
AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Found 575 products of "AChR"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
SIB 1508Y maleate
CAS:<p>neuronal nicotinic ACh receptor agonist</p>Formula:C16H18N2O4Purity:98%Color and Shape:SolidMolecular weight:302.33LRE1
CAS:<p>LRE1 is a specific and allosteric soluble adenylyl cyclase inhibitor.</p>Formula:C12H13ClN4SPurity:>99.99%Color and Shape:SolidMolecular weight:280.78Terodiline
CAS:<p>Terodiline is an orally available selective muscarinic M1 receptor and calcium channel antagonist for the study of diseases caused by abnormal bladder function.</p>Formula:C20H27NPurity:98.20% - 99.59%Color and Shape:SolidMolecular weight:281.44Methacholine bromide
CAS:<p>Methacholine bromide is a potent M3 agonist for diagnosing asthma by identifying bronchial hyperresponsiveness.</p>Formula:C8H18BrNO2Color and Shape:SolidMolecular weight:240.141Nuvenzepine
CAS:<p>Nuvenzepine is an antagonist of mAChR. It has the potential for gastrospasm treatment.</p>Formula:C19H20N4O2Purity:98%Color and Shape:SolidMolecular weight:336.39DA 4626
CAS:<p>DA 4626 is an H2-receptor antagonist with KB values akin to those in standard assays.</p>Formula:C14H18N4Purity:98%Color and Shape:SolidMolecular weight:242.32Telenzepine
CAS:<p>Telenzepine is a potent and selective M1 antimuscarinic.</p>Formula:C19H22N4O2SPurity:98%Color and Shape:SolidMolecular weight:370.47AC260584
CAS:AC260584 is an M1 muscarinic receptor allosteric agonist (pEC50: 7.6).Formula:C20H29FN2O2Color and Shape:SolidMolecular weight:348.45Neramexane Mesylate
CAS:<p>Neramexane: NMDA & nicotinic receptor blocker with neuroprotective, antidepressant, and cognitive-enhancing effects.</p>Formula:C12H27NO3SPurity:98%Color and Shape:SolidMolecular weight:265.41Chlorisondamine diiodide
CAS:<p>long lasting nicotinic antagonist</p>Formula:C14H20Cl4I2N2Color and Shape:SolidMolecular weight:611.94ML381
CAS:<p>ML381 is a M5-orthosteric antagonist with a high selectivity of muscarinic subtype.</p>Formula:C21H21N3O4Color and Shape:SolidMolecular weight:379.41ML169
CAS:<p>ML169 is a selective and brain penetrant M1 positive allosteric modulator (PAM).</p>Formula:C21H17BrFN3O4SPurity:98%Color and Shape:SolidMolecular weight:506.34Zamifenacin
CAS:<p>Zamifenacin obviously decreases colonic motility in irritable bowel syndrome. Zamifenacin is an effective gut-selective muscarinic M3 receptor antagonist.</p>Formula:C27H29NO3Purity:98%Color and Shape:SolidMolecular weight:415.52BNC375
CAS:<p>BNC375 is a α7 nAChRs type I positive allosteric modulator (EC50: 1.9 μM).</p>Formula:C19H23ClN2O3SPurity:98%Color and Shape:SolidMolecular weight:394.92(R,R)-Reboxetine mesylate
CAS:<p>(R,R)-Reboxetine mesylate: Antidepressant, high bioavailability, (R,R) enantiomer, selective for noradrenaline, low toxicity.</p>Formula:C20H27NO6SColor and Shape:SolidMolecular weight:409.5M1 ligand 1
CAS:<p>Compound 3b-b: N-desmethyl arecoline derivative, muscarinic M1 ligand, potential PET radiotracer.</p>Formula:C20H21NO2Color and Shape:SolidMolecular weight:307.39Benzatropine
CAS:<p>Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.</p>Formula:C21H25NOPurity:98%Color and Shape:SolidMolecular weight:307.43Muscarine iodide
CAS:<p>Muscarinic acetylcholine receptor agonist</p>Formula:C9H20INO2Purity:98%Color and Shape:SolidMolecular weight:301.17Tridihexethyl chloride
CAS:<p>Tridihexethyl is an anticholinergic, antimuscarinic, and antispasmolytic drug, which can be used to treat acquired nystagmus or peptic ulcer disease.</p>Formula:C21H36ClNOColor and Shape:SolidMolecular weight:353.97TC 2559 difumarate
CAS:<p>partial agonist of α4β2 nicotinic acetylcholine receptor</p>Formula:C12H18N2OC4H404Purity:98%Color and Shape:SolidMolecular weight:380.39
