AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Found 574 products of "AChR"
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Darenzepine
CAS:<p>Darenzepine is a muscarinic receptor inhibitor.</p>Formula:C21H21N3O2Purity:99.87%Color and Shape:SolidMolecular weight:347.41UB 165 fumarate
CAS:<p>UB 165 fumarate is a nAChR agonist, α4β2 partial, α3β2 full, with a 0.27 nM Ki for [3H]-nicotine in rat brain.</p>Formula:C17H19ClN2O4Purity:99.72%Color and Shape:SolidMolecular weight:350.8CDD0102
CAS:<p>CDD0102 is a potent agonist of M1 Muscarinic receptor.</p>Formula:C8H12N4OPurity:98%Color and Shape:SolidMolecular weight:180.215-Iodo-A-85380 dihydrochloride
CAS:<p>α4β2 and α6β2 nicotinic acetylcholine receptors agonist</p>Formula:C9H13Cl2IN2OPurity:98%Color and Shape:SolidMolecular weight:363.02Dimethyl-W84 (dibromide)
CAS:<p>Dimethyl-W84, selective M2 muscarinic receptor modulator; slows N-methylscopolamine release, EC50=3 nM.</p>Formula:C34H48Br2N4O4Color and Shape:SolidMolecular weight:736.59LY 2087101
CAS:<p>Allosteric potentiator of α7, α4β2 and α4β4 nAChRs</p>Formula:C15H11FN2OS2Purity:98%Color and Shape:SolidMolecular weight:318.39AR-R 17779 hydrochloride
CAS:<p>AR-R17779 hydrochloride: potent α7 nAChR agonist; K i : 92 nM (α7), 16,000 nM (α4β2); enhances rat cognition; anxiolytic; anti-inflammatory.</p>Formula:C9H15ClN2O2Color and Shape:SolidMolecular weight:218.68Elucaine
CAS:<p>Elucaine is an antagonist of the muscarinic acetylcholine receptor. It has anti-ulcerative activity.</p>Formula:C19H23NO2Purity:98%Color and Shape:SolidMolecular weight:297.39(R,R)-Glycopyrrolate
CAS:<p>(R,R)-Glycopyrrolate is an agent of anticholinergic, has the ability to reduce the frequency of drooling in vivo with developmental disabilities.</p>Formula:C19H28BrNO3Purity:98%Color and Shape:SolidMolecular weight:398.34SIB 1508Y maleate
CAS:<p>neuronal nicotinic ACh receptor agonist</p>Formula:C16H18N2O4Purity:98%Color and Shape:SolidMolecular weight:302.33LRE1
CAS:<p>LRE1 is a specific and allosteric soluble adenylyl cyclase inhibitor.</p>Formula:C12H13ClN4SPurity:>99.99%Color and Shape:SolidMolecular weight:280.78Terodiline
CAS:<p>Terodiline is an orally available selective muscarinic M1 receptor and calcium channel antagonist for the study of diseases caused by abnormal bladder function.</p>Formula:C20H27NPurity:98.20% - 99.59%Color and Shape:SolidMolecular weight:281.44Methacholine bromide
CAS:<p>Methacholine bromide is a potent M3 agonist for diagnosing asthma by identifying bronchial hyperresponsiveness.</p>Formula:C8H18BrNO2Color and Shape:SolidMolecular weight:240.141Nuvenzepine
CAS:<p>Nuvenzepine is an antagonist of mAChR. It has the potential for gastrospasm treatment.</p>Formula:C19H20N4O2Purity:98%Color and Shape:SolidMolecular weight:336.39DA 4626
CAS:<p>DA 4626 is an H2-receptor antagonist with KB values akin to those in standard assays.</p>Formula:C14H18N4Purity:98%Color and Shape:SolidMolecular weight:242.32Telenzepine
CAS:<p>Telenzepine is a potent and selective M1 antimuscarinic.</p>Formula:C19H22N4O2SPurity:98%Color and Shape:SolidMolecular weight:370.47AC260584
CAS:<p>AC260584 is an M1 muscarinic receptor allosteric agonist (pEC50: 7.6).</p>Formula:C20H29FN2O2Color and Shape:SolidMolecular weight:348.45Neramexane Mesylate
CAS:<p>Neramexane: NMDA & nicotinic receptor blocker with neuroprotective, antidepressant, and cognitive-enhancing effects.</p>Formula:C12H27NO3SPurity:98%Color and Shape:SolidMolecular weight:265.41Chlorisondamine diiodide
CAS:<p>long lasting nicotinic antagonist</p>Formula:C14H20Cl4I2N2Color and Shape:SolidMolecular weight:611.94ML381
CAS:<p>ML381 is a M5-orthosteric antagonist with a high selectivity of muscarinic subtype.</p>Formula:C21H21N3O4Color and Shape:SolidMolecular weight:379.41ML169
CAS:<p>ML169 is a selective and brain penetrant M1 positive allosteric modulator (PAM).</p>Formula:C21H17BrFN3O4SPurity:98%Color and Shape:SolidMolecular weight:506.34Zamifenacin
CAS:<p>Zamifenacin obviously decreases colonic motility in irritable bowel syndrome. Zamifenacin is an effective gut-selective muscarinic M3 receptor antagonist.</p>Formula:C27H29NO3Purity:98%Color and Shape:SolidMolecular weight:415.52BNC375
CAS:<p>BNC375 is a α7 nAChRs type I positive allosteric modulator (EC50: 1.9 μM).</p>Formula:C19H23ClN2O3SPurity:98%Color and Shape:SolidMolecular weight:394.92(R,R)-Reboxetine mesylate
CAS:<p>(R,R)-Reboxetine mesylate: Antidepressant, high bioavailability, (R,R) enantiomer, selective for noradrenaline, low toxicity.</p>Formula:C20H27NO6SColor and Shape:SolidMolecular weight:409.5M1 ligand 1
CAS:<p>Compound 3b-b: N-desmethyl arecoline derivative, muscarinic M1 ligand, potential PET radiotracer.</p>Formula:C20H21NO2Color and Shape:SolidMolecular weight:307.39Benzatropine
CAS:<p>Benzatropine: Central muscarinic blocker, inhibits dopamine uptake, treats Parkinson's symptoms.</p>Formula:C21H25NOPurity:98%Color and Shape:SolidMolecular weight:307.43Muscarine iodide
CAS:<p>Muscarinic acetylcholine receptor agonist</p>Formula:C9H20INO2Purity:98%Color and Shape:SolidMolecular weight:301.17Tridihexethyl chloride
CAS:<p>Tridihexethyl is an anticholinergic, antimuscarinic, and antispasmolytic drug, which can be used to treat acquired nystagmus or peptic ulcer disease.</p>Formula:C21H36ClNOColor and Shape:SolidMolecular weight:353.97TC 2559 difumarate
CAS:<p>partial agonist of α4β2 nicotinic acetylcholine receptor</p>Formula:C12H18N2OC4H404Purity:98%Color and Shape:SolidMolecular weight:380.39TC299423
CAS:<p>TC299423 is a novel agonist for nicotinic acetylcholine receptors (nAChRs). TC299423 modestly selectively targets α6β2 subtype.</p>Formula:C11H15N3Color and Shape:SolidMolecular weight:189.26SM-21 maleate
CAS:<p>Increases release of acetylcholine,σ2 antagonist</p>Formula:C22H28ClNO7Purity:98%Color and Shape:SolidMolecular weight:453.91TC 1698 dihydrochloride
CAS:<p>nicotinic α7 receptor agonist</p>Formula:C13H18N2Purity:98%Color and Shape:SolidMolecular weight:202.3Beperidium iodide
CAS:<p>Beperidium iodide is a competitive antagonist of the acetylcholine receptor (pA2: 7.93).</p>Formula:C23H34IN3O3Color and Shape:SolidMolecular weight:527.44WIN 62,577
CAS:<p>WIN 62,577 is a allosteric antagonist of mAChR.</p>Formula:C29H31N3OPurity:98%Color and Shape:SolidMolecular weight:437.58Benzamide Derivative 1
CAS:<p>Benzamide Derivative 1 Benzamide derivative with gastrokinetic activity.Benzamide Derivative 1 can be used in the study of gastrointestinal diseases.</p>Formula:C22H34ClN3O3Purity:>99.99%Color and Shape:SolidMolecular weight:423.98Alvameline
CAS:<p>Alvameline (Lu25-109) is a partial M1 agonist. Alvameline (Lu25-109) also is a M2/M3 antagonist.</p>Formula:C9H15N5Purity:98%Color and Shape:SolidMolecular weight:193.25Muscarine chloride
CAS:<p>Muscarine chloride is a toxic alkaloid found in Amanita muscaria and other fungi of the Inocybe species.</p>Formula:C9H20ClNO2Color and Shape:SolidMolecular weight:209.71Quifenadine
CAS:<p>Quifenadine, an H1-histamine receptor blocker, has antiarrhythmic properties.</p>Formula:C20H23NOPurity:98%Color and Shape:SolidMolecular weight:293.4DAU 5884 hydrochloride
CAS:<p>muscarinic M3 receptor antagonist</p>Formula:C17H22ClN3O3Purity:98%Color and Shape:SolidMolecular weight:351.83Nelonicline
CAS:<p>Nelonicline is a selective agonist of neuronal nicotinic receptors.</p>Formula:C17H19N3OSPurity:98%Color and Shape:SolidMolecular weight:313.42BTM-1086
CAS:<p>BTM-1086 is a potent gastric secretory inhibitor and an anti-ulcer agent.</p>Formula:C21H25N3OSPurity:98%Color and Shape:SolidMolecular weight:367.51CP-601932
CAS:<p>CP-601932 (free base) is a selective base α( 4) β( 2) Nicotinic acetylcholine receptor agonist.</p>Formula:C12H12F3NColor and Shape:SolidMolecular weight:227.23Eucatropine
CAS:<p>Eucatropine, an anticholinergic agent, acts as a potent inhibitor of the muscarinic acetylcholine receptor (mAChR) with an IC 50 value of 0.583 μM.</p>Formula:C17H25NO3Color and Shape:SolidMolecular weight:291.39Thiochrome
CAS:<p>Thiochrome is a selective enhancer of M4 muscarinic receptor of acetylcholine (ACh) affinity.</p>Formula:C12H14N4OSPurity:98%Color and Shape:SolidMolecular weight:262.33VU0090157
CAS:<p>VU0090157, a novel allosteric potentiators of M1 muscarinic receptor, may provide novel treatments for schizophrenia and Alzheimer's disease.</p>Formula:C19H21N3O7Purity:98%Color and Shape:SolidMolecular weight:403.39S-(+)-Mecamylamine hydrochloride
CAS:<p>Dexmecamylamine( TC-5214, NIH-11008) is used as a nicotinic channel modulator with antidepressant activity.</p>Formula:C11H22ClNColor and Shape:SolidMolecular weight:203.75T761-0184
CAS:<p>T761-0184 is a potent antagonist of α7 nicotinic receptor (nAChR) [1].</p>Formula:C16H20FN3OColor and Shape:SolidMolecular weight:289.35Revatropate
CAS:<p>Revatropate, a selective muscarinic antagonist, is an antimuscarinic drug.</p>Formula:C19H27NO4SColor and Shape:SolidMolecular weight:365.49Rispenzepine
CAS:<p>Rispenzepine, a novel mAChRs M1/M3 antagonist, treats immune, infections, and respiratory issues.</p>Formula:C19H20N4O2Purity:98%Color and Shape:SolidMolecular weight:336.39Milameline
CAS:<p>Milameline is a muscarinic receptor agonist that improves cognition.</p>Formula:C8H14N2OColor and Shape:SolidMolecular weight:154.21
