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Opioid Receptor

Opioid Receptor

Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.

Found 296 products of "Opioid Receptor"

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  • Neuropeptide AF (human)
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    Neuropeptide AF (human)

    CAS:
    <p>Neuropeptide AF (93-110), Human is an endogenous antiopioid peptide.</p>
    Formula:C90H132N26O25
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1978.17

    Ref: TM-TP1082

  • Neurotransmitter Receptor Compound Library
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    Neurotransmitter Receptor Compound Library

    <p>A unique collection of 1513 neurotransmitter receptor compounds, can be used for HTS and HCS screening；</p>
    Color and Shape:Odour Solid

    Ref: TM-L2610

  • Ro 64-6198
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    Ro 64-6198

    CAS:
    <p>Ro 64-6198: Nonpeptide, selective NOP agonist, high brain uptake, EC50=25.6 nM, 100x NOP&gt;opioid affinity.</p>
    Formula:C26H31N3O
    Purity:98%
    Color and Shape:Solid
    Molecular weight:401.54

    Ref: TM-T16772

  • [DPro10] Dynorphin A (1-11)acetate,porcine
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    [DPro10] Dynorphin A (1-11)acetate,porcine

    <p>[DPro10] Dynorphin A (1-11)acetate,porcine is a highly potent κ-opioid receptor agonist with a Ki value of 0.13 nM.</p>
    Formula:C65H107N21O15
    Purity:99.05%
    Color and Shape:Soild
    Molecular weight:1422.7

    Ref: TM-T76341L

  • U-54494A hydrochloride
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    U-54494A hydrochloride

    CAS:
    <p>U-54494A hydrochloride is a benzamide derivative related to kappa opioid receptor agonists. U-54494A hydrochloride has anticonvulsant activity.</p>
    Formula:C18H25Cl3N2O
    Color and Shape:Solid
    Molecular weight:391.76

    Ref: TM-T36372

  • Akuammicine
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    Akuammicine

    CAS:
    <p>Akuammicine, as an indole alkaloid from Catharanthus roseus, can be used in cancer cell eradication.</p>
    Formula:C20H22N2O2
    Color and Shape:Solid
    Molecular weight:322.408

    Ref: TM-T29805

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    β-Endorphin, equine TFA

    <p>β-Endorphin, equine TFA, an endogenous opioid peptide, demonstrates high affinity binding to μ/δ opioid receptors and possesses analgesic properties [1] [2] [3</p>
    Formula:C156H249F3N42O46S
    Color and Shape:Solid
    Molecular weight:3537.96

    Ref: TM-T76027

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    Frakefamide TFA

    <p>Frakefamide TFA: potent, peripherally active μ-opioid agonist; doesn't cross blood-brain barrier.</p>
    Formula:C32H35F4N5O7
    Color and Shape:Solid
    Molecular weight:677.64

    Ref: TM-T73655

  • PL-017
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    PL-017

    CAS:
    <p>μ opioid receptor agonist; IC50: 5.5 nM (μ), &gt;10,000 nM (δ). Induces reversible analgesia, catalepsy, hyperthermia in rats.</p>
    Formula:C29H37N5O5
    Purity:98%
    Color and Shape:Solid
    Molecular weight:535.64

    Ref: TM-TP1958

  • DAMGO (TFA)
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    DAMGO (TFA)

    CAS:
    <p>DAMGO is a selective peptide agonist of the µ-opioid receptor .</p>
    Formula:C28H36F3N5O8
    Purity:98%
    Color and Shape:Solid
    Molecular weight:627.61

    Ref: TM-TP1607

  • Orphanin FQ(1-11)
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    Orphanin FQ(1-11)

    CAS:
    <p>Nociceptin peptide fragment (1-11) with potent ORL1/KOR-3 receptor agonism (Ki = 55 nM), no opioid receptor affinity, and analgesic in mice.</p>
    Formula:C49H75N15O14
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1098.2

    Ref: TM-TP1882

  • Biphalin TFA
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    Biphalin TFA

    CAS:
    <p>Biphalin TFA is an opioid peptide analog that penetrates the blood-brain barrier (BBB) and encompasses two active enkephalin pharmacophores.</p>
    Formula:C46H56N10O10·xC2HF3O2
    Purity:98%
    Color and Shape:Solid
    Molecular weight:909.00 (free base)

    Ref: TM-T80074

  • Dermorphin
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    Dermorphin

    CAS:
    <p>Dermorphin is agonist of μ-opioid receptor (MOR) agonist.</p>
    Formula:C40H50N8O10
    Purity:98.82%
    Color and Shape:Solid
    Molecular weight:802.87

    Ref: TM-T7404

  • ICI 174,864
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    ICI 174,864

    CAS:
    <p>Selective δ opioid antagonist. Exhibits partial agonist in vitro activity at δ receptors at high concentrations.</p>
    Formula:C38H53N5O7
    Purity:98%
    Color and Shape:White Solid
    Molecular weight:691.87

    Ref: TM-TP2013

  • Ac-RYYRIK-NH2
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    Ac-RYYRIK-NH2

    CAS:
    <p>NOP site high affinity ligand (Ki=1.5 nM); blocks nociceptin effects in rat brain/heart; agonist in vivo, reduces mouse movement.</p>
    Formula:C44H70N14O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:939.12

    Ref: TM-TP1940

  • [(pF)Phe4]Nociceptin(1-13)NH2
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    [(pF)Phe4]Nociceptin(1-13)NH2

    CAS:
    <p>Potent, selective OP4 agonist; pKi=10.68, pEC50=9.80. &gt;8000x selectivity vs other opioid receptors; long-lasting in vivo effects.</p>
    Formula:C61H99FN22O15
    Purity:98%
    Color and Shape:Solid
    Molecular weight:1399.6

    Ref: TM-TP1885

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    HINT1-IN-1

    <p>HINT1-IN-1 (compound 8) is an inhibitor of histidine triad nucleotide-binding protein 1 (HINT1) with a Ki of 1.14 μM. It influences the cross-regulation between μ-opioid receptors (MOR) and NMDA receptors (NMDAR).</p>
    Formula:C23H24N8O5
    Color and Shape:Solid
    Molecular weight:492.49

    Ref: TM-T205282

  • SNC 80
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    SNC 80

    CAS:
    <p>SNC 80, a non-peptide δ-opioid agonist (Ki=1.78 nM, IC50=2.73 nM), also targets μ-δ heteromers (EC50=52.8 nM), with analgesic and antidepressant potential.</p>
    Formula:C28H39N3O2
    Purity:99.65%
    Color and Shape:Solid
    Molecular weight:449.63

    Ref: TM-T8414

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    KOR agonist 4

    <p>KOR agonist 4 (compound 39) is an agonist targeting the κ opioid receptor (Kappa Opioid Receptor) and activates G protein signaling. It has an EC50 of 14 nM and an Emax of 83% for binding to GTPγS. This compound demonstrates moderate to high intrinsic clearance in human liver cells and shows selectivity for the κ opioid receptor over the μ (MOR) and δ (DOR) opioid receptors by factors of 60 and 810, respectively. KOR agonist 4 is useful for research into central nervous system (CNS) disorders.</p>
    Formula:C21H25N3
    Color and Shape:Solid
    Molecular weight:319.44

    Ref: TM-T205240

  • Nociceptin(1-7)
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    Nociceptin(1-7)

    CAS:
    <p>Bioactive metabolite of nociceptin, antagonist of nociceptin-induced hyperalgesia</p>
    Formula:C31H41N7O9
    Purity:98%
    Color and Shape:Solid
    Molecular weight:655.709

    Ref: TM-T23076