AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Found 645 products of "AChR"
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Milameline hydrochloride
CAS:Milameline hydrochloride is a Muscarinic receptor agonist.Formula:C8H15ClN2OPurity:98%Color and Shape:SolidMolecular weight:190.67Cycrimine
CAS:Cycrimine: oral M1 mAChR blocker, lowers acetylcholine, antispasmodic, for Parkinson's and mental disorder studies.Formula:C19H29NOColor and Shape:SolidMolecular weight:287.44Parapenzolate bromide
CAS:Parapenzolate bromide is an orally active mAChR antagonist. parapenzolate bromide is an anticholinergic and antitussive agent.Formula:C21H26BrNO3Color and Shape:SolidMolecular weight:420.347Darenzepine
CAS:Darenzepine is a muscarinic receptor inhibitor.Formula:C21H21N3O2Purity:99.87%Color and Shape:SolidMolecular weight:347.41Ref: TM-T10961
1mg203.00€5mg404.00€10mg567.00€25mg842.00€50mg1,125.00€100mg1,521.00€1mL*10mM (DMSO)447.00€DPNB-ABT594
DPNB-ABT594, a nitrobenzyl-caged ABT594, selectively activates α4β2 over α7 nAChRs; used to study Ca²⁺ signaling in MHb.Formula:C31H46ClN3O11Color and Shape:SolidMolecular weight:672.16Tarafenacin
CAS:Tarafenacin is a highly selective M3 muscarinic receptor antagonist (Ki= 0.19 nM), ~200 fold selectivity over the M2 receptor.Formula:C21H20F4N2O2Purity:98%Color and Shape:SolidMolecular weight:408.39AFDX384
CAS:AFDX384 is potent M2/M4 selective antagonist.Formula:C28H42N6O5SColor and Shape:SolidMolecular weight:574.74VU 6008667
CAS:VU 6008667 is a selective negative allosteric M5 NAM modulator (IC50s: 1.2 μM and 1.6 μM for human M5 and rat M5, respectively).Formula:C24H17ClF2N2O2Purity:98%Color and Shape:SolidMolecular weight:438.85TC 1698 dihydrochloride
CAS:nicotinic α7 receptor agonistFormula:C13H18N2Purity:98%Color and Shape:SolidMolecular weight:202.3(S)-VQW-765
(S)-VQW-765, oral α7 nAChR partial agonist, may improve cognition in Alzheimer's and schizophrenia.Formula:C19H22N2OColor and Shape:SolidMolecular weight:294.39Mazaticol
CAS:Mazaticol: an anticholinergic, blocks muscarinic receptors, inhibits dopamine uptake, used in Parkinson's research.Formula:C21H27NO3S2Color and Shape:SolidMolecular weight:405.57J-104129 fumarate
CAS:J-104129 fumarate is a potent M3 muscarinic receptor antagonist.Formula:C28H40N2O6Color and Shape:SolidMolecular weight:500.63BMS-902483
CAS:BMS-902483: potent α7 partial agonist; enhances rodent cognition; α7 EC50=9.3nM; 5-HT3A IC50=480nM.Formula:C18H20N4OPurity:98%Color and Shape:SolidMolecular weight:308.38RLH 033
CAS:RLH 033 is a selective ligand for the sigma 1 recognition site.Formula:C25H31ClN2O4Purity:98%Color and Shape:SolidMolecular weight:458.98Talsaclidine
CAS:Talsaclidine: full M1 agonist, partial M2/M3 agonist with neuron-stimulating effects.Formula:C10H15NOPurity:98%Color and Shape:SolidMolecular weight:165.23A-85380 HCl
CAS:A-85380 is an agonist of nicotinic acetylcholine receptor.Formula:C9H14Cl2N2OColor and Shape:SolidMolecular weight:237.13AR-R 17779 hydrochloride
CAS:AR-R17779 hydrochloride: potent α7 nAChR agonist; K i : 92 nM (α7), 16,000 nM (α4β2); enhances rat cognition; anxiolytic; anti-inflammatory.Formula:C9H15ClN2O2Color and Shape:SolidMolecular weight:218.68Phenglutarimid
CAS:Phenglutarimid is an anticholinergic. It is used as an antiparkinsonian agent.Formula:C17H24N2O2Purity:98%Color and Shape:SolidMolecular weight:288.38Pirenzepine
CAS:Pirenzepine targets M1 mAChR, curbs acid secretion, eases spasms, and has anti-cancer properties.Formula:C19H21N5O2Color and Shape:SolidMolecular weight:351.4Elucaine
CAS:Elucaine is an antagonist of the muscarinic acetylcholine receptor. It has anti-ulcerative activity.Formula:C19H23NO2Purity:98%Color and Shape:SolidMolecular weight:297.39ENS-163 phosphate
CAS:Ens-163 phosphate is a muscarinic M1 receptor agonist. It is selective.Formula:C11H19N2O5PSPurity:98%Color and Shape:SolidMolecular weight:322.32TMPH hydrochloride
CAS:neuronal nicotinic ACh receptors (nAChRs) antagonistFormula:C16H32ClNO2Purity:98%Color and Shape:SolidMolecular weight:305.88Beperidium iodide
CAS:Beperidium iodide is a competitive antagonist of the acetylcholine receptor (pA2: 7.93).Formula:C23H34IN3O3Color and Shape:SolidMolecular weight:527.449-CP-Ade Mesylate
CAS:9-CP-Ade Mesylate (9 CP Ade Mesylate) is a cell-permeable, stable and non-competitive inhibitor of adenylate cyclase.Formula:C11H17N5O3SPurity:99.81%Color and Shape:SolidMolecular weight:299.35Arecaidine but-2-ynyl ester tosylate
CAS:mAChR M2 agonistFormula:C18H23NO5SPurity:98%Color and Shape:SolidMolecular weight:365.44GSK575594A
CAS:GSK575594A is a selective agonist of GPR55.Formula:C24H23F2N3O3SColor and Shape:SolidMolecular weight:471.52(R)-Oxybutynin
CAS:(R)-Oxybutynin: oral muscarinic blocker with antispasmodic effects, used in neurogenic bladder research.Formula:C22H31NO3Color and Shape:SolidMolecular weight:357.49AC-42
CAS:AC-42 is an allosteric agonist of M1 muscarinic receptor.
Formula:C20H31NOColor and Shape:SolidMolecular weight:301.47α7 nAchR-JAK2-STAT3 agonist 1
CAS:α7 nAchR-JAK2-STAT3 agonist 1 is a potent inhibitor of the α7 nAchR-JAK2-STAT3 pathway that acts on nitric oxide (NO) (IC50: 0.32 μM).Formula:C25H30O6Color and Shape:SolidMolecular weight:426.5Ethybenztropine
CAS:Ethybenztropine is an anticholinergic used as an antiparkinsonian agent and may also act as a dopamine reuptake inhibitor.Formula:C22H27NOPurity:98%Color and Shape:SolidMolecular weight:321.46Anabasine hydrochloride
CAS:neuronal nicotinic ACh receptor partial agonistFormula:C10H15ClN2Purity:98%Color and Shape:White To Off-White SolidMolecular weight:198.693Flupyrimin
CAS:Flupyrimin is the insect nicotinic acetylcholine receptor (nAChR) antagonist [1].Formula:C13H9ClF3N3OColor and Shape:SolidMolecular weight:315.68(R,R)-Glycopyrrolate
CAS:(R,R)-Glycopyrrolate is an agent of anticholinergic, has the ability to reduce the frequency of drooling in vivo with developmental disabilities.Formula:C19H28BrNO3Purity:98%Color and Shape:SolidMolecular weight:398.34Bibn 99
CAS:Bibn 99, a lipophilic and selective muscarinic M2 receptor antagonist, has applications in cognitive performance and Alzheimer's Disease.Formula:C31H42ClN5O3Color and Shape:SolidMolecular weight:568.15Adenylyl cyclase type 2 agonist-1
CAS:Potent AC2 agonist with an EC50 of 90 nM, potential for respiratory disease treatment.Formula:C27H17BrClNO5Color and Shape:SolidMolecular weight:550.78SCH 57790
CAS:SCH 57790: selective muscarinic M2 blocker, boosts acetylcholine & cognition, may treat Alzheimer's.Formula:C25H31N3O2SPurity:99.12% - 99.69%Color and Shape:SolidMolecular weight:437.6RJR-2403 oxalate
CAS:RJR-2403 oxalate is a highly selective agonist of α4β2 subtype nicotinic receptor.Formula:C14H18N2O4Purity:98%Color and Shape:SolidMolecular weight:278.308Bibn 140
CAS:Bibn 140 is a highly selective M2 antagonist, it is used to treat Alzheimer's disease and other cognitive disorders.Formula:C32H44N4O3Purity:98%Color and Shape:SolidMolecular weight:532.72GAT107
CAS:GAT107, a strong α7 nicotinic receptor modulator, aids inflammation and neuropathic pain in mice.Formula:C18H17BrN2O2SPurity:99.33%Color and Shape:SolidMolecular weight:405.31AZD 0328
CAS:AZD 0328 is a nicotinic receptor agonist for α7 neurons.Formula:C13H16N2OColor and Shape:SolidMolecular weight:216.28Nelonicline citrate
CAS:Nelonicline citrate (ABT-126) is a selective α7 nAChR agonist with a Ki of 12.3 nM, studied for schizophrenia and Alzheimer's.Formula:C23H27N3O8SColor and Shape:SolidMolecular weight:505.54TC-T 6000
CAS:TC-T 6000 (hENT4-IN-1) is an ENT4 inhibitor with vasodilator activity that inhibits hENT1 and hENT2 for the study of cancer and cardiovascular damage.Formula:C26H48N8O2Purity:98.14%Color and Shape:SolidMolecular weight:504.71SIB 1508Y maleate
CAS:neuronal nicotinic ACh receptor agonistFormula:C16H18N2O4Purity:98%Color and Shape:SolidMolecular weight:302.33N-0861 racemate
CAS:N-0861 racemate is the racemate of N-0861.Formula:C13H17N5Purity:98%Color and Shape:SolidMolecular weight:243.31Bradanicline
CAS:Bradanicline: potent α7 nAChR agonist, EC50=17 nM, Ki=1.4 nM, used in cognitive disorder research.Formula:C22H23N3O2Color and Shape:SolidMolecular weight:361.44DBO-83
CAS:DBO-83, an agonist of nicotinic acetylcholine receptors (nAChRs), has anti-amnesic and antinociceptive activities.Formula:C10H15Cl3N4Purity:98%Color and Shape:SolidMolecular weight:297.61ADX-10061
CAS:ADX-10061 is a dopamine D1 receptor antagonist.Formula:C19H20N2O4Color and Shape:SolidMolecular weight:340.37JN403
CAS:JN403 is a selective agonist of nicotinic acetylcholine receptor alpha7.Formula:C16H21FN2O2Color and Shape:SolidMolecular weight:292.35Telenzepine
CAS:Telenzepine is a potent and selective M1 antimuscarinic.Formula:C19H22N4O2SPurity:98%Color and Shape:SolidMolecular weight:370.47AC260584
CAS:AC260584 is an M1 muscarinic receptor allosteric agonist (pEC50: 7.6).Formula:C20H29FN2O2Color and Shape:SolidMolecular weight:348.45
