NMDAR
N-Methyl-D-Aspartate Receptor (NMDAR) inhibitors are compounds that block the activity of NMDARs, a subtype of glutamate receptors that play a critical role in synaptic plasticity, learning, and memory. Overactivation of NMDARs is implicated in excitotoxicity, which can lead to neuronal damage and is associated with conditions such as stroke, traumatic brain injury, and neurodegenerative diseases. NMDAR inhibitors are essential tools for studying excitotoxicity and for developing neuroprotective therapies. At CymitQuimica, we offer a range of NMDAR inhibitors to support your research in synaptic function, neuroprotection, and cognitive disorders.
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Flutriafol
CAS:76674-21-0
Flutriafol is a pesticide, demethylation inhibitor, and NMDA receptor agonist
Formula:
C16H13F2N3O
Purity:
98.75%
Color and Shape:
Solid
Molecular weight:
301.29
Ref: TM-T7867
| 1g | 262.00 € | ||
| 25mg | 46.00 € | ||
| 50mg | 59.00 € | ||
| 100mg | 82.00 € | ||
| 200mg | 95.00 € | ||
| 500mg | 174.00 € | ||
| 1mL*10mM (DMSO) | 47.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
PEAQX
CAS:459836-30-7
PEAQX (NVP-AAM077) is an oral NMDA antagonist, inhibits 1A/2A receptors (IC50: 270 nM), less so …
Formula:
C17H17BrN3O5P
Purity:
100% - ≥98%
Color and Shape:
Solid
Molecular weight:
454.21
Ref: TM-T4171
| 1mg | 33.00 € | ||
| 2mg | 44.00 € | ||
| 5mg | 72.00 € | ||
| 10mg | 120.00 € | ||
| 25mg | 208.00 € | ||
| 50mg | 323.00 € | ||
| 100mg | 451.00 € | ||
| 200mg | 651.00 € | ||
| 1mL*10mM (DMSO) | 93.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
1-Aminocyclobutanecarboxylic acid
CAS:22264-50-2
1-Aminocyclobutanecarboxylic acid (ACBC) is a NMDA receptor partial agonist. 1-Aminocyclobutanecarboxylic acid act at the glycine …
Formula:
C5H9NO2
Purity:
99.94%
Color and Shape:
White To Tan Powder Crystals Crystalline Powder And/Or With Chunks
Molecular weight:
115.13
Ref: TM-T22542
| 10mg | 48.00 € | ||
| 25mg | 89.00 € | ||
| 50mg | 119.00 € | ||
| 100mg | 172.00 € | ||
| 200mg | 251.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
Ro 8-4304
CAS:195988-65-9
Ro 8-4304 Hydrochloride is an antagonist of NMDA receptor with IC50 of 0.4 μM
Formula:
C21H23FN2O3
Purity:
98%
Color and Shape:
Solid
Molecular weight:
370.42
Ref: TM-T8447
| 25mg | 633.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
GNE-8324
CAS:1698901-76-6
GNE-8324 is a GluN2A selective positive allosteric modulator that enhances NMDAR-mediated synaptic responses in inhibitory, …
Formula:
C18H18FN3OS
Purity:
98.68% - 99.34%
Color and Shape:
Solid
Molecular weight:
343.42
Ref: TM-T31981
| 25mg | 1,437.00 € | ||
| 50mg | 1,872.00 € | ||
| 100mg | 2,364.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
MDL-29951
CAS:130798-51-5
MDL-29951 is a novel glycine antagonist of NMDA receptor activation.
Formula:
C12H9Cl2NO4
Purity:
99.07% - 99.49%
Color and Shape:
Solid
Molecular weight:
302.11
Ref: TM-T1897
| 1mg | 50.00 € | ||
| 5mg | 101.00 € | ||
| 10mg | 174.00 € | ||
| 25mg | 315.00 € | ||
| 50mg | 452.00 € | ||
| 100mg | 621.00 € | ||
| 200mg | 837.00 € | ||
| 1mL*10mM (DMSO) | 105.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Gacyclidine
CAS:68134-81-6
Gacyclidine (OTO311), an NMDA receptor blocker, treats tinnitus and injuries in the brain and spinal …
Formula:
C16H25NS
Purity:
100% - 99%
Color and Shape:
Solid
Molecular weight:
263.44
Ref: TM-T27397
| 1mg | 92.00 € | ||
| 5mg | 196.00 € | ||
| 10mg | 288.00 € | ||
| 25mg | 544.00 € | ||
| 50mg | 728.00 € | ||
| 100mg | 1,012.00 € | ||
| 500mg | 2,023.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
N20C hydrochloride
CAS:1177583-87-7
N20C hydrochloride (2-((3,3-diphenylpropyl)amino)acetamide hydrochloride) is a non-competitive NMDA receptor open-channel blocker.
Formula:
C17H21ClN2O
Purity:
98.58%
Color and Shape:
Solid
Molecular weight:
304.81
Ref: TM-T23048
| 1mg | 51.00 € | ||
| 2mg | 81.00 € | ||
| 5mg | 107.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 273.00 € | ||
| 50mg | 397.00 € | ||
| 100mg | 542.00 € | ||
| 200mg | 717.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Aptiganel
CAS:137159-92-3
Aptiganel (CNS-1102) is a non-competitive NMDA antagonist, a peptide that may be used to study …
Formula:
C20H21N3
Purity:
98.19% - 98.90%
Color and Shape:
Solid
Molecular weight:
303.4
Ref: TM-T26645
| 1mg | 277.00 € | ||
| 5mg | 681.00 € | ||
| 10mg | 931.00 € | ||
| 25mg | 1,434.00 € | ||
| 50mg | 1,867.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
CGP 37849
CAS:127910-31-0
CGP 37849: oral NMDA antagonist (Ki=35 nM), anticonvulsant, with antidepressant/anxiolytic effects.
Formula:
C6H12NO5P
Purity:
99.87%
Color and Shape:
White Solid
Molecular weight:
209.14
Ref: TM-T7720
| 1mg | 124.00 € | ||
| 5mg | 276.00 € | ||
| 10mg | 423.00 € | ||
| 25mg | 680.00 € | ||
| 50mg | 916.00 € | ||
| 100mg | 1,262.00 € | ||
| 1mL*10mM (DMSO) | 275.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
RPR104632
CAS:154106-92-0
RPR104632 is a novel and potent antagonist located at the NMDA glycine site with neuroprotective …
Formula:
C15H11BrCl2N2O4S
Purity:
99.06%
Color and Shape:
Solid
Molecular weight:
466.13
Ref: TM-T16797
| 1mg | 654.00 € | ||
| 5mg | 1,672.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
GV-196771A
CAS:166974-23-8
GV-196771A A novel NMDA receptor glycine site antagonist with potent antinociceptive activity.
Formula:
C20H13Cl2N2NaO3
Purity:
96.43%
Color and Shape:
Solid
Molecular weight:
423.23
Ref: TM-T11516
| 1mg | 654.00 € | ||
| 5mg | 1,671.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Ro 25-6981
CAS:169274-78-6
Ro 25-6981: potent, selective NMDA receptor blocker (NR2B), IC50: 0.009 μM (NR1C/NR2B), 52 μM (NR1C/NR2A), …
Formula:
C22H29NO2
Purity:
99.44%
Color and Shape:
Solid
Molecular weight:
339.47
Ref: TM-T12758
| 1mg | 52.00 € | ||
| 2mg | 73.00 € | ||
| 5mg | 88.00 € | ||
| 10mg | 125.00 € | ||
| 25mg | 258.00 € | ||
| 50mg | 406.00 € | ||
| 100mg | 600.00 € | ||
| 1mL*10mM (DMSO) | 95.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
L-Cysteine S-sulfate
CAS:1637-71-4
L-Cysteine S-sulfate (S-Sulfo-L-cysteine) is an effective N-methyl-d-aspartate (NMDA) glutamatergic receptors agonist.
Formula:
C3H7NO5S2
Purity:
98.92%
Color and Shape:
Solid
Molecular weight:
201.22
Ref: TM-T60237
| 50mg | 54.00 € | ||
| 500mg | 66.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
UK-240455
CAS:178908-09-3
UK-240455: Potent NMDA glycine antagonist with neuroprotection and motor function benefits in Parkinson's.
Formula:
C11H11Cl2N3O5S
Purity:
98.34% - 99.83%
Color and Shape:
Solid
Molecular weight:
368.19
Ref: TM-T13248
| 1mg | 327.00 € | ||
| 5mg | 769.00 € | ||
| 10mg | 1,056.00 € | ||
| 25mg | 1,476.00 € | ||
| 50mg | 1,838.00 € | ||
| 100mg | 2,320.00 € | ||
| 500mg | 4,549.00 € | ||
| 1mL*10mM (DMSO) | 676.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
L-701252
CAS:151057-13-5
L-701252, a potent glycine site NMDA receptor antagonist, exhibits an inhibition concentration (IC50) of 420 …
Formula:
C13H10ClNO3
Purity:
98.53%
Color and Shape:
White Crystalline Solid
Molecular weight:
263.68
Ref: TM-T22900
| 1mg | 38.00 € | ||
| 5mg | 73.00 € | ||
| 10mg | 87.00 € | ||
| 25mg | 139.00 € | ||
| 50mg | 185.00 € | ||
| 100mg | 278.00 € | ||
| 500mg | 679.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Dizocilpine
CAS:77086-21-6
MK-801 (Dizocilpine (MK-801)) is a potent N-methyl-D-aspartate (NMDA) receptor antagonist with Ki of 30.5 nM.
Formula:
C16H15N
Purity:
99.75% - 99.97%
Color and Shape:
Solid
Molecular weight:
221.3
Ref: TM-T6259
| 1mg | 35.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 94.00 € | ||
| 25mg | 148.00 € | ||
| 50mg | 234.00 € | ||
| 100mg | 376.00 € | ||
| 500mg | 895.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
CNS-5161 hydrochloride
CAS:160756-38-7
CNS-5161 hydrochloride (CNS 5161A) is a new antagonist of NMDA ion-channel.
Formula:
C16H19Cl2N3S2
Purity:
99.53%
Color and Shape:
Solid
Molecular weight:
388.38
Ref: TM-T10852
| 1mg | 471.00 € | ||
| 5mg | 924.00 € | ||
| 10mg | 1,256.00 € | ||
| 25mg | 1,866.00 € | ||
| 50mg | 2,503.00 € | ||
| 1mL*10mM (DMSO) | 1,063.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
AV-101
CAS:153152-32-0
AV-101 (4-Cl-KYN) is a prodrug antagonist at the glycine site of the NMDA receptor with …
Formula:
C10H11ClN2O3
Purity:
97.84% - 98%
Color and Shape:
Solid
Molecular weight:
242.66
Ref: TM-T26686
| 1mg | 180.00 € | ||
| 5mg | 449.00 € | ||
| 10mg | 643.00 € | ||
| 25mg | 1,011.00 € | ||
| 50mg | 1,386.00 € | ||
| 100mg | 1,835.00 € | ||
| 500mg | 3,669.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
Gavestinel sodium
CAS:153436-38-5
Gavestinel (GV 150526): potent, selective oral NMDA antagonist; binds glycine site, pKi 8.5; studied for …
Formula:
C18H11Cl2N2NaO3
Purity:
99.04%
Color and Shape:
Solid
Molecular weight:
397.19
Ref: TM-T22798
| 1mg | 45.00 € | ||
| 5mg | 96.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 231.00 € | ||
| 50mg | 343.00 € | ||
| 100mg | 507.00 € |
Estimated delivery in United States, on Wednesday 22 Jan 2025
