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GABA Receptor

GABA Receptor

GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.

Found 336 products of "GABA Receptor"

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  • Muscimol HBr

    CAS:
    <p>Muscimol HBr (Agarin HBr) is an agonist of GABAA receptor.</p>
    Formula:C4H7BrN2O2
    Purity:98.13%
    Color and Shape:Off-White Powder
    Molecular weight:195.01
  • DSP-0565

    CAS:
    <p>DSP-0565 is a broad-spectrum anti-epileptic with a high safety margin and effectiveness in several convulsant models.</p>
    Formula:C14H12FNO
    Purity:99.51% - 99.56%
    Color and Shape:Solid
    Molecular weight:229.25
  • CGP 55845 hydrochloride

    CAS:
    <p>CGP55845 hydrochloride is a potent and selective GABAB receptor antagonist with an IC 50 of 6 nM which can be used in neurological research [1] [2].</p>
    Formula:C18H23Cl3NO3P
    Color and Shape:Solid
    Molecular weight:438.71
  • FGIN-1-27

    CAS:
    <p>FGIN-1-27 is a high-affinity agonist of the translocator protein and a specific peripheral benzodiazepine receptor (PBR) ligand(Ki = 5.0 nM).</p>
    Formula:C28H37FN2O
    Purity:99.86%
    Color and Shape:Solid
    Molecular weight:436.6
  • GMA-839

    CAS:
    <p>GMA-839 is a selective modulator of gamma-aminobutyric acid(A) receptors.</p>
    Formula:C21H31F3O3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:388.46
  • NO-711ME

    CAS:
    <p>NO-711ME (N-O711 Methyl ester) is a prodrug of NO-711. It also is a potent and selective GABA uptake inhibitor.</p>
    Formula:C22H24N2O3
    Purity:99.54%
    Color and Shape:Solid
    Molecular weight:364.44
  • U 89843A

    CAS:
    <p>U 89843A is a positive allosteric modulator of gamma-aminobutyric acid (GABA)A receptors.</p>
    Formula:C16H23N5
    Purity:99.62%
    Color and Shape:Solid
    Molecular weight:285.39
  • (+)-Bicuculline methiodide

    CAS:
    <p>(+)-Bicuculline methiodide is a GABAA receptor blocker that blocks epileptogens and may be used in the study of neurological disorders.</p>
    Formula:C21H20INO6
    Purity:99.24%
    Color and Shape:Solid
    Molecular weight:509.29
  • CP-409092

    CAS:
    <p>CP-409092 is a partial GABAA receptor agonist. It has anti-anxiety activity.</p>
    Formula:C17H19N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:297.35
  • mGAT3/4-IN-2

    CAS:
    <p>mGAT3/4-IN-2 are potent inhibitors of mGAT3/mGAT4 with their pIC50 values of 5.44 and 5.25, respectively.</p>
    Formula:C26H32ClN3OS2
    Color and Shape:Solid
    Molecular weight:502.13
  • COR659

    CAS:
    <p>COR659: suppresses alcohol/chocolate intake in rats; enhances GABAB receptor, blocks CB1 receptor.</p>
    Formula:C16H16ClNO3S
    Purity:99.75%
    Color and Shape:Solid
    Molecular weight:337.82
  • Diproqualone

    CAS:
    <p>Diproqualone, analogous to methaqualone, exhibits sedative, anxiolytic, anti-inflammatory, and analgesic properties [1].</p>
    Formula:C12H14N2O3
    Color and Shape:Solid
    Molecular weight:234.255
  • ADX71441

    CAS:
    <p>ADX71441, a GABAB PAM, lengthens urinary latencies, lessens events &amp; volume, and may aid in alcoholism and bladder pain.</p>
    Formula:C19H15ClF2N4O4
    Color and Shape:Solid
    Molecular weight:436.8
  • Adipiplon

    CAS:
    <p>Adipiplon(NG2-73, NG273) is a novel selective gamma-aminobutyric acid (GABA) partial agonist.</p>
    Formula:C18H18FN7
    Color and Shape:Solid
    Molecular weight:351.38
  • PZ-II-029

    CAS:
    <p>PZ-II-029 is a modulator of α6β3γ2-selective GABAA channel.</p>
    Formula:C18H15N3O3
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:321.33
  • CGP 64213

    CAS:
    <p>CGP 64213 is a GABAb receptor agonist.</p>
    Formula:C26H36IN2O7P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:646.45
  • (-)-Bicuculline methochloride

    CAS:
    <p>(-)-Bicuculline methochloride is a potent antagonist of GABAA receptor.</p>
    Formula:C21H20ClNO6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:417.84
  • GABAA receptor agent 2 TFA

    CAS:
    <p>Potent GABAA antagonist; IC50: 24 nM (α1β2γ2), Ki: 28 nM (rat); inactive on human GABA transporters.</p>
    Formula:C22H22F3N3O3
    Color and Shape:Solid
    Molecular weight:433.42
  • JM-1232

    CAS:
    <p>JM-1232 is a sedative and hypnotic drug being researched as a potential anesthetic.</p>
    Formula:C24H27N3O2
    Color and Shape:Solid
    Molecular weight:389.49
  • CGP-54626 free base

    CAS:
    <p>CGP-54626 is a selective antagonist of the GABAB receptor (IC50 = 4 nM ).</p>
    Formula:C18H28Cl2NO3P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:408.3