GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
Found 373 products of "GABA Receptor"
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DS1
CAS:DS1 is a GABAA receptor agonist which can stimulate gonadotropin subunit gene expression in mouse.Formula:C18H10Br2ClN3OSColor and Shape:SolidMolecular weight:511.623α,21-Dihydroxy-5α-pregnan-20-one
CAS:3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.Formula:C21H34O3Purity:98.00%Color and Shape:SolidMolecular weight:334.49GABAA receptor agent 6
CAS:GABAA receptor agent 6 (compound 2027) is a potent γ-GABAAR antagonist with low cellular membrane permeability (Ki = 0.56 μM) [1].Formula:C18H25N3O2Color and Shape:SolidMolecular weight:315.41SCH-50910 free base
CAS:SCH-50910 is an antagonist of GABAB receptor.Formula:C8H15NO3Color and Shape:SolidMolecular weight:173.21GABAA receptor agent 4
CAS:Compound 1e is a potent γ-GABAAR antagonist with a Ki of 0.18 µM, offering immunomodulatory effects on T cell proliferation.Formula:C17H24N2OColor and Shape:SolidMolecular weight:272.39Profadol hydrochloride
CAS:Profadol hydrochloride acts as a mixed agonist-antagonist of the μ-opioid receptor with analgesic activity.Formula:C14H22ClNOPurity:98%Color and Shape:SolidMolecular weight:255.783-Methyl-GABA
CAS:3-Methyl-GABA activates GABA aminotransferase, fits GABAaR, stimulates GAD, and acts as an anticonvulsant.Formula:C20H30N2O10S2Purity:98%Color and Shape:SolidMolecular weight:522.59Ro15-4513
CAS:Ro15-4513 is imidazobenzodiazepinone derivative and is a partial inverse agonist of benzodiazepine receptors. Ro15-4513 is an effective ethanol antagonist.Formula:C15H14N6O3Purity:98%Color and Shape:SolidMolecular weight:326.31Ro 14-7437
CAS:Ro 14-7437 is an antagonist of GABA-benzodiazepine receptor.Formula:C15H15N3O3Color and Shape:SolidMolecular weight:285.3Phaclofen
CAS:GABAB antagonistFormula:C9H13ClNO3PPurity:99.32%Color and Shape:White SolidMolecular weight:249.63Adinazolam Mesylate
CAS:Adinazolam Mesylate is an anxiolytic and antidepressant agent. Adinazolam Mesylate binds to peripheral-type benzodiazepine receptors that interact allosterically with GABA receptors as an agonist to produce inhibitory effects.Formula:C20H22ClN5O3SPurity:98%Color and Shape:SolidMolecular weight:447.94Ro 15-1310
CAS:Ro 15-3505, a benzodiazepine receptor partial inverse agonist, has shown the ability to improve impaired recent memory of aged mice.Formula:C15H14ClN3O3Color and Shape:SolidMolecular weight:319.74mGAT3/4-IN-1
CAS:mGAT3/4-IN-1 inhibits mGAT3/4 with pIC50: 5.31/5.24, reduces neuropathic pain in diabetic mice.Formula:C26H31ClN2O2S2Color and Shape:SolidMolecular weight:503.12GABA-AT-IN-1
CAS:GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.Formula:C23H18N2O6Color and Shape:SolidMolecular weight:418.4AZD 3043
CAS:AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.Formula:C19H29NO5Purity:98.19% - 99.55%Color and Shape:SolidMolecular weight:351.44CCD-3693
CAS:CCD-3693 is a gamma-aminobutyric acid (GABA) receptor agonist.Formula:C21H31F3O2Purity:98%Color and Shape:SolidMolecular weight:372.462-Hydroxysaclofen
CAS:2-Hydroxysaclofen is a GABAB receptor antagonist.Formula:C9H12ClNO4SPurity:98.56%Color and Shape:White SolidMolecular weight:265.71CGS 20625
CAS:partial agonist for the benzodiazepine binding site of the GABAA receptorFormula:C18H19N3O2Purity:99.61%Color and Shape:SolidMolecular weight:309.36SX-3228
CAS:SX-3228 is a selective agonist of benzodiazepine1 (BZ1) receptor(IC50 of 17 nM).Formula:C18H18N4O3Purity:98%Color and Shape:SolidMolecular weight:338.36NO 711
CAS:NO 711（NNC-711 free acid） is a selective inhibitor of GAT-1, which enhances non-rapid eye movement sleep, and prevents paclitaxel-induced neuropathic pain.Formula:C21H22N2O3Purity:99.70%Color and Shape:SolidMolecular weight:350.41
