AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Found 574 products of "AChR"
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Biricodar dicitrate
CAS:<p>Biricodar dicitrate (VX-710) is a potent MDR inhibitor with no anticancer activity and can be used to study prostate cancer.</p>Formula:C46H57N3O21Purity:97.78% - 99.78%Color and Shape:SolidMolecular weight:987.95Sofiniclin
CAS:<p>Sofiniclin (ABT 894) is an agonist of nicotinic acetylcholine receptor (nAChR). It is used for the research for attention-deficit/hyperactivity disorder (ADHD).</p>Formula:C10H11Cl2N3Purity:98%Color and Shape:SolidMolecular weight:244.12Bibn 99
CAS:<p>Bibn 99, a lipophilic and selective muscarinic M2 receptor antagonist, has applications in cognitive performance and Alzheimer's Disease.</p>Formula:C31H42ClN5O3Color and Shape:SolidMolecular weight:568.15VU 6008667
CAS:VU 6008667 is a selective negative allosteric M5 NAM modulator (IC50s: 1.2 μM and 1.6 μM for human M5 and rat M5, respectively).Formula:C24H17ClF2N2O2Purity:98%Color and Shape:SolidMolecular weight:438.85Rivanicline
CAS:<p>Rivanicline is a selective α4β2 nicotinic receptor agonist (Ki=26 nM), with >1,000x less affinity for α7 receptors.</p>Formula:C10H14N2Purity:98%Color and Shape:SolidMolecular weight:162.23Rapacuronium bromide
CAS:<p>Rapacuronium bromide is an allosteric muscarinic acetylcholine receptor (mAChR) modulator.</p>Formula:C37H61BrN2O4Purity:98%Color and Shape:SolidMolecular weight:677.8ML375
CAS:<p>ML375 is a potent, selective and CNS penetrant M5 negative allosteric modulator (NAM).</p>Formula:C23H15ClF2N2O2Color and Shape:SolidMolecular weight:424.83CP-601927
CAS:<p>CP-601927 is a nicotinic acetylcholine receptor (NACHR) agonist with permeability, high affinity, and selectivity.</p>Formula:C12H12F3NColor and Shape:SolidMolecular weight:227.23Arecaidine propargyl ester tosylate
CAS:<p>Arecaidine propargyl ester tosylate is a muscarinic receptor agonist.</p>Formula:C17H21NO5SPurity:98%Color and Shape:SolidMolecular weight:351.42VMY-2-95
CAS:<p>VMY-2-95 is an α4β2 nicotinic acetylcholine receptors (nAChRs) selective desensitizer.</p>Formula:C17H16N2OColor and Shape:SolidMolecular weight:264.32RJR 2429 dihydrochloride
CAS:<p>nAChR agonist that displays selectivity for α4β2</p>Formula:C12H18Cl2N2Purity:98%Color and Shape:SolidMolecular weight:261.19J 104129 fumarate
CAS:<p>M3 muscarinic receptor antagonist</p>Formula:C24H36N2O2Purity:98%Color and Shape:SolidMolecular weight:384.55Alvameline maleate
CAS:<p>Alvameline maleate is used as a Partial M1 Agonist and M2/M3 Antagonist.</p>Formula:C13H19N5O4Color and Shape:SolidMolecular weight:309.32Vinconate
CAS:<p>Vinconate is an indolonaphthyridine derivative and can stimulate the muscarinic acetylcholine receptor.</p>Formula:C18H20N2O2Purity:98%Color and Shape:SolidMolecular weight:296.36AT-1001
CAS:<p>AT-1001 is an α3β4 nAChR partial agonist reducing nicotine relapse and withdrawal with negligible impact on food response and dopamine release.</p>Formula:C15H21BrN2Color and Shape:SolidMolecular weight:309.24Rivanicline oxalate
CAS:<p>Rivanicline oxalate is an agonist of neuronal nicotinic receptor, showing high selectivity for the α4β2 subtype (Ki=26 nM).</p>Formula:C12H16N2O4Purity:98%Color and Shape:SolidMolecular weight:252.27Bradanicline HCl
CAS:<p>Bradanicline(TC-5619) is the agonist of Alpha-7 Nicotinic Receptor.</p>Formula:C22H24ClN3O2Color and Shape:SolidMolecular weight:397.9DREADD agonist 21 dihydrochloride
CAS:<p>DREADD agonist 21 dihydrochloride is a potent human muscarinic acetylcholine M3 receptors ( hM3Dq ) agonist with EC 50 of 1.7 nM [1].</p>Formula:C17H20Cl2N4Purity:98%Color and Shape:SolidMolecular weight:351.27BPIPP
CAS:<p>guanylyl cyclase (GC) and adenylyl cyclase (AC) inhibitor</p>Formula:C22H16BrN3O3Purity:98%Color and Shape:SolidMolecular weight:450.28Procyclidine
CAS:<p>Procyclidine is an anticholinergic, muscarinic and NMDA antagonist used in Parkinson's and psychiatric disorder studies.</p>Formula:C19H29NOColor and Shape:SolidMolecular weight:287.44Oxybutynin R-isomer HCl
CAS:<p>Aroxybutynin, R-isomer of oxybutynin, is a muscarinic antagonist with antispasmodic effects on bladder muscle, weaker than atropine.</p>Formula:C22H32ClNO3Color and Shape:SolidMolecular weight:393.95VU0455691
CAS:<p>VU0455691 is a selective M1 Muscarinic Receptor Allosteric Modulators.</p>Formula:C24H25N5O3SPurity:98%Color and Shape:SolidMolecular weight:463.55Ambutonium bromide
CAS:<p>Ambutonium bromide is an antagonist of acetylcholine.</p>Formula:C20H27BrN2OPurity:98%Color and Shape:SolidMolecular weight:391.35(±)-Muscarine chloride
CAS:<p>(±)-Muscarine chloride is the racemate of Muscarine chloride. Muscarine is a prototypical agonist for the muscarinic acetylcholine receptor [1] [2].</p>Formula:C9H20ClNO2Color and Shape:SolidMolecular weight:209.71Methapyrilene
CAS:<p>Methapyrilene is a histamine H1 antagonist with sedative action.</p>Formula:C14H19N3SColor and Shape:Liquid Physical Description Clear Colorless Liquid (Ntp 1992)Molecular weight:261.39Milameline hydrochloride
CAS:<p>Milameline hydrochloride is a Muscarinic receptor agonist.</p>Formula:C8H15ClN2OPurity:98%Color and Shape:SolidMolecular weight:190.67Cycrimine
CAS:<p>Cycrimine: oral M1 mAChR blocker, lowers acetylcholine, antispasmodic, for Parkinson's and mental disorder studies.</p>Formula:C19H29NOColor and Shape:SolidMolecular weight:287.44Parapenzolate bromide
CAS:<p>Parapenzolate bromide is an orally active mAChR antagonist. parapenzolate bromide is an anticholinergic and antitussive agent.</p>Formula:C21H26BrNO3Color and Shape:SolidMolecular weight:420.347DPNB-ABT594
<p>DPNB-ABT594, a nitrobenzyl-caged ABT594, selectively activates α4β2 over α7 nAChRs; used to study Ca²⁺ signaling in MHb.</p>Formula:C31H46ClN3O11Color and Shape:SolidMolecular weight:672.16AFDX384
CAS:<p>AFDX384 is potent M2/M4 selective antagonist.</p>Formula:C28H42N6O5SColor and Shape:SolidMolecular weight:574.74(S)-VQW-765
<p>(S)-VQW-765, oral α7 nAChR partial agonist, may improve cognition in Alzheimer's and schizophrenia.</p>Formula:C19H22N2OColor and Shape:SolidMolecular weight:294.39Mazaticol
CAS:<p>Mazaticol: an anticholinergic, blocks muscarinic receptors, inhibits dopamine uptake, used in Parkinson's research.</p>Formula:C21H27NO3S2Color and Shape:SolidMolecular weight:405.57J-104129 fumarate
CAS:<p>J-104129 fumarate is a potent M3 muscarinic receptor antagonist.</p>Formula:C28H40N2O6Color and Shape:SolidMolecular weight:500.63BMS-902483
CAS:<p>BMS-902483: potent α7 partial agonist; enhances rodent cognition; α7 EC50=9.3nM; 5-HT3A IC50=480nM.</p>Formula:C18H20N4OPurity:98%Color and Shape:SolidMolecular weight:308.38RLH 033
CAS:<p>RLH 033 is a selective ligand for the sigma 1 recognition site.</p>Formula:C25H31ClN2O4Purity:98%Color and Shape:SolidMolecular weight:458.98Talsaclidine
CAS:<p>Talsaclidine: full M1 agonist, partial M2/M3 agonist with neuron-stimulating effects.</p>Formula:C10H15NOPurity:98%Color and Shape:SolidMolecular weight:165.23A-85380 HCl
CAS:<p>A-85380 is an agonist of nicotinic acetylcholine receptor.</p>Formula:C9H14Cl2N2OColor and Shape:SolidMolecular weight:237.13Phenglutarimid
CAS:<p>Phenglutarimid is an anticholinergic. It is used as an antiparkinsonian agent.</p>Formula:C17H24N2O2Purity:98%Color and Shape:SolidMolecular weight:288.38Pirenzepine
CAS:<p>Pirenzepine targets M1 mAChR, curbs acid secretion, eases spasms, and has anti-cancer properties.</p>Formula:C19H21N5O2Color and Shape:SolidMolecular weight:351.4ENS-163 phosphate
CAS:<p>Ens-163 phosphate is a muscarinic M1 receptor agonist. It is selective.</p>Formula:C11H19N2O5PSPurity:98%Color and Shape:SolidMolecular weight:322.32TMPH hydrochloride
CAS:<p>neuronal nicotinic ACh receptors (nAChRs) antagonist</p>Formula:C16H32ClNO2Purity:98%Color and Shape:SolidMolecular weight:305.889-CP-Ade Mesylate
CAS:<p>9-CP-Ade Mesylate (9 CP Ade Mesylate) is a cell-permeable, stable and non-competitive inhibitor of adenylate cyclase.</p>Formula:C11H17N5O3SPurity:99.81%Color and Shape:SolidMolecular weight:299.35Arecaidine but-2-ynyl ester tosylate
CAS:<p>mAChR M2 agonist</p>Formula:C18H23NO5SPurity:98%Color and Shape:SolidMolecular weight:365.44GSK575594A
CAS:<p>GSK575594A is a selective agonist of GPR55.</p>Formula:C24H23F2N3O3SColor and Shape:SolidMolecular weight:471.52(R)-Oxybutynin
CAS:<p>(R)-Oxybutynin: oral muscarinic blocker with antispasmodic effects, used in neurogenic bladder research.</p>Formula:C22H31NO3Color and Shape:SolidMolecular weight:357.49AC-42
CAS:<p>AC-42 is an allosteric agonist of M1 muscarinic receptor.</p>Formula:C20H31NOColor and Shape:SolidMolecular weight:301.47α7 nAchR-JAK2-STAT3 agonist 1
CAS:<p>α7 nAchR-JAK2-STAT3 agonist 1 is a potent inhibitor of the α7 nAchR-JAK2-STAT3 pathway that acts on nitric oxide (NO) (IC50: 0.32 μM).</p>Formula:C25H30O6Color and Shape:SolidMolecular weight:426.5Ethybenztropine
CAS:<p>Ethybenztropine is an anticholinergic used as an antiparkinsonian agent and may also act as a dopamine reuptake inhibitor.</p>Formula:C22H27NOPurity:98%Color and Shape:SolidMolecular weight:321.46Anabasine hydrochloride
CAS:<p>neuronal nicotinic ACh receptor partial agonist</p>Formula:C10H15ClN2Purity:98%Color and Shape:White To Off-White SolidMolecular weight:198.693Flupyrimin
CAS:<p>Flupyrimin is the insect nicotinic acetylcholine receptor (nAChR) antagonist [1].</p>Formula:C13H9ClF3N3OColor and Shape:SolidMolecular weight:315.68
