Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Found 327 products of "Opioid Receptor"
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ADL-5859
CAS:ADL-5859 HCl is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for theFormula:C24H28N2O3·HClPurity:98.78% - 99.11%Color and Shape:SolidMolecular weight:428.95Ref: TM-T6175
1mg49.00€2mg66.00€5mg90.00€10mg166.00€25mg319.00€50mg492.00€100mg710.00€500mg1,468.00€1mL*10mM (DMSO)108.00€Orphanin FQ(1-11) acetate(178249-41-7 free base)
Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.Formula:C51H79N15O16Purity:95.54%Color and Shape:SolidMolecular weight:1158.26BMS-986122
CAS:BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1Formula:C16H15BrClNO3S2Purity:98.42%Color and Shape:SolidMolecular weight:448.78Ref: TM-T26869
1mg46.00€5mg90.00€10mg152.00€25mg295.00€50mg447.00€100mg623.00€200mg880.00€1mL*10mM (DMSO)90.00€Leuphasyl TFA
CAS:Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.Formula:C31H40F3N5O9Purity:98.79%Color and Shape:SolidMolecular weight:683.67Methylnaltrexone bromide
CAS:Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.Formula:C21H26BrNO4Purity:99.02%Color and Shape:SolidMolecular weight:436.35GRT2932Q
CAS:GRT2932Q is a nonpeptidic agonist of the opioid receptor-like 1 (ORL1) [1].Formula:C25H26ClN3OColor and Shape:SolidMolecular weight:419.95Viminol
CAS:Viminol is an opioid analgesic. Viminol is based on the α-pyrryl-2-aminoethanol structure, unlike any other class of opioids.Formula:C21H31ClN2OPurity:98%Color and Shape:SolidMolecular weight:362.94CR-665 Acetate
CAS:CR-665, a kappa-opioid agonist, is used potentially for the treatment of postoperative pain.Formula:C38H53N9O6Color and Shape:SolidMolecular weight:731.899GSK1521498 free base
CAS:GSK1521498 free base is an effective and selective μ-opioid receptor antagonist with potential applications in obesity, alcoholism, and drug addiction.Formula:C24H20F2N4Purity:99.85%Color and Shape:SolidMolecular weight:402.44Ref: TM-T11478L
1mg118.00€5mg282.00€10mg516.00€25mg1,007.00€50mg1,583.00€100mg2,322.00€1mL*10mM (DMSO)310.00€GSK1521498
CAS:GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).Formula:C24H23F2N4O4PPurity:98%Color and Shape:SolidMolecular weight:500.43ADL-5859 HCl
CAS:ADL-5859 is a delta-opioid receptor agonist.Formula:C24H28N2O3Purity:98%Color and Shape:SolidMolecular weight:392.49AZD7268
CAS:AZD7268 is a potent, selective, reversible, and orally bioavailable agonist of δ-opioid receptor with CNS penetration.Formula:C29H30N4O2SColor and Shape:SolidMolecular weight:498.64AT-076
CAS:AT-076: κ-opioid (Ki=1.14 nM) & nociceptin (Ki=1.75 nM) noncompetitive antagonist; μ-opioid (Ki=1.67 nM) & δ-opioid (Ki=19.6 nM) competitive antagonist.Formula:C26H35N3O3Color and Shape:SolidMolecular weight:437.57ML 190
CAS:ML 190 is a potent and selective κ opioid receptor (KOR) antagonist (Ki=129 nM), exhibiting an IC50=150 nM in β-arrestin assays, drug addiction.Formula:C27H32N6O3Purity:99.88%Color and Shape:SolidMolecular weight:488.58Ref: TM-T22995
1mg63.00€5mg137.00€10mg205.00€25mg447.00€50mg715.00€100mg964.00€1mL*10mM (DMSO)147.00€LY2048978
CAS:LY2048978: orally-active kappa antagonist, shows promise for mood and addiction in animal studies.Formula:C19H24N2O2Purity:98%Color and Shape:SolidMolecular weight:312.41Dup 747
CAS:Dup 747 is an analgesic that binds with high affinity and selectivity to the kappa-opioid receptor.Formula:C24H28Cl2N2O2Purity:98%Color and Shape:SolidMolecular weight:447.4Opioid receptor modulator 1
CAS:Opioid receptor modulator 1 is a modulator of opioid receptor.Formula:C18H23NO2Purity:98%Color and Shape:SolidMolecular weight:285.38ORL1 antagonist 1
CAS:ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).Formula:C20H22ClN5Purity:98.92%Color and Shape:SolidMolecular weight:367.88Ref: TM-T12320
1mg50.00€5mg105.00€10mg155.00€25mg224.00€50mg315.00€100mg424.00€200mg560.00€1mL*10mM (DMSO)108.00€TIPP
CAS:TIPP is an agent of delta opioid antagonist.Formula:C37H38N4O6Purity:98%Color and Shape:SolidMolecular weight:634.72SCH 221510
CAS:SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.Formula:C28H31NOPurity:99.74%Color and Shape:SolidMolecular weight:397.55μ opioid receptor agonist 2
CAS:μ opioid receptor agonist 2 （Compound H-3）is a MOR receptor agonist. μ opioid receptor agonist 2 can be used for the research of pain and pain related diseases.Formula:C25H34N4OColor and Shape:SolidMolecular weight:406.56Enadoline (Free Base)
CAS:Enadoline is a K-opioid agonist with visual and dissociative effects, studied for pain but dropped due to dysphoria.Formula:C24H32N2O3Color and Shape:SolidMolecular weight:396.52Azoenkephalin
CAS:Azoenkephalin is the azo bridge between tyrosine & phenylalanine of enkephalin molecule.Formula:C28H35N7O7Color and Shape:SolidMolecular weight:581.62ML138
CAS:ML138 is a probe for MLPCN, an agonist of the κ opioid receptor.Formula:C19H14Cl2N4OSColor and Shape:SolidMolecular weight:417.31Norbinaltorphimine
CAS:nor-Binaltorphimine dihydrochloride is a long-acting potent and highly selective kappa opioid receptor antagonist.Formula:C40H43N3O6Color and Shape:SolidMolecular weight:661.79σ1 Receptor/μ Opioid receptor modulator 1
CAS:σ 1 Receptor/ μ Opioid receiver modulator 1 (Compound 44) is an effective σ 1 receptor antagonist (Ki=1.86 nM) and μ Opioid receptor agonists (Ki=2.1 nM).Formula:C24H31FN2O2Color and Shape:SolidMolecular weight:398.51LY 164929
CAS:LY 164929 is a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding site.Formula:C28H41N5O4Color and Shape:SolidMolecular weight:511.66SR8993
CAS:SR8993 is a highly selective, brain-penetrant agonist of the nociceptin receptor.Formula:C25H37FN4Purity:98%Color and Shape:SolidMolecular weight:412.59BMS-986124
CAS:BMS-986124 is an allosteric modulator of the μ-Opioid Receptor.Formula:C16H15BrClNO3S2Color and Shape:SolidMolecular weight:448.78DDD028
CAS:DDD-028 is a potential non-opioid and non-cannabinoid analgesic. It was used for treating neuropathic and inflammatory pain.Formula:C20H20N2Purity:98%Color and Shape:SolidMolecular weight:288.39CP-866087
CAS:CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.Formula:C24H28N2O2Purity:99.56% - >99.99%Color and Shape:SoildMolecular weight:376.49Anrikefon
CAS:Anrikefon (HSK21542) is a kappa opioid receptor agonist with analgesic effect .Formula:C39H57N7O5Molecular weight:703.91GSK1521498 free base (hydrochloride)
CAS:GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).Formula:C24H21ClF2N4Purity:98%Color and Shape:SolidMolecular weight:438.9Ici 174865
CAS:Ici 174865 is a delta opioid receptor antagonist agent.Formula:C38H53N5O7Color and Shape:SolidMolecular weight:691.86LY 281217
CAS:LY 281217, an organic opioid agonist, can produce analgesic effects in mice.Formula:C32H42N4O6Purity:98%Color and Shape:SolidMolecular weight:578.7BW 373U86
CAS:BW373U86 (SNC86), a δ-opioid receptor agonist, demonstrates potent activity with an IC50 value of 1.49 nM and has shown to exhibit antidepressant-like effects [Formula:C27H37N3O2Color and Shape:SolidMolecular weight:435.6DIPPA hydrochloride
CAS:κ receptor antagonistFormula:C22H24Cl3N3OSPurity:98%Color and Shape:SolidMolecular weight:484.87JTC-801 free base
CAS:JTC-801 is a selective antagonist of the opioid receptor-like1 receptor (Ki: 8.2 nM).Formula:C26H25N3O2Purity:98%Color and Shape:SolidMolecular weight:411.5ICI 154,129
CAS:Selective δ opioid antagonistFormula:C34H46N4O6SPurity:98%Color and Shape:SolidMolecular weight:638.82Endomorphin 1 acetate
CAS:Endomorphin 1 acetate is a μ-opioid receptor agonist with antinociceptive and analgesic effects and can be used to study neurological diseases.Formula:C36H42N6O7Purity:99.74%Color and Shape:SolidMolecular weight:670.75Axomadol
CAS:Axomadol (EN3324) is a centrally active analgesic compound. It has opioid agonistic properties and inhibitory effects on the reuptake of monoamines.Formula:C16H25NO3Purity:98%Color and Shape:SolidMolecular weight:279.37Diallyl G
CAS:Diallyl G is a delta-opioid receptor antagonist agent.Formula:C38H53N5O8Color and Shape:SolidMolecular weight:707.86PF-4455242 HCl
CAS:PF-4455242 HCl is a selective and orally available κ-opioid receptor antagonist that exhibiting antidepressant effects.Formula:C21H29ClN2O2SPurity:99.59%Color and Shape:SolidMolecular weight:408.99Loperamide oxide
CAS:Loperamide oxide (R 58425) is a secreted antidiarrheal agent that increases peristalsis and inhibits intestinal absorption of water and ions.Formula:C29H33ClN2O3Color and Shape:SolidMolecular weight:493.04LY2444296
CAS:LY2444296 (FP3FBZ) is an orally active and selective antagonist of kappa opioid receptor(Ki = 1 nM).Formula:C24H22F2N2O2Purity:99.18%Color and Shape:SolidMolecular weight:408.44AT-121
CAS:AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, respectively).Formula:C24H38N4O3SPurity:98.49% - 99.97%Color and Shape:SolidMolecular weight:462.65Ref: TM-T37610
1mg333.00€5mg787.00€10mg1,074.00€25mg1,510.00€50mg1,882.00€100mg2,375.00€500mg4,655.00€IPAG
CAS:IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.Formula:C17H22IN3Purity:99.65%Color and Shape:SolidMolecular weight:395.28ICI 204,448
CAS:ICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of neurological diseases.Formula:C23H27Cl3N2O4Purity:>99.99%Color and Shape:SolidMolecular weight:501.83GR 89696 fumarate
CAS:GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.Formula:C23H29Cl2N3O7Purity:99.84%Color and Shape:SolidMolecular weight:530.4NNC 63-0532
CAS:NNC 63-0532 is a potentnociceptin receptor agonist, Ki=7.3 nM, EC50=305 nM.Formula:C27H29N3O3Purity:99.53%Color and Shape:SolidMolecular weight:443.54ADL-5747
CAS:ADL-5747 (ADL-5747 (free base)) (free base) is a delta opioid receptor agonist used in the treatment of neurological disorders, skin and musculoskeletalFormula:C24H28N2O3Purity:98.94% - 99.74%Color and Shape:SolidMolecular weight:392.49ML-335
CAS:ML-335, a μ-δ targeted agonist and MOR/DOR ligand, may lead to isomer-biased drugs with pain-relief properties.Formula:C25H32N2O3Purity:98.58%Color and Shape:SolidMolecular weight:408.53Ref: TM-T23002
5mg44.00€10mg64.00€25mg112.00€50mg175.00€100mg253.00€200mg359.00€1mL*10mM (DMSO)33.00€JNJ-20788560
CAS:JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective for DOR than for mu opioid receptors (MOR).
Formula:C25H28N2O2Purity:98.02%Color and Shape:SolidMolecular weight:388.5Bevenopran
CAS:Bevenopran (CB-5945) is a peripheral antagonist of μ-opioid receptor and can be used in studies about the treatment of opioid-induced bowel dysfunction.Formula:C20H26N4O4Purity:98.69% - 98.9%Color and Shape:SolidMolecular weight:386.44Ref: TM-T14551
1mg62.00€5mg130.00€10mg187.00€25mg299.00€50mg408.00€100mg532.00€200mg705.00€1mL*10mM (DMSO)142.00€SCH-486757
CAS:SCH-486757 is an agonist of nociceptin-1 (NOP1) and orphanin FQ peptide receptors and is used in the study of cough.Formula:C24H23Cl2N3OPurity:99.53% - >99.99%Color and Shape:SolidMolecular weight:440.37Trimebutine CTB salt
CAS:Trimebutine CTB salt (GIC-1001) is an opioid receptor agonist used in the study of pain.Formula:C29H36N2O8S2Purity:99.85% - >99.99%Color and Shape:SolidMolecular weight:604.74ICI 199,441 hydrochloride
CAS:ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.Formula:C21H25Cl3N2OPurity:99.57%Color and Shape:SolidMolecular weight:427.8Ref: TM-T22849
2mg33.00€5mg52.00€10mg75.00€25mg138.00€50mg215.00€100mg314.00€200mg442.00€1mL*10mM (DMSO)58.00€Frakefamide
CAS:Frakefamide: potent analgesic, μ-selective agonist, non-CNS penetrating.Formula:C30H34FN5O5Purity:98%Color and Shape:SolidMolecular weight:563.62Mu opioid receptor antagonist 7
CAS:Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid receptor (µOR) antagonist with an inhibitory concentration (Formula:C22H27ClN2O2Purity:98%Color and Shape:SolidMolecular weight:386.91μ opioid receptor agonist 3
CAS:Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM.Formula:C22H28N2O2Purity:98%Color and Shape:SolidMolecular weight:352.47ICI 204448
CAS:ICI 204448 is a potent and peripherally selective κ-opioid agonist.Formula:C23H26Cl2N2O4Color and Shape:SolidMolecular weight:465.37Icalcaprant
CAS:Icalcaprant is a kappa-opioid receptor antagonist [1].Formula:C23H26N4O3Purity:98%Color and Shape:SolidMolecular weight:406.48DPI-3290
CAS:DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potentFormula:C30H34FN3O2Purity:98%Color and Shape:SolidMolecular weight:487.61CYT-1010
CAS:CYT-1010, a mu-opioid receptor agonist; EC50: β-arrestin, 13.1 nM; cAMP, 0.0053 nM. Extracted from patent WO2013173730A2.Formula:C35H40N6O5Purity:98%Color and Shape:SolidMolecular weight:624.73N-Benzylnaltrindole hydrochloride
CAS:δ2 opioid receptor antagonistFormula:C33H33ClN2O3Purity:98%Color and Shape:SolidMolecular weight:541.08Deltakephalin
CAS:Deltakephalin is a synthetic, potent specific opiate delta receptors agonist.Formula:C34H48N6O10Purity:98%Color and Shape:SolidMolecular weight:700.78MR2034
CAS:MR2034 is an agonist of kappa-Opioid receptor. MR2034 stimulates hypothalamic-pituitary-adrenal axis.Formula:C19H27NO2Color and Shape:SolidMolecular weight:301.42Naloxonazine
CAS:Naloxonazine, a potent, selective opiate mu-1 (μ1) antagonist, also influences leishmania through the modulation of host coding function.Formula:C38H42N4O6Color and Shape:SolidMolecular weight:650.76ADL-08-0011
CAS:ADL-08-0011 is an metabolite of alvimopan.Formula:C23H29NO3Color and Shape:SolidMolecular weight:367.49R-84760 hydrochloride
CAS:R-84760, a potent κ-opioid receptor agonist, relieves tonic pain via supraspinal/spinal pathways, activating noradrenergic descent.Formula:C19H25Cl3N2OSColor and Shape:SolidMolecular weight:435.84Trap-101 hydrochloride
CAS:nociceptin/orphanin FQ (NOP) receptor antagonistFormula:C24H36ClN3O2Purity:98%Color and Shape:SolidMolecular weight:434.02μ opioid receptor agonist 1
CAS:μ opioid receptor agonist 1 (Compound H-1a) is an optically pure oxyheterocyclic substituted pyrroloxypyrazole derivative and an MOR receptor agonist that canFormula:C26H38N4OColor and Shape:SolidMolecular weight:422.61Ro 48-6791
CAS:Ro 48-6791, a GABA receptor agonist, is used potentially for anesthesia.Formula:C21H25FN6O2Color and Shape:SolidMolecular weight:412.46ADL 08-0011 HCl
CAS:ADL 08-0011, a μ-opioid antagonist with Ki 0.25 nM, is derived from alvimopan by gut microbes and counteracts loperamide effects in rats.Formula:C23H30ClNO3Color and Shape:SolidMolecular weight:403.947Salvinorin A Carbamate
CAS:Salvinorin A carbamate, a potent κ-opioid receptor (KOR) full agonist, exhibits nearly the same potency as salvinorin A, with EC50 values of 6.2 and 4.5 nM, respectively, for activating the human KOR to augment the binding of [35S]GTPγS. Enhancing biological stability, the addition of a carbamate group to salvinorin A reduces deacetylation.Formula:C22H27NO8Color and Shape:SolidMolecular weight:433.457Prodilidine hydrochloride
CAS:Prodilidine hydrochloride is an opioid analgesic.Formula:C15H22ClNO2Color and Shape:SolidMolecular weight:283.79PD 117302
CAS:PD 117302: nonpeptide, kappa-opioid agonist, anti-arrhythmic, anticonvulsant, impacts locomotion, diuresis.Formula:C21H28N2OSColor and Shape:SolidMolecular weight:356.52Naloxonazine dihydrochloride
CAS:μ1 receptor antagonistFormula:C38H43ClN4O6Purity:98%Color and Shape:SolidMolecular weight:687.22SNC 162
CAS:SNC 162 is a potent and selective delta-opioid receptor (δ-opioid) agonist with analgesic, antidepressant and antiarrhythmic effects.Formula:C27H37N3OPurity:98%Color and Shape:SolidMolecular weight:419.6FK 33-824
CAS:FK 33-824, a stable synthetic analog of methionine enkephalin, reversible with naloxone.Formula:C29H41N5O7SPurity:98%Color and Shape:SolidMolecular weight:603.73Naldemedine tosylate
CAS:Naldemedine (S-297995) tosylate, a PAMORA, targets μ-, δ-, κ-opioid receptors, aiding OIC research, may bind to SARS-CoV2's 3CL pro.Formula:C39H42N4O9SColor and Shape:SolidMolecular weight:742.84DS34942424
DS34942424 is an orally potent analgesic which did not exhibit mu opioid receptor agonist activity.Formula:C15H17FN2OColor and Shape:SolidMolecular weight:260.31BU72
CAS:BU72 is a potent, long-lasting agonist for μ and κ opioid receptors, with partial agonistic activity at the δ opioid receptor (EC50 values of 0.054, 0.033, and 0.58 nM, respectively). It provides strong, enduring analgesic effects primarily mediated through μ opioid receptors. BU72 also exhibits a prolonged duration of activity and can partially reverse morphine-induced analgesia. It is applicable in studies of opioid dependence.Formula:C28H32N2O2Color and Shape:SolidMolecular weight:428.57Mu opioid receptor antagonist 5
Compound NAP: MOR antagonist, crosses blood-brain barrier, EC50: 1.14 nM, Ki: 0.37 nM, useful for OUD research.Formula:C26H29N3O4Color and Shape:SolidMolecular weight:447.53σ1 Receptor/μ Opioid receptor modulator 2
CAS:Compound 4x, also known as σ1 Receptor/μOpioid receptormodulator 2, acts as a μOR agonist and a σ1R antagonist, exhibiting a potent μOR EC50 of 0.6 nM and strong σ1R inhibitory activity (Ki: 363.7 nM). It demonstrates significant analgesic effects in various pain models.Formula:C23H31N3OMolecular weight:365.51Daeatal
CAS:Dynorphin A ethylamide (1-9), the opioid activities were examined in the bioassays.Formula:C56H93N19O10Purity:98%Color and Shape:SolidMolecular weight:1192.46BNTX maleate
CAS:δ1 opioid receptor antagonistFormula:C31H31NO8Purity:98%Color and Shape:SolidMolecular weight:545.58BW 443C
CAS:BW 443C is a selective agonist of mu-opioid receptor.Formula:C33H46N10O10Color and Shape:SolidMolecular weight:742.791Mu opioid receptor antagonist 2
Compound 25: potent, selective MOR antagonist, crosses blood-brain barrier (Ki: 0.37 nM, EC50: 0.44 nM), for OUD research.Formula:C25H28N2O4SColor and Shape:SolidMolecular weight:452.57Salvinorin A Propionate
CAS:Salvinorin A propionate: partial KOR agonist, Ki=32.6 nM, EC50=4.7 nM; ignores μ/δ/ORL-1, non-opioid receptors; less potent analgesic vs. salvinorin A.Formula:C24H30O8Color and Shape:SolidMolecular weight:446.49Phenethyl 4-ANPP
CAS:Phenethyl 4-ANPP is a MOR (μ-opioid receptor) agonist with a structure similar to known opioids.Formula:C27H32N2Color and Shape:SolidMolecular weight:384.56SB-612111
CAS:SB-612111: potent ORL-1 antagonist, Ki=0.33 nM; μ-, κ-, δ-receptor Ki=57.6, 160.5, 2109 nM; blocks nociceptin's pain effect.Formula:C24H29Cl2NOColor and Shape:SolidMolecular weight:418.40CCG258747
CAS:CCG258747 is a novel, selective inhibitor of the GRK2 subfamily.Formula:C28H27FN4O4Color and Shape:SolidMolecular weight:502.54Sunobinop
CAS:Sunobinop (S 117957) is an opioid receptor-like orphan receptor (ORL1) modulator.Formula:C26H33N3O3Color and Shape:SolidMolecular weight:435.56NOP agonist-1
CAS:NOP agonist-1 (compound 4) is a nociceptin opioid receptor (NOP) partial agonist that attenuates Parkinsonian disabilities in 6-OHDA hemilesioned rats [1].Formula:C22H34N2Molecular weight:326.52Mu opioid receptor antagonist 4
Compound 31: Potent, selective MOR antagonist; crosses blood-brain barrier; Ki & EC50: 0.38 nM; useful for OUD research.Formula:C25H28N2O4SColor and Shape:SolidMolecular weight:452.57SB-612111 hydrochloride
SB-612111 is a potent ORL-1 antagonist, with high affinity (Ki: 0.33 nM) and µ-receptor activity (Ki: 57.6 nM), blocking Nociceptin-induced pain.Formula:C24H30Cl3NOColor and Shape:SolidMolecular weight:454.86MTI013
MTI013 is a selective inhibitor of SARS-CoV-2 nsp14 Mtase (IC50: 2.98 µM) and an antiviral agent (IC50: 10.33 µM in HCoV-229E infected Huh7 cells). Additionally, MTI013 demonstrates synergistic antiviral effects when used in conjunction with the RdRp inhibitor SHEN26.Formula:C24H26N6O4SColor and Shape:SolidMolecular weight:494.57RX 809055AX
CAS:RX 809055AX is a long lasting opioid antagonist at mu and delta receptors.Formula:C29H29ClN2O4Color and Shape:SolidMolecular weight:505SC13
CAS:SC13, a novel mitragynine analog, exhibits low-efficacy agonism at Mu opioid receptors and provides antinociception while minimizing adverse effects.Formula:C26H30N2O5Color and Shape:SolidMolecular weight:450.53
