolecular weight:165.62MK-0343
CAS:MK0343 is an orally bioavailable GABAA receptor subtype-selective partial agonist and is a non-sedating anxiolytic.Formula:C19H17F2N7OPurity:98%Color and Shape:SolidMolecular weight:397.3817-PA
CAS:17-PA is a GABAA receptor antagonist.Formula:C25H34OPurity:98%Color and Shape:SolidMolecular weight:350.54Bifenazate
CAS:Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.Formula:C17H20N2O3Purity:99.62%Color and Shape:Solid CrystallineMolecular weight:300.35CGP11952
CAS:CGP11952 is same the benzodiazepines in its pharmacological action and it also is an experimental benzodiazepine derivative.Formula:C21H21Cl2N5O2Purity:98%Color and Shape:SolidMolecular weight:446.33E2730
CAS:E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.Formula:C9H8F4N2O2SPurity:98.22% - 98.54%Color and Shape:SolidMolecular weight:284.23U-89843A
CAS:U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].Formula:C16H24ClN5Purity:98%Color and Shape:SolidMolecular weight:321.85(R)-Baclofen hydrochloride
CAS:Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.Formula:C10H13Cl2NO2Purity:98%Color and Shape:SolidMolecular weight:250.12NO 711
CAS:NO 711（NNC-711 free acid） is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.Formula:C21H22N2O3Purity:99.70%Color and Shape:SolidMolecular weight:350.41AZD 3043
CAS:AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.Formula:C19H29NO5Purity:98.19% - 99.55%Color and Shape:SolidMolecular weight:351.44mGAT3/4-IN-1
CAS:mGAT3/4-IN-1 inhibits mGAT3/4 with pIC50: 5.31/5.24, reduces neuropathic pain in diabetic mice.Formula:C26H31ClN2O2S2Color and Shape:SolidMolecular weight:503.12GABAA receptor agent 4
CAS:Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.Formula:C17H24N2OColor and Shape:SolidMolecular weight:272.39Ro 19-4603
CAS:Benzodiazepine inverse agonistFormula:C15H17N3O3SPurity:98%Color and Shape:SolidMolecular weight:319.38GABAA receptor agent 6
CAS:GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with low cellular membrane permeability (Ki = 0.56 μM) [1].Formula:C18H25N3O2Color and Shape:SolidMolecular weight:315.41TB 21007
CAS:GABAA receptor inverse agonistFormula:C15H17NO2S3Purity:98%Color and Shape:SolidMolecular weight:339.5SL-651498
CAS:SL-651498, a GABAA receptor agonist, is used potentially for the treatment of anxiety.Formula:C23H20FN3O2Purity:98%Color and Shape:SolidMolecular weight:389.42Bamaluzole
CAS:Bamaluzole is an agonist of GABA receptor.Formula:C14H12ClN3OPurity:98%Color and Shape:SolidMolecular weight:273.72NAP-1
CAS:NAP-1 is an anesthetic that enhances CA1 brain inhibition in rats and causes tadpole sedation (EC50 = 0.53 μM).Formula:C20H18ClNO2Color and Shape:SolidMolecular weight:339.82GABAA receptor agent 7
CAS:Compound 5c, a GABAA receptor modulator with anticonvulsant properties and low neurotoxicity, is promising for epilepsy research.Formula:C18H13ClN4OColor and Shape:SolidMolecular weight:336.77MRK-623
CAS:MRK-623 (14k) is an oral GABA A agonist with high affinity for α1/α2/α3/α5 subunits and anxiolytic properties.Formula:C20H17FN4OColor and Shape:SolidMolecular weight:348.37Lesogaberan
CAS:Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity (Ki 1.4 μM).Formula:C3H9FNO2PPurity:98%Color and Shape:SolidMolecular weight:141.08FG8119
CAS:FG8119 is a novel benzodiazepine agonist with potential anticonvulsant and antiepileptic activity for the study of neurological disorders.Formula:C17H15N5O2Purity:>99.99%Color and Shape:SolidMolecular weight:321.33TG41
CAS:TG41 is a GABAA receptors positive modulator.Formula:C18H13BrCl2N2O2Purity:98%Color and Shape:SolidMolecular weight:440.12Etbicyphat
CAS:Etbicyphat: potent GABA(A) antagonist, induces epileptiform activity, binds to GABA/benzodiazepine receptors.Formula:C6H11O4PColor and Shape:SolidMolecular weight:178.12TCS 1105
CAS:TCS 1105 is a GABAA BZR ligand, blocking Sema3A and altering mouse anxiety, aggression, and social dominance.Formula:C17H13FN2O2Purity:99.75%Color and Shape:SolidMolecular weight:296.3Pipazethate
CAS:Pipipyrazine is a nonnarcotic oral cough suppressant, cough suppressant.Formula:C21H25N3O3SColor and Shape:SolidMolecular weight:399.51NNC052090
CAS:NNC052090 inhibits GABA uptake, favoring hBGT-1 (Ki=1.4μM), affects α1/D2 receptors (IC50=266/1632nM).Formula:C27H30N2O2Color and Shape:SolidMolecular weight:414.54RU 33965
CAS:RU 33965, a 3-cyclopropyl carbonyl imidazobenzodiazepine, act as a low-efficacy benzodiazepine receptor inverse agonist.Formula:C16H15N3O2Purity:98%Color and Shape:SolidMolecular weight:281.31NCS-382
CAS:γ-Hydroxybutyric acid antagonistFormula:C13H14O3Purity:98%Color and Shape:SolidMolecular weight:218.25ZAPA sulfate
CAS:GABAA receptors agonistFormula:C4H8N2O6S2Purity:98%Color and Shape:SolidMolecular weight:244.25ZK93423
CAS:ZK93423: potent benzodiazepine agonist, IC50=1nM, non-selective, Ki=4.1-6nM for α1-α5 GABAA subunits.Formula:C23H22N2O4Color and Shape:SolidMolecular weight:390.43β-CCB
CAS:benzodiazepine receptor ligandFormula:C16H16N2O2Purity:98%Color and Shape:SolidMolecular weight:268.31GABAA receptor modulator-2
CAS:Compound 20: Selective, oral α5-GABAAR inhibitor, Ki: 4.1 nM. High stability, CNS safe.Formula:C22H22FN3O5SColor and Shape:SolidMolecular weight:459.49Carburazepam
CAS:Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.Formula:C17H16ClN3O2Purity:98%Color and Shape:SolidMolecular weight:329.78UMB68 sodium
CAS:UMB-68 is a GHB receptor ligand with no affinity (IC(50) >100 microM) at GABA(A) or GABA(B) receptors.Formula:C6H12NaO3Color and Shape:SolidMolecular weight:155.149Pregabalin arenacarbil
CAS:Pregabalin arenacarbil is a gabamimetic.Formula:C15H27NO6Color and Shape:SolidMolecular weight:317.38GABAA receptor agent 8
CAS:Compound 5e, a GABAA receptor modulator, shows potent anticonvulsant effects with low neurotoxicity for epilepsy research.Formula:C19H16N4OColor and Shape:SolidMolecular weight:316.36Tracazolate hydrochloride
CAS:Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.Formula:C16H25ClN4O2Purity:99.52%Color and Shape:SolidMolecular weight:340.85CGP 36216 hydrochloride
CAS:CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).Formula:C5H14NO2PPurity:98%Color and Shape:SolidMolecular weight:151.14(+)-Nipecotic acid
CAS:(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.Formula:C6H11NO2Purity:99.38%Color and Shape:SolidMolecular weight:129.16GABA-AT-IN-1
CAS:GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.Formula:C23H18N2O6Color and Shape:SolidMolecular weight:418.4(S)-SNAP5114
CAS:(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.Formula:C30H35NO6Purity:98.20%Color and Shape:SolidMolecular weight:505.6Ref: TM-T16831
5mg49.00€10mg73.00€25mg152.00€50mg213.00€100mg309.00€200mg423.00€1mL*10mM (DMSO)49.00€Radequinil
CAS:Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).Formula:C18H14N4O3Purity:98%Color and Shape:SolidMolecular weight:334.33Phaclofen
CAS:GABAB antagonistFormula:C9H13ClNO3PPurity:99.32%Color and Shape:White SolidMolecular weight:249.633α,21-Dihydroxy-5α-pregnan-20-one
CAS:3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.Formula:C21H34O3Purity:98.00%Color and Shape:SolidMolecular weight:334.49HZ166
CAS:HZ-166 is a positive GABAA receptor modulator and a GABAA receptor subtype-selective benzodiazepine site ligand.Formula:C21H16N4O2Purity:98%Color and Shape:SolidMolecular weight:356.38CCD-3693
CAS:CCD-3693 is a gamma-aminobutyric acid (GABA) receptor agonist.Formula:C21H31F3O2Purity:98%Color and Shape:SolidMolecular weight:372.46Chlormethiazole edisylate
CAS:Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic.Formula:C8H14ClNO6S3Purity:98%Color and Shape:SolidMolecular weight:351.85COR628
CAS:COR628 is the GABA(B) receptor positive allosteric modulator.Formula:C16H23NO3SColor and Shape:SolidMolecular weight:309.42trans-4-Hydroxycrotonic acid
CAS:ligand of γ-hydroxybutyric acid (GHB) receptorFormula:C4H6O3Purity:99.19%Color and Shape:SolidMolecular weight:102.09LY 81067
CAS:LY 81067, a new anticonvulsant, prevents PTZ- and picrotoxin-induced seizures in mice via picrotoxin site interaction.Formula:C22H24N4OColor and Shape:SolidMolecular weight:360.45U 90042
CAS:GABAA receptor ligandFormula:C17H13ClN6OPurity:98%Color and Shape:SolidMolecular weight:352.78COR627
CAS:COR627 is the GABA receptor positive allosteric modulator.Formula:C20H27NO3SPurity:98%Color and Shape:SolidMolecular weight:361.5CPP-115
CAS:CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.Formula:C7H9F2NO2Color and Shape:SolidMolecular weight:177.15JY-XHe-053
CAS:JY-XHe-053 is a selective modulator of GABAA receptors.Formula:C22H16FN3O2Purity:98%Color and Shape:SolidMolecular weight:373.38HIE-124
CAS:HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.Formula:C10H12N2O3SPurity:98%Color and Shape:SolidMolecular weight:240.28Suclofenide
CAS:Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.Formula:C16H13ClN2O4SPurity:98%Color and Shape:SolidMolecular weight:364.8(S)-Baclofen
CAS:(S)-Baclofen may treat hyperacusis and tinnitus by reducing auditory pathway excitation.Formula:C10H12ClNO2Purity:98%Color and Shape:SolidMolecular weight:213.66Lirequinil
CAS:Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.Formula:C26H25ClN2O3Purity:98.54%Color and Shape:SolidMolecular weight:448.94NNC 05-711
CAS:NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.Formula:C21H23ClN2O3Purity:99.92%Color and Shape:SolidMolecular weight:386.87Divaplon
CAS:Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.Formula:C17H17N3O2Purity:97.44% - 98.25%Color and Shape:SolidMolecular weight:295.34Ru-32514
CAS:Ru-32514 is a benzodiazepine receptor agonist.Formula:C18H17N3O2Purity:99.21%Color and Shape:SolidMolecular weight:307.35Sarmazenil
CAS:Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.Formula:C15H14ClN3O3Purity:99.46%Color and Shape:SolidMolecular weight:319.74Muscimol HBr
CAS:Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.Formula:C4H7BrN2O2Purity:98.13%Color and Shape:Off-White PowderMolecular weight:195.01Ref: TM-T20657
1mg113.00€2mg169.00€5mg240.00€10mg385.00€25mg622.00€50mg898.00€100mg1,198.00€500mg2,422.00€1mL*10mM (DMSO)205.00€Golexanolone
CAS:Golexanolone can be used to study neurological diseases.Formula:C21H31NO2Purity:99.90% - 99.99%Color and Shape:SolidMolecular weight:329.48Riluzole hydrochloride
CAS:Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).Formula:C8H6ClF3N2OSPurity:99.76%Color and Shape:SolidMolecular weight:270.66Saripidem
CAS:Saripidem (SL-85.0274) is a compound with anxiolytic activity.Formula:C19H20ClN3OPurity:98.42%Color and Shape:SolidMolecular weight:341.83NS-2710
CAS:NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.Formula:C22H20N4OPurity:99.7% - 99.82%Color and Shape:SolidMolecular weight:356.42L-838417
CAS:L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disordersFormula:C19H19F2N7OPurity:98.12% - 99.70%Color and Shape:SolidMolecular weight:399.4DMCM hydrochloride
CAS:DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.Formula:C17H19ClN2O4Purity:99.56%Color and Shape:SolidMolecular weight:350.8Ref: TM-T11061
1mg34.00€2mg50.00€5mg80.00€10mg105.00€25mg236.00€50mg439.00€100mg620.00€1mL*10mM (DMSO)88.00€ELB-139
CAS:ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.Formula:C14H16ClN3OPurity:>99.99%Color and Shape:SolidMolecular weight:277.75DSP-0565
CAS:DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.Formula:C14H12FNOPurity:99.51% - 99.56%Color and Shape:SolidMolecular weight:229.25Ref: TM-T11106
1mg109.00€2mg163.00€5mg241.00€10mg354.00€25mg532.00€50mg745.00€100mg1,018.00€500mg2,035.00€1mL*10mM (DMSO)208.00€
