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Opioid Receptor

Opioid Receptor

Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.

Found 296 products of "Opioid Receptor"

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  • ORL1 antagonist 1

    CAS:
    <p>ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).</p>
    Formula:C20H22ClN5
    Purity:98.92%
    Color and Shape:Solid
    Molecular weight:367.88
  • ICI 154,129

    CAS:
    <p>Selective δ opioid antagonist</p>
    Formula:C34H46N4O6S
    Purity:98%
    Color and Shape:Solid
    Molecular weight:638.82
  • JTC-801 free base

    CAS:
    <p>JTC-801 is a selective antagonist of the opioid receptor-like1 receptor (Ki: 8.2 nM).</p>
    Formula:C26H25N3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:411.5
  • LY 164929

    CAS:
    <p>LY 164929 is a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding site.</p>
    Formula:C28H41N5O4
    Color and Shape:Solid
    Molecular weight:511.66
  • SR8993

    CAS:
    <p>SR8993 is a highly selective, brain-penetrant agonist of the nociceptin receptor.</p>
    Formula:C25H37FN4
    Purity:98%
    Color and Shape:Solid
    Molecular weight:412.59
  • BMS-986124

    CAS:
    <p>BMS-986124 is an allosteric modulator of the μ-Opioid Receptor.</p>
    Formula:C16H15BrClNO3S2
    Color and Shape:Solid
    Molecular weight:448.78
  • DDD028

    CAS:
    <p>DDD-028 is a potential non-opioid and non-cannabinoid analgesic. It was used for treating neuropathic and inflammatory pain.</p>
    Formula:C20H20N2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:288.39
  • Viminol

    CAS:
    <p>Viminol is an opioid analgesic. Viminol is based on the α-pyrryl-2-aminoethanol structure, unlike any other class of opioids.</p>
    Formula:C21H31ClN2O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:362.94
  • Ici 174865

    CAS:
    <p>Ici 174865 is a delta opioid receptor antagonist agent.</p>
    Formula:C38H53N5O7
    Color and Shape:Solid
    Molecular weight:691.86
  • Endomorphin 1 acetate

    CAS:
    <p>Endomorphin 1 acetate is a μ-opioid receptor agonist with antinociceptive and analgesic effects and can be used to study neurological diseases.</p>
    Formula:C36H42N6O7
    Color and Shape:Solid
    Molecular weight:670.75
  • Axomadol

    CAS:
    <p>Axomadol (EN3324) is a centrally active analgesic compound. It has opioid agonistic properties and inhibitory effects on the reuptake of monoamines.</p>
    Formula:C16H25NO3
    Purity:98%
    Color and Shape:Solid
    Molecular weight:279.37
  • LY 281217

    CAS:
    <p>LY 281217, an organic opioid agonist, can produce analgesic effects in mice.</p>
    Formula:C32H42N4O6
    Purity:98%
    Color and Shape:Solid
    Molecular weight:578.7
  • Diallyl G

    CAS:
    <p>Diallyl G is a delta-opioid receptor antagonist agent.</p>
    Formula:C38H53N5O8
    Color and Shape:Solid
    Molecular weight:707.86
  • Loperamide oxide

    CAS:
    <p>Loperamide oxide (R 58425) is a secreted antidiarrheal agent that increases peristalsis and inhibits intestinal absorption of water and ions.</p>
    Formula:C29H33ClN2O3
    Color and Shape:Solid
    Molecular weight:493.04
  • CR-665 Acetate

    CAS:
    <p>CR-665, a kappa-opioid agonist, is used potentially for the treatment of postoperative pain.</p>
    Formula:C38H53N9O6
    Color and Shape:Solid
    Molecular weight:731.899
  • AZD7268

    CAS:
    <p>AZD7268 is a potent, selective, reversible, and orally bioavailable agonist of δ-opioid receptor with CNS penetration.</p>
    Formula:C29H30N4O2S
    Color and Shape:Solid
    Molecular weight:498.64
  • AT-076

    CAS:
    <p>AT-076: κ-opioid (Ki=1.14 nM) &amp; nociceptin (Ki=1.75 nM) noncompetitive antagonist; μ-opioid (Ki=1.67 nM) &amp; δ-opioid (Ki=19.6 nM) competitive antagonist.</p>
    Formula:C26H35N3O3
    Color and Shape:Solid
    Molecular weight:437.57
  • GSK1521498

    CAS:
    <p>GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).</p>
    Formula:C24H23F2N4O4P
    Purity:98%
    Color and Shape:Solid
    Molecular weight:500.43
  • Dup 747

    CAS:
    <p>Dup 747 is an analgesic that binds with high affinity and selectivity to the kappa-opioid receptor.</p>
    Formula:C24H28Cl2N2O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:447.4
  • σ1 Receptor/μ Opioid receptor modulator 1

    CAS:
    <p>σ 1 Receptor/ μ Opioid receiver modulator 1 (Compound 44) is an effective σ 1 receptor antagonist (Ki=1.86 nM) and μ Opioid receptor agonists (Ki=2.1 nM).</p>
    Formula:C24H31FN2O2
    Color and Shape:Solid
    Molecular weight:398.51