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Serine Protease

Serine Protease

Serine protease inhibitors are compounds that target and inhibit serine proteases, a group of enzymes characterized by a serine residue at their active site. These proteases are involved in numerous physiological processes, including digestion, immune response, blood coagulation, and inflammation. Serine protease inhibitors are important for studying diseases where these enzymes are dysregulated, such as cardiovascular diseases, cancer, and inflammatory conditions. At CymitQuimica, we provide serine protease inhibitors to support your research in enzymology, disease mechanisms, and therapeutic interventions.

Found 82 products for "Serine Protease".

products per page.
  • Chlorobenzothiazolinone

    CAS:
    Chlorobenzothiazolinone blocks human chymase at 90 μM, assessed by fluorescence using a specific peptide substrate after 1 hr.
    Formula:C7H4ClNOS
    Purity:99.42% - 99.77%
    Color and Shape:Solid
    Molecular weight:185.63

    Ref: TM-T0577

    1mL*10mM (DMSO)
    33.00€
    1g
    37.00€
  • BAY-85-8501

    CAS:
    BAY-85-8501 is a selective, reversible and potent inhibitor of Human Neutrophil Elastase (HNE; IC50 of 65 pM)
    Formula:C22H17F3N4O3S
    Purity:99.16%
    Color and Shape:Solid
    Molecular weight:474.46

    Ref: TM-T12613L

    1mg
    92.00€
    2mg
    122.00€
    5mg
    200.00€
    1mL*10mM (DMSO)
    208.00€
    10mg
    298.00€
    25mg
    535.00€
    50mg
    750.00€
    100mg
    1,035.00€
  • TAO Kinase inhibitor 2

    CAS:
    TAO Kinase inhibitor 2 is a TAO kinase inhibitor with an IC50 of 50-500 nM. TAO Kinase inhibitor 2 inhibits KIAA1361 and JIK with IC50s of 50-500 nM.
    Formula:C25H24N2O3
    Purity:98.58%
    Color and Shape:Solid
    Molecular weight:400.47

    Ref: TM-T77501

    1mg
    34.00€
    5mg
    71.00€
    10mg
    105.00€
    25mg
    170.00€
    50mg
    255.00€
    100mg
    378.00€
    500mg
    858.00€
  • α-Methyl-DL-aspartic acid

    CAS:
    α-Methyl-DL-aspartic acid specifically inhibits argininosuccinate synthase (ASS), the rate-limiting enzyme in 1-citrulline-to-1-arginine recycling.
    Formula:C5H9NO4
    Purity:99.91%
    Color and Shape:Solid
    Molecular weight:147.129

    Ref: TM-T78044

    5mg
    33.00€
    10mg
    46.00€
    25mg
    84.00€
    50mg
    120.00€
    100mg
    178.00€
  • Tiprelestat

    CAS:
    Tiprelestat: strong inhibitor of human neutrophil elastase, anti-inflammatory, antimicrobial, used in inflammation/immune research.
    Formula:C254H416N72O75S10
    Color and Shape:Solid
    Molecular weight:5999.09

    Ref: TM-T73657

    5mg
    To inquire
    50mg
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  • SFTI-1

    CAS:
    SFTI-1, a cyclic peptide trypsin inhibitor comprising 14 amino acid residues, is a potent Bowman-Birk inhibitor.
    Formula:C67H104N18O18S2
    Color and Shape:Solid
    Molecular weight:1513.78

    Ref: TM-TP2622

    10mg
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    50mg
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  • Roseltide rT1

    CAS:
    Roseltide rT1 is a neutrophil elastase inhibitor (IC50=0.47 μM) and is rich in cysteine, classified as one of the Roseltides (rT1-rT8). It has the potential to inhibit related diseases by improving neutrophil elastase-stimulated cAMP accumulation in vitro.
    Formula:C110H177N31O31S6
    Color and Shape:Solid
    Molecular weight:2622.16

    Ref: TM-TP3226

    10mg
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    50mg
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  • Lonodelestat TFA


    Lonodelestat TFA, an oral peptide, selectively inhibits hNE, potentially aiding in CF research.
    Formula:C73H112F3N15O21
    Color and Shape:Solid
    Molecular weight:1592.75

    Ref: TM-T76216

    5mg
    To inquire
    50mg
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  • α 1 Antichymotrypsin, Human Plasma

    CAS:
    Alpha 1 Antichymotrypsin, Human Plasma is an inhibitor of serine proteases. This compound is present in amyloid lesions associated with Alzheimer's disease and can be utilized in Alzheimer's research.
    Color and Shape:Solid

    Ref: TM-TP3129

    10mg
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    50mg
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  • Kallikrein 5-IN-2 TFA


    Kallikrein5-IN-2 TFA is the trifluoroacetate salt form of Kallikrein5-IN-2. It acts as a selective inhibitor of kallikrein5 (KLK5), with a pIC50 value of 7.1. Kallikrein5-IN-2 TFA exhibits no phototoxicity at 100 μg/mL and is non-irritating. The compound remains stable in non-oxidative conditions within a pH range of 4 to 8. Kallikrein5-IN-2 shows potential for improving Netherton syndrome.
    Formula:C25H23F3N6O3
    Color and Shape:Solid
    Molecular weight:512.17837

    Ref: TM-T209910

    10mg
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    50mg
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  • hCAXII-IN-10


    hCAXII-IN-10 (Compound 18b) acts as a dual inhibitor of human carbonic anhydrase isoenzyme XII (hCAXII) and cathepsin B, with a Ki value of 2.2 nM. It inhibits the function of hCAXII in creating a pH microenvironment conducive to tumor growth, showing promise for use in cancer research.
    Color and Shape:Odour Solid

    Ref: TM-T89066

    10mg
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    50mg
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  • Chymotrypsinogen

    CAS:
    Chymotrypsinogen is an inactive precursor of Chymotrypsin . Chymotrypsin is a serine protease produced by the pancreas [1] [2] .
    Color and Shape:Solid

    Ref: TM-T76157

    5mg
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    50mg
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  • Z-APF-CMK

    CAS:
    Z-APF-CMK is a selective inhibitor of the calcium (Ca2+)-regulated nuclear scaffold protease (CRNSP), as reported in reference [1].
    Formula:C26H30ClN3O5
    Color and Shape:Solid
    Molecular weight:499.99

    Ref: TM-T80743

    5mg
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    50mg
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  • Suc-AAP-Abu-pNA

    CAS:
    Suc-AAP-Abu-pNA is a specific substrate for pancreatic elastase (Km = 100 μM; Kcat/Km = 35,300 s-1 M-1 for rat pancreatic elastase; Km = 30 μM; Kcat/Km = 351,
    Formula:C25H34N6O9
    Color and Shape:Solid
    Molecular weight:562.57

    Ref: TM-T36351

    1mg
    132.00€
  • Protease Inhibitor Library


    A unique collection of xnum protease and proteasome inhibitors for research in chemical genomics, and drug screening;
    Color and Shape:Odour Solid

    Ref: TM-L1100

    1mg
    To inquire
    10μL*10mM (DMSO)
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    20μL*10mM (DMSO)
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    30μL*10mM (DMSO)
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    50μL*10mM (DMSO)
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    100μL*10mM (DMSO)
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    250μL*10mM (DMSO)
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  • MeOSuc-AAPA-CMK


    MeOSuc-AAPA-CMK is a potent inhibitor of human neutrophil elastase (HNE) [1].
    Formula:C20H31ClN4O8
    Color and Shape:Solid
    Molecular weight:490.94

    Ref: TM-T80553

    5mg
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    50mg
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  • Safflower oil (from Carthamus tinctorius seed)

    CAS:
    Safflower oil (from Carthamus tinctorius seed) contains unsaturated fatty acids, tocopherols and phenolic compounds, which has antioxidant and lipid metabolism regulating activities, can scavenge free radicals and inhibit collagenase and elastase activities, and is often used in skin aging, atherosclerosis and functional oil-related research.

    Ref: TM-T217594

    25g
    33.00€
  • KKI-5

    CAS:
    KKI 5: Serine protease inhibitor, blocks kallikrein & plasmin, potential for cancer therapy & angioedema treatment.
    Formula:C35H55N11O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:773.88

    Ref: TM-TP1792

    1mg
    60.00€
    5mg
    163.00€
    10mg
    284.00€
  • CDD-3290


    CDD-3290 serves as a functional therapeutic tool specifically designed to enable the precise detection and inhibition of the proteolytic activity of PSA which plays a pivotal role in the progression of prostate cancer during strictly monitored laboratory observation periods and molecular investigations to evaluate the pharmacological potential of targeted kallikrein inhibition in specialized preclinical research environments.
    Formula:C17H14N6O2
    Purity:99.06% - 99.13%
    Color and Shape:White Solid
    Molecular weight:334.33

    Ref: TM-T89314

    5mg
    To inquire
    25mg
    To inquire
    100mg
    To inquire
    1mL*10mM (DMSO)
    To inquire
    1mg
    172.00€
    10mg
    565.00€
    50mg
    1,288.00€
  • Tilpisertib fosmecarbil TFA

    CAS:
    Tilpisertib fosmecarbil TFA, the TFA salt form of Tilpisertib, acts as an inhibitor of serine/threonine kinases. This compound also exhibits anti-inflammatory activity.
    Formula:C37H37ClF3N8O9P
    Color and Shape:Solid
    Molecular weight:861.16

    Ref: TM-T88817

    10mg
    To inquire
    50mg
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