Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Found 327 products of "Opioid Receptor"
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ADL-5859
CAS:ADL-5859 HCl is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for theFormula:C24H28N2O3·HClPurity:98.78% - 99.11%Color and Shape:SolidMolecular weight:428.95Ref: TM-T6175
1mg49.00€2mg66.00€5mg90.00€1mL*10mM (DMSO)108.00€10mg166.00€25mg319.00€50mg492.00€100mg710.00€500mg1,468.00€Orphanin FQ(1-11) acetate(178249-41-7 free base)
Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.Formula:C51H79N15O16Purity:95.54%Color and Shape:SolidMolecular weight:1158.26BMS-986122
CAS:BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1Formula:C16H15BrClNO3S2Purity:98.42%Color and Shape:SolidMolecular weight:448.78Ref: TM-T26869
1mg46.00€5mg90.00€1mL*10mM (DMSO)90.00€10mg152.00€25mg295.00€50mg447.00€100mg623.00€200mg880.00€Leuphasyl TFA
CAS:Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.Formula:C31H40F3N5O9Purity:98.79%Color and Shape:SolidMolecular weight:683.67Methylnaltrexone bromide
CAS:Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.Formula:C21H26BrNO4Purity:99.02%Color and Shape:SolidMolecular weight:436.35GRT2932Q
CAS:GRT2932Q is a nonpeptidic agonist of the opioid receptor-like 1 (ORL1) [1].Formula:C25H26ClN3OColor and Shape:SolidMolecular weight:419.95Viminol
CAS:Viminol is an opioid analgesic. Viminol is based on the α-pyrryl-2-aminoethanol structure, unlike any other class of opioids.Formula:C21H31ClN2OPurity:98%Color and Shape:SolidMolecular weight:362.94CR-665 Acetate
CAS:CR-665, a kappa-opioid agonist, is used potentially for the treatment of postoperative pain.Formula:C38H53N9O6Color and Shape:SolidMolecular weight:731.899GSK1521498 free base
CAS:GSK1521498 free base is an effective and selective μ-opioid receptor antagonist with potential applications in obesity, alcoholism, and drug addiction.Formula:C24H20F2N4Purity:99.85%Color and Shape:SolidMolecular weight:402.44Ref: TM-T11478L
1mg118.00€5mg282.00€1mL*10mM (DMSO)310.00€10mg516.00€25mg1,007.00€50mg1,583.00€100mg2,322.00€GSK1521498
CAS:GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).Formula:C24H23F2N4O4PPurity:98%Color and Shape:SolidMolecular weight:500.43ADL-5859 HCl
CAS:ADL-5859 is a delta-opioid receptor agonist.Formula:C24H28N2O3Purity:98%Color and Shape:SolidMolecular weight:392.49AZD7268
CAS:AZD7268 is a potent, selective, reversible, and orally bioavailable agonist of δ-opioid receptor with CNS penetration.Formula:C29H30N4O2SColor and Shape:SolidMolecular weight:498.64AT-076
CAS:AT-076: κ-opioid (Ki=1.14 nM) & nociceptin (Ki=1.75 nM) noncompetitive antagonist; μ-opioid (Ki=1.67 nM) & δ-opioid (Ki=19.6 nM) competitive antagonist.Formula:C26H35N3O3Color and Shape:SolidMolecular weight:437.57ML 190
CAS:ML 190 is a potent and selective κ opioid receptor (KOR) antagonist (Ki=129 nM), exhibiting an IC50=150 nM in β-arrestin assays, drug addiction.Formula:C27H32N6O3Purity:99.88%Color and Shape:SolidMolecular weight:488.58Ref: TM-T22995
1mg63.00€5mg137.00€1mL*10mM (DMSO)147.00€10mg205.00€25mg447.00€50mg715.00€100mg964.00€LY2048978
CAS:LY2048978: orally-active kappa antagonist, shows promise for mood and addiction in animal studies.Formula:C19H24N2O2Purity:98%Color and Shape:SolidMolecular weight:312.41Dup 747
CAS:Dup 747 is an analgesic that binds with high affinity and selectivity to the kappa-opioid receptor.Formula:C24H28Cl2N2O2Purity:98%Color and Shape:SolidMolecular weight:447.4Opioid receptor modulator 1
CAS:Opioid receptor modulator 1 is a modulator of opioid receptor.Formula:C18H23NO2Purity:98%Color and Shape:SolidMolecular weight:285.38ORL1 antagonist 1
CAS:ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).Formula:C20H22ClN5Purity:98.92%Color and Shape:SolidMolecular weight:367.88Ref: TM-T12320
1mg50.00€5mg105.00€1mL*10mM (DMSO)108.00€10mg155.00€25mg224.00€50mg315.00€100mg424.00€200mg560.00€TIPP
CAS:TIPP is an agent of delta opioid antagonist.Formula:C37H38N4O6Purity:98%Color and Shape:SolidMolecular weight:634.72SCH 221510
CAS:SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.Formula:C28H31NOPurity:99.74%Color and Shape:SolidMolecular weight:397.55
