HER
HER inhibitors are compounds that block the activity of Human Epidermal Growth Factor Receptors, particularly HER2, which is overexpressed in certain breast cancers and other malignancies. Inhibition of HER signaling pathways is a key strategy in targeted cancer therapies. At CymitQuimica, we offer HER inhibitors to support your research in oncology, targeted therapies, and cell signaling.
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Varlitinib
CAS:845272-21-1
Varlitinib (ASLAN001) is a potent, reversible, small molecule pan-EGFR inhibitor with IC50s of 7, 2, …
Formula:
C22H19ClN6O2S
Purity:
99.7%
Color and Shape:
Solid
Molecular weight:
466.94
Ref: TM-T6719
| 1mg | 35.00 € | ||
| 5mg | 62.00 € | ||
| 10mg | 99.00 € | ||
| 25mg | 165.00 € | ||
| 50mg | To inquire | ||
| 1mL*10mM (DMSO) | 72.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
BMS-599626 2HCL(714971-09-2 Free base)
CAS:1781932-33-9
BMS-599626 2HCL (AC480 2HCl) is a BMS-599626 derivative.
Formula:
C27H29Cl2FN8O3
Purity:
98%
Color and Shape:
Soild
Molecular weight:
603.47
Ref: TM-T2610L
| 1mg | 93.00 € | ||
| 5mg | 148.00 € | ||
| 10mg | 278.00 € | ||
| 25mg | 477.00 € | ||
| 50mg | 690.00 € | ||
| 100mg | 979.00 € | ||
| 1mL*10mM (DMSO) | 330.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Panomifene HCl
Panomifene HCl is a selective anti-estrogenic compound with antitumor activity for the treatment of breast …
Formula:
C25H25ClF3NO2
Purity:
99.09%
Color and Shape:
Soild
Molecular weight:
463.92
Ref: TM-T33876L
| 1mg | 183.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Sulcardine 2HCl
CAS:343935-48-8
Sulcardine 2HCl is a multi-ion channel blocker that blocks the properties of hERG and hNav1.5 …
Formula:
C24H35Cl2N3O4S
Purity:
98.45% - 99.51%
Color and Shape:
Soild
Molecular weight:
532.523
Ref: TM-T83979
| 1mg | 184.00 € | ||
| 5mg | 455.00 € | ||
| 10mg | 651.00 € | ||
| 25mg | 1,016.00 € | ||
| 50mg | 1,401.00 € |
Estimated delivery in United States, on Thursday 5 Dec 2024
Tucatinib hemiethanolate
CAS:1429755-56-5
Tucatinib (Irbinitinib) hemiethanolate is a potent, orally active and selective HER2 inhibitor with an IC50 …
Formula:
C54H54N16O5
Purity:
99.76%
Color and Shape:
Solid
Molecular weight:
1007.11
Ref: TM-T36648
| 5mg | 48.00 € | ||
| 10mg | 67.00 € | ||
| 25mg | 96.00 € | ||
| 50mg | 136.00 € | ||
| 100mg | 187.00 € | ||
| 1mL*10mM (DMSO) | 52.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
BI-4142
CAS:2682003-36-5
BI-4142 is a HER2 inhibitor that inhibits cancer cell proliferation, suppresses her2-dependent cell lines and …
Formula:
C28H27N9O2
Purity:
97.21% - 98.09%
Color and Shape:
Liquid
Molecular weight:
521.57
Ref: TM-T63643
| 1mg | 214.00 € | ||
| 5mg | 530.00 € | ||
| 10mg | 833.00 € | ||
| 25mg | 1,368.00 € | ||
| 50mg | 1,867.00 € | ||
| 1mL*10mM (DMSO) | 604.00 € |
Estimated delivery in United States, on Tuesday 10 Dec 2024
BMS 599626 2HCl (873837-23-1(HCl))
CAS:1781932-33-9
BMS 599626 2HCl (873837-23-1(HCl)) (AC480 dihydrochloride) is a selective inhibitor of HER1 and HER2 (IC50s: …
Formula:
C27H29FN8O3Cl2
Purity:
99.94%
Color and Shape:
Soild
Molecular weight:
603.48
Ref: TM-T5398
| 1mg | 54.00 € | ||
| 5mg | 109.00 € | ||
| 10mg | 171.00 € | ||
| 25mg | 351.00 € | ||
| 50mg | 521.00 € | ||
| 100mg | 736.00 € | ||
| 1mL*10mM (DMSO) | 272.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
ICA-105574
CAS:316146-57-3
ICA-105574 activates hERG, enhancing peak current and shortening action potential, while modulating activation kinetics.
Formula:
C19H14N2O4
Purity:
98.89%
Color and Shape:
Solid
Molecular weight:
334.33
Ref: TM-T9009
| 1mg | 42.00 € | ||
| 5mg | 90.00 € | ||
| 10mg | 142.00 € | ||
| 25mg | 291.00 € | ||
| 50mg | 461.00 € | ||
| 100mg | 672.00 € | ||
| 500mg | 1,411.00 € | ||
| 1mL*10mM (DMSO) | 124.00 € |
Estimated delivery in United States, on Wednesday 11 Dec 2024
BMS-599626 Hydrochloride
CAS:873837-23-1
BMS-599626 HCl (AC480 HCl) is an oral inhibitor of HER1, HER2, HER4 kinases, potentially blocking …
Formula:
C27H28ClFN8O3
Purity:
100%
Color and Shape:
Solid
Molecular weight:
567.01
Ref: TM-T5390
| 1mg | 43.00 € | ||
| 5mg | 94.00 € | ||
| 10mg | 129.00 € | ||
| 25mg | 236.00 € | ||
| 50mg | 415.00 € | ||
| 100mg | 612.00 € | ||
| 1mL*10mM (DMSO) | 106.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
MCHR1 antagonist 2
CAS:863115-70-2
MCHR1 antagonist 2 is an antagonist of melanin-concentratin hormone receptor 1(MCH1-R, IC50 = 65 nM) …
Formula:
C23H21FN2O5
Purity:
97.16%
Color and Shape:
Solid
Molecular weight:
424.42
Ref: TM-T11966
| 1mg | 49.00 € | ||
| 5mg | 102.00 € | ||
| 10mg | 172.00 € | ||
| 25mg | 360.00 € | ||
| 50mg | 575.00 € | ||
| 100mg | 922.00 € | ||
| 1mL*10mM (DMSO) | 123.00 € |
Estimated delivery in United States, on Wednesday 5 Feb 2025
AZD-5672
CAS:780750-65-4
AZD-5672 is an antagonist of CCR5 with an IC50 of 0.32 nM.
Formula:
C32H38F2N2O5S2
Purity:
95.58%
Color and Shape:
Solid
Molecular weight:
632.78
Ref: TM-T30260
| 1mg | 198.00 € | ||
| 5mg | 449.00 € | ||
| 10mg | 628.00 € | ||
| 25mg | 916.00 € | ||
| 50mg | 1,281.00 € | ||
| 100mg | 1,744.00 € | ||
| 1mL*10mM (DMSO) | 547.00 € |
Estimated delivery in United States, on Wednesday 5 Mar 2025
