
GluR
Glutamate Receptor inhibitors are compounds that block the activity of glutamate receptors, which are the main excitatory neurotransmitter receptors in the brain. These receptors play a pivotal role in synaptic transmission, plasticity, learning, and memory. Dysregulation of glutamate signaling is associated with various neurological disorders, including epilepsy, stroke, and neurodegenerative diseases. GluR inhibitors are essential for investigating the mechanisms of excitotoxicity and developing neuroprotective strategies. At CymitQuimica, we offer a range of glutamate receptor inhibitors to support your research in synaptic function, neuroprotection, and cognitive disorders.
Found 265 products of "GluR"
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VU0418506
CAS:VU0418506 is a positive allosteric modulator (PAM) of the metabotropic glutamate receptor 4 (mGlu4).Formula:C12H8ClFN4Purity:98%Color and Shape:SolidMolecular weight:262.67ACDPP hydrochloride
CAS:mGlu5 receptor antagonistFormula:C12H13ClN6OPurity:98%Color and Shape:SolidMolecular weight:292.72Ro 64-5229
CAS:mGlu2 antagonistFormula:C17H19Cl2N3OPurity:98%Color and Shape:SolidMolecular weight:352.26DL-AP4 Sodium salt
CAS:Broad spectrum EAA ligandFormula:C4H10NNaO5PPurity:98%Color and Shape:SolidMolecular weight:206.09VU6001966
CAS:VU6001966: potent, selective mGlu2 inhibitor (IC50=78 nM), negative modulator, with good CNS penetration.Formula:C17H15FN4O2Purity:98%Color and Shape:SolidMolecular weight:326.33VU6010572
CAS:VU6010572: potent, selective mGlu3 modulator, IC50 245 nM, high CNS penetration.Formula:C20H18FNO3Color and Shape:SolidMolecular weight:339.36VU0463841
CAS:VU0463841 is a mGlu5 negative allosteric modulators.Formula:C13H8ClFN4OColor and Shape:SolidMolecular weight:290.68VU 0360172 hydrochloride
CAS:positive allosteric modulator of mGlu5 receptorsFormula:C18H16ClFN2OPurity:98%Color and Shape:SolidMolecular weight:330.78ACPT-II
CAS:metabotropic receptor antagonistFormula:C8H11NO6Purity:98%Color and Shape:SolidMolecular weight:217.18mGluR2 modulator 4
CAS:Compound 47 is a potent mGluR2 enhancer with an EC50 of 0.8 μM, potentially useful for antipsychotic research.Formula:C18H18BrN3Color and Shape:SolidMolecular weight:356.26VU0400195
CAS:VU0400195 is a oral effective, positive allosteric modulator of the metabotropic glutamate receptor 4 (mGlu(4)).Formula:C21H16ClN3O3Purity:98%Color and Shape:SolidMolecular weight:393.82VU0404251
CAS:VU0404251 is a positive allosteric modulator of mGlu5.Formula:C19H23FN2O2Color and Shape:SolidMolecular weight:330.4VU0364289
CAS:VU0364289 is a positive allosteric modulator of mGlu5.Formula:C20H21N3O2Color and Shape:SolidMolecular weight:335.4VU0361747
CAS:VU0361747 is a positive allosteric modulators (PAM) of metabotropic glutamate receptor subtype 5 (mGlu5).Formula:C19H17FN2O2Color and Shape:SolidMolecular weight:324.35MSOP
CAS:MSOP is a selective antagonist of group III metabotropic glutamate receptor (KD of 51 μM for the L-AP4-sensitive presynaptic mGluR).Formula:C4H10NO6PPurity:98%Color and Shape:SolidMolecular weight:199.1LY487379 hydrochloride
CAS:Positive allosteric modulator of mGlu2 receptorsFormula:C21H20ClF3N2O4SPurity:98%Color and Shape:SolidMolecular weight:488.91AZ12216052
CAS:AZ12216052 is a GRP8 antagonist with anxiolytic and anti-inflammatory activity and can be used to study obesity and metabolic disorders.Formula:C19H22BrNOSPurity:99.29%Color and Shape:SolidMolecular weight:392.35CFMMC
CAS:CFMMC is an allosteric mGluR1 antagonist agent.
Formula:C22H28FNO4Color and Shape:SolidMolecular weight:389.46YM 230888
CAS:Selective mGlu1 antagonistFormula:C19H28N4OSPurity:98%Color and Shape:SolidMolecular weight:360.52LY2607540
CAS:LY2607540 is a metabotropic glutamate 2 potentiator with potential anxiolytic/antidepressant properties (EC(50) = 23 and 13 nM, respectively).Formula:C24H24F3N3O4Purity:98%Color and Shape:SolidMolecular weight:475.46
