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GABA Receptor

GABA Receptor

GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.

Found 336 products of "GABA Receptor"

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  • Pipazethate

    CAS:
    <p>Pipipyrazine is a nonnarcotic oral cough suppressant, cough suppressant.</p>
    Formula:C21H25N3O3S
    Color and Shape:Solid
    Molecular weight:399.51
  • NNC052090

    CAS:
    <p>NNC052090 inhibits GABA uptake, favoring hBGT-1 (Ki=1.4μM), affects α1/D2 receptors (IC50=266/1632nM).</p>
    Formula:C27H30N2O2
    Color and Shape:Solid
    Molecular weight:414.54
  • RU 33965

    CAS:
    <p>RU 33965, a 3-cyclopropyl carbonyl imidazobenzodiazepine, act as a low-efficacy benzodiazepine receptor inverse agonist.</p>
    Formula:C16H15N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:281.31
  • ZK93423

    CAS:
    <p>ZK93423: potent benzodiazepine agonist, IC50=1nM, non-selective, Ki=4.1-6nM for α1-α5 GABAA subunits.</p>
    Formula:C23H22N2O4
    Color and Shape:Solid
    Molecular weight:390.43
  • GABAA receptor modulator-2

    CAS:
    <p>Compound 20: Selective, oral α5-GABAAR inhibitor, Ki: 4.1 nM. High stability, CNS safe.</p>
    Formula:C22H22FN3O5S
    Color and Shape:Solid
    Molecular weight:459.49
  • Carburazepam

    CAS:
    <p>Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.</p>
    Formula:C17H16ClN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:329.78
  • UMB68 sodium

    CAS:
    <p>UMB-68 is a GHB receptor ligand with no affinity (IC(50) &gt;100 microM) at GABA(A) or GABA(B) receptors.</p>
    Formula:C6H12NaO3
    Color and Shape:Solid
    Molecular weight:155.149
  • (+)-Nipecotic acid

    CAS:
    <p>(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.</p>
    Formula:C6H11NO2
    Purity:99.38%
    Color and Shape:Solid
    Molecular weight:129.16
  • (S)-SNAP5114

    CAS:
    <p>(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.</p>
    Formula:C30H35NO6
    Purity:97%
    Color and Shape:Solid
    Molecular weight:505.6
  • Radequinil

    CAS:
    <p>Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).</p>
    Formula:C18H14N4O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:334.33
  • 3α,21-Dihydroxy-5α-pregnan-20-one

    CAS:
    <p>3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.</p>
    Formula:C21H34O3
    Purity:98.00%
    Color and Shape:Solid
    Molecular weight:334.49
  • Chlormethiazole edisylate

    CAS:
    <p>Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic.</p>
    Formula:C8H14ClNO6S3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:351.85
  • COR628

    CAS:
    <p>COR628 is the GABA(B) receptor positive allosteric modulator.</p>
    Formula:C16H23NO3S
    Color and Shape:Solid
    Molecular weight:309.42
  • trans-4-Hydroxycrotonic acid

    CAS:
    <p>ligand of γ-hydroxybutyric acid (GHB) receptor</p>
    Formula:C4H6O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:102.09
  • LY 81067

    CAS:
    <p>LY 81067, a new anticonvulsant, prevents PTZ- and picrotoxin-induced seizures in mice via picrotoxin site interaction.</p>
    Formula:C22H24N4O
    Color and Shape:Solid
    Molecular weight:360.45
  • U 90042

    CAS:
    <p>GABAA receptor ligand</p>
    Formula:C17H13ClN6O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:352.78
  • COR627

    CAS:
    <p>COR627 is the GABA receptor positive allosteric modulator.</p>
    Formula:C20H27NO3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:361.5
  • CPP-115

    CAS:
    <p>CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.</p>
    Formula:C7H9F2NO2
    Color and Shape:Solid
    Molecular weight:177.15
  • JY-XHe-053

    CAS:
    <p>JY-XHe-053 is a selective modulator of GABAA receptors.</p>
    Formula:C22H16FN3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:373.38
  • HIE-124

    CAS:
    <p>HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.</p>
    Formula:C10H12N2O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:240.28