AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Found 574 products of "AChR"
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Angiopeptin TFA
CAS:<p>Angiopeptin TFA: somatostatin analogue, sst2/sst5 partial agonist (IC50: 0.26/6.92 nM), suppresses GH & IGF-1, for atherosclerosis research.</p>Formula:C58H73F6N11O14S2Color and Shape:SolidMolecular weight:1326.39[Tyr22] Calcitonin Gene Related Peptide, (22-37), rat
CAS:<p>[Tyr22] CGRP (22-37), rat is a fragment of rat CGRP, targeting its receptor and adenylate cyclase, produced by thyroid and stored in the nervous system.</p>Formula:C82H120N20O25Color and Shape:SolidMolecular weight:1785.95Small Cardioactive Peptide B (SCPB)
CAS:<p>SCPB: neurally active peptide, boosts adenylate cyclase in heart/gills, EC50s: 0.1 μM (heart), 1.0 μM (gills).</p>Formula:C52H80N14O11S2Purity:98%Color and Shape:SolidMolecular weight:1141.41(-)-OPC-51803
CAS:<p>(-)-OPC-51803 is an antidiuretic hormone V2 receptor agonist used in the treatment of nocturia and urinary incontinence.</p>Formula:C26H32ClN3O2Purity:98.73% - 99.59%Color and Shape:SoildMolecular weight:454LtIA-F
<p>LtIA-F, a fluorescent LtIA derivative, aids study of α3β2 nAChR's structure, distribution, and binding domain.</p>Formula:C86H121N25O22S4Color and Shape:SolidMolecular weight:1985.31Aceclidine (hydrochloride)
CAS:<p>agonist of muscarinic receptors</p>Formula:C9H16ClNO2Purity:98%Color and Shape:SolidMolecular weight:205.68R-(+)-Cotinine
CAS:<p>R-(+)-Cotinine, an inactive nicotine metabolite, boosts Ach-induced current in human α7 nAChRs.</p>Formula:C10H12N2OColor and Shape:SolidMolecular weight:176.22nAChR modulator-2
CAS:<p>nAChR modulator-2, a insecticide, is a insect nAChR orthosteric modulator [1] .</p>Formula:C12H8ClN3O2Color and Shape:SolidMolecular weight:261.66nAChR modulator-1
CAS:<p>nAChR modulator-1, a insecticide, is a insect nAChR orthosteric modulator [1] .</p>Formula:C12H8ClN3O2Color and Shape:SolidMolecular weight:261.66Octamylamine
CAS:<p>Octamylamine is a bioactive chemical.</p>Formula:C13H29NColor and Shape:SolidMolecular weight:199.3761sabcomeline
CAS:<p>Sabcomeline: potent, selective M1 agonist; boosts cognition; for Alzheimer's study.</p>Formula:C10H15N3OColor and Shape:SolidMolecular weight:193.25Bencycloquidium Bromide
CAS:<p>Bencycloquidium bromide is an M3 muscarinic antagonist that reduces nasal secretion in allergic rhinitis and has high affinity for M3 receptors.</p>Formula:C21H32BrNO2Color and Shape:SolidMolecular weight:410.39nAChR agonist 2
CAS:<p>Compound 8, identified as a selective alpha4beta2 (α4β2) neuronal acetylcholine receptor (nAChR) agonist, demonstrates a dissociation constant (Kd) of 26 nM,</p>Formula:C11H16N2Color and Shape:SolidMolecular weight:176.263NNC 11-1607
CAS:<p>NNC 11-1607 is a functionally selective agonist of M(1)/M(4) mAChR.</p>Formula:C30H32N6O2S2Color and Shape:SolidMolecular weight:572.74(Rac)-5-Carboxy tolterodine
CAS:<p>(Rac)-5-Carboxy tolterodine is an inactive metabolite of Tolterodine, which acts as a muscarinic acetylcholine receptor antagonist.</p>Formula:C22H29NO3Color and Shape:SolidMolecular weight:355.47Perindoprilat
CAS:<p>Perindoprilat (Perindoprilate) is an angiotensin-converting enzyme inhibitor.</p>Formula:C17H28N2O5Purity:99.48%Color and Shape:SolidMolecular weight:340.41Methylatropine (nitrate)
CAS:<p>Methylatropine: Muscarinic antagonist, <0.1 nM IC50, atropine derivative, lowers ACh's effect on BP, affects salivation, pupil dilation, heart rate.</p>Formula:C18H26N2O6Color and Shape:SolidMolecular weight:366.414Navafenterol saccharinate
CAS:<p>AZD-8871 saccharinate is a dual-acting bronchodilator which may be useful in the treatment of Chronic Obstructive Pulmonary Disease (COPD).</p>Formula:C45H47N7O9S3Color and Shape:SolidMolecular weight:926.09M4 mAChR agonist-1
CAS:<p>M4 mAChR agonist-1 (4-Piperidinecarboxamide, 1-(5,6-dimethylthieno[2,3-d]pyrimidin-4-yl)-) is an effective agonist of M4 mAChR (EC50 >10 μM).</p>Formula:C14H18N4OSPurity:99.14%Color and Shape:SolidMolecular weight:290.38Epiboxidine
CAS:<p>Epiboxidine: Potent, selective nAChR agonist; Ki 0.46/1.2 nM for rat/human α4β2; analogous to Epibatidine and ABT 418.</p>Formula:C10H14N2OColor and Shape:SolidMolecular weight:178.23
![[Tyr22] Calcitonin Gene Related Peptide, (22-37), rat](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FT76363.webp&w=3840&q=75)
