P450
Cytochrome P450 enzymes are a large family of enzymes involved in the metabolism of various endogenous and exogenous compounds, including drugs, toxins, and hormones. P450 inhibitors are widely used to study drug metabolism, pharmacokinetics, and the role of these enzymes in disease states such as cancer and liver disorders. At CymitQuimica, we provide a broad selection of P450 inhibitors to support your research in pharmacology, toxicology, and metabolic regulation.
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Oteseconazole
CAS:1340593-59-0
Oteseconazole (VT-1161) is an orally active anti-fungal agent.
Formula:
C23H16F7N5O2
Purity:
99.07%
Color and Shape:
Solid
Molecular weight:
527.39
Ref: TM-T16412
| 1mg | 91.00 € | ||
| 2mg | 134.00 € | ||
| 5mg | 215.00 € | ||
| 10mg | 351.00 € | ||
| 25mg | 537.00 € | ||
| 50mg | 742.00 € | ||
| 100mg | 1,009.00 € | ||
| 200mg | 1,348.00 € | ||
| 1mL*10mM (DMSO) | 253.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
β-Tetralone
CAS:530-93-8
β-Tetralone (2-Tetralone) is a vital drug synthesis precursor with complex pharmacological properties in combating neurological …
Formula:
C10H10O
Purity:
97.26% - 99.18%
Color and Shape:
Clear To Yellow Liquid
Molecular weight:
146.19
Ref: TM-T0660
| 10mg | 35.00 € | ||
| 25mg | 48.00 € | ||
| 50mg | 70.00 € | ||
| 100mg | 92.00 € | ||
| 500mg | 182.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Topiroxostat
CAS:577778-58-6
Topiroxostat (FYX-051) is a selective xanthine oxidase inhibitor developed for treatment and management of hyperuricemia …
Formula:
C13H8N6
Purity:
98.95%
Color and Shape:
Solid
Molecular weight:
248.24
Ref: TM-T2397
| 25mg | 45.00 € | ||
| 50mg | 64.00 € | ||
| 100mg | 99.00 € | ||
| 200mg | 128.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Gemfibrozil
CAS:25812-30-0
Gemfibrozil, a fibric acid derivative, stimulates PPARalpha, boosts fatty acid oxidation, LPL, lowers VLDL-C, apoC-III, …
Formula:
C15H22O3
Purity:
98.59% - 99.9%
Color and Shape:
Crystals From Hexane Solid
Molecular weight:
250.33
Ref: TM-T1415
| 25mg | 35.00 € | ||
| 50mg | 45.00 € | ||
| 100mg | 54.00 € | ||
| 200mg | 68.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Piperine
CAS:94-62-2
Piperine (Bioperine) , a alkaloid, has been used in trials studying the treatment of multiple …
Formula:
C17H19NO3
Purity:
100% - 97.79%
Color and Shape:
Solid
Molecular weight:
285.34
Ref: TM-T3002
| 100mg | 23.00 € | ||
| 1mL*10mM (DMSO) | 36.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Alizarin
CAS:72-48-0
Alizarin, red dye from madder roots, inhibits CYP1A1 (IC50=6.2μM), CYP1A2 (IC50=10μM), CYP1B1 (IC50=2.7μM).
Formula:
C14H8O4
Purity:
98.14%
Color and Shape:
Orange-Red Crystals Or Powder
Molecular weight:
240.21
Ref: TM-T2949
| 1g | 51.00 € | ||
| 500mg | 46.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
ε-Viniferin
CAS:62218-08-0
ε-Viniferin (epsilon-Viniferin) a dimer of resveratrol, shows the inhibitory effects of epsilon-viniferin on human CYP1A1, …
Formula:
C28H22O6
Purity:
98% - 99.73%
Color and Shape:
Solid
Molecular weight:
454.47
Ref: TM-T11218
| 1mg | 291.00 € | ||
| 5mg | 713.00 € | ||
| 10mg | 1,003.00 € | ||
| 25mg | 1,468.00 € | ||
| 50mg | 1,995.00 € | ||
| 100mg | 2,673.00 € | ||
| 1mL*10mM (DMSO) | 932.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Liarozole
CAS:115575-11-6
Liarozole dihydrochloride inhibits CYP450, estrogen, androgen synthesis; an oral drug for prostate cancer/skin disorders.
Formula:
C17H13ClN4
Purity:
98.31%
Color and Shape:
Solid
Molecular weight:
308.76
Ref: TM-T11847L
| 1mg | 83.00 € | ||
| 5mg | 186.00 € | ||
| 10mg | 308.00 € | ||
| 25mg | 524.00 € | ||
| 50mg | 739.00 € | ||
| 100mg | 1,051.00 € | ||
| 1mL*10mM (DMSO) | 212.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Naringenin
CAS:480-41-1
Naringenin (NSC-11855) is a bioactive flavanone with antioxidant, anti-inflammatory properties, aids in carbohydrate metabolism, immunity, …
Formula:
C15H12O5
Purity:
98.2% - 99.55%
Color and Shape:
Solid
Molecular weight:
272.25
Ref: TM-T2838
| 1g | 116.00 € | ||
| 50mg | 54.00 € | ||
| 100mg | 58.00 € | ||
| 500mg | 87.00 € | ||
| 1mL*10mM (DMSO) | 62.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Clarithromycin
CAS:81103-11-9
Clarithromycin (A-56268), a macrolide antibiotic, inhibits Cytochrome P450 3A4 and P-Glycoprotein.
Formula:
C38H69NO13
Purity:
99.89% - 99.89%
Color and Shape:
White To Off-White Crystalline Powder
Molecular weight:
747.95
Ref: TM-T1434
| 100mg | 59.00 € | ||
| 200mg | 67.00 € | ||
| 500mg | 80.00 € | ||
| 1mL*10mM (DMSO) | 59.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Isoasatone A
CAS:67451-73-4
Isoasatone A acts against S.
Formula:
C24H32O8
Purity:
99.21%
Color and Shape:
Solid
Molecular weight:
448.51
Ref: TM-T11680
| 1mg | 61.00 € | ||
| 2mg | 85.00 € | ||
| 5mg | 120.00 € | ||
| 10mg | 169.00 € | ||
| 25mg | 280.00 € | ||
| 50mg | 428.00 € | ||
| 100mg | 616.00 € | ||
| 500mg | 1,273.00 € | ||
| 1mL*10mM (DMSO) | 140.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Abiraterone
CAS:154229-19-3
Abiraterone (CB-7598) (CB-7598) is an effective steroidal cytochrome P450 17alpha-hydroxylase-17, 20-lyase (CYP17) inhibitor (IC50: 4 …
Formula:
C24H31NO
Purity:
98.95% - 99.87%
Color and Shape:
White Solid
Molecular weight:
349.51
Ref: TM-T6216
| 1g | 150.00 € | ||
| 5mg | 45.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 71.00 € | ||
| 50mg | 77.00 € | ||
| 100mg | 93.00 € | ||
| 200mg | 103.00 € | ||
| 500mg | 121.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Climbazole
CAS:38083-17-9
Climbazole (BAY-e 6975) is a broad-spectrum imidazole antifungal agent with anti-dandruff benefits.
Formula:
C15H17ClN2O2
Purity:
98.1%
Color and Shape:
White Solid Crystalline
Molecular weight:
292.76
Ref: TM-T1403
| 1g | 66.00 € | ||
| 5g | 142.00 € | ||
| 500mg | 48.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Fenofibrate
CAS:49562-28-9
Fenofibrate (Lipanthyl) is a PPARα agonist. Fenofibrate inhibits cytochrome P450 isoforms. Fenofibrate exhibits antihyperlipidemic activity. …
Formula:
C20H21ClO4
Purity:
99.13% - 99.95%
Color and Shape:
Crystals From Isopropanol Solid
Molecular weight:
360.83
Ref: TM-T1149
| 100mg | 38.00 € | ||
| 200mg | 49.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Licopyranocoumarin
CAS:117038-80-9
Licopyranocoumarin could as a potent neuroprotective drug via markedly blocked MPP+-induced neuronal PC12D cell death …
Formula:
C21H20O7
Purity:
98%
Color and Shape:
Solid
Molecular weight:
384.38
Ref: TM-TN4435
| 5mg | 718.00 € | ||
| 1mL*10mM (DMSO) | 736.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Methysticin
CAS:20697-20-5
Methysticin, a major kavalactone extracted from kava, can induce CYP1A1.
Formula:
C15H14O5
Purity:
98%
Color and Shape:
Solid
Molecular weight:
274.27
Ref: TM-TQ0276
| 5mg | 659.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
2-Hydroxy-1-Methoxyaporphine
CAS:33770-27-3
2-Hydroxy-1-Methoxyaporphine can inhibit CYP2D6 activity, it also increase the glucose consumption significantly as rosiglitazone.
Formula:
C18H19NO2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
281.355
Ref: TM-TN1210
| 10mg | 414.00 € | ||
| 1mL*10mM (DMSO) | 292.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Schizandrin A
CAS:61281-38-7
Schisandrin A, a primary active component extracted from the traditional Eastern medicine Schisandra chinensis, inhibits …
Formula:
C24H32O6
Purity:
99.91%
Color and Shape:
Liquid
Molecular weight:
416.51
Ref: TM-T2926
| 10mg | 42.00 € | ||
| 25mg | 61.00 € | ||
| 50mg | 85.00 € | ||
| 1mL*10mM (DMSO) | 46.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
4,5-Dimethoxycanthin-6-one
CAS:18110-87-7
Alkaloid from Picrasma quassioides with antimicrobial, anti-cancer properties; inhibits CYP1A2 and cAMP phosphodiesterase. IC50: 1.7 …
Formula:
C16H12N2O3
Purity:
98.84%
Color and Shape:
Solid
Molecular weight:
280.28
Ref: TM-TN3013
| 1mg | 79.00 € | ||
| 5mg | 172.00 € | ||
| 10mg | 291.00 € | ||
| 25mg | 490.00 € | ||
| 50mg | 698.00 € | ||
| 1mL*10mM (DMSO) | 212.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Guanfu base A
CAS:1394-48-5
Guanfu base A is a potent noncompetitive CYP2D6 inhibitor (Ki: 1.20 μM in HLMs; Ki: …
Formula:
C24H31NO6
Purity:
99.71% - 99.85%
Color and Shape:
Solid
Molecular weight:
429.5
Ref: TM-T8182
| 1mg | 87.00 € | ||
| 5mg | 180.00 € | ||
| 10mg | 269.00 € | ||
| 25mg | 454.00 € | ||
| 50mg | 648.00 € | ||
| 100mg | 898.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
