GABA Receptor
GABA receptors are the primary inhibitory neurotransmitter receptors in the central nervous system, playing a critical role in regulating neuronal excitability and maintaining the balance between excitation and inhibition. GABA receptor dysfunction is implicated in various neurological and psychiatric disorders, including epilepsy, anxiety, and depression. At CymitQuimica, we provide a comprehensive range of GABA receptor modulators to support your research in neurobiology, mental health, and therapeutic development.
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L-838417
CAS:286456-42-6
L-838417 is a GABAA receptor subtype-selective benzodiazepine site-selective ligand and GABAA receptor-positive modulator used in …
Formula:
C19H19F2N7O
Purity:
98.12% - 99.82%
Color and Shape:
Solid
Molecular weight:
399.4
Ref: TM-T19702
| 1mg | 56.00 € | ||
| 5mg | 212.00 € | ||
| 10mg | 339.00 € | ||
| 25mg | 742.00 € | ||
| 50mg | 1,183.00 € | ||
| 100mg | 1,893.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
Bifenazate
CAS:149877-41-8
Bifenazate is a positive allosteric modulator of GABA receptor. Bifenazate is an acaricide that controls …
Formula:
C17H20N2O3
Purity:
99.44%
Color and Shape:
Solid Crystalline
Molecular weight:
300.35
Ref: TM-T14571
| 25mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
(R)-Baclofen hydrochloride
CAS:63701-55-3
Arbaclofen HCl, a GABA-B agonist, treats spasticity from spinal injury by reducing excitatory transmission.
Formula:
C10H13Cl2NO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
250.12
Ref: TM-T17306
| 10mg | 96.00 € | ||
| 25mg | 200.00 € | ||
| 50mg | 328.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
Pipequaline
CAS:77472-98-1
Pipequaline (PK-8165) is an anticonflict & anticonvulsant quinoline derivative. It is an anxiolytic drug that …
Formula:
C22H24N2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
316.44
Ref: TM-T4655
| 5mg | 49.00 € | ||
| 25mg | 121.00 € | ||
| 50mg | 219.00 € | ||
| 100mg | 379.00 € | ||
| 1ml*10 (DMSO) | 50.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
GABAB receptor antagonist 1
CAS:797-17-1
(E)-GABAB receptor antagonist 1 decreases GABA-induced IP3 (inositol trisphosphate) production with IC50 of 37.9 μM.GABAB …
Formula:
C18H24O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
304.38
Ref: TM-T11350
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
AZD 3043
CAS:579494-66-9
AZD 3043 (THRX 918661) is a modulator of the gamma-aminobutyric acid type A receptor, a …
Formula:
C19H29NO5
Purity:
98.19% - ≥98%
Color and Shape:
Solid
Molecular weight:
351.44
Ref: TM-T30248
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
(E)-GABAB receptor antagonist 1
CAS:1611483-29-4
(E)-GABAB antagonist 1 inhibits GABA IP3 production, with an IC50 of 37.9 μM and acts …
Formula:
C18H24O4
Purity:
95.26%
Color and Shape:
Solid
Molecular weight:
304.38
Ref: TM-T11137
| 1mg | 115.00 € | ||
| 5mg | 255.00 € | ||
| 10mg | 375.00 € | ||
| 25mg | 562.00 € | ||
| 50mg | 787.00 € | ||
| 100mg | 1,074.00 € | ||
| 200mg | 1,454.00 € | ||
| 1mL*10mM (DMSO) | 246.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
Ru-32514
CAS:90807-98-0
Ru-32514 is a benzodiazepine receptor agonist.
Formula:
C18H17N3O2
Purity:
98.74%
Color and Shape:
Solid
Molecular weight:
307.35
Ref: TM-T12779
| 1mg | 279.00 € | ||
| 2mg | 414.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
Golexanolone
CAS:2089238-18-4
Golexanolone can be used to study neurological diseases.
Formula:
C21H31NO2
Purity:
98.81% - 99.98%
Color and Shape:
Solid
Molecular weight:
329.48
Ref: TM-T25458
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
NS-2710
CAS:184220-36-8
NS-2710, a GABA receptor agonist, is used potentially for the treatment of anxiety.
Formula:
C22H20N4O
Purity:
98.10% - 99.82%
Color and Shape:
Solid
Molecular weight:
356.42
Ref: TM-T28197
| 1mg | 279.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
Radequinil
CAS:219846-31-8
Radequinil is a benzodiazepine receptor partial inverse agonist. Rade quinil binds to GABA(-) and GABA(+) …
Formula:
C18H14N4O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
334.33
Ref: TM-T16717
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
(S)-SNAP5114
CAS:157604-55-2
(S)-SNAP5114 is a selective inhibitor of GABA transport with IC50s of 5 μM for hGAT-3 …
Formula:
C30H35NO6
Purity:
97%
Color and Shape:
Solid
Molecular weight:
505.6
Ref: TM-T16831
| 1mg | 35.00 € | ||
| 5mg | 80.00 € | ||
| 10mg | 116.00 € | ||
| 25mg | 259.00 € | ||
| 50mg | 375.00 € | ||
| 100mg | 545.00 € | ||
| 500mg | 1,093.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
ELB-139
CAS:188116-08-7
ELB-139 is a GABA A receptor agonist. ELB139 increases 5-HT in the striatum and prefrontal …
Formula:
C14H16ClN3O
Purity:
100%
Color and Shape:
Solid
Molecular weight:
277.75
Ref: TM-T27252
| 1mg | 279.00 € | ||
| 2mg | 414.00 € | ||
| 5mg | 685.00 € | ||
| 10mg | 938.00 € | ||
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
Divaplon
CAS:90808-12-1
Divaplon is a GABA receptor agonist (IC50: 0.056 µM) that displays non-sedating anxiolytic behavioral characteristics …
Formula:
C17H17N3O2
Purity:
96.90% - 97.49%
Color and Shape:
Solid
Molecular weight:
295.34
Ref: TM-T27186
| 1mg | 143.00 € | ||
| 5mg | 333.00 € | ||
| 10mg | 504.00 € | ||
| 25mg | 817.00 € | ||
| 50mg | 1,121.00 € | ||
| 100mg | 1,510.00 € | ||
| 500mg | 3,030.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
Lesogaberan
CAS:344413-67-8
Lesogaberan: selective GABAB agonist, EC50 8.6 nM, Ki 5.1 nM in rats, weak GABAA affinity …
Formula:
C3H9FNO2P
Purity:
98%
Color and Shape:
Solid
Molecular weight:
141.08
Ref: TM-T15737
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
Alpidem
CAS:82626-01-5
Alpidem (Ananxyl), a non-sedative imidazopyridine anxiolytic, treats anxiety with high benzodiazepine receptor affinity.
Formula:
C21H23Cl2N3O
Purity:
100% - 99.49%
Color and Shape:
White To Off-White Solid
Molecular weight:
404.33
Ref: TM-T26600
| 1mg | 62.00 € | ||
| 5mg | 144.00 € | ||
| 10mg | 235.00 € | ||
| 25mg | 398.00 € | ||
| 50mg | 565.00 € | ||
| 100mg | 818.00 € | ||
| 1mL*10mM (DMSO) | 168.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
Bamaluzole
CAS:87034-87-5
Bamaluzole is an agonist of GABA receptor.
Formula:
C14H12ClN3O
Purity:
98%
Color and Shape:
Solid
Molecular weight:
273.72
Ref: TM-T10456
| 25mg | 1,444.00 € | ||
| 50mg | 1,882.00 € | ||
| 100mg | 2,375.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
Tracazolate hydrochloride
CAS:1135210-68-2
Tracazolate hydrochloride (Tracazolate (hydrochloride)) is a modulator of the GABAA receptor with anxiolytic and anticonvulsant …
Formula:
C16H25ClN4O2
Purity:
99.07%
Color and Shape:
Solid
Molecular weight:
340.85
Ref: TM-T23470
| 10mg | 116.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire |
Estimated delivery in United States, on Tuesday 3 Jun 2025
BPDBA
CAS:312281-74-6
BPDBA is an effective, selective, and non-competitive inhibitor of the betaine/GABA transporter (BGT-1), displaying inhibitory …
Formula:
C19H20Cl2N2O
Purity:
99.24% - 99.86%
Color and Shape:
Solid
Molecular weight:
363.28
Ref: TM-T26891
| 5mg | 40.00 € | ||
| 10mg | 58.00 € | ||
| 25mg | 109.00 € | ||
| 50mg | 170.00 € | ||
| 100mg | 273.00 € | ||
| 200mg | 378.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
Suriclone
CAS:53813-83-5
Suriclone (RP 31264), a cyclic pyrrolidone for anxiety, modulates GABA-A receptors without major sedation.
Formula:
C20H20ClN5O3S2
Purity:
98.17% - 98.52%
Color and Shape:
Solid
Molecular weight:
477.99
Ref: TM-T28887
| 1mg | 143.00 € | ||
| 5mg | 333.00 € | ||
| 10mg | 504.00 € | ||
| 25mg | 817.00 € | ||
| 50mg | 1,121.00 € | ||
| 100mg | 1,510.00 € |
Estimated delivery in United States, on Tuesday 3 Jun 2025
