P450
Cytochrome P450 enzymes are a large family of enzymes involved in the metabolism of various endogenous and exogenous compounds, including drugs, toxins, and hormones. P450 inhibitors are widely used to study drug metabolism, pharmacokinetics, and the role of these enzymes in disease states such as cancer and liver disorders. At CymitQuimica, we provide a broad selection of P450 inhibitors to support your research in pharmacology, toxicology, and metabolic regulation.
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TAK-700
CAS:426219-18-3
TAK-700 (Orteronel) is a selective 17, 20-lyase inhibitor, IC50 38 nM, with >1000x specificity vs …
Formula:
C18H17N3O2
Purity:
97.26%
Color and Shape:
Solid
Molecular weight:
307.35
Ref: TM-T6050
| 1mg | 40.00 € | ||
| 2mg | 52.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 134.00 € | ||
| 25mg | 260.00 € | ||
| 50mg | 417.00 € | ||
| 100mg | 603.00 € | ||
| 200mg | 824.00 € | ||
| 1mL*10mM (DMSO) | 87.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Lasiodin
CAS:28957-08-6
Lasiodin from Camellia sinensis has antitumor, antioxidant, antibacterial properties; halts NPC cell growth.
Formula:
C22H30O7
Purity:
99.90%
Color and Shape:
Solid
Molecular weight:
406.47
Ref: TM-TN1854
| 1mg | 142.00 € | ||
| 5mg | 346.00 € | ||
| 10mg | 500.00 € | ||
| 25mg | 794.00 € | ||
| 50mg | 1,067.00 € | ||
| 100mg | 1,438.00 € | ||
| 1mL*10mM (DMSO) | 389.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
CDD3506
CAS:197913-15-8
CDD3506 (1-TRITYL-1H-IMIDAZOL-4-AMINE) increases high-density lipoprotein cholesterol by targeting hepatic CYP3A.
Formula:
C22H19N3
Purity:
98.67%
Color and Shape:
Solid
Molecular weight:
325.41
Ref: TM-T13601
| 1mg | 42.00 € | ||
| 5mg | 93.00 € | ||
| 10mg | 135.00 € | ||
| 25mg | 263.00 € | ||
| 50mg | 381.00 € | ||
| 100mg | 543.00 € | ||
| 200mg | 717.00 € | ||
| 1mL*10mM (DMSO) | 92.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
AS1810722
CAS:909561-15-5
AS1810722, a fused bicyclic pyrimidine derivative, is an orally active and potent inhibitor of STAT6, …
Formula:
C25H25F2N7O
Purity:
99.13%
Color and Shape:
Solid
Molecular weight:
477.51
Ref: TM-T9043
| 1mg | 101.00 € | ||
| 5mg | 230.00 € | ||
| 10mg | 341.00 € | ||
| 25mg | 580.00 € | ||
| 50mg | 817.00 € | ||
| 1mL*10mM (DMSO) | 245.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
7-Ethoxyresorufin
CAS:5725-91-7
7-Ethoxyresorufin (Resorufin ethyl ether) (7-ER) is a fluorometric substrate for and competitive inhibitor of cytochrome …
Formula:
C14H11NO3
Purity:
99.09% - 99.35%
Color and Shape:
Red Solid
Molecular weight:
241.24
Ref: TM-T21507
| 1mg | 35.00 € | ||
| 2mg | 45.00 € | ||
| 5mg | 66.00 € | ||
| 10mg | 98.00 € | ||
| 25mg | 192.00 € | ||
| 50mg | 344.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Pyributicarb
CAS:88678-67-5
Pyributicarb (TSH-888) is a potent activator of both CYP3A4 gene and human pregnane X receptor …
Formula:
C18H22N2O2S
Purity:
≥95%
Color and Shape:
Solid
Molecular weight:
330.44
Ref: TM-T7618
| 25mg | 48.00 € | ||
| 50mg | 68.00 € | ||
| 100mg | 96.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Corydaline
CAS:518-69-4
Corydaline: an isoquinoline alkaloid that aids digestion, has anti-inflammatory and pain relief properties, and inhibits …
Formula:
C22H27NO4
Purity:
98.01% - 99.86%
Color and Shape:
Solid
Molecular weight:
369.45
Ref: TM-T5S2360
| 5mg | 60.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 143.00 € | ||
| 50mg | 204.00 € | ||
| 100mg | 303.00 € | ||
| 1mL*10mM (DMSO) | 67.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Stiripentol
CAS:49763-96-4
Stiripentol (BCX2600) (STP) is an anticonvulsant agent, which can inhibit N-demethylation of CLB to NCLB …
Formula:
C14H18O3
Purity:
99.93%
Color and Shape:
White Solid
Molecular weight:
234.29
Ref: TM-T4498
| 5mg | 51.00 € | ||
| 10mg | 81.00 € | ||
| 25mg | 147.00 € | ||
| 50mg | 202.00 € | ||
| 100mg | 341.00 € | ||
| 200mg | 504.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Bergapten
CAS:484-20-8
Bergapten (5-Methoxypsoralen), a psoralen, inhibits cell replication.
Formula:
C12H8O4
Purity:
99.48% - ≥95%
Color and Shape:
Needles From Alcohol; Soln In Sulfuric Acid Is Yellow-Gold Physical Description Grayish-White Micr°Crystalline Powder Or Yellow Fluffy Solid (Ntp 1992)
Molecular weight:
216.19
Ref: TM-T2143
| 1g | 96.00 € | ||
| 100mg | 35.00 € | ||
| 500mg | 73.00 € | ||
| 1mL*10mM (DMSO) | 51.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Tienilic Acid
CAS:40180-04-9
Tienilic Acid is a uricosuric diuretic with certain hepatotoxicity
Formula:
C13H8Cl2O4S
Purity:
99.61%
Color and Shape:
Solid
Molecular weight:
331.17
Ref: TM-T36125
| 5mg | 46.00 € | ||
| 10mg | 78.00 € | ||
| 25mg | 142.00 € | ||
| 50mg | 203.00 € | ||
| 100mg | 302.00 € | ||
| 200mg | 449.00 € | ||
| 500mg | 720.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
TETRAHYDROPIPERINE
CAS:23434-88-0
Tetrahydropiperine (Cosmoperine) is a natural product derived from piperine, can be used to treat convulsion, …
Formula:
C17H23NO3
Purity:
98.04% - 99.51%
Color and Shape:
Off-White Low Melting Solid With Characteristic Odour
Molecular weight:
289.37
Ref: TM-T5786
| 25mg | 42.00 € | ||
| 50mg | 57.00 € | ||
| 100mg | 79.00 € | ||
| 200mg | 103.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Pradefovir mesylate
CAS:625095-61-6
Pradefovir mesylate (Hepavir B) is converted to 9-(2-phosphonylmethoxyethyl)adenine (PMEA) in human liver microsomes with Km …
Formula:
C18H23ClN5O7PS
Purity:
98%
Color and Shape:
Solid
Molecular weight:
519.9
Ref: TM-T19526
| 1mg | 132.00 € | ||
| 5mg | 320.00 € | ||
| 10mg | 514.00 € | ||
| 25mg | 813.00 € | ||
| 50mg | 1,088.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Schisandrol B
CAS:58546-54-6
Schisandrol B fights neuroinflammation, liver/renal damage, and reduces cell growth via multiple signaling pathways.
Formula:
C23H28O7
Purity:
99.14% - 99.32%
Color and Shape:
Solid
Molecular weight:
416.46
Ref: TM-T6S1917
| 5mg | 71.00 € | ||
| 10mg | 95.00 € | ||
| 25mg | 199.00 € | ||
| 50mg | 299.00 € | ||
| 100mg | 447.00 € | ||
| 500mg | 1,016.00 € | ||
| 1mL*10mM (DMSO) | 78.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
3-(2-Naphthalenyl)-1-(3-pyridinyl)-2-propen-1-one
CAS:1031063-36-1
DMU2105 is a specific CYP1B1 inhibitor(CYP1B1 and CYP1A1 with IC50 of 10 nM and 742 …
Formula:
C18H13NO
Purity:
99.84%
Color and Shape:
Solid
Molecular weight:
259.3
Ref: TM-T8729
| 1mg | 49.00 € | ||
| 2mg | 67.00 € | ||
| 5mg | 87.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 223.00 € | ||
| 50mg | 335.00 € | ||
| 100mg | 502.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Ginsenoside F1
CAS:53963-43-2
Ginsenoside F1, a derivative of Rg1, inhibits CYP3A4 strongly and CYP2D6 weakly.
Formula:
C36H62O9
Purity:
98% - 99.86%
Color and Shape:
Solid
Molecular weight:
638.87
Ref: TM-T3401
| 5mg | 62.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 170.00 € | ||
| 50mg | 276.00 € | ||
| 1mL*10mM (DMSO) | 89.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Naloxegol oxalate
CAS:1354744-91-4
Naloxegol oxalate (NKTR-118) is a peripherally-selective opioid antagonist for the treatment of opioid-induced constipation.
Formula:
C36H55NO15
Purity:
100% - 99.82%
Color and Shape:
Solid
Molecular weight:
741.83
Ref: TM-T3355
| 5mg | 47.00 € | ||
| 10mg | 61.00 € | ||
| 25mg | 89.00 € | ||
| 50mg | 128.00 € | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
AMG-208
CAS:1002304-34-8
AMG-208 is a highly selective c-Met inhibitor with IC50 of 9 nM. Phase 1.
Formula:
C22H17N5O2
Purity:
99.27%
Color and Shape:
Solid
Molecular weight:
383.4
Ref: TM-T6260
| 2mg | 38.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 93.00 € | ||
| 25mg | 152.00 € | ||
| 50mg | 246.00 € | ||
| 100mg | 355.00 € | ||
| 200mg | 506.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Humantenmine
CAS:82354-38-9
1. Humantenmine is a toxic compound isolated from Gelsemium elegans Benth . 2. Humantenmine and …
Formula:
C19H22N2O3
Purity:
99.13% - 99.51%
Color and Shape:
Solid
Molecular weight:
326.39
Ref: TM-T2S0663
| 1mg | 47.00 € | ||
| 5mg | 138.00 € | ||
| 10mg | 212.00 € | ||
| 25mg | 361.00 € | ||
| 1mL*10mM (DMSO) | 134.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Gomisin G
CAS:62956-48-3
Gomisin G is a natural compound and exhibits potent anti-HIV activity (EC50: 0.006 μg/mL; therapeutic …
Formula:
C30H32O9
Purity:
98% - 99.95%
Color and Shape:
Solid
Molecular weight:
536.57
Ref: TM-TQ0217
| 1mg | 69.00 € | ||
| 5mg | 166.00 € | ||
| 10mg | 252.00 € | ||
| 25mg | 429.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 186.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
Uniconazole
CAS:83657-22-1
Uniconazole is a plant growth regulator that inhibit cytochrome P450 707As (Ki=68 nM).
Formula:
C15H18ClN3O
Purity:
99.94%
Color and Shape:
White-Light Brown Crystalline
Molecular weight:
291.78
Ref: TM-T21482
| 1g | 51.00 € | ||
| 5g | 109.00 € | ||
| 10g | 159.00 € | ||
| 500mg | 38.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
