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AChR

AChR

Acetylcholine Receptor (AChR) inhibitors are compounds that block the activity of acetylcholine receptors, which are critical for neurotransmission in the central and peripheral nervous systems. AChRs play a vital role in muscle contraction, memory, and cognitive functions. Inhibitors of AChRs are used to study conditions such as myasthenia gravis, Alzheimer's disease, and other neurological disorders. By modulating AChR activity, these inhibitors can help unravel the complexities of cholinergic signaling in the brain. At CymitQuimica, we provide a range of AChR inhibitors to support your research in neuroscience, pharmacology, and neurodegenerative disease.

Found 575 products of "AChR"

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  • Milameline
    Targetmol
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    Milameline

    CAS:
    <p>Milameline is a muscarinic receptor agonist that improves cognition.</p>
    Formula:C8H14N2O
    Color and Shape:Solid
    Molecular weight:154.21

    Ref: TM-T70772

  • Biricodar dicitrate
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    Biricodar dicitrate

    CAS:
    <p>Biricodar dicitrate (VX-710) is a potent MDR inhibitor with no anticancer activity and can be used to study prostate cancer.</p>
    Formula:C46H57N3O21
    Purity:97.78% - 99.78%
    Color and Shape:Solid
    Molecular weight:987.95

    Ref: TM-T67790

  • Sofiniclin
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    Sofiniclin

    CAS:
    <p>Sofiniclin (ABT 894) is an agonist of nicotinic acetylcholine receptor (nAChR). It is used for the research for attention-deficit/hyperactivity disorder (ADHD).</p>
    Formula:C10H11Cl2N3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:244.12

    Ref: TM-T10226

  • PD-102807
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    PD-102807

    CAS:
    <p>PD-102807 is a selective and competitive M4 muscarinic receptor antagonist for Parkinson's disease research, inhibit airway smooth muscle (ASM) contraction.</p>
    Formula:C23H24N2O4
    Purity:98.90%
    Color and Shape:Solid
    Molecular weight:392.45

    Ref: TM-T23124

  • S 24795
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    S 24795

    CAS:
    <p>S 24795 (Catestatin acetate(142211-96-9 free base)) is an α7 nAChR partial agonist.</p>
    Formula:C14H13BrINO
    Purity:99.934%
    Color and Shape:Solid
    Molecular weight:418.07

    Ref: TM-T23286

  • Bibn 99
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    Bibn 99

    CAS:
    <p>Bibn 99, a lipophilic and selective muscarinic M2 receptor antagonist, has applications in cognitive performance and Alzheimer's Disease.</p>
    Formula:C31H42ClN5O3
    Color and Shape:Solid
    Molecular weight:568.15

    Ref: TM-T26799

  • VU 6008667
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    VU 6008667

    CAS:
    VU 6008667 is a selective negative allosteric M5 NAM modulator (IC50s: 1.2 μM and 1.6 μM for human M5 and rat M5, respectively).
    Formula:C24H17ClF2N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:438.85

    Ref: TM-T13315

  • Rivanicline
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    Rivanicline

    CAS:
    <p>Rivanicline is a selective α4β2 nicotinic receptor agonist (Ki=26 nM), with &gt;1,000x less affinity for α7 receptors.</p>
    Formula:C10H14N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:162.23

    Ref: TM-T12738L

  • Rapacuronium bromide
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    Rapacuronium bromide

    CAS:
    Rapacuronium bromide is an allosteric muscarinic acetylcholine receptor (mAChR) modulator.
    Formula:C37H61BrN2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:677.8

    Ref: TM-T12690

  • ML375
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    ML375

    CAS:
    <p>ML375 is a potent, selective and CNS penetrant M5 negative allosteric modulator (NAM).</p>
    Formula:C23H15ClF2N2O2
    Color and Shape:Solid
    Molecular weight:424.83

    Ref: TM-T28068

  • CP-601927
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    CP-601927

    CAS:
    <p>CP-601927 is a nicotinic acetylcholine receptor (NACHR) agonist with permeability, high affinity, and selectivity.</p>
    Formula:C12H12F3N
    Color and Shape:Solid
    Molecular weight:227.23

    Ref: TM-T31066

  • Arecaidine propargyl ester tosylate
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    Arecaidine propargyl ester tosylate

    CAS:
    <p>Arecaidine propargyl ester tosylate is a muscarinic receptor agonist.</p>
    Formula:C17H21NO5S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:351.42

    Ref: TM-T22585

  • VMY-2-95
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    VMY-2-95

    CAS:
    <p>VMY-2-95 is an α4β2 nicotinic acetylcholine receptors (nAChRs) selective desensitizer.</p>
    Formula:C17H16N2O
    Color and Shape:Solid
    Molecular weight:264.32

    Ref: TM-T35068

  • RJR 2429 dihydrochloride
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    RJR 2429 dihydrochloride

    CAS:
    <p>nAChR agonist that displays selectivity for α4β2</p>
    Formula:C12H18Cl2N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:261.19

    Ref: TM-T23236

  • J 104129 fumarate
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    J 104129 fumarate

    CAS:
    <p>M3 muscarinic receptor antagonist</p>
    Formula:C24H36N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:384.55

    Ref: TM-T22876

  • Alvameline maleate
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    Alvameline maleate

    CAS:
    <p>Alvameline maleate is used as a Partial M1 Agonist and M2/M3 Antagonist.</p>
    Formula:C13H19N5O4
    Color and Shape:Solid
    Molecular weight:309.32

    Ref: TM-T14197L

  • Vinconate
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    Vinconate

    CAS:
    <p>Vinconate is an indolonaphthyridine derivative and can stimulate the muscarinic acetylcholine receptor.</p>
    Formula:C18H20N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:296.36

    Ref: TM-T13959

  • AT-1001
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    AT-1001

    CAS:
    <p>AT-1001 is an α3β4 nAChR partial agonist reducing nicotine relapse and withdrawal with negligible impact on food response and dopamine release.</p>
    Formula:C15H21BrN2
    Color and Shape:Solid
    Molecular weight:309.24

    Ref: TM-T70987

  • Rivanicline oxalate
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    Rivanicline oxalate

    CAS:
    <p>Rivanicline oxalate is an agonist of neuronal nicotinic receptor, showing high selectivity for the α4β2 subtype (Ki=26 nM).</p>
    Formula:C12H16N2O4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:252.27

    Ref: TM-T12739

  • Bradanicline HCl
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    Bradanicline HCl

    CAS:
    <p>Bradanicline(TC-5619) is the agonist of Alpha-7 Nicotinic Receptor.</p>
    Formula:C22H24ClN3O2
    Color and Shape:Solid
    Molecular weight:397.9

    Ref: TM-T30574