
AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Found 645 products of "AChR"
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Muscarine
CAS:Muscarine is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.Formula:C9H20NO2Purity:98%Color and Shape:SolidMolecular weight:174.26Emraclidine
CAS:Emraclidine (CVL-231) is a novel, highly selective allosteric modulator of the muscarinic M4 receptor positive receptor.Cost-effective and quality-assured.Formula:C20H21F3N4OPurity:99.63% - 99.96%Color and Shape:SolidMolecular weight:390.4Ref: TM-T9694
1mg120.00€2mg170.00€5mg289.00€10mg467.00€25mg835.00€50mg1,134.00€100mg1,504.00€1mL*10mM (DMSO)319.00€Rocuronium
CAS:Rocuronium is an blocker of aminosteroid non-depolarizing neuromuscular.Formula:C32H53N2O4Purity:98%Color and Shape:SolidMolecular weight:529.77N-Ethyl-N-(3-pyridylmethyl)amine
CAS:N-Ethyl-N-(3-pyridylmethyl)amine has affinity for nAChR (Ki = 0.97 µM) and can be used in related research in the field of life sciences.Formula:C8H12N2Purity:99.65%Color and Shape:SolidMolecular weight:136.19[Ala2,8,9,11,19,22,24,25,27,28]-VIP
CAS:[Ala2,8,9,11,19,22,24,25,27,28]-VIP can be used for related research in the field of life sciences. Its product number is T36637 and CAS number is 866552-34-3.Formula:C131H219N41O33SColor and Shape:SolidMolecular weight:2928.51Bencycloquidium Bromide
CAS:Bencycloquidium bromide is an M3 muscarinic antagonist that reduces nasal secretion in allergic rhinitis and has high affinity for M3 receptors.Formula:C21H32BrNO2Color and Shape:SolidMolecular weight:410.39TDI-10229
CAS:TDI-10229: potent oral sAC inhibitor, IC50=195 nM. Good mouse pharmacokinetics for in vivo use.Formula:C16H16ClN5Purity:99.85% - 99.89%Color and Shape:SoildMolecular weight:313.78Ref: TM-T64355
1mg39.00€5mg157.00€10mg224.00€25mg409.00€50mg615.00€100mg888.00€200mg1,198.00€1mL*10mM (DMSO)167.00€M1/M4 muscarinic agonist 2
Compound 40 is a selective M1/M4 muscarinic antagonist with an IC50 of 19 nM for M1 receptors and 42 nM for M4 receptors [1].Color and Shape:Odour SolidBTMPS
CAS:BTMPS is a usage-dependent nicotinic antagonist capable of reducing acute withdrawal symptoms associated with morphine use.Formula:C28H52N2O4Purity:98.1%Color and Shape:SolidMolecular weight:480.72VU6028418
CAS:VU6028418 is a highly selective, potent, orally active M4mAChR antagonist that acts on hM4 (IC50: 4.1 nM).Formula:C23H27F3N4OColor and Shape:SolidMolecular weight:432.491M3/PDE4 modulator-1
M3/PDE4 Modulator-1 (compound 10f) serves as a bifunctional entity functioning both as an M3 mAChR antagonist and a PDE4 inhibitor.Formula:C38H41Cl2N3O8SColor and Shape:SolidMolecular weight:770.72DSPE-PEG2000-RVG29
DSPE-PEG2000-RVG29 is a PEG compound composed of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 specifically binds to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and can traverse the BBB.Color and Shape:Odour SolidBr-PBTC
CAS:Br-PBTC modulates nAChRs; targets α2/β2,4 subtypes; potent with 0.1-0.6 μM EC50; binds α subunit c-tail.Formula:C14H15BrN2OSColor and Shape:SolidMolecular weight:339.25(rel)-Asperparaline A
CAS:Aspergillimide, from A. japonicus, inhibits silkworm neuron nAChRs (IC50s: 20.2/39.6 nM), not affecting chicken nAChRs, and paralyzes silkworm larvae.
Formula:C20H29N3O3Color and Shape:SolidMolecular weight:359.47Rivanicline 2HCl
Rivanicline 2HCl is a selective neuronal nicotinic receptor inhibitor with a high affinity for the α4β2 subtype.Formula:C10H16Cl2N2Purity:99.4%Color and Shape:SoildMolecular weight:235.15Ref: TM-T12738L1
1mg34.00€5mg71.00€10mg100.00€25mg234.00€50mg420.00€100mg617.00€1mL*10mM (DMSO)110.00€Albanin A
Albanin A is a useful organic compound for research related to life sciences and the catalog number is T124310.Formula:C20H18O6Color and Shape:SolidMolecular weight:354.358Ebiratide
CAS:Ebiratide is an analog of ACTH 4-9.Formula:C48H73N11O10SPurity:98%Color and Shape:SolidMolecular weight:996.23Lupanine perchlorate
CAS:Lupanine perchlorate is a bioactive chemical.Formula:C15H25ClN2O5Color and Shape:SolidMolecular weight:348.82AC1-IN-1
CAS:AC1-IN-1 is a selective inhibitor of adenylyl cyclase type 1 (AC1, IC50 = 0.54 µM).
Formula:C18H18FN5O2Purity:99.89%Color and Shape:SolidMolecular weight:355.37(Rac)-Sabcomeline
CAS:(Rac)-Sabcomeline ((Rac)-SB-202026) is an M1/M4 muscarinic agonist used in the study of neurologic disorders such as schizophrenia.Formula:C10H15N3OPurity:99.14%Color and Shape:SolidMolecular weight:193.25Ref: TM-T68135L1
1mg109.00€2mg160.00€5mg261.00€10mg374.00€25mg583.00€50mg803.00€100mg1,063.00€200mg1,431.00€

