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AChR

AChR

Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.

Found 575 products of "AChR"

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  • Procyclidine
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    Procyclidine

    CAS:
    <p>Procyclidine is an anticholinergic, muscarinic and NMDA antagonist used in Parkinson's and psychiatric disorder studies.</p>
    Formula:C19H29NO
    Color and Shape:Solid
    Molecular weight:287.44

    Ref: TM-T60578

  • Oxybutynin R-isomer HCl
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    Oxybutynin R-isomer HCl

    CAS:
    <p>Aroxybutynin, R-isomer of oxybutynin, is a muscarinic antagonist with antispasmodic effects on bladder muscle, weaker than atropine.</p>
    Formula:C22H32ClNO3
    Color and Shape:Solid
    Molecular weight:393.95

    Ref: TM-T71236

  • VU0455691
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    VU0455691

    CAS:
    <p>VU0455691 is a selective M1 Muscarinic Receptor Allosteric Modulators.</p>
    Formula:C24H25N5O3S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:463.55

    Ref: TM-T26328

  • Ambutonium bromide
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    Ambutonium bromide

    CAS:
    <p>Ambutonium bromide is an antagonist of acetylcholine.</p>
    Formula:C20H27BrN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:391.35

    Ref: TM-T14206

  • (±)-Muscarine chloride
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    (±)-Muscarine chloride

    CAS:
    <p>(±)-Muscarine chloride is the racemate of Muscarine chloride. Muscarine is a prototypical agonist for the muscarinic acetylcholine receptor [1] [2].</p>
    Formula:C9H20ClNO2
    Color and Shape:Solid
    Molecular weight:209.71

    Ref: TM-T60253

  • Methapyrilene
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    Methapyrilene

    CAS:
    <p>Methapyrilene is a histamine H1 antagonist with sedative action.</p>
    Formula:C14H19N3S
    Color and Shape:Liquid Physical Description Clear Colorless Liquid (Ntp 1992)
    Molecular weight:261.39

    Ref: TM-T28026

  • Milameline hydrochloride
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    Milameline hydrochloride

    CAS:
    <p>Milameline hydrochloride is a Muscarinic receptor agonist.</p>
    Formula:C8H15ClN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:190.67

    Ref: TM-T22979

  • Cycrimine
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    Cycrimine

    CAS:
    <p>Cycrimine: oral M1 mAChR blocker, lowers acetylcholine, antispasmodic, for Parkinson's and mental disorder studies.</p>
    Formula:C19H29NO
    Color and Shape:Solid
    Molecular weight:287.44

    Ref: TM-T60577

  • Parapenzolate bromide
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    Parapenzolate bromide

    CAS:
    <p>Parapenzolate bromide is an orally active mAChR antagonist. parapenzolate bromide is an anticholinergic and antitussive agent.</p>
    Formula:C21H26BrNO3
    Color and Shape:Solid
    Molecular weight:420.347

    Ref: TM-T62218

  • DPNB-ABT594
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    DPNB-ABT594

    <p>DPNB-ABT594, a nitrobenzyl-caged ABT594, selectively activates α4β2 over α7 nAChRs; used to study Ca²⁺ signaling in MHb.</p>
    Formula:C31H46ClN3O11
    Color and Shape:Solid
    Molecular weight:672.16

    Ref: TM-T72982

  • AFDX384
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    AFDX384

    CAS:
    <p>AFDX384 is potent M2/M4 selective antagonist.</p>
    Formula:C28H42N6O5S
    Color and Shape:Solid
    Molecular weight:574.74

    Ref: TM-T71311

  • (S)-VQW-765
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    (S)-VQW-765

    <p>(S)-VQW-765, oral α7 nAChR partial agonist, may improve cognition in Alzheimer's and schizophrenia.</p>
    Formula:C19H22N2O
    Color and Shape:Solid
    Molecular weight:294.39

    Ref: TM-T73055

  • Mazaticol
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    Mazaticol

    CAS:
    <p>Mazaticol: an anticholinergic, blocks muscarinic receptors, inhibits dopamine uptake, used in Parkinson's research.</p>
    Formula:C21H27NO3S2
    Color and Shape:Solid
    Molecular weight:405.57

    Ref: TM-T62008

  • J-104129 fumarate
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    J-104129 fumarate

    CAS:
    <p>J-104129 fumarate is a potent M3 muscarinic receptor antagonist.</p>
    Formula:C28H40N2O6
    Color and Shape:Solid
    Molecular weight:500.63

    Ref: TM-T69576

  • BMS-902483
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    BMS-902483

    CAS:
    <p>BMS-902483: potent α7 partial agonist; enhances rodent cognition; α7 EC50=9.3nM; 5-HT3A IC50=480nM.</p>
    Formula:C18H20N4O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:308.38

    Ref: TM-T26862

  • RLH 033
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    RLH 033

    CAS:
    <p>RLH 033 is a selective ligand for the sigma 1 recognition site.</p>
    Formula:C25H31ClN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:458.98

    Ref: TM-T26100

  • Talsaclidine
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    Talsaclidine

    CAS:
    <p>Talsaclidine: full M1 agonist, partial M2/M3 agonist with neuron-stimulating effects.</p>
    Formula:C10H15NO
    Purity:98%
    Color and Shape:Solid
    Molecular weight:165.23

    Ref: TM-T13071

  • A-85380 HCl
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    A-85380 HCl

    CAS:
    <p>A-85380 is an agonist of nicotinic acetylcholine receptor.</p>
    Formula:C9H14Cl2N2O
    Color and Shape:Solid
    Molecular weight:237.13

    Ref: TM-T26489

  • Phenglutarimid
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    Phenglutarimid

    CAS:
    <p>Phenglutarimid is an anticholinergic. It is used as an antiparkinsonian agent.</p>
    Formula:C17H24N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:288.38

    Ref: TM-T16521

  • Pirenzepine
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    Pirenzepine

    CAS:
    <p>Pirenzepine targets M1 mAChR, curbs acid secretion, eases spasms, and has anti-cancer properties.</p>
    Formula:C19H21N5O2
    Color and Shape:Solid
    Molecular weight:351.4

    Ref: TM-T61228