NMDAR
N-Methyl-D-Aspartate Receptor (NMDAR) inhibitors are compounds that block the activity of NMDARs, a subtype of glutamate receptors that play a critical role in synaptic plasticity, learning, and memory. Overactivation of NMDARs is implicated in excitotoxicity, which can lead to neuronal damage and is associated with conditions such as stroke, traumatic brain injury, and neurodegenerative diseases. NMDAR inhibitors are essential tools for studying excitotoxicity and for developing neuroprotective therapies. At CymitQuimica, we offer a range of NMDAR inhibitors to support your research in synaptic function, neuroprotection, and cognitive disorders.
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1-Aminocyclobutanecarboxylic acid
CAS:22264-50-2
1-Aminocyclobutanecarboxylic acid (ACBC) is a NMDA receptor partial agonist. 1-Aminocyclobutanecarboxylic acid act at the glycine …
Formula:
C5H9NO2
Purity:
99.94%
Color and Shape:
White To Tan Powder Crystals Crystalline Powder And/Or With Chunks
Molecular weight:
115.13
Ref: TM-T22542
| 10mg | 48.00 € | ||
| 25mg | 89.00 € | ||
| 50mg | 119.00 € | ||
| 100mg | 168.00 € | ||
| 200mg | 254.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Traxoprodil
CAS:134234-12-1
Traxoprodil (CP101606) is a selective NMDA antagonist and protects hippocampal neurons (IC50: 10 nM).
Formula:
C20H25NO3
Purity:
99.89%
Color and Shape:
Solid
Molecular weight:
327.42
Ref: TM-TQ0233
| 5mg | 51.00 € | ||
| 10mg | 70.00 € | ||
| 25mg | To inquire | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 57.00 € |
Estimated delivery in United States, on Friday 16 May 2025
DNQX disodium salt
CAS:1312992-24-7
DNQX disodium salt is a water-soluble form of selective antagonist of non-NMDA receptor
Formula:
C8H2N4Na2O6
Purity:
98.93%
Color and Shape:
Solid
Molecular weight:
296.1
Ref: TM-T8459
| 1mg | 88.00 € | ||
| 5mg | 170.00 € | ||
| 10mg | 259.00 € | ||
| 25mg | 425.00 € | ||
| 50mg | 598.00 € | ||
| 100mg | 810.00 € | ||
| 200mg | 1,074.00 € | ||
| 1mL*10mM (DMSO) | 170.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Dizocilpine Maleate
CAS:77086-22-7
Dizocilpine Maleate (MK 801) is a potent noncompetitive antagonist of the NMDA receptor with Kd …
Formula:
C20H19NO4
Purity:
99% - 99.96%
Color and Shape:
White Solid
Molecular weight:
337.38
Ref: TM-T3320
| 5mg | 38.00 € | ||
| 10mg | 55.00 € | ||
| 25mg | 89.00 € | ||
| 50mg | 145.00 € | ||
| 100mg | 255.00 € | ||
| 200mg | 420.00 € | ||
| 1mL*10mM (DMSO) | 55.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Flupirtine maleate
CAS:75507-68-5
Flupirtine maleate (Katadolon maleate), a centrally acting non-opioid analgesia, is the salt form of Flupirtine. …
Formula:
C15H17FN4O2·C4H4O4
Purity:
99.50% - 99.9%
Color and Shape:
Off-White Crystalline Powder
Molecular weight:
420.39
Ref: TM-T6504
| 10mg | 49.00 € | ||
| 50mg | 62.00 € | ||
| 100mg | 85.00 € | ||
| 200mg | 120.00 € | ||
| 500mg | 281.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Friday 16 May 2025
5,7-Dichlorokynurenic acid
CAS:131123-76-7
5,7-Dichlorokynurenic acid (5,7-dichlorokynurenic acid sodium) is an NMDA receptor antagonist.
Formula:
C10H5Cl2NO3
Purity:
99.56%
Color and Shape:
Solid
Molecular weight:
258.06
Ref: TM-T22517
| 5mg | 47.00 € | ||
| 10mg | 74.00 € | ||
| 25mg | 145.00 € | ||
| 50mg | 246.00 € | ||
| 100mg | 368.00 € | ||
| 500mg | 852.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Co 101244 hydrochloride
CAS:193356-17-1
Co 101244 hydrochloride (4-Piperidinol, 1-[2-(4-hydroxyphenoxy)ethyl]-4-[(4-Methylphenyl)Methyl]-,hydrochloride) is an NR2B-containing NMDA receptor antagonist.
Formula:
C21H28ClNO3
Purity:
98.44%
Color and Shape:
Solid
Molecular weight:
377.9
Ref: TM-T22674
| 2mg | 42.00 € | ||
| 5mg | 64.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 183.00 € | ||
| 50mg | 283.00 € |
Estimated delivery in United States, on Friday 16 May 2025
DQP 1105
CAS:380560-89-4
DQP 1105 is a NMDA receptor antagonist.
Formula:
C29H24BrN3O4
Purity:
98.77%
Color and Shape:
Solid
Molecular weight:
558.42
Ref: TM-T22748
| 2mg | 34.00 € | ||
| 5mg | 52.00 € | ||
| 10mg | 96.00 € | ||
| 25mg | 178.00 € | ||
| 50mg | 253.00 € |
Estimated delivery in United States, on Friday 16 May 2025
BZAD01
CAS:305339-41-7
BZAD01 is a selective NMDA NR1A/2B receptor antagonist.
Formula:
C16H12F6N2O
Purity:
99.51% - 99.78%
Color and Shape:
Solid
Molecular weight:
362.27
Ref: TM-T25196
| 5mg | 50.00 € | ||
| 10mg | 84.00 € | ||
| 25mg | 150.00 € | ||
| 50mg | 226.00 € | ||
| 100mg | 375.00 € | ||
| 200mg | 523.00 € | ||
| 1mL*10mM (DMSO) | 71.00 € |
Estimated delivery in United States, on Friday 16 May 2025
TCN 213
CAS:556803-08-8
TCN 213 is an antagonist of NMDA receptor that has a selective for NR1/NR2A over …
Formula:
C18H24N4OS2
Purity:
99.68%
Color and Shape:
Solid
Molecular weight:
376.54
Ref: TM-T8450
| 5mg | 43.00 € | ||
| 10mg | 65.00 € | ||
| 25mg | 117.00 € | ||
| 50mg | 187.00 € | ||
| 100mg | 306.00 € | ||
| 200mg | 442.00 € | ||
| 1mL*10mM (DMSO) | 35.00 € |
Estimated delivery in United States, on Friday 16 May 2025
ZL006
CAS:1181226-02-7
ZL006 is an effective inhibitor of nNOS/PSD-95 interaction. ZL006 also inhibits NMDA receptor-mediated NO synthesis.
Formula:
C14H11Cl2NO4
Purity:
98.29%
Color and Shape:
Solid
Molecular weight:
328.15
Ref: TM-T17293
| 5mg | 50.00 € | ||
| 10mg | 66.00 € | ||
| 25mg | 117.00 € | ||
| 50mg | 180.00 € | ||
| 100mg | 306.00 € | ||
| 200mg | 444.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Friday 16 May 2025
L-701324
CAS:142326-59-8
L-701324 is an NMDA receptor with high affinity and selectivity for the glycine site, used …
Formula:
C21H14ClNO3
Purity:
100% - 98.63%
Color and Shape:
Solid
Molecular weight:
363.79
Ref: TM-T1909
| 5mg | 40.00 € | ||
| 10mg | 62.00 € | ||
| 25mg | 97.00 € | ||
| 50mg | 163.00 € | ||
| 100mg | 235.00 € | ||
| 200mg | 341.00 € | ||
| 1mL*10mM (DMSO) | 44.00 € |
Estimated delivery in United States, on Friday 16 May 2025
TCN 201
CAS:852918-02-6
TCN 201 is a selective antagonist of NMDA receptors containing the NR2A subunit.
Formula:
C21H17ClFN3O4S
Purity:
98.50%
Color and Shape:
Solid
Molecular weight:
461.89
Ref: TM-T7870
| 5mg | 65.00 € | ||
| 10mg | 97.00 € | ||
| 25mg | 172.00 € | ||
| 50mg | 303.00 € | ||
| 100mg | 563.00 € |
Estimated delivery in United States, on Friday 16 May 2025
DL-AP5
CAS:76326-31-3
DL-AP5 is the racemic form of a selective N-methyl-D-aspartate (NMDA) receptor antagonist with anticonvulsant effects.
Formula:
C5H12NO5P
Purity:
99.33%
Color and Shape:
White Fine Crystalline Powder
Molecular weight:
197.13
Ref: TM-T22733
| 1mg | 35.00 € | ||
| 5mg | 74.00 € | ||
| 10mg | 111.00 € | ||
| 25mg | 216.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 522.00 € |
Estimated delivery in United States, on Friday 16 May 2025
UBP551
CAS:89-35-0
UBP551 is a potent and selective NMDA receptors modulator.
Formula:
C11H8O4
Purity:
98.69%
Color and Shape:
Solid
Molecular weight:
204.18
Ref: TM-T8351
| 5mg | 55.00 € | ||
| 10mg | 82.00 € | ||
| 25mg | 126.00 € | ||
| 50mg | 182.00 € | ||
| 100mg | 273.00 € | ||
| 200mg | 409.00 € | ||
| 500mg | 677.00 € | ||
| 1mL*10mM (DMSO) | 64.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Eliprodil
CAS:119431-25-3
Eliprodil (SL-820715), NR2B-NMDA receptor blocker (IC50: 1 uM), less potent on NR2A/NR2C (IC50>100 uM), …
Formula:
C20H23ClFNO
Purity:
97.56% - 99.77%
Color and Shape:
Solid
Molecular weight:
347.85
Ref: TM-T1751
| 5mg | 34.00 € | ||
| 10mg | 60.00 € | ||
| 25mg | 104.00 € | ||
| 50mg | 188.00 € | ||
| 100mg | 283.00 € | ||
| 200mg | 408.00 € | ||
| 1mL*10mM (DMSO) | 34.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Radiprodil
CAS:496054-87-6
Radiprodil (RGH-896) is an oral NMDA NR2B antagonist for potential DPNP neuropathic pain treatment.
Formula:
C21H20FN3O4
Purity:
99.74%
Color and Shape:
Solid
Molecular weight:
397.4
Ref: TM-T5385
| 1mg | 48.00 € | ||
| 2mg | 65.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 153.00 € | ||
| 25mg | 240.00 € | ||
| 50mg | 354.00 € | ||
| 100mg | 532.00 € | ||
| 1mL*10mM (DMSO) | 96.00 € |
Estimated delivery in United States, on Friday 16 May 2025
UBP710
CAS:1333111-40-2
UBP710 is an effective and selective NMDA receptor modulator.
Formula:
C18H14O2
Purity:
98.39%
Color and Shape:
Solid
Molecular weight:
262.3
Ref: TM-T24918
| 1mg | 87.00 € | ||
| 2mg | 124.00 € | ||
| 5mg | 187.00 € | ||
| 10mg | 284.00 € | ||
| 25mg | 452.00 € | ||
| 50mg | 645.00 € | ||
| 100mg | 867.00 € | ||
| 200mg | 1,159.00 € | ||
| 1mL*10mM (DMSO) | 177.00 € |
Estimated delivery in United States, on Friday 16 May 2025
Rapastinel Trifluoroacetate
CAS:1435786-04-1
Rapastinel Trifluoroacetate (GLYX-13 Trifluoroacetate) is an NMDA receptor modulator with glycine-site partial agonist properties.
Formula:
C20H32F3N5O8
Purity:
99.01% - 99.77%
Color and Shape:
Solid
Molecular weight:
527.49
Ref: TM-T5819
| 1mg | 39.00 € | ||
| 5mg | 101.00 € | ||
| 10mg | 170.00 € | ||
| 25mg | 305.00 € | ||
| 50mg | 419.00 € | ||
| 100mg | 562.00 € | ||
| 200mg | 743.00 € | ||
| 1mL*10mM (DMSO) | 116.00 € |
Estimated delivery in United States, on Friday 16 May 2025
(RS)-(Tetrazol-5-yl)glycine
CAS:138199-51-6
(RS)-(Tetrazol-5-yl)glycine (LY 285265) is a selective NMDA receptor agonist with EC50 of 99 nM (GluN1/GluN2D) …
Formula:
C3H5N5O2
Purity:
95.00%
Color and Shape:
Solid
Molecular weight:
143.1
Ref: TM-T16801
| 5mg | 43.00 € | ||
| 10mg | 64.00 € | ||
| 25mg | 140.00 € | ||
| 50mg | 235.00 € | ||
| 100mg | 335.00 € | ||
| 200mg | 470.00 € |
Estimated delivery in United States, on Friday 16 May 2025
