GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
Found 372 products of "GABA Receptor"
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Gabaculine HCl
CAS:Gabaculine, an irreversible GABA-T inhibitor (Ki: 2.9 μM), impacts plastid development and affects DPOR/GluTR levels.Formula:C7H10ClNO2Color and Shape:SolidMolecular weight:175.61S-8510 phosphate
CAS:S-8510 phosphate is an agonist of inverse Benzodiazepine (BDZ) receptor(Kis of 34.6 nM, 36.2 nM for –GABA and +GABA respectively).Formula:C12H13N4O6PPurity:98%Color and Shape:SolidMolecular weight:340.23GABA-IN-4
CAS:GABA-IN-4 (Compound 17) is a derivative of N-(indol-3-ylglyoxylyl)benzylamine. It exhibits high affinity for the benzodiazepine receptor (BzR), the binding site within the GABAA receptor complex, with a Ki value of 67 nM. Benzodiazepines are widely used as anxiolytic, sedative-hypnotic, and anticonvulsant agents.Formula:C17H13ClN2O2Color and Shape:SolidMolecular weight:312.75GABAA receptor agonist 1
Compound 3e, a potent GABAA agonist, targets GABA sites and has potential anti-depressive effects in mice.Formula:C20H30O3Color and Shape:SolidMolecular weight:318.45Tuclazepam
CAS:Tuclazepam (KC 1956) is a derivative of the benzodiazepine class of drugs, exhibiting anti-anxiety and sedative properties.Formula:C17H16Cl2N2OColor and Shape:SolidMolecular weight:335.23SGE-516
CAS:SGE516: neuroactive steroid, enhances GABAA, lowers neuronal activity, protects from seizures.Formula:C23H35N3O2Purity:98%Color and Shape:SolidMolecular weight:385.54ZK 93426 hydrochloride
CAS:benzodiazepine receptor antagonist,competitiveFormula:C18H21ClN2O3Purity:98%Color and Shape:SolidMolecular weight:348.82TP003
CAS:TP003 is a novel non-selective GABAA receptor benzodiazepine site agonist with affinity for α1β2gam2, α2β3gam2, α3β3gam2, α5β2gam2, EC50 of 20.3, 10.6, 3.24, 5.
Formula:C23H16F3N3OPurity:99.17%Color and Shape:SolidMolecular weight:407.39Fletazepam
CAS:Fletazepam, a benzodiazepine derivative, exhibits sedative, anti-anxiety, and muscle-relaxant properties. It is utilized in neurological research.Formula:C17H13ClF4N2Color and Shape:SolidMolecular weight:356.74Thiomuscimol hydrobromide
CAS:Thiomuscimol hydrobromide is an agonist of GABAA receptor.Formula:C4H6N2OSPurity:98%Color and Shape:SolidMolecular weight:130.17GABAA receptor agonist 2
Compound 4c, a potent GABAA agonist with anti-depressive effects in mouse FST/TST, shows promise in depression research.Formula:C22H36O5Color and Shape:SolidMolecular weight:380.52Refisolone
CAS:Refisolone is an antagonist of the GABAA receptor.Formula:C18H24O3Color and Shape:SolidMolecular weight:288.381EF1502 free base
CAS:EF1502 is a potent and selective GABA transporter inhibitor.Formula:C22H26N2O2S2Purity:98%Color and Shape:SolidMolecular weight:414.58(-)-Bicuculline methobromide
CAS:(-)-Bicuculline methobromide is a potent antagonist of GABAA receptor .Formula:C21H20BrNO6Color and Shape:WhiteMolecular weight:462.29Alfadolone acetate
CAS:Alfadolone acetate is a gamma-aminobutyric acid (GABA) receptor agonist.Formula:C23H34O5Color and Shape:SolidMolecular weight:390.512-AEMP TFA
CAS:2-AEMP TFA is a potent and rapidly acting antagonist of GABA(A)-ρ1 receptors. 2-AEMP is an analog of GABA.Formula:C3H10NO3PPurity:98%Color and Shape:SolidMolecular weight:139.0913-Methylglutaconic acid
CAS:3-Methylglutaconic acid, a primary metabolite accumulating in 3-Methylglutaconic aciduria (MGTA), induces lipid and protein oxidation, while diminishing non-enzymatic antioxidant defenses in cerebral cortex supernatants, thereby promoting oxidative stress in the cerebral cortex. This compound is utilized in research concerning brain damage diseases [1].Formula:C6H8O4Purity:98%Color and Shape:SolidMolecular weight:144.13Pipequaline
CAS:Pipequaline (PK-8165) is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that was never marketed. It possesses a novel chemical structure that is not closely related to other drugs of this type. The drug has a similar pharmacological profile to the benzodiazepine family of drugs, but with mainly anxiolytic properties and very little sedative, amnestic or anticonvulsant effects, and so is classified as a nonbenzodiazepine anxiolytic.Formula:C22H24N2Purity:98%Color and Shape:SolidMolecular weight:316.44Ref: TM-T4655
Discontinued productPazinaclone
CAS:Pazinaclone is a non-benzodiazepine (GABAA) partial agonist with sedative and anxiolytic activity.Formula:C25H23ClN4O4Purity:97.79% - 98.65%Color and Shape:SolidMolecular weight:478.93CGP 44532
CAS:CGP 44532 a GABAB receptor agonist.Formula:C4H12NO3PPurity:98%Color and Shape:SolidMolecular weight:153.12CGP 56999A
CAS:CGP 56999A is a GABA(B) receptor antagonist; it boosts BDNF and reduces dopamine loss in rat striatum.Formula:C19H30NO5PPurity:98%Color and Shape:SolidMolecular weight:383.42Xilmenolone
CAS:Xilmenolone acts as a positive allosteric modulator of the GABA_A receptor [1].
Formula:C26H37N3O2Purity:98%Color and Shape:SolidMolecular weight:423.59
