
AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Found 575 products of "AChR"
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Milameline
CAS:<p>Milameline is a muscarinic receptor agonist that improves cognition.</p>Formula:C8H14N2OColor and Shape:SolidMolecular weight:154.21Biricodar dicitrate
CAS:<p>Biricodar dicitrate (VX-710) is a potent MDR inhibitor with no anticancer activity and can be used to study prostate cancer.</p>Formula:C46H57N3O21Purity:97.78% - 99.78%Color and Shape:SolidMolecular weight:987.95Sofiniclin
CAS:<p>Sofiniclin (ABT 894) is an agonist of nicotinic acetylcholine receptor (nAChR). It is used for the research for attention-deficit/hyperactivity disorder (ADHD).</p>Formula:C10H11Cl2N3Purity:98%Color and Shape:SolidMolecular weight:244.12Bibn 99
CAS:<p>Bibn 99, a lipophilic and selective muscarinic M2 receptor antagonist, has applications in cognitive performance and Alzheimer's Disease.</p>Formula:C31H42ClN5O3Color and Shape:SolidMolecular weight:568.15VU 6008667
CAS:VU 6008667 is a selective negative allosteric M5 NAM modulator (IC50s: 1.2 μM and 1.6 μM for human M5 and rat M5, respectively).Formula:C24H17ClF2N2O2Purity:98%Color and Shape:SolidMolecular weight:438.85Rivanicline
CAS:<p>Rivanicline is a selective α4β2 nicotinic receptor agonist (Ki=26 nM), with >1,000x less affinity for α7 receptors.</p>Formula:C10H14N2Purity:98%Color and Shape:SolidMolecular weight:162.23Rapacuronium bromide
CAS:Rapacuronium bromide is an allosteric muscarinic acetylcholine receptor (mAChR) modulator.Formula:C37H61BrN2O4Purity:98%Color and Shape:SolidMolecular weight:677.8ML375
CAS:<p>ML375 is a potent, selective and CNS penetrant M5 negative allosteric modulator (NAM).</p>Formula:C23H15ClF2N2O2Color and Shape:SolidMolecular weight:424.83CP-601927
CAS:<p>CP-601927 is a nicotinic acetylcholine receptor (NACHR) agonist with permeability, high affinity, and selectivity.</p>Formula:C12H12F3NColor and Shape:SolidMolecular weight:227.23Arecaidine propargyl ester tosylate
CAS:<p>Arecaidine propargyl ester tosylate is a muscarinic receptor agonist.</p>Formula:C17H21NO5SPurity:98%Color and Shape:SolidMolecular weight:351.42VMY-2-95
CAS:<p>VMY-2-95 is an α4β2 nicotinic acetylcholine receptors (nAChRs) selective desensitizer.</p>Formula:C17H16N2OColor and Shape:SolidMolecular weight:264.32RJR 2429 dihydrochloride
CAS:<p>nAChR agonist that displays selectivity for α4β2</p>Formula:C12H18Cl2N2Purity:98%Color and Shape:SolidMolecular weight:261.19J 104129 fumarate
CAS:<p>M3 muscarinic receptor antagonist</p>Formula:C24H36N2O2Purity:98%Color and Shape:SolidMolecular weight:384.55Alvameline maleate
CAS:<p>Alvameline maleate is used as a Partial M1 Agonist and M2/M3 Antagonist.</p>Formula:C13H19N5O4Color and Shape:SolidMolecular weight:309.32Vinconate
CAS:<p>Vinconate is an indolonaphthyridine derivative and can stimulate the muscarinic acetylcholine receptor.</p>Formula:C18H20N2O2Purity:98%Color and Shape:SolidMolecular weight:296.36AT-1001
CAS:<p>AT-1001 is an α3β4 nAChR partial agonist reducing nicotine relapse and withdrawal with negligible impact on food response and dopamine release.</p>Formula:C15H21BrN2Color and Shape:SolidMolecular weight:309.24Rivanicline oxalate
CAS:<p>Rivanicline oxalate is an agonist of neuronal nicotinic receptor, showing high selectivity for the α4β2 subtype (Ki=26 nM).</p>Formula:C12H16N2O4Purity:98%Color and Shape:SolidMolecular weight:252.27Bradanicline HCl
CAS:<p>Bradanicline(TC-5619) is the agonist of Alpha-7 Nicotinic Receptor.</p>Formula:C22H24ClN3O2Color and Shape:SolidMolecular weight:397.9DREADD agonist 21 dihydrochloride
CAS:<p>DREADD agonist 21 dihydrochloride is a potent human muscarinic acetylcholine M3 receptors ( hM3Dq ) agonist with EC 50 of 1.7 nM [1].</p>Formula:C17H20Cl2N4Purity:98%Color and Shape:SolidMolecular weight:351.27BPIPP
CAS:<p>guanylyl cyclase (GC) and adenylyl cyclase (AC) inhibitor</p>Formula:C22H16BrN3O3Purity:98%Color and Shape:SolidMolecular weight:450.28
