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AChR

AChR

Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.

Found 645 products of "AChR"

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  • Muscarine

    CAS:
    Muscarine is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.
    Formula:C9H20NO2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:174.26

    Ref: TM-T24507

    5mg
    1,144.00€
  • Emraclidine

    CAS:
    Emraclidine (CVL-231) is a novel, highly selective allosteric modulator of the muscarinic M4 receptor positive receptor.Cost-effective and quality-assured.
    Formula:C20H21F3N4O
    Purity:99.63% - 99.96%
    Color and Shape:Solid
    Molecular weight:390.4

    Ref: TM-T9694

    1mg
    120.00€
    2mg
    170.00€
    5mg
    289.00€
    10mg
    467.00€
    25mg
    835.00€
    50mg
    1,134.00€
    100mg
    1,504.00€
    1mL*10mM (DMSO)
    319.00€
  • Rocuronium

    CAS:
    Rocuronium is an blocker of aminosteroid non-depolarizing neuromuscular.
    Formula:C32H53N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:529.77

    Ref: TM-T12748

    25mg
    1,369.00€
  • N-Ethyl-N-(3-pyridylmethyl)amine

    CAS:
    N-Ethyl-N-(3-pyridylmethyl)amine has affinity for nAChR (Ki = 0.97 µM) and can be used in related research in the field of life sciences.
    Formula:C8H12N2
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:136.19

    Ref: TM-TN9660

    50mg
    42.00€
    100mg
    57.00€
  • [Ala2,8,9,11,19,22,24,25,27,28]-VIP

    CAS:
    [Ala2,8,9,11,19,22,24,25,27,28]-VIP can be used for related research in the field of life sciences. Its product number is T36637 and CAS number is 866552-34-3.
    Formula:C131H219N41O33S
    Color and Shape:Solid
    Molecular weight:2928.51

    Ref: TM-T36637

    1mg
    190.00€
  • Bencycloquidium Bromide

    CAS:
    Bencycloquidium bromide is an M3 muscarinic antagonist that reduces nasal secretion in allergic rhinitis and has high affinity for M3 receptors.
    Formula:C21H32BrNO2
    Color and Shape:Solid
    Molecular weight:410.39

    Ref: TM-T26770

    25mg
    3,615.00€
    50mg
    4,708.00€
    100mg
    5,943.00€
  • TDI-10229

    CAS:
    TDI-10229: potent oral sAC inhibitor, IC50=195 nM. Good mouse pharmacokinetics for in vivo use.
    Formula:C16H16ClN5
    Purity:99.85% - 99.89%
    Color and Shape:Soild
    Molecular weight:313.78

    Ref: TM-T64355

    1mg
    39.00€
    5mg
    157.00€
    10mg
    224.00€
    25mg
    409.00€
    50mg
    615.00€
    100mg
    888.00€
    200mg
    1,198.00€
    1mL*10mM (DMSO)
    167.00€
  • M1/M4 muscarinic agonist 2


    Compound 40 is a selective M1/M4 muscarinic antagonist with an IC50 of 19 nM for M1 receptors and 42 nM for M4 receptors [1].
    Color and Shape:Odour Solid

    Ref: TM-T81893

    5mg
    To inquire
    50mg
    To inquire
  • BTMPS

    CAS:
    BTMPS is a usage-dependent nicotinic antagonist capable of reducing acute withdrawal symptoms associated with morphine use.
    Formula:C28H52N2O4
    Purity:98.1%
    Color and Shape:Solid
    Molecular weight:480.72

    Ref: TM-T203537

    10g
    36.00€
  • VU6028418

    CAS:
    VU6028418 is a highly selective, potent, orally active M4mAChR antagonist that acts on hM4 (IC50: 4.1 nM).
    Formula:C23H27F3N4O
    Color and Shape:Solid
    Molecular weight:432.491

    Ref: TM-T71675

    5mg
    931.00€
    25mg
    1,458.00€
    50mg
    1,839.00€
    100mg
    2,322.00€
  • M3/PDE4 modulator-1


    M3/PDE4 Modulator-1 (compound 10f) serves as a bifunctional entity functioning both as an M3 mAChR antagonist and a PDE4 inhibitor.
    Formula:C38H41Cl2N3O8S
    Color and Shape:Solid
    Molecular weight:770.72

    Ref: TM-T79618

    5mg
    To inquire
    50mg
    To inquire
  • DSPE-PEG2000-RVG29


    DSPE-PEG2000-RVG29 is a PEG compound composed of DSPE and rabies virus glycoprotein 29 (RVG29). RVG29 specifically binds to nicotinic acetylcholine receptors (nAChR) at the blood-brain barrier (BBB) and can traverse the BBB.
    Color and Shape:Odour Solid

    Ref: TM-TCL-01083

    10mg
    To inquire
    50mg
    To inquire
  • Br-PBTC

    CAS:
    Br-PBTC modulates nAChRs; targets α2/β2,4 subtypes; potent with 0.1-0.6 μM EC50; binds α subunit c-tail.
    Formula:C14H15BrN2OS
    Color and Shape:Solid
    Molecular weight:339.25

    Ref: TM-T39286

    5mg
    922.00€
  • (rel)-Asperparaline A

    CAS:

    Aspergillimide, from A. japonicus, inhibits silkworm neuron nAChRs (IC50s: 20.2/39.6 nM), not affecting chicken nAChRs, and paralyzes silkworm larvae.

    Formula:C20H29N3O3
    Color and Shape:Solid
    Molecular weight:359.47

    Ref: TM-T37609

    1mg
    251.00€
    5mg
    938.00€
  • Rivanicline 2HCl


    Rivanicline 2HCl is a selective neuronal nicotinic receptor inhibitor with a high affinity for the α4β2 subtype.
    Formula:C10H16Cl2N2
    Purity:99.4%
    Color and Shape:Soild
    Molecular weight:235.15

    Ref: TM-T12738L1

    1mg
    34.00€
    5mg
    71.00€
    10mg
    100.00€
    25mg
    234.00€
    50mg
    420.00€
    100mg
    617.00€
    1mL*10mM (DMSO)
    110.00€
  • Albanin A


    Albanin A is a useful organic compound for research related to life sciences and the catalog number is T124310.
    Formula:C20H18O6
    Color and Shape:Solid
    Molecular weight:354.358

    Ref: TM-T124310

    1mg
    To inquire
    5mg
    To inquire
  • Ebiratide

    CAS:
    Ebiratide is an analog of ACTH 4-9.
    Formula:C48H73N11O10S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:996.23

    Ref: TM-TP2379

    100mg
    To inquire
    500mg
    To inquire
  • Lupanine perchlorate

    CAS:
    Lupanine perchlorate is a bioactive chemical.
    Formula:C15H25ClN2O5
    Color and Shape:Solid
    Molecular weight:348.82

    Ref: TM-T32964

    1mg
    269.00€
    5mg
    1,189.00€
  • AC1-IN-1

    CAS:

    AC1-IN-1 is a selective inhibitor of adenylyl cyclase type 1 (AC1, IC50 = 0.54 µM).

    Formula:C18H18FN5O2
    Purity:99.89%
    Color and Shape:Solid
    Molecular weight:355.37

    Ref: TM-T60003

    1mg
    90.00€
    5mg
    188.00€
    10mg
    316.00€
    25mg
    512.00€
    50mg
    702.00€
    100mg
    940.00€
    500mg
    1,872.00€
  • (Rac)-Sabcomeline

    CAS:
    (Rac)-Sabcomeline ((Rac)-SB-202026) is an M1/M4 muscarinic agonist used in the study of neurologic disorders such as schizophrenia.
    Formula:C10H15N3O
    Purity:99.14%
    Color and Shape:Solid
    Molecular weight:193.25

    Ref: TM-T68135L1

    1mg
    109.00€
    2mg
    160.00€
    5mg
    261.00€
    10mg
    374.00€
    25mg
    583.00€
    50mg
    803.00€
    100mg
    1,063.00€
    200mg
    1,431.00€