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AChR

AChR

Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.

Found 574 products of "AChR"

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  • ADX-10061
    Targetmol
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    ADX-10061

    CAS:
    <p>ADX-10061 is a dopamine D1 receptor antagonist.</p>
    Formula:C19H20N2O4
    Color and Shape:Solid
    Molecular weight:340.37

    Ref: TM-T26568

  • JN403
    Targetmol
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    JN403

    CAS:
    <p>JN403 is a selective agonist of nicotinic acetylcholine receptor alpha7.</p>
    Formula:C16H21FN2O2
    Color and Shape:Solid
    Molecular weight:292.35

    Ref: TM-T27657

  • Tebanicline tosylate
    Targetmol
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    Tebanicline tosylate

    CAS:
    <p>Tebanicline: synthetic, potent, non-opioid analgesic, less toxic than epibatidine; relieves neuropathic pain, acts on α3β4 and α4β2 nicotinic receptors.</p>
    Formula:C16H19ClN2O4S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:370.85

    Ref: TM-T3694L

  • Terodiline hydrochloride
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    Terodiline hydrochloride

    CAS:
    <p>Terodiline hydrochloride is an antagonist of M1-selective muscarinic receptor (mAChR)(Kbs of 15, 160, 280, and 198 nM in rabbit vas deferens (M1), atria (M2),</p>
    Formula:C20H28ClN
    Purity:98%
    Color and Shape:Solid
    Molecular weight:317.9

    Ref: TM-T13129

  • YM-46303
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    YM-46303

    CAS:
    <p>YM-46303 is a selective and potent muscarinic receptor antagonist that exhibits high affinity for the M3 receptor.YM-46303 can be used to study bradycardia in</p>
    Formula:C20H23ClN2O2
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:358.86

    Ref: TM-T13370

  • CHF5407
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    CHF5407

    CAS:
    <p>CHF5407（SVT-47060） is a potent and selective muscarinic M3 receptor antagonist with prolonged action at muscarinic receptors.CHF5407 has an effect on</p>
    Formula:C27H25BrF4N2O3S
    Purity:>99.99%
    Color and Shape:Solid
    Molecular weight:613.46

    Ref: TM-T13992

  • YM-58790
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    YM-58790

    CAS:
    <p>YM-58790 is a potent mAChR blocker with Ki values of 28 nM (M1), 260 nM (M2), 15 nM (M3), and reduces bladder contractions in rats.</p>
    Formula:C27H31N3O2
    Purity:98.59%
    Color and Shape:Soild
    Molecular weight:429.55

    Ref: TM-T72038

  • Metixene hydrochloride
    Targetmol
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    Metixene hydrochloride

    CAS:
    <p>Metixene hydrochloride is an anticholinergic antiparkinsonian agent.</p>
    Formula:C20H24ClNS
    Purity:98%
    Color and Shape:Solid
    Molecular weight:345.93

    Ref: TM-T12020

  • PQCA
    Targetmol
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    PQCA

    CAS:
    <p>PQCA is a selective M1 receptor modulator with EC50s of 49 nM (monkey) and 135 nM (human), potential for Alzheimer's treatment.</p>
    Formula:C22H20N4O3
    Purity:99.88%
    Color and Shape:Solid
    Molecular weight:388.42

    Ref: TM-T12531

  • Penehyclidine hydrochloride
    Targetmol
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    Penehyclidine hydrochloride

    CAS:
    <p>Penehyclidine hydrochloride: M1/M3 antagonist, activates NF-κB, anti-inflammatory, anticholinergic.</p>
    Formula:C20H30ClNO2
    Purity:99.79%
    Color and Shape:Solid
    Molecular weight:351.91

    Ref: TM-T61233

  • PD-102807
    Targetmol
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    PD-102807

    CAS:
    <p>PD-102807 is a selective and competitive M4 muscarinic receptor antagonist for Parkinson's disease research, inhibit airway smooth muscle (ASM) contraction.</p>
    Formula:C23H24N2O4
    Purity:98.90%
    Color and Shape:Solid
    Molecular weight:392.45

    Ref: TM-T23124

  • S 24795
    Targetmol
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    S 24795

    CAS:
    <p>S 24795 (Catestatin acetate(142211-96-9 free base)) is an α7 nAChR partial agonist.</p>
    Formula:C14H13BrINO
    Purity:99.934%
    Color and Shape:Solid
    Molecular weight:418.07

    Ref: TM-T23286

  • S16961
    Targetmol
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    S16961

    CAS:
    <p>S16961 (S169611) is an agonist of nicotinic receptor.</p>
    Formula:C41H71NO6
    Purity:99.69%
    Color and Shape:Solid
    Molecular weight:674.01

    Ref: TM-T12820

  • Afacifenacin
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    Afacifenacin

    CAS:
    <p>Afacifenacin (SMP-986) fumarate is an M3-selective antagonist for ischemic heart disease and urinary disorders.</p>
    Formula:C27H26F3N3O2
    Purity:99.83%
    Color and Shape:Solid
    Molecular weight:481.51

    Ref: TM-T29687

  • UP202-56
    Targetmol
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    UP202-56

    CAS:
    <p>UP202-56 is an adenosinergic agonist and is an adenosine analog.</p>
    Formula:C33H37N7O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:595.69

    Ref: TM-T13256

  • CB-7921220
    Targetmol
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    CB-7921220

    CAS:
    <p>CB-7921220 (6-[2-(4-Aminophenyl)vinyl]-2-pyridinecarboxylic acid) is an inhibitor of adenylate cyclase.</p>
    Formula:C14H12N2O2
    Purity:99.59%
    Color and Shape:Solid
    Molecular weight:240.26

    Ref: TM-T14880

  • Cimetropium Bromide
    Targetmol
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    Cimetropium Bromide

    CAS:
    <p>Cimetropium Bromide is a mAChR antagonist used for long-term treatment of irritable bowel syndrome.</p>
    Formula:C21H28BrNO4
    Color and Shape:Solid
    Molecular weight:438.36

    Ref: TM-T14966

  • GP531
    Targetmol
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    GP531

    CAS:
    <p>GP531, a second-gen adenosine regulator, is inactive at rest but boosts adenosine in ischemia.</p>
    Formula:C16H21N5O4
    Color and Shape:Solid
    Molecular weight:347.37

    Ref: TM-T13713

  • GAT107
    Targetmol
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    GAT107

    CAS:
    <p>GAT107, a strong α7 nicotinic receptor modulator, aids inflammation and neuropathic pain in mice.</p>
    Formula:C18H17BrN2O2S
    Purity:99.33%
    Color and Shape:Solid
    Molecular weight:405.31

    Ref: TM-T27404

  • SCH 57790
    Targetmol
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    SCH 57790

    CAS:
    <p>SCH 57790: selective muscarinic M2 blocker, boosts acetylcholine &amp; cognition, may treat Alzheimer's.</p>
    Formula:C25H31N3O2S
    Purity:99% - 99.12%
    Color and Shape:Solid
    Molecular weight:437.6

    Ref: TM-T28722