AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Found 643 products of "AChR"
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Solifenacin succinate
CAS:Solifenacin succinate (YM905) is a quinuclidine and tetrahydroisoquinoline derivative and selective M3 muscarinic antagonist, which is used as a urologic agent.Formula:C23H26N2O2·C4H6O4Purity:99.85% - 99.98%Color and Shape:SolidMolecular weight:480.56Diphenmanil methylsulfate
CAS:Diphenmanil methylsulfate (Diphemanil mesylate), a quaternary ammonium anticholinergic, binds muscarinic acetylcholine receptors.Formula:C20H24N·CH3O4SPurity:98% - 99.27%Color and Shape:SolidMolecular weight:389.51Pirenzepine dihydrochloride
CAS:Pirenzepine dihydrochloride (LS519) is a selective M1 muscarinic receptor antagonist, inhibiting gastric secretion.Formula:C19H21N5O2·2HClPurity:99.48% - 99.62%Color and Shape:White PowderMolecular weight:424.32Carbetapentane citrate
CAS:Carbetapentane citrate (Pentoxyverine citrate) , an antitussive (cough suppressant), is frequently used for a cough related to illnesses like the common cold.Formula:C20H31NO3·C6H8O7Purity:99.46%Color and Shape:White To Off-White SolidMolecular weight:525.59Primidone
CAS:Primidone (NCI-C56360) is a potent anticonvulsant agent.Formula:C12H14N2O2Purity:99.91%Color and Shape:Crystals (Ntp 1992)Molecular weight:218.25Droperidol
CAS:Droperidol (Dehydrobenzperidol) is a Dopamine-2 Receptor Antagonist. The mechanism of action of droperidol is as a Dopamine D2 Antagonist.Formula:C22H22FN3O2Purity:97.16% - 98%Color and Shape:SolidMolecular weight:379.43VU 0365114
CAS:VU 0365114 is a positive allosteric modulator of mAChR M5 and increases ACh-induced calcium mobilization(EC50: 2.7 μM).Formula:C22H14F3NO3Purity:99.86%Color and Shape:SolidMolecular weight:397.35Ref: TM-T13325
2mg35.00€5mg55.00€10mg78.00€25mg130.00€50mg212.00€100mg318.00€200mg444.00€1mL*10mM (DMSO)62.00€Dibucaine
CAS:Dibucaine (Cinchocaine), a local anesthetic of the amide type, is now usually used for surface anesthesia.Formula:C20H29N3O2Purity:99.698% - 99.88%Color and Shape:Colorless Or Almost Colorless Powder SolidMolecular weight:343.46Orphenadrine Citrate
CAS:Orphenadrine Citrate (Flexon) is a skeletal muscle relaxant, it acts in the central nervous system to produce its muscle relaxant effects.Formula:C18H23NO·C6H8O7Purity:99.58%Color and Shape:White SolidMolecular weight:461.5MK-7622
CAS:MK-7622 (M1 receptor modulator) is a modulator of muscarinic M1 receptor positive allosteric.Formula:C25H25N3O2Purity:99.77% - 99.8%Color and Shape:SolidMolecular weight:399.48Carbachol
CAS:Carbachol (Carbamoylcholine chloride), an analog of acetylcholine, serves as a valuable tool in the investigation of various physiological responses mediated by nicotinic (nAChR) and muscarinic (mAChR) acetylcholine receptors. These responses include smooth muscle contraction, gut motility, and neuronal signaling. Known for its agonistic properties, Carbachol activates both nAChR and mAChR, with reported Ki values ranging from 10 to 10,000 nM for different receptor types and experimental preparations.Formula:C6H15ClN2O2Purity:>99.99%Color and Shape:SolidMolecular weight:182.65MN58b
CAS:MN58b is a selective inhibitor of choline kinase α (CHKα).Formula:C32H40Br2N4Purity:97.23%Color and Shape:SolidMolecular weight:640.49Ref: TM-T12085
1mg279.00€5mg683.00€10mg888.00€25mg1,395.00€50mg1,783.00€100mg2,512.00€1mL*10mM (DMSO)862.00€Procainamide hydrochloride
CAS:Procainamide Hydrochloride (Procapan) is the hydrochloride salt form of procainamide, an amide derivative exhibiting class 1A antiarrhythmic property and analogFormula:C13H21N3O·HClPurity:99.83% - 99.97%Color and Shape:White To Slightly Yellow PowderMolecular weight:271.79Dequalinium chloride
CAS:Dequalinium chloride: topical bacteriostat, blocks apamin-sensitive K+ channels, used for wounds, oral infections, potential antifungal, risk of skin ulcers.
Formula:C30H40Cl2N4Purity:99.79% - 99.9%Color and Shape:SolidMolecular weight:527.59Benztropine mesylate
CAS:Benztropine mesylate (Benztropine methanesulfonate) is a centrally active muscarinic antagonist that has been used in the symptomatic treatment of PARKINSON
Formula:C21H25NO·CH4SO3Purity:98.41% - 99.96%Color and Shape:White Crystalline Powder; Odourless Or Almost OdourlessMolecular weight:403.53Lysipressin acetate(50-57-7(fb_acetate))
CAS:Lysipressin acetate (50-57-7), triggers rabbit bladder contraction & activates adenylate cyclase, is an antidiuretic in pigs & marsupials.
Formula:C48H69N13O14S2Purity:98.08%Color and Shape:SolidMolecular weight:1116.28(Rac)-ABT-202 dihydrochloride
CAS:(Rac)-ABT-202 dihydrochloride is a racemate of ABT-202. ABT-202 is an nicotinic acetylcholine receptors (nAChRs) agonist and can be used as an analgesic.Formula:C9H15Cl2N3Purity:97.4%Color and Shape:SolidMolecular weight:236.142Nebracetam hydrochloride
CAS:Nebracetam HCl (WEB 1881 FU) is an M1-muscarinic agonist nootropic, increasing intracellular Ca2+ with an EC50 of 1.59 mM.Formula:C12H17ClN2OPurity:99.23%Color and Shape:SolidMolecular weight:240.729Pyrantel tartrate
CAS:Pyrantel tartrate (Banminth) is broad spectrum anthelmintic for livestock.Formula:C15H20N2O6SPurity:99.96%Color and Shape:White CrystalsMolecular weight:356.39Flavoxate hydrochloride
CAS:Flavoxate hydrochloride (DW61) , a muscarinic AChR antagonist, is used in the therapy of various urinary syndromes and as an antispasmodic.Formula:C24H26ClNO4Purity:99.78%Color and Shape:White SolidMolecular weight:427.92
