AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Found 645 products of "AChR"
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Syn-Ake acetate
CAS:Syn-Ake acetate (Dipeptide diaminobutyroyl benzylamide) is a muscarinic acetylcholine receptor antagonist.Formula:C19H29N5O3·2(C2H4O2)Purity:99.60%Color and Shape:SolidMolecular weight:495.58α-Conotoxin MII acetate
α-Conotoxin MII acetate is a 16-amino acid peptide from the venom of the marine snail Conus magus.Formula:C69H107N23O24S4Purity:94.82% - 97.79%Color and Shape:SolidMolecular weight:1770.99VU0152099
CAS:VU0152099 is a potent and selective M4 mAChR allosteric potentiator(EC50 = 380 ± 93 nM).Formula:C18H17N3O3SPurity:98.46%Color and Shape:SolidMolecular weight:355.41Bestim
CAS:Bestim is an immunomodulatory dipeptide that is synthetic.Formula:C16H19N3O5Purity:99.76%Color and Shape:SolidMolecular weight:333.34Ref: TM-T25146
1mg84.00€5mg168.00€10mg245.00€25mg404.00€50mg567.00€100mg767.00€200mg1,018.00€1mL*10mM (DMSO)172.00€Oxyphenonium bromide
CAS:Oxyphenonium bromide is an anticholinergic used to study and treat ulcers and relieve visceral spasms.
Formula:C21H34BrNO3Purity:98.96%Color and Shape:SolidMolecular weight:428.404Pozanicline dihydrochloride
CAS:Pozanicline dihydrochloride (ABT-089 dihydrochloride) is an orally bioavailable agonist of nicotinic acetylcholine receptor (nAChR) (Ki = 16.7 nM)Formula:C11H18Cl2N2OPurity:98%Color and Shape:SolidMolecular weight:265.18SEN12333
CAS:SEN12333 is an α7 nicotinic acetylcholine receptor (nAChR) agonistFormula:C20H25N3O2Purity:99.02%Color and Shape:SolidMolecular weight:339.43Ref: TM-T23348
2mg37.00€5mg54.00€10mg90.00€25mg164.00€50mg255.00€100mg409.00€200mg590.00€1mL*10mM (DMSO)59.00€NS9283
CAS:NS9283, a positive allosteric modulator selective for the α4β2 form, reduces ethanol consumption.
Formula:C14H8N4OPurity:99.12%Color and Shape:SolidMolecular weight:248.24W-84 dibromide
CAS:W-84 dibromide (HDMPPA) is a M2-receptor selective modulator.Formula:C32H44Br2N4O4Purity:95.56%Color and Shape:SolidMolecular weight:708.524BP-TQS
CAS:4BP-TQS is an allosteric agonist of α7 nAChRs.Formula:C18H17BrN2O2SPurity:99.96%Color and Shape:SolidMolecular weight:405.31ST034307
CAS:ST034307 is an effective and selective inhibitor of adenylyl cyclase 1 (IC50: 2.3 μM).Formula:C10H4Cl4O2Purity:99.28%Color and Shape:SolidMolecular weight:297.95Ref: TM-T16938
1mg35.00€2mg50.00€5mg77.00€10mg109.00€25mg224.00€50mg353.00€100mg567.00€200mg797.00€1mL*10mM (DMSO)84.00€Irsogladine
CAS:Irsogladine (Dicloguamine) is an anti-ulcer agent that promotes gap junction intercellular communication via M1 muscarinic acetylcholine receptor binding.Formula:C9H7Cl2N5Purity:99.74% - 99.91%Color and Shape:White Or Colorless Crystal Or Crystalline Powder Odorless Slightly BitterMolecular weight:256.09PHA 543613 hydrochloride
CAS:PHA-543613 hydrochloride, a potent α7 nicotinic receptor agonist, may treat schizophrenia-related cognitive deficits.Formula:C15H18ClN3O2Color and Shape:SolidMolecular weight:307.78A 582941 HCl (848591-90-2(free base))
A-582941 is a alpha7 neuronal nicotinic receptor agonist with broad spectrum cognition-enhancing propertiesFormula:C17H21ClN4Purity:99.83%Color and Shape:SolidMolecular weight:316.83Ref: TM-T8725
1mg58.00€5mg118.00€10mg172.00€25mg281.00€50mg396.00€100mg537.00€200mg712.00€1mL*10mM (DMSO)116.00€Dicyclomine
CAS:Dicyclomine: oral muscarinic antagonist, eases GI muscle spasms, high affinity for M1/M2 receptors, Ki of 5.1 nM/54.6 nM.Formula:C19H35NO2Color and Shape:SolidMolecular weight:309.49CCMI
CAS:CCMI (AVL-3288) is a potent and selective modulator of α7 nAChR-positive allosteric.Formula:C19H15Cl2N3O2Purity:>99.99%Color and Shape:SolidMolecular weight:388.25TBPB
CAS:TBPB is an allosteric M1 mAChR agonist.
Formula:C25H32N4OPurity:97.87% - 99.9%Color and Shape:SolidMolecular weight:404.55α-Conotoxin PIA acetate
α-Conotoxin PIA acetate is an antagonist of nicotinic acetylcholine receptor (nAChR) mainly targeting α6 and α3 subunits.Purity:98%Color and Shape:LiquidMolecular weight:N/A9-Ethyladenine
CAS:9-Ethyladenine (6-Amino-9-ethylpurine) is a partially potent APRT (adenine phosphoribosyltransferase) inhibitor [1].Formula:C7H9N5Purity:99.35% - 99.37%Color and Shape:SolidMolecular weight:163.18Mecamylamine hydrochloride
CAS:Mecamylamine hydrochloride (Mevasin) is a nicotinic antagonist, used as a ganglionic blocker in hypertension.Formula:C11H22ClNPurity:99.76% - >99.99%Color and Shape:White SolidMolecular weight:203.75
