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AChR

AChR

Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.

Found 575 products of "AChR"

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  • Nitrobenzylthioinosine
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    Nitrobenzylthioinosine

    CAS:
    <p>Nitrobenzylthioinosine (NBMPR) is an inhibitor of ENT1 transporter that binds to ENT1 transporter with high affinity.</p>
    Formula:C17H17N5O6S
    Purity:99.69% - 99.74%
    Color and Shape:Off-White Solid
    Molecular weight:419.41

    Ref: TM-T8551

  • Monepantel
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    Monepantel

    CAS:
    <p>Monepantel (AAD1566) is an organic anthelmintic and an antagonist of nAChRs from roundworms and esophageostomy.</p>
    Formula:C20H13F6N3O2S
    Purity:99.83%
    Color and Shape:White Powder
    Molecular weight:473.39

    Ref: TM-T16126

  • Velufenacin
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    Velufenacin

    CAS:
    <p>Velufenacin is an antagonist of muscarinic receptor[1].</p>
    Formula:C19H20ClFN2O2
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:362.83

    Ref: TM-T9771

  • Pentoxyverine
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    Pentoxyverine

    CAS:
    <p>Pentoxyverine (Carbetapentan) is an orally available cough suppressant, an antagonist of muscarinic receptor M1 and an agonist of the σ1 receptor.</p>
    Formula:C20H31NO3
    Purity:97.11%
    Color and Shape:Solid
    Molecular weight:333.47

    Ref: TM-T22284

  • Xanomeline tartrate
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    Xanomeline tartrate

    CAS:
    <p>Xanomeline tartrate (LY 246708 tartrate) 是 M1和 M4 mAChR 激动剂，具有抗精神病样活性，可改善认知，可用于研究精神分裂症和阿尔茨海默病。</p>
    Formula:C18H29N3O7S
    Purity:99.19%
    Color and Shape:Solid
    Molecular weight:431.5

    Ref: TM-T39010

  • AF-710B
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    AF-710B

    CAS:
    <p>AF710B is an enantiomer of AF710. AF-710B is also a sigma and M1 muscarinic receptors agonist.</p>
    Formula:C20H27N3OS
    Purity:98.62% - 99.89%
    Color and Shape:Solid
    Molecular weight:357.51

    Ref: TM-T23649

  • Mepenzolate Bromide
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    Mepenzolate Bromide

    CAS:
    <p>Mepenzolate Bromide (Colibantil) is a muscarinic antagonist used to treat gastrointestinal conditions.</p>
    Formula:C21H26BrNO3
    Purity:95.73% - 99.21%
    Color and Shape:Solid
    Molecular weight:420.34

    Ref: TM-T0794

  • Pipecuronium bromide
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    Pipecuronium bromide

    CAS:
    <p>Pipecuronium bromide (RGH-1106) is an nAChR antagonist that also acts as a non-depolarising steroidal neuromuscular blocker that causes muscle relaxation.</p>
    Formula:C35H62Br2N4O4
    Purity:>99.99%
    Color and Shape:Powder
    Molecular weight:762.7

    Ref: TM-T12481

  • Varenicline
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    Varenicline

    CAS:
    <p>Varenicline (CP 526555) is a selective partial agonist of the α4β2 nAChR and a full agonist of the α3β4 nAChR and α7 nAChR.</p>
    Formula:C13H13N3
    Purity:99.76%
    Color and Shape:Solid
    Molecular weight:211.26

    Ref: TM-T4246L

  • Atropine hydrobromide
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    Atropine hydrobromide

    CAS:
    <p>Atropine hydrobromide is a biochemical.</p>
    Formula:C17H24BrNO3
    Color and Shape:Solid
    Molecular weight:370.28

    Ref: TM-T30206

  • Anatabine dicitrate
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    Anatabine dicitrate

    <p>Anatabine dicitrate is a tobacco alkaloid that can cross the blood-brain barrier.</p>
    Formula:C22H28N2O14
    Purity:98%
    Color and Shape:Solid
    Molecular weight:544.46

    Ref: TM-T10318

  • Pyrantel
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    Pyrantel

    CAS:
    <p>Pyrantel: Nicotinic agonist; causes spastic paralysis in nematodes by depolarizing block.</p>
    Formula:C11H14N2S
    Purity:98%
    Color and Shape:Crystals From Methanol Yellowish Crystalline Powder
    Molecular weight:206.31

    Ref: TM-T0395L

  • Flavoxate
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    Flavoxate

    CAS:
    <p>Flavoxate is an anticholinergic with antimuscarinic effects.</p>
    Formula:C24H25NO4
    Color and Shape:Solid
    Molecular weight:391.46

    Ref: TM-T0703L

  • CymitQuimica logo
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    (±)-Atropine-d3 (N-methyl-d3)

    CAS:
    (±)-Atropine-d3 (N-methyl-d3) is a deuterated compound of (±)-Atropine. (±)-Atropine has a CAS number of 51-55-8. Atropine Sulfate is the sulfate salt of atropine, a naturally-occurring alkaloid isolated from the plant Atropa belladonna. Atropine functions as a sympathetic, competitive antagonist of muscarinic cholinergic receptors, thereby abolishing the effects of parasympathetic stimulation.
    Formula:C17H20D3NO3
    Molecular weight:292.39

    Ref: TM-TMID-0258

  • Oxantel
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    Oxantel

    CAS:
    <p>Oxantel is a fumarate reductase inhibitor with anthelmintic activity.</p>
    Formula:C13H16N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:216.28

    Ref: TM-T0323L

  • Aprofene
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    Aprofene

    CAS:
    <p>Aprofene blocks acetylcholine receptors, used for peptic ulcers, endarteritis, cholecystitis, and colitis.</p>
    Formula:C21H27NO2
    Color and Shape:Solid
    Molecular weight:325.44

    Ref: TM-T25104

  • Catestatin
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    Catestatin

    CAS:
    <p>Non-competitive inhibitor of nicotinic receptors; blocks cationic signalling and catecholamine release; stimulates histamine release. IC50 ~200-250nM.</p>
    Formula:C107H173N37O26S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:2425.84

    Ref: TM-TP2058

  • Dianicline dihydrochloride
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    Dianicline dihydrochloride

    CAS:
    <p>Dianicline dihydrochloride is a partial agonist of α4β2 nicotinic acetylcholine receptor. It increases cessation rates in a dose-dependent manner.</p>
    Formula:C13H16N2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:216.28

    Ref: TM-T15112

  • Biperiden lactate
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    Biperiden lactate

    CAS:
    <p>Biperiden lactate is a biochemical.</p>
    Formula:C24H35NO4
    Color and Shape:Solid
    Molecular weight:401.54

    Ref: TM-T30456

  • VU0029767
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    VU0029767

    CAS:
    <p>VU0029767 is an allosteric enhancer of the M1 muscarinic receptor, capable of modulating the receptor's activity. This compound enhances M1 receptor activity by increasing agonist affinity. However, VU0029767 demonstrates distinct characteristics from other compounds, particularly under varying experimental conditions such as its interaction with mutated M1 receptors and its effects on downstream signaling pathways.</p>
    Formula:C21H21N3O3
    Color and Shape:Solid
    Molecular weight:363.41

    Ref: TM-T200818