AChR
Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.
Found 644 products of "AChR"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
Camylofine
CAS:Camylofine (Avacan) is an antimuscarinic, used for relaxing smooth muscle.Formula:C19H32N2O2·2HClPurity:98%Color and Shape:SolidMolecular weight:393.4(Rac)-VU 6008667
CAS:(Rac)-VU 6008667 is a selective M5 NAM with IC50 of 1.8 μM, high CNS penetration.Formula:C24H17ClF2N2O2Purity:99.82%Color and Shape:SolidMolecular weight:438.85DA 4626
CAS:DA 4626 is an H2-receptor antagonist with KB values akin to those in standard assays.Formula:C14H18N4Purity:98%Color and Shape:SolidMolecular weight:242.32Pentolinium Tartrate
CAS:Pentolinium Tartrate (Pendine) is a nicotinic antagonist that has been used as a ganglionic blocking agent in hypertension.Formula:C15H32N2·2C4H5O6Purity:98%Color and Shape:SolidMolecular weight:538.6AF-DX 384 free base
CAS:AF-DX 384 free base is an M2 mAChR and M4 mAChR antagonist, useful in research on neurodivisions and diseases such as Parkinson's.Formula:C27H38N6O2Purity:98%Color and Shape:SolidMolecular weight:478.63Pozanicline
CAS:Pozanicline, a selective α4β2 nAChR partial agonist (Ki=16 nM), may treat nicotine addiction by reversing cognitive deficits.Formula:C11H16N2OPurity:98%Color and Shape:SolidMolecular weight:192.26CB-6673567
CAS:CB-6673567 is a selective inhibitor of adenylyl cyclase.Formula:C19H14N4O3Color and Shape:SolidMolecular weight:346.34NGX-267
CAS:NGX-267, a muscarinic M1 agonist, is used potentially for the treatment of Xerostomia, Alzheimer's disease and cognitive.Formula:C10H18N2OSColor and Shape:SolidMolecular weight:214.33Dac 5945
CAS:DAC 5945 is a more effective muscarinic antagonist in the airways than in the heart.Formula:C19H30ClN3OPurity:98%Color and Shape:SolidMolecular weight:351.91Hexocyclium metilsulfate
CAS:Hexocyclium metilsulfate has anti-gastric secretory effects in humans.Formula:C21H36N2O5SPurity:98%Color and Shape:SolidMolecular weight:428.59GS 283
CAS:GS 283 is a Ca(2+) antagonist. GS 283 is also a weak histamine and muscarinic receptor blocker in rat and guinea pig tracheal smooth muscles.Formula:C17H17NO3Color and Shape:SolidMolecular weight:283.32(R)-VU 6008667
CAS:(R)-VU 6008667 is devoid of M5 NAM activity (IC50>10 μM).Formula:C24H17ClF2N2O2Color and Shape:SolidMolecular weight:438.85Anisodine hydrobromide
CAS:Anisodine hydrobromide is an inhibitor of adenosine kinase.Formula:C17H22BrNO5Color and Shape:White Crystals Or Crystalline PowderMolecular weight:400.27TC 2559 difumarate
CAS:partial agonist of α4β2 nicotinic acetylcholine receptorFormula:C12H18N2OC4H404Purity:98%Color and Shape:SolidMolecular weight:380.39TC299423
CAS:TC299423 is a novel agonist for nicotinic acetylcholine receptors (nAChRs). TC299423 modestly selectively targets α6β2 subtype.Formula:C11H15N3Color and Shape:SolidMolecular weight:189.26CDD0102
CAS:CDD0102 is a potent agonist of M1 Muscarinic receptor.Formula:C8H12N4OPurity:98%Color and Shape:SolidMolecular weight:180.215-Iodo-A-85380 dihydrochloride
CAS:α4β2 and α6β2 nicotinic acetylcholine receptors agonistFormula:C9H13Cl2IN2OPurity:98%Color and Shape:SolidMolecular weight:363.02Dimethyl-W84 (dibromide)
CAS:Dimethyl-W84, selective M2 muscarinic receptor modulator; slows N-methylscopolamine release, EC50=3 nM.Formula:C34H48Br2N4O4Color and Shape:SolidMolecular weight:736.59Sulfoxaflor
CAS:Sulfoxaflor (GF 2032) is an agonist of nAChR1 and nAChR2 subtypes and a systemic insecticide. Cost-effective and quality-assured.Formula:C10H10F3N3OSPurity:99.56% - 99.98%Color and Shape:SolidMolecular weight:277.27Ref: TM-T19940
1mg100.00€5mg275.00€10mg384.00€25mg572.00€50mg780.00€100mg1,018.00€250mg2,080.00€1mL*10mM (DMSO)245.00€LY 2087101
CAS:Allosteric potentiator of α7, α4β2 and α4β4 nAChRsFormula:C15H11FN2OS2Purity:98%Color and Shape:SolidMolecular weight:318.39GAT107
CAS:GAT107, a strong α7 nicotinic receptor modulator, aids inflammation and neuropathic pain in mice.Formula:C18H17BrN2O2SPurity:99.33%Color and Shape:SolidMolecular weight:405.31Rapacuronium bromide
CAS:Rapacuronium bromide is an allosteric muscarinic acetylcholine receptor (mAChR) modulator.Formula:C37H61BrN2O4Purity:98%Color and Shape:SolidMolecular weight:677.8ML375
CAS:ML375 is a potent, selective and CNS penetrant M5 negative allosteric modulator (NAM).Formula:C23H15ClF2N2O2Color and Shape:SolidMolecular weight:424.83Penehyclidine hydrochloride
CAS:Penehyclidine hydrochloride: M1/M3 antagonist, activates NF-κB, anti-inflammatory, anticholinergic.Formula:C20H30ClNO2Purity:99.79% - 99.91%Color and Shape:SolidMolecular weight:351.91CP-601927
CAS:CP-601927 is a nicotinic acetylcholine receptor (NACHR) agonist with permeability, high affinity, and selectivity.Formula:C12H12F3NColor and Shape:SolidMolecular weight:227.23CP-601932
CAS:CP-601932 (free base) is a selective base α( 4) β( 2) Nicotinic acetylcholine receptor agonist.Formula:C12H12F3NColor and Shape:SolidMolecular weight:227.23Arecaidine propargyl ester tosylate
CAS:Arecaidine propargyl ester tosylate is a muscarinic receptor agonist.Formula:C17H21NO5SPurity:98%Color and Shape:SolidMolecular weight:351.42VMY-2-95
CAS:VMY-2-95 is an α4β2 nicotinic acetylcholine receptors (nAChRs) selective desensitizer.Formula:C17H16N2OColor and Shape:SolidMolecular weight:264.32RJR 2429 dihydrochloride
CAS:nAChR agonist that displays selectivity for α4β2Formula:C12H18Cl2N2Purity:98%Color and Shape:SolidMolecular weight:261.19SR 16584
CAS:α3β4 nAChR antagonistFormula:C17H22N2OPurity:99.84%Color and Shape:SolidMolecular weight:270.37J 104129 fumarate
CAS:M3 muscarinic receptor antagonistFormula:C24H36N2O2Purity:98%Color and Shape:SolidMolecular weight:384.55Alvameline maleate
CAS:Alvameline maleate is used as a Partial M1 Agonist and M2/M3 Antagonist.Formula:C13H19N5O4Color and Shape:SolidMolecular weight:309.32Vinconate
CAS:Vinconate is an indolonaphthyridine derivative and can stimulate the muscarinic acetylcholine receptor.Formula:C18H20N2O2Purity:98%Color and Shape:SolidMolecular weight:296.36AT-1001
CAS:AT-1001 is an α3β4 nAChR partial agonist reducing nicotine relapse and withdrawal with negligible impact on food response and dopamine release.Formula:C15H21BrN2Color and Shape:SolidMolecular weight:309.24SM-21 maleate
CAS:Increases release of acetylcholine,σ2 antagonistFormula:C22H28ClNO7Purity:98%Color and Shape:SolidMolecular weight:453.91Rivanicline oxalate
CAS:Rivanicline oxalate is an agonist of neuronal nicotinic receptor, showing high selectivity for the α4β2 subtype (Ki=26 nM).Formula:C12H16N2O4Purity:98%Color and Shape:SolidMolecular weight:252.27Bradanicline HCl
CAS:Bradanicline(TC-5619) is the agonist of Alpha-7 Nicotinic Receptor.Formula:C22H24ClN3O2Color and Shape:SolidMolecular weight:397.9DREADD agonist 21 dihydrochloride
CAS:DREADD agonist 21 dihydrochloride is a potent human muscarinic acetylcholine M3 receptors ( hM3Dq ) agonist with EC 50 of 1.7 nM [1].Formula:C17H20Cl2N4Purity:98%Color and Shape:SolidMolecular weight:351.27BPIPP
CAS:guanylyl cyclase (GC) and adenylyl cyclase (AC) inhibitorFormula:C22H16BrN3O3Purity:98%Color and Shape:SolidMolecular weight:450.28Procyclidine
CAS:Procyclidine is an anticholinergic, muscarinic and NMDA antagonist used in Parkinson's and psychiatric disorder studies.Formula:C19H29NOColor and Shape:SolidMolecular weight:287.44Oxybutynin R-isomer HCl
CAS:Aroxybutynin, R-isomer of oxybutynin, is a muscarinic antagonist with antispasmodic effects on bladder muscle, weaker than atropine.Formula:C22H32ClNO3Color and Shape:SolidMolecular weight:393.95VU0455691
CAS:VU0455691 is a selective M1 Muscarinic Receptor Allosteric Modulators.Formula:C24H25N5O3SPurity:98%Color and Shape:SolidMolecular weight:463.55Sch412348
CAS:Sch412348: potent A2A receptor antagonist, Ki=0.6 nM, >1000-fold selectivity vs. other adenosine receptors.Formula:C22H21F2N9OPurity:98%Color and Shape:SolidMolecular weight:465.46Eucatropine
CAS:Eucatropine, an anticholinergic agent, acts as a potent inhibitor of the muscarinic acetylcholine receptor (mAChR) with an IC 50 value of 0.583 μM.Formula:C17H25NO3Color and Shape:SolidMolecular weight:291.39Rivanicline
CAS:Rivanicline is a selective α4β2 nicotinic receptor agonist (Ki=26 nM), with >1,000x less affinity for α7 receptors.Formula:C10H14N2Purity:98%Color and Shape:SolidMolecular weight:162.23Bradanicline
CAS:Bradanicline: potent α7 nAChR agonist, EC50=17 nM, Ki=1.4 nM, used in cognitive disorder research.Formula:C22H23N3O2Color and Shape:SolidMolecular weight:361.44Ambutonium bromide
CAS:Ambutonium bromide is an antagonist of acetylcholine.Formula:C20H27BrN2OPurity:98%Color and Shape:SolidMolecular weight:391.35PD-102807
CAS:PD-102807 is a selective and competitive M4 muscarinic receptor antagonist for Parkinson's disease research, inhibit airway smooth muscle (ASM) contraction.Formula:C23H24N2O4Purity:98.90%Color and Shape:SolidMolecular weight:392.45(±)-Muscarine chloride
CAS:(±)-Muscarine chloride is the racemate of Muscarine chloride. Muscarine is a prototypical agonist for the muscarinic acetylcholine receptor [1] [2].Formula:C9H20ClNO2Color and Shape:SolidMolecular weight:209.71S 24795
CAS:S 24795 (Catestatin acetate(142211-96-9 free base)) is an α7 nAChR partial agonist.Formula:C14H13BrINOPurity:99.934%Color and Shape:SolidMolecular weight:418.07Ref: TM-T23286
5mg44.00€10mg66.00€25mg138.00€50mg215.00€100mg338.00€200mg480.00€1mL*10mM (DMSO)48.00€
