P450
Cytochrome P450 enzymes are a large family of enzymes involved in the metabolism of various endogenous and exogenous compounds, including drugs, toxins, and hormones. P450 inhibitors are widely used to study drug metabolism, pharmacokinetics, and the role of these enzymes in disease states such as cancer and liver disorders. At CymitQuimica, we provide a broad selection of P450 inhibitors to support your research in pharmacology, toxicology, and metabolic regulation.
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Climbazole
CAS:38083-17-9
Climbazole (BAY-e 6975) is a broad-spectrum imidazole antifungal agent with anti-dandruff benefits.
Formula:
C15H17ClN2O2
Purity:
98.23%
Color and Shape:
White Solid Crystalline
Molecular weight:
292.76
Ref: TM-T1403
| 1g | 66.00 € | ||
| 5g | 142.00 € | ||
| 500mg | 48.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 15 Apr 2025
Methysticin
CAS:20697-20-5
Methysticin, a major kavalactone extracted from kava, can induce CYP1A1.
Formula:
C15H14O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
274.27
Ref: TM-TQ0276
| 5mg | 663.00 € |
Estimated delivery in United States, on Wednesday 16 Apr 2025
Licopyranocoumarin
CAS:117038-80-9
Licopyranocoumarin could as a potent neuroprotective drug via markedly blocked MPP+-induced neuronal PC12D cell death …
Formula:
C21H20O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
384.38
Ref: TM-TN4435
| 5mg | 722.00 € | ||
| 1mL*10mM (DMSO) | 742.00 € |
Estimated delivery in United States, on Wednesday 16 Apr 2025
BI 653048
CAS:1198784-72-3
BI 653048 is a selective and orally active agonist of nonsteroidal glucocorticoid (IC50: 55 nM). …
Formula:
C23H25F4N3O4S
Purity:
98%
Color and Shape:
Solid
Molecular weight:
515.52
Ref: TM-T10535
| 25mg | 2,585.00 € | ||
| 50mg | 3,402.00 € | ||
| 100mg | 4,655.00 € |
Estimated delivery in United States, on Wednesday 16 Apr 2025
Humantenirine
CAS:82375-30-2
Humantenirine is a natural product of Gelsemium, Loganiaceae.
Formula:
C21H26N2O4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
370.44
Ref: TM-TN1748
| 5mg | 627.00 € | ||
| 1mL*10mM (DMSO) | 637.00 € |
Estimated delivery in United States, on Wednesday 16 Apr 2025
15-Hydroxydehydroabietic acid
CAS:54113-95-0
15-Hydroxydehydroabietic acid exhibits a promising alpha-glucosidase inhibitory activity, it also shows significant antibacterial activities.
Formula:
C20H28O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
316.441
Ref: TM-TMA0164
| 5mg | 457.00 € | ||
| 1mL*10mM (DMSO) | 465.00 € |
Estimated delivery in United States, on Wednesday 16 Apr 2025
6',7'-Dihydroxybergamottin
CAS:264234-05-1
6',7'-Dihydroxybergamottin (DHB) inhibits CYP3A4 and POR; affects nifedipine oxidation.
Formula:
C21H24O6
Purity:
98%
Color and Shape:
Solid
Molecular weight:
372.41
Ref: TM-TN3147
| 10mg | 2,855.00 € |
Estimated delivery in United States, on Wednesday 16 Apr 2025
Dipterocarpol
CAS:471-69-2
Dipterocarpol is a dammarane-type triterpenoid, as are the major bioactive compounds of ginseng.
Formula:
C30H50O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
442.728
Ref: TM-TN3875
| 5mg | 590.00 € | ||
| 1mL*10mM (DMSO) | 598.00 € |
Estimated delivery in United States, on Wednesday 16 Apr 2025
2-Hydroxy-1-Methoxyaporphine
CAS:33770-27-3
2-Hydroxy-1-Methoxyaporphine can inhibit CYP2D6 activity, it also increase the glucose consumption significantly as rosiglitazone.
Formula:
C18H19NO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
281.355
Ref: TM-TN1210
| 10mg | 419.00 € | ||
| 1mL*10mM (DMSO) | 294.00 € |
Estimated delivery in United States, on Wednesday 16 Apr 2025
Canadine
CAS:5096-57-1
Canadine has antioxidant activity with low-toxic effect.
Formula:
C20H21NO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
339.39
Ref: TM-TN3574
| 1mg | 71.00 € | ||
| 5mg | 259.00 € | ||
| 10mg | 457.00 € |
Estimated delivery in United States, on Wednesday 16 Apr 2025
BI 653048 phosphate
CAS:1198784-97-2
BI 653048 phosphate is a selective and orally active agonist of nonsteroidal glucocorticoid (GC)(IC50 : …
Formula:
C23H28F4N3O8PS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
613.52
Ref: TM-T10535L
| 25mg | 3,496.00 € | ||
| 50mg | 4,854.00 € | ||
| 100mg | 5,824.00 € |
Estimated delivery in United States, on Wednesday 16 Apr 2025
Corydalmine
CAS:30413-84-4
Corydalmine exhibits antibacterial activities against Staphylococcus aureus and methicillin-resistant S.
Formula:
C20H23NO4
Purity:
98%
Color and Shape:
Solid
Molecular weight:
341.4
Ref: TM-TN1526
| 1mg | 266.00 € | ||
| 5mg | 598.00 € | ||
| 10mg | 893.00 € | ||
| 25mg | 1,520.00 € | ||
| 50mg | 2,280.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
2,3',4,6-Tetrahydroxybenzophenone
CAS:26271-33-0
2,3',4,6-Tetrahydroxybenzophenone possesses significant antioxidant activity.
Formula:
C13H10O5
Color and Shape:
Solid
Molecular weight:
246.22
Ref: TM-TN2687
| 5mg | 1,586.00 € | ||
| 1mL*10mM (DMSO) | 1,943.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
N-Nornuciferine
CAS:4846-19-9
N-Nornuciferine, an aporphine alkaloid in lotus leaf, significantly inhibits CYP2D6 (IC50: 3.76 μM, Ki: 2.34 …
Formula:
C18H19NO2
Color and Shape:
Solid
Molecular weight:
281.35
Ref: TM-TQ0296
| 20mg | 758.00 € |
Estimated delivery in United States, on Monday 21 Apr 2025
GSK-25
CAS:874119-56-9
GSK-25 maintains good selectivity against a panel of 31 kinases, as well as RSK1 and …
Formula:
C24H16Cl2F2N6O
Purity:
98.59%
Color and Shape:
Solid
Molecular weight:
513.33
Ref: TM-T4488
| 1mg | 47.00 € | ||
| 2mg | 59.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 117.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 271.00 € | ||
| 100mg | 454.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Norfluoxetine Hydrochloride
CAS:57226-68-3
Norfluoxetine Hydrochloride (Norfluoxetine HCl) is an active metabolite of fluoxetine. Fluoxetine is an antidepressant drug.
Formula:
C16H17ClF3NO
Purity:
99.75%
Color and Shape:
Solid
Molecular weight:
331.76
Ref: TM-T21029
| 1mg | 48.00 € | ||
| 2mg | 74.00 € | ||
| 5mg | 163.00 € | ||
| 10mg | 229.00 € | ||
| 25mg | 378.00 € | ||
| 50mg | 502.00 € | ||
| 100mg | 727.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
(S)-Mephenytoin
CAS:70989-04-7
(S)-Mephenytoin: (+)-enantiomer, anticonvulsant, CYP2C19 substrate for analyzing CYP450 metabolism.
Formula:
C12H14N2O2
Purity:
99.05% - 99.82%
Color and Shape:
Solid
Molecular weight:
218.25
Ref: TM-T21529
| 1mg | 56.00 € | ||
| 5mg | 119.00 € | ||
| 10mg | 187.00 € | ||
| 25mg | 376.00 € | ||
| 50mg | 562.00 € | ||
| 100mg | 802.00 € | ||
| 1mL*10mM (DMSO) | 131.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Uniconazole
CAS:83657-22-1
Uniconazole is a plant growth regulator that inhibit cytochrome P450 707As (Ki=68 nM).
Formula:
C15H18ClN3O
Purity:
99.94%
Color and Shape:
White-Light Brown Crystalline
Molecular weight:
291.78
Ref: TM-T21482
| 1g | 52.00 € | ||
| 5g | 113.00 € | ||
| 10g | 165.00 € | ||
| 500mg | 39.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
Cephaeline dihydrochloride
CAS:5853-29-2
(-)-Cephaeline (dihydrochloride) is an enantiomer of Cephaeline. Cephaeline is a selective CYP2D6 inhibitor (IC50: 121 …
Formula:
C28H40Cl2N2O4
Color and Shape:
Solid
Molecular weight:
539.54
Ref: TM-TQ0109
| 2mg | 78.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
1-Ethynylpyrene
CAS:34993-56-1
1-Ethynylpyrene is an aryl acetylenic inhibitor of CYTP450 1A1(IC50=0.18 μM), 1A2(IC50 = 0.32 μM), and …
Formula:
C18H10
Purity:
98.89%
Color and Shape:
Solid
Molecular weight:
226.27
Ref: TM-T9704
| 200mg | 34.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 22 Apr 2025
