GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
Found 336 products of "GABA Receptor"
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Bifenazate
CAS:<p>Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls 100% of mites at a concentration of 25 ppm.</p>Formula:C17H20N2O3Purity:99.62%Color and Shape:Solid CrystallineMolecular weight:300.35E2730
CAS:<p>E2730 is a non-competitive GABA transporter 1 (GAT1) inhibitor with anti-epileptic activity, useful in studying neurological disorders.</p>Formula:C9H8F4N2O2SPurity:98.22% - 98.54%Color and Shape:SolidMolecular weight:284.23U-89843A
CAS:<p>U-89843A is an allosteric modulator of the GABA_A receptor, known to enhance GABA-induced Cl^- currents [1].</p>Formula:C16H24ClN5Purity:98%Color and Shape:SolidMolecular weight:321.85(R)-Baclofen hydrochloride
CAS:<p>Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.</p>Formula:C10H13Cl2NO2Purity:98%Color and Shape:SolidMolecular weight:250.12Lesogaberan
CAS:<p>Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity (Ki 1.4 μM).</p>Formula:C3H9FNO2PPurity:98%Color and Shape:SolidMolecular weight:141.08Tracazolate hydrochloride
CAS:<p>Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant activity.</p>Formula:C16H25ClN4O2Purity:99.52%Color and Shape:SolidMolecular weight:340.85RO 4938581
CAS:<p>RO 4938581: potent GABAA α5 inverse agonist (Ki 4.6 nM); lower affinity for α1β3γ2a, α2β3γ2a, α3β3γ2a (Ki: 174, 185, 80 nM).</p>Formula:C13H8BrF2N5Purity:98%Color and Shape:SolidMolecular weight:352.14AZD 3043
CAS:<p>AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a novel sedative-hypnotic, and a potential short-acting anesthetic.</p>Formula:C19H29NO5Purity:98.19% - 99.55%Color and Shape:SolidMolecular weight:351.44Phaclofen
CAS:<p>GABAB antagonist</p>Formula:C9H13ClNO3PPurity:99.32%Color and Shape:White SolidMolecular weight:249.63Panadiplon
CAS:<p>Panadiplon (FG 10571) is a selective gamma-aminobutyric acid receptor agonist and partial agonist of 5GABAA, a benzodiazepine receptor, used in the treatment of</p>Formula:C18H17N5O2Purity:98.30% - 98.94%Color and Shape:SolidMolecular weight:335.36Cirsimaritin
CAS:<p>Cirsimaritin has anti-bacterial, anti-inflammatory, anti-tumor, antioxidant effects, and protects kidneys; it weakly targets GABAA receptors.</p>Formula:C17H14O6Purity:99.9%Color and Shape:SolidMolecular weight:314.29Progabide
CAS:<p>Progabide (SL 76002) is an agonist of the gamma-aminobutyric acid receptor.</p>Formula:C17H16ClFN2O2Purity:99.68%Color and Shape:SolidMolecular weight:334.77Saripidem
CAS:<p>Saripidem (SL-85.0274) is a compound with anxiolytic activity.</p>Formula:C19H20ClN3OPurity:99.45%Color and Shape:SolidMolecular weight:341.83NS-2710
CAS:<p>NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.</p>Formula:C22H20N4OPurity:99.7% - 99.82%Color and Shape:SolidMolecular weight:356.42ELB-139
CAS:<p>ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal cortex of rats.</p>Formula:C14H16ClN3OPurity:>99.99%Color and Shape:SolidMolecular weight:277.75Ru-32514
CAS:<p>Ru-32514 is a benzodiazepine receptor agonist.</p>Formula:C18H17N3O2Purity:99.21%Color and Shape:SolidMolecular weight:307.35Fengabine
CAS:<p>Fengabine (SL-79229) is a GABA receptor agonist with antidepressant activity and is used to treat depression.</p>Formula:C17H17Cl2NOPurity:99%Color and Shape:SolidMolecular weight:322.23Nerisopam
CAS:<p>Nerisopam is an agonist of gamma-aminobutyric acid (GABA) receptor.</p>Formula:C18H19N3O2Purity:97.07%Color and Shape:SolidMolecular weight:309.36DMCM hydrochloride
CAS:<p>DMCM hydrochloride is a non-selective fully inverse agonist of benzodiazepine.</p>Formula:C17H19ClN2O4Purity:99.56%Color and Shape:SolidMolecular weight:350.8Suriclone
CAS:<p>Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.</p>Formula:C20H20ClN5O3S2Purity:99.21% - 99.73%Color and Shape:SolidMolecular weight:477.99NNC 05-711
CAS:<p>NNC 05-711 (NO-711 hydrochloride) is a potent and selective inhibitor of GAT-1 (GABA transporter 1), exerting anticonvulsant and analgesic effects.</p>Formula:C21H23ClN2O3Purity:99.92%Color and Shape:SolidMolecular weight:386.87Riluzole hydrochloride
CAS:<p>Riluzole hydrochloride, an anticonvulsant Na+ channel blocker, inhibits GABA uptake (IC50: 43 µM).</p>Formula:C8H6ClF3N2OSPurity:99.76%Color and Shape:SolidMolecular weight:270.66BPDBA
CAS:<p>BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory activity against human BGT-1 and</p>Formula:C19H20Cl2N2OPurity:99.37% - 99.95%Color and Shape:SolidMolecular weight:363.28RWJ-51204
CAS:<p>RWJ-51204: potent adenosine A2A blocker, GABA(A) partial agonist (IC50: 0.2-2 nM), neuroprotective, may treat Parkinson's.</p>Formula:C21H19F2N3O3Purity:99.57% - 99.95%Color and Shape:SolidMolecular weight:399.39Lirequinil
CAS:<p>Lirequinil (Ro 41-3696) is a small molecule GABAA receptor agonist used to study neurological disorders.</p>Formula:C26H25ClN2O3Purity:98.54%Color and Shape:SolidMolecular weight:448.94L-838417
CAS:<p>L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in the study of anxiety disorders</p>Formula:C19H19F2N7OPurity:98.12% - 99.70%Color and Shape:SolidMolecular weight:399.4Divaplon
CAS:<p>Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics in a rat model of anxiety.</p>Formula:C17H17N3O2Purity:97.44% - 98.25%Color and Shape:SolidMolecular weight:295.34Alpidem
CAS:<p>Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.</p>Formula:C21H23Cl2N3OPurity:99.56% - 99.97%Color and Shape:White To Off-White SolidMolecular weight:404.33Sarmazenil
CAS:<p>Sarmazenil (Ro 15-3505) is a partial inverse agonist at the benzodiazepine receptor and is used in the study of chronic hepatic encephalopathy.</p>Formula:C15H14ClN3O3Purity:99.46%Color and Shape:SolidMolecular weight:319.74Golexanolone
CAS:<p>Golexanolone can be used to study neurological diseases.</p>Formula:C21H31NO2Purity:99.90% - 99.99%Color and Shape:SolidMolecular weight:329.48Muscimol HBr
CAS:<p>Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.</p>Formula:C4H7BrN2O2Purity:98.13%Color and Shape:Off-White PowderMolecular weight:195.01DSP-0565
CAS:<p>DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.</p>Formula:C14H12FNOPurity:99.51% - 99.56%Color and Shape:SolidMolecular weight:229.25CGP 55845 hydrochloride
CAS:<p>CGP55845 hydrochloride is a potent and selective GABAB receptor antagonist with an IC 50 of 6 nM which can be used in neurological research [1] [2].</p>Formula:C18H23Cl3NO3PColor and Shape:SolidMolecular weight:438.71FGIN-1-27
CAS:<p>FGIN-1-27 is a high-affinity agonist of the translocator protein and a specific peripheral benzodiazepine receptor (PBR) ligand(Ki = 5.0 nM).</p>Formula:C28H37FN2OPurity:99.86%Color and Shape:SolidMolecular weight:436.6GMA-839
CAS:<p>GMA-839 is a selective modulator of gamma-aminobutyric acid(A) receptors.</p>Formula:C21H31F3O3Purity:98%Color and Shape:SolidMolecular weight:388.46NO-711ME
CAS:<p>NO-711ME (N-O711 Methyl ester) is a prodrug of NO-711. It also is a potent and selective GABA uptake inhibitor.</p>Formula:C22H24N2O3Purity:99.54%Color and Shape:SolidMolecular weight:364.44U 89843A
CAS:<p>U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.</p>Formula:C16H23N5Purity:99.62%Color and Shape:SolidMolecular weight:285.39(+)-Bicuculline methiodide
CAS:<p>(+)-Bicuculline methiodide is a GABAA receptor blocker that blocks epileptogens and may be used in the study of neurological disorders.</p>Formula:C21H20INO6Purity:99.24%Color and Shape:SolidMolecular weight:509.29CP-409092
CAS:<p>CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.</p>Formula:C17H19N3O2Purity:98%Color and Shape:SolidMolecular weight:297.35mGAT3/4-IN-2
CAS:<p>mGAT3/4-IN-2 are potent inhibitors of mGAT3/mGAT4 with their pIC50 values of 5.44 and 5.25, respectively.</p>Formula:C26H32ClN3OS2Color and Shape:SolidMolecular weight:502.13COR659
CAS:<p>COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.</p>Formula:C16H16ClNO3SPurity:99.75%Color and Shape:SolidMolecular weight:337.82Diproqualone
CAS:<p>Diproqualone, analogous to methaqualone, exhibits sedative, anxiolytic, anti-inflammatory, and analgesic properties [1].</p>Formula:C12H14N2O3Color and Shape:SolidMolecular weight:234.255ADX71441
CAS:<p>ADX71441, a GABAB PAM, lengthens urinary latencies, lessens events & volume, and may aid in alcoholism and bladder pain.</p>Formula:C19H15ClF2N4O4Color and Shape:SolidMolecular weight:436.8Adipiplon
CAS:<p>Adipiplon(NG2-73, NG273) is a novel selective gamma-aminobutyric acid (GABA) partial agonist.</p>Formula:C18H18FN7Color and Shape:SolidMolecular weight:351.38PZ-II-029
CAS:<p>PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.</p>Formula:C18H15N3O3Purity:99.79%Color and Shape:SolidMolecular weight:321.33CGP 64213
CAS:<p>CGP 64213 is a GABAb receptor agonist.</p>Formula:C26H36IN2O7PPurity:98%Color and Shape:SolidMolecular weight:646.45(-)-Bicuculline methochloride
CAS:<p>(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.</p>Formula:C21H20ClNO6Purity:98%Color and Shape:SolidMolecular weight:417.84GABAA receptor agent 2 TFA
CAS:<p>Potent GABAA antagonist; IC50: 24 nM (α1β2γ2), Ki: 28 nM (rat); inactive on human GABA transporters.</p>Formula:C22H22F3N3O3Color and Shape:SolidMolecular weight:433.42JM-1232
CAS:<p>JM-1232 is a sedative and hypnotic drug being researched as a potential anesthetic.</p>Formula:C24H27N3O2Color and Shape:SolidMolecular weight:389.49CGP-54626 free base
CAS:<p>CGP-54626 is a selective antagonist of the GABAB receptor (IC50 = 4 nM ).</p>Formula:C18H28Cl2NO3PPurity:98%Color and Shape:SolidMolecular weight:408.3
