AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Found 643 products of "AChR"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Pirenzepine dihydrochloride
CAS:Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.Formula:C19H21N5O2·2HClPurity:99.48% - 99.62%Color and Shape:White PowderMolecular weight:424.32DL-trihexyphenidyl hydrochloride
CAS:DL-trihexyphenidyl hydrochloride (Trihexyphenidyl HCl) is a muscarinic antagonist.Formula:C20H32ClNOPurity:99.63% - 99.71%Color and Shape:SolidMolecular weight:337.93Nefiracetam
CAS:Nefiracetam (DM9384), in Phase 2 trials, enhances GABA, choline, monoamine systems, and treats Ro 5-4864 convulsions.Formula:C14H18N2O2Purity:97.37%Color and Shape:White To Off-White Crystalline PowderMolecular weight:246.3Fesoterodine fumarate
CAS:Fesoterodine fumarate (Toviaz) is a competitive muscarinic receptor antagonist with muscle relaxant and urinary antispasmodic properties.Formula:C26H37NO3·C4H4O4Purity:99.16%Color and Shape:White SolidMolecular weight:527.65Ref: TM-T1475
2mg34.00€5mg50.00€10mg71.00€25mg100.00€50mg137.00€100mg205.00€500mg396.00€1mL*10mM (DMSO)54.00€Solifenacin succinate
CAS:Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.Formula:C23H26N2O2·C4H6O4Purity:99.85% - 99.98%Color and Shape:SolidMolecular weight:480.56Temephos
CAS:Temephos is an organothiophosphate insecticide and cholinesterase inhibitor for treating water with disease-carrying insects.
Formula:C16H20O6P2S3Purity:≥95%Color and Shape:White Crystalline Solid Or LiquidMolecular weight:466.47Valethamate bromide
CAS:Valethamate bromide (Resitan) is an anticholinergic agent that has antispasmodic effects and inhibits glandular secretion.Formula:C19H32BrNO2Purity:>99.99%Color and Shape:SolidMolecular weight:386.37(Rac)-ABT-202 dihydrochloride
CAS:(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.Formula:C9H15Cl2N3Purity:97.4%Color and Shape:SolidMolecular weight:236.142Procainamide hydrochloride
CAS:Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analogFormula:C13H21N3O·HClPurity:99.83% - 99.97%Color and Shape:White To Slightly Yellow PowderMolecular weight:271.79Droperidol
CAS:Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.Formula:C22H22FN3O2Purity:97.16% - 98%Color and Shape:SolidMolecular weight:379.43Acetamiprid
CAS:Acetamiprid: nAChR agonist, global neonicotinoid insecticide linked to neuromuscular/reproductive issues.Formula:C10H11ClN4Purity:99.66%Color and Shape:White PowderMolecular weight:222.67Rocuronium bromide
CAS:Rocuronium bromide (ORG 9426) is a muscle relaxant or aminosteroid non-depolarizing neuromuscular blocker, which is used to provide skeletal muscle relaxation.Formula:C32H53BrN2O4Purity:99.77% - >99.99%Color and Shape:White Or Off-White PowderMolecular weight:609.68MK-7622
CAS:MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.Formula:C25H25N3O2Purity:99.77% - 99.8%Color and Shape:SolidMolecular weight:399.48Nebracetam hydrochloride
CAS:Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.Formula:C12H17ClN2OPurity:99.23%Color and Shape:SolidMolecular weight:240.729Dicyclomine hydrochloride
CAS:Dicyclomine hydrochloride is a muscarinic antagonist used as an antispasmodic and in urinary incontinence.Formula:C19H36ClNO2Purity:99.81%Color and Shape:SolidMolecular weight:345.95Pyrantel tartrate
CAS:Pyrantel tartrate (Banminth) is broad spectrum anthelmintic for livestock.Formula:C15H20N2O6SPurity:99.96%Color and Shape:White CrystalsMolecular weight:356.39Carbachol
CAS:Carbachol (Carbamoylcholine chloride), an analog of acetylcholine, serves as a valuable tool in the investigation of various physiological responses mediated by nicotinic (nAChR) and muscarinic (mAChR) acetylcholine receptors. These responses include smooth muscle contraction, gut motility, and neuronal signaling. Known for its agonistic properties, Carbachol activates both nAChR and mAChR, with reported Ki values ranging from 10 to 10,000 nM for different receptor types and experimental preparations.Formula:C6H15ClN2O2Purity:>99.99%Color and Shape:SolidMolecular weight:182.65TAK-071
CAS:TAK-071 is a potent, novel and highly selective modulator of muscarinic acetylcholine receptor 1 (M1R) positive allosteric(EC50 : 520 nM).
Formula:C24H24FN3O3Purity:98.02%Color and Shape:SolidMolecular weight:421.46Bethanechol chloride
CAS:Bethanechol chloride: muscarinic agonist, boosts smooth muscle tone, used post-abdominal surgery & for urinary retention; may cause hypotension & bronchospasm.Formula:C7H17N2O2·ClPurity:95% - 99.73%Color and Shape:White CrystallineMolecular weight:196.68Ribavirin
CAS:Ribavirin (Tribavirin) is a synthetic nucleoside analog of ribofuranose with activity against hepatitis C virus and other RNA viruses.Formula:C8H12N4O5Purity:99.09% - 99.83%Color and Shape:Less Solid Colourless SolidMolecular weight:244.20
