GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
Found 373 products of "GABA Receptor"
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L-838417
CAS:L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disordersFormula:C19H19F2N7OPurity:98.12% - 99.70%Color and Shape:SolidMolecular weight:399.4DMCM hydrochloride
CAS:DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.Formula:C17H19ClN2O4Purity:99.56%Color and Shape:SolidMolecular weight:350.8Ref: TM-T11061
1mg34.00€2mg50.00€5mg80.00€1mL*10mM (DMSO)88.00€10mg105.00€25mg236.00€50mg439.00€100mg620.00€Alpidem
CAS:Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.Formula:C21H23Cl2N3OPurity:99.56% - 99.97%Color and Shape:White To Off-White SolidMolecular weight:404.33Ref: TM-T26600
1mg58.00€1mL*10mM (DMSO)122.00€5mg137.00€10mg207.00€25mg371.00€50mg522.00€100mg747.00€500mg1,513.00€NNC 05-2090 hydrochloride
CAS:NNC 05-2090 HCl: BGT-1 inhibitor, IC50 = 10.6 μM, potential for epilepsy, neurological research.Formula:C27H31ClN2O2Purity:99.11%Color and Shape:SolidMolecular weight:451Cirsimaritin
CAS:Cirsimaritin has anti-bacterial, anti-inflammatory, anti-tumor, antioxidant effects, and protects kidneys; it weakly targets GABAA receptors.
Formula:C17H14O6Purity:99.9%Color and Shape:SolidMolecular weight:314.29NNC 05-711
CAS:NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.Formula:C21H23ClN2O3Purity:99.92%Color and Shape:SolidMolecular weight:386.87Ru-32514
CAS:Ru-32514 is a benzodiazepine receptor agonist.Formula:C18H17N3O2Purity:99.21%Color and Shape:SolidMolecular weight:307.35Golexanolone
CAS:Golexanolone can be used to study neurological diseases.Formula:C21H31NO2Purity:99.90% - 99.99%Color and Shape:SolidMolecular weight:329.48NS-2710
CAS:NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.Formula:C22H20N4OPurity:99.7% - 99.82%Color and Shape:SolidMolecular weight:356.42ELB-139
CAS:ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.Formula:C14H16ClN3OPurity:>99.99%Color and Shape:SolidMolecular weight:277.75RWJ-51204
CAS:RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.
Formula:C21H19F2N3O3Purity:99.57% - 99.95%Color and Shape:SolidMolecular weight:399.39Ref: TM-T16811
1mg333.00€5mg787.00€10mg1,074.00€25mg1,510.00€50mg1,882.00€100mg2,375.00€500mg4,655.00€SCS
CAS:SCS is a GABAA receptor antagonist.Formula:C14H12N2O3Purity:99.73%Color and Shape:SolidMolecular weight:256.26GABA-IN-2
CAS:GABA-IN-2 (Compound 5), a GABA inhibitor, exhibits both larvicidal and insecticidal properties, achieving an 87% mortality rate at a concentration of 50 mg/L [1Formula:C12H4Cl2F6N4SeColor and Shape:SolidMolecular weight:468.04GABAA receptor agent 2 TFA
CAS:Potent GABAA antagonist; IC50: 24 nM (α1β2γ2), Ki: 28 nM (rat); inactive on human GABA transporters.Formula:C22H22F3N3O3Color and Shape:SolidMolecular weight:433.42RPC425 free base
CAS:RPC425 is a noncompetitive inhibitors of the Betaine-γ-Aminobutyric Acid Transporter 1 (BGT1).Formula:C22H27NO2S2Purity:98%Color and Shape:SolidMolecular weight:401.59(R)-4-Amino-3-hydroxybutyric Acid
CAS:(R)-4-Amino-3-hydroxybutyric acid, also known as (R)-GABOB, acts as a modulator of GABA receptors, specifically binding to both GABAA and GABAB receptors and blocking GABA reuptake in rat brain synaptosomes. Additionally, it serves as a GABAC receptor agonist, triggering currents in patch-clamp assays with Xenopus oocytes that express the human receptor. In vivo studies reveal its capability to suppress electrical discharges in the amygdala in cats undergoing N-amidinobenzamide-triggered seizures, indicating its potential therapeutic application in managing seizure disorders.Formula:C4H9NO3Color and Shape:SolidMolecular weight:119.12Org-21465
CAS:Org-21465, a gamma-aminobutyric acid (GABA) receptor agonist, is used potentially for the use of anesthesia.Formula:C27H43NO4Purity:98%Color and Shape:SolidMolecular weight:445.63CGP36216 hydrochloride
CAS:CGP36216 hydrochloride acts as a selective antagonist at the presynaptic GABA receptor, specifically binding to the GABAB receptor with a Ki value of 0.3 μM. This compound is leveraged in research focused on anxiety and trauma-related disorders [1] [2].Formula:C5H15ClNO2PColor and Shape:SolidMolecular weight:187.6(-)-Bicuculline methochloride
CAS:(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.
Formula:C21H20ClNO6Purity:98%Color and Shape:SolidMolecular weight:417.84CGP 55845 hydrochloride
CAS:CGP55845 hydrochloride is a potent and selective GABAB receptor antagonist with an IC 50 of 6 nM which can be used in neurological research [1] [2].Formula:C18H23Cl3NO3PColor and Shape:SolidMolecular weight:438.71
