P450
Cytochrome P450 enzymes are a large family of enzymes involved in the metabolism of various endogenous and exogenous compounds, including drugs, toxins, and hormones. P450 inhibitors are widely used to study drug metabolism, pharmacokinetics, and the role of these enzymes in disease states such as cancer and liver disorders. At CymitQuimica, we provide a broad selection of P450 inhibitors to support your research in pharmacology, toxicology, and metabolic regulation.
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TMS
CAS:24144-92-1
TMS (2,3',4,5'-Tetramethoxystilbene) is a very selective and potent competitive inhibitor of P450 1B1 (CYP1A1).
Formula:
C18H20O4
Purity:
99.42% - 99.56%
Color and Shape:
Solid
Molecular weight:
300.35
Ref: TM-T3585
| 5mg | 51.00 € | ||
| 10mg | 83.00 € | ||
| 25mg | 147.00 € | ||
| 50mg | 260.00 € | ||
| 100mg | 386.00 € | ||
| 500mg | 874.00 € | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Lofemizole
CAS:65571-68-8
Lofemizole is an antagonist of CYP1A2.
Formula:
C10H9ClN2
Purity:
97.11%
Color and Shape:
Solid
Molecular weight:
192.64
Ref: TM-T50053
| 1mg | 47.00 € | ||
| 5mg | 92.00 € | ||
| 10mg | 139.00 € | ||
| 25mg | 227.00 € | ||
| 50mg | 339.00 € | ||
| 100mg | 482.00 € | ||
| 200mg | 662.00 € | ||
| 1mL*10mM (DMSO) | 88.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Guan-fu base A hydrochloride(1394-48-5 free base)
CAS:618094-85-2
Guanfu base A HCl, an antiarrhythmic from Aconitum coreanum, inhibits CYP2D6 in humans, monkeys, and …
Formula:
C24H32NO6Cl
Purity:
99.90%
Color and Shape:
Solid
Molecular weight:
465.97
Ref: TM-T8182L
| 1mg | 128.00 € | ||
| 5mg | 283.00 € | ||
| 10mg | 421.00 € | ||
| 25mg | 697.00 € | ||
| 50mg | 975.00 € | ||
| 100mg | 1,319.00 € | ||
| 500mg | 2,627.00 € | ||
| 1mL*10mM (DMSO) | 159.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
DMU-2139
CAS:104890-70-2
DMU2139 is a specific CYP1B1 inhibitor (CYP1B1 and CYP1A1 with IC50 of 9 nM and …
Formula:
C19H15NO2
Purity:
98.88%
Color and Shape:
Solid
Molecular weight:
289.33
Ref: TM-T8728
| 1mg | 38.00 € | ||
| 5mg | 79.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 224.00 € | ||
| 50mg | 331.00 € | ||
| 100mg | 491.00 € | ||
| 200mg | 710.00 € | ||
| 1mL*10mM (DMSO) | 79.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Chrysosplenetin
CAS:603-56-5
Chrysosplenetin is a metabolic inhibitor of artemisinin.
Formula:
C19H18O8
Purity:
97.43% - 98.53%
Color and Shape:
Solid
Molecular weight:
374.34
Ref: TM-TJS1159
| 1mg | 59.00 € | ||
| 5mg | 125.00 € | ||
| 10mg | 185.00 € | ||
| 25mg | 341.00 € | ||
| 50mg | 501.00 € | ||
| 100mg | 715.00 € | ||
| 500mg | 1,451.00 € | ||
| 1mL*10mM (DMSO) | 225.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Soticlestat
CAS:1429505-03-2
Soticlestat (OV935) is a potent, selective and orally active cholesterol 24-hydroxylase (CYP46A1) inhibitor.
Formula:
C23H23N3O2
Purity:
99.95%
Color and Shape:
Solid
Molecular weight:
373.45
Ref: TM-T8937
| 1mg | 65.00 € | ||
| 5mg | 142.00 € | ||
| 10mg | 222.00 € | ||
| 25mg | 447.00 € | ||
| 50mg | 639.00 € | ||
| 100mg | 925.00 € | ||
| 1mL*10mM (DMSO) | 159.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ranitidine
CAS:66357-35-5
Ranitidine (HSDB 3925) is a non-imidazole blocker of those histamine receptors that mediate gastric secretion …
Formula:
C13H22N4O3S
Purity:
99.1%
Color and Shape:
Solid Solid
Molecular weight:
314.4
Ref: TM-T3610
| 5mg | 41.00 € | ||
| 10mg | 49.00 € | ||
| 25mg | 89.00 € | ||
| 50mg | 105.00 € | ||
| 100mg | 124.00 € | ||
| 200mg | 217.00 € | ||
| 500mg | 362.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Germacrone
CAS:6902-91-6
Germacrone, a major active component found in Curcuma zedoaria oil product, shows anti-inflammatory, antiandrogenic, and …
Formula:
C15H22O
Purity:
98.81% - 99.95%
Color and Shape:
Solid
Molecular weight:
218.33
Ref: TM-T2945
| 5mg | 48.00 € | ||
| 10mg | 80.00 € | ||
| 25mg | 122.00 € | ||
| 50mg | 156.00 € | ||
| 100mg | 196.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Cephaeline dihydrochloride
CAS:5853-29-2
(-)-Cephaeline (dihydrochloride) is an enantiomer of Cephaeline. Cephaeline is a selective CYP2D6 inhibitor (IC50: 121 …
Formula:
C28H40Cl2N2O4
Color and Shape:
Solid
Molecular weight:
539.54
Ref: TM-TQ0109
| 2mg | 76.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
GSK-25
CAS:874119-56-9
GSK-25 maintains good selectivity against a panel of 31 kinases, as well as RSK1 and …
Formula:
C24H16Cl2F2N6O
Purity:
98.59%
Color and Shape:
Solid
Molecular weight:
513.33
Ref: TM-T4488
| 1mg | 46.00 € | ||
| 2mg | 58.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 115.00 € | ||
| 25mg | 168.00 € | ||
| 50mg | 267.00 € | ||
| 100mg | 444.00 € | ||
| 1mL*10mM (DMSO) | 94.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Orteronel
CAS:566939-85-3
Orteronel ((S)-Orteronel)(TAK-700) was selected as a candidate for clinical evaluation.
Formula:
C18H17N3O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
307.35
Ref: TM-T6051
| 50mg | To inquire | ||
| 100mg | To inquire |
Estimated delivery in United States, on Thursday 19 Dec 2024
Verapamil
CAS:52-53-9
Verapamil (CP-16533-1), an oral calcium channel blocker, inhibits P-gp and CYP3A4, used for hypertension, arrhythmias, …
Formula:
C27H38N2O4
Purity:
99.53%
Color and Shape:
Oil
Molecular weight:
454.6
Ref: TM-T20656
| 10mg | 35.00 € | ||
| 25mg | 51.00 € | ||
| 50mg | 72.00 € | ||
| 100mg | 99.00 € | ||
| 200mg | 142.00 € | ||
| 500mg | 226.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Dehydroabiethylamine
CAS:1446-61-3
Dehydroabiethylamine (NSC-2955) boosts liver CYP2B, blocks PDKs & cholesterol transport, and has anti-tumor effects.
Formula:
C20H31N
Purity:
97.24%
Color and Shape:
Pale Yellow Viscous Liquid /Technical Grade/ Viscous Colorless To Amber Liquid
Molecular weight:
285.47
Ref: TM-T19783
| 1g | 38.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 7 Jan 2025
Azalanstat
CAS:143393-27-5
Azalanstat (RS 21607) is a mammalian lanosterol 14-alpha-demethylase inhibitor with hypocholesterolemic activity.
Formula:
C22H24ClN3O2S
Purity:
99.07% - 99.82%
Color and Shape:
Solid
Molecular weight:
429.96
Ref: TM-T25127
| 25mg | 1,397.00 € | ||
| 50mg | 1,820.00 € | ||
| 100mg | 2,297.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
LY 43578
CAS:26766-35-8
LY 43578 is an orally active aromatase inhibitor.
Formula:
C17H12Cl2N2O
Purity:
99.62%
Color and Shape:
Solid
Molecular weight:
331.2
Ref: TM-T27918
| 2mg | 36.00 € | ||
| 5mg | 53.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 124.00 € | ||
| 50mg | 177.00 € | ||
| 100mg | 263.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
MCH-1 antagonist 1
CAS:1039825-68-7
MCH-1 antagonist 1 also inhibits CYP3A4 (IC50: 10μM).MCH-1 antagonist 1 is a potent melanin concentrating …
Formula:
C25H26N4O2
Purity:
98%
Color and Shape:
Solid
Molecular weight:
414.5
Ref: TM-T11964
| 25mg | 1,410.00 € | ||
| 50mg | 1,852.00 € | ||
| 100mg | 2,338.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Seviteronel
CAS:1610537-15-9
Seviteronel (VT-464) is a novel CYP17 cleavage enzyme inhibitor and androgen receptor antagonist for the …
Formula:
C18H17F4N3O3
Purity:
100% - 99.98%
Color and Shape:
Solid
Molecular weight:
399.34
Ref: TM-T13312L
| 1mg | 109.00 € | ||
| 5mg | 253.00 € | ||
| 10mg | 361.00 € | ||
| 25mg | 616.00 € | ||
| 50mg | 874.00 € | ||
| 100mg | 1,167.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
Omeprazole Sodium
CAS:95510-70-6
Omeprazole Sodium is a proton pump inhibitor(PPI) and suppresses gastric acid secretion.
Formula:
C17H18N3NaO3S
Purity:
99.57%
Color and Shape:
Clear In Water
Molecular weight:
367.4
Ref: TM-T22391
| 100mg | 48.00 € | ||
| 200mg | 63.00 € | ||
| 500mg | 95.00 € | ||
| 1mL*10mM (DMSO) | 49.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
4'-Methylchrysoeriol
CAS:4712-12-3
4'-Methylchrysoeriol (3',4'-dimethoxyluteolin) is a P450 inhibitor and can be used in the study of neurological …
Formula:
C17H14O6
Purity:
98.4%
Color and Shape:
Solid
Molecular weight:
314.29
Ref: TM-T10163
| 1mg | 111.00 € | ||
| 5mg | 264.00 € | ||
| 10mg | 422.00 € | ||
| 25mg | 750.00 € | ||
| 50mg | 1,175.00 € | ||
| 100mg | 1,894.00 € | ||
| 1mL*10mM (DMSO) | 45.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
NP10679
CAS:2914889-88-4
NP10679 is a N-methyl-D-aspartate (NMDA) receptor inhibitor of the GluN2B subunit that inhibits histamine H1, …
Formula:
C23H26F3N3O3
Purity:
99.43%
Color and Shape:
Liquid
Molecular weight:
449.47
Ref: TM-T73447
| 1mg | 273.00 € | ||
| 5mg | 673.00 € | ||
| 10mg | 920.00 € | ||
| 25mg | 1,416.00 € | ||
| 50mg | 1,845.00 € | ||
| 100mg | 2,329.00 € |
Estimated delivery in United States, on Tuesday 21 Jan 2025
