GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
Found 371 products of "GABA Receptor"
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Etbicyphat
CAS:Etbicyphat: potent GABA(A) antagonist, induces epileptiform activity, binds to GABA/benzodiazepine receptors.Formula:C6H11O4PColor and Shape:SolidMolecular weight:178.12TCS 1105
CAS:TCS 1105 is a GABAA BZR ligand, blocking Sema3A and altering mouse anxiety, aggression, and social dominance.Formula:C17H13FN2O2Purity:99.75%Color and Shape:SolidMolecular weight:296.3Pipazethate
CAS:Pipipyrazine is a nonnarcotic oral cough suppressant, cough suppressant.Formula:C21H25N3O3SColor and Shape:SolidMolecular weight:399.51NNC052090
CAS:NNC052090 inhibits GABA uptake, favoring hBGT-1 (Ki=1.4μM), affects α1/D2 receptors (IC50=266/1632nM).Formula:C27H30N2O2Color and Shape:SolidMolecular weight:414.54RU 33965
CAS:RU 33965, a 3-cyclopropyl carbonyl imidazobenzodiazepine, act as a low-efficacy benzodiazepine receptor inverse agonist.Formula:C16H15N3O2Purity:98%Color and Shape:SolidMolecular weight:281.31NCS-382
CAS:γ-Hydroxybutyric acid antagonistFormula:C13H14O3Purity:98%Color and Shape:SolidMolecular weight:218.25ZAPA sulfate
CAS:GABAA receptors agonistFormula:C4H8N2O6S2Purity:98%Color and Shape:SolidMolecular weight:244.25ZK93423
CAS:ZK93423: potent benzodiazepine agonist, IC50=1nM, non-selective, Ki=4.1-6nM for α1-α5 GABAA subunits.Formula:C23H22N2O4Color and Shape:SolidMolecular weight:390.43β-CCB
CAS:benzodiazepine receptor ligandFormula:C16H16N2O2Purity:98%Color and Shape:SolidMolecular weight:268.31GABAA receptor modulator-2
CAS:Compound 20: Selective, oral α5-GABAAR inhibitor, Ki: 4.1 nM. High stability, CNS safe.Formula:C22H22FN3O5SColor and Shape:SolidMolecular weight:459.49Carburazepam
CAS:Carburazepam is a derivate of benzodiazepines. Benzodiazepines are a class of psychoactive drugs.Formula:C17H16ClN3O2Purity:98%Color and Shape:SolidMolecular weight:329.78UMB68 sodium
CAS:UMB-68 is a GHB receptor ligand with no affinity (IC(50) >100 microM) at GABA(A) or GABA(B) receptors.Formula:C6H12NaO3Color and Shape:SolidMolecular weight:155.149Pregabalin arenacarbil
CAS:Pregabalin arenacarbil is a gabamimetic.Formula:C15H27NO6Color and Shape:SolidMolecular weight:317.38GABAA receptor agent 8
CAS:Compound 5e, a GABAA receptor modulator, shows potent anticonvulsant effects with low neurotoxicity for epilepsy research.Formula:C19H16N4OColor and Shape:SolidMolecular weight:316.36Tracazolate hydrochloride
CAS:Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.Formula:C16H25ClN4O2Purity:99.52%Color and Shape:SolidMolecular weight:340.85CGP 36216 hydrochloride
CAS:CGP 36216 hydrochloride is a potent and selective antagonist of GABAB receptors (IC50: 43 μM).Formula:C5H14NO2PPurity:98%Color and Shape:SolidMolecular weight:151.14(+)-Nipecotic acid
CAS:(+)-Nipecotic acid ((+)-β-Homoproline) is a specific inhibitor of GABA transport and uptake, capable of activating GABAA receptors.Formula:C6H11NO2Purity:99.38%Color and Shape:SolidMolecular weight:129.16GABA-AT-IN-1
CAS:GABA-AT-IN-1 (Compound 6) is an inhibitor of γ-aminobutyric acid transaminase (GABA-AT) that crosses the blood-brain barrier.Formula:C23H18N2O6Color and Shape:SolidMolecular weight:418.4(S)-SNAP5114
CAS:(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 and 21 μM for rGAT-2. (S)-SNAP5114 has anticonvulsant properties.Formula:C30H35NO6Purity:98.20%Color and Shape:SolidMolecular weight:505.6Ref: TM-T16831
5mg49.00€10mg73.00€25mg152.00€50mg213.00€100mg309.00€200mg423.00€1mL*10mM (DMSO)49.00€Radequinil
CAS:Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) ligand (Kis: 5.15 and 6.11 nM, respectively).Formula:C18H14N4O3Purity:98%Color and Shape:SolidMolecular weight:334.33Phaclofen
CAS:GABAB antagonistFormula:C9H13ClNO3PPurity:99.32%Color and Shape:White SolidMolecular weight:249.633α,21-Dihydroxy-5α-pregnan-20-one
CAS:3α,21-Dihydroxy-5α-pregnan-20-one (5alpha-THDOC) is a GABAA modulator that can be used in the study of Alzheimer's-like neurological diseases.Formula:C21H34O3Purity:98.00%Color and Shape:SolidMolecular weight:334.49HZ166
CAS:HZ-166 is a positive GABAA receptor modulator and a GABAA receptor subtype-selective benzodiazepine site ligand.Formula:C21H16N4O2Purity:98%Color and Shape:SolidMolecular weight:356.38CCD-3693
CAS:CCD-3693 is a gamma-aminobutyric acid (GABA) receptor agonist.Formula:C21H31F3O2Purity:98%Color and Shape:SolidMolecular weight:372.46Chlormethiazole edisylate
CAS:Chlormethiazole edisylate is a positive allosteric modulator of the GABAA receptor. Chlormethiazole edisylate is a sedative and hypnotic.Formula:C8H14ClNO6S3Purity:98%Color and Shape:SolidMolecular weight:351.85COR628
CAS:COR628 is the GABA(B) receptor positive allosteric modulator.Formula:C16H23NO3SColor and Shape:SolidMolecular weight:309.42trans-4-Hydroxycrotonic acid
CAS:ligand of γ-hydroxybutyric acid (GHB) receptorFormula:C4H6O3Purity:99.19%Color and Shape:SolidMolecular weight:102.09LY 81067
CAS:LY 81067, a new anticonvulsant, prevents PTZ- and picrotoxin-induced seizures in mice via picrotoxin site interaction.Formula:C22H24N4OColor and Shape:SolidMolecular weight:360.45U 90042
CAS:GABAA receptor ligandFormula:C17H13ClN6OPurity:98%Color and Shape:SolidMolecular weight:352.78COR627
CAS:COR627 is the GABA receptor positive allosteric modulator.Formula:C20H27NO3SPurity:98%Color and Shape:SolidMolecular weight:361.5CPP-115
CAS:CPP-115 is a GABA-aminotransferase inhibitor and a high-affinity vigabatrin analogue.Formula:C7H9F2NO2Color and Shape:SolidMolecular weight:177.15JY-XHe-053
CAS:JY-XHe-053 is a selective modulator of GABAA receptors.Formula:C22H16FN3O2Purity:98%Color and Shape:SolidMolecular weight:373.38HIE-124
CAS:HIE-124 is a central cervous system active anticonvulsant and ultra-short acting hypnotic.Formula:C10H12N2O3SPurity:98%Color and Shape:SolidMolecular weight:240.28Suclofenide
CAS:Suclofenide: a benzenesulfonamide anticonvulsant, effective in mouse seizure models, with side effects like lethargy and diarrhea.Formula:C16H13ClN2O4SPurity:98%Color and Shape:SolidMolecular weight:364.8(S)-Baclofen
CAS:(S)-Baclofen may treat hyperacusis and tinnitus by reducing auditory pathway excitation.Formula:C10H12ClNO2Purity:98%Color and Shape:SolidMolecular weight:213.66Lirequinil
CAS:Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.Formula:C26H25ClN2O3Purity:98.54%Color and Shape:SolidMolecular weight:448.94NNC 05-711
CAS:NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.Formula:C21H23ClN2O3Purity:99.92%Color and Shape:SolidMolecular weight:386.87Divaplon
CAS:Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.Formula:C17H17N3O2Purity:97.44% - 98.25%Color and Shape:SolidMolecular weight:295.34Ru-32514
CAS:Ru-32514 is a benzodiazepine receptor agonist.Formula:C18H17N3O2Purity:99.21%Color and Shape:SolidMolecular weight:307.35Sarmazenil
CAS:Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.Formula:C15H14ClN3O3Purity:99.46%Color and Shape:SolidMolecular weight:319.74Muscimol HBr
CAS:Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.Formula:C4H7BrN2O2Purity:98.13%Color and Shape:Off-White PowderMolecular weight:195.01Ref: TM-T20657
1mg113.00€2mg169.00€5mg240.00€10mg385.00€25mg622.00€50mg898.00€100mg1,198.00€500mg2,422.00€1mL*10mM (DMSO)205.00€Golexanolone
CAS:Golexanolone can be used to study neurological diseases.Formula:C21H31NO2Purity:99.90% - 99.99%Color and Shape:SolidMolecular weight:329.48Riluzole hydrochloride
CAS:Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).Formula:C8H6ClF3N2OSPurity:99.76%Color and Shape:SolidMolecular weight:270.66Saripidem
CAS:Saripidem (SL-85.0274) is a compound with anxiolytic activity.Formula:C19H20ClN3OPurity:98.42%Color and Shape:SolidMolecular weight:341.83NS-2710
CAS:NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.Formula:C22H20N4OPurity:99.7% - 99.82%Color and Shape:SolidMolecular weight:356.42L-838417
CAS:L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disordersFormula:C19H19F2N7OPurity:98.12% - 99.70%Color and Shape:SolidMolecular weight:399.4DMCM hydrochloride
CAS:DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.Formula:C17H19ClN2O4Purity:99.56%Color and Shape:SolidMolecular weight:350.8Ref: TM-T11061
1mg34.00€2mg50.00€5mg80.00€10mg105.00€25mg236.00€50mg439.00€100mg620.00€1mL*10mM (DMSO)88.00€ELB-139
CAS:ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.Formula:C14H16ClN3OPurity:>99.99%Color and Shape:SolidMolecular weight:277.75DSP-0565
CAS:DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.Formula:C14H12FNOPurity:99.51% - 99.56%Color and Shape:SolidMolecular weight:229.25Ref: TM-T11106
1mg109.00€2mg163.00€5mg241.00€10mg354.00€25mg532.00€50mg745.00€100mg1,018.00€500mg2,035.00€1mL*10mM (DMSO)208.00€
