Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Found 327 products of "Opioid Receptor"
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DPI-287
CAS:DPI-287, a selective delta-opioid receptor (DOP) agonist, has a K\(_i\) value of 0.39 nM and is applicable for pain research [1].Formula:C31H39N3O2Molecular weight:485.66Naldemedine
CAS:Naldemedine (S 297995), developed by Shionogi, is a drug for opioid side effects like constipation. It's well tolerated with minor GI issues.Formula:C32H34N4O6Color and Shape:SolidMolecular weight:570.64N-Acetyl-α-Endorphin
CAS:N-Acetyl-α-Endorphin is a chemical compound consisting of α-Endorphin that has been acetylated at the N-terminal.Formula:C79H122N18O27SPurity:98%Color and Shape:SolidMolecular weight:1787.98[Phe1Ψ(CH2-NH)Gly2]Nociceptin(1-13)NH2
CAS:Potent agonist of the nociceptin (ORL1) receptor, demonstrated both in vitro and in vivo.Formula:C61H102N22O14Purity:98%Color and Shape:SolidMolecular weight:1367.6HINT1-IN-1
HINT1-IN-1 (compound 8) is an inhibitor of histidine triad nucleotide-binding protein 1 (HINT1) with a Ki of 1.14 μM. It influences the cross-regulation between μ-opioid receptors (MOR) and NMDA receptors (NMDAR).Formula:C23H24N8O5Color and Shape:SolidMolecular weight:492.49Deltorphin acetate
Deltorphin acetate is a substance obtained from the skin secretions of a frog, Phyllomedusa bicolor and shows high selectivity and affinity for δ-opioidFormula:C46H66N10O12S2Purity:98.93%Color and Shape:SolidMolecular weight:1015.21Ref: TM-T20166L
1mg175.00€5mg394.00€10mg590.00€25mg1,060.00€50mg1,591.00€100mg2,387.00€200mg3,580.00€Neuropeptide AF (human) acetate
Neuropeptide AF (human) acetate (Neuropeptide AF (human) acetate (192387-38-5 Free base)) is an anti-opioid neuropeptide, a Neuropeptide AF (human) derivative,
Purity:99.89%Color and Shape:Soild[Arg14,Lys15]Nociceptin
CAS:Potent NOP agonist (EC50 = 1 nM), >875x selective vs opioid receptors; outperforms nociceptin in vivo, increases pain perception, reduces movement.Formula:C82H137N31O22Purity:98%Color and Shape:SolidMolecular weight:1909.18β-Endorphin, equine TFA
β-Endorphin, equine TFA, an endogenous opioid peptide, demonstrates high affinity binding to μ/δ opioid receptors and possesses analgesic properties [1] [2] [3Formula:C156H249F3N42O46SColor and Shape:SolidMolecular weight:3537.96Dynorphin B (1-13) (TFA)
Dynorphin B (1-13) TFA acts as an agonist on opioid κ-receptor .Formula:C76H116N21F3O19Color and Shape:SolidMolecular weight:1684.86β-Endorphin (1-27) (human) acetate
β-Endorphin (1-27) (human) acetate, existing in the hypophysis cerebri and hypothalamus, exhibits antinociception activity.
Formula:C141H221N33O42SPurity:96.52%Color and Shape:SolidMolecular weight:3082.52Akuammicine
CAS:Akuammicine, as an indole alkaloid from Catharanthus roseus, can be used in cancer cell eradication.Formula:C20H22N2O2Color and Shape:SolidMolecular weight:322.408MT-7716 hydrochloride
CAS:MT-7716 hydrochloride is a selective agonist of non-peptide nociceptin receptor (NOP)Formula:C27H29ClN4O2Purity:98%Color and Shape:SolidMolecular weight:477(S,S)-J-113397
CAS:(S,S)-J-113397 is an isomer of J-113397 . J-113397 is an Opioid Receptor antagonist [1] .Formula:C24H37N3O2Color and Shape:SolidMolecular weight:399.57[(pF)Phe4]Nociceptin(1-13)NH2
CAS:Potent, selective OP4 agonist; pKi=10.68, pEC50=9.80. >8000x selectivity vs other opioid receptors; long-lasting in vivo effects.Formula:C61H99FN22O15Purity:98%Color and Shape:SolidMolecular weight:1399.6DPDPE
CAS:DPDPE is selective δ-opioid receptor agonist peptide.Formula:C30H39N5O7S2Purity:98%Color and Shape:SolidMolecular weight:645.79Clocinnamox mesylate
CAS:Clocinnamox mesylate: irreversible μ-opioid blocker; Ki: 0.7 nM (mouse μ), 1.9 nM (δ), 5.7 nM (κ).Formula:C30H33ClN2O7SColor and Shape:SolidMolecular weight:601.11Dermorphin Analog
Dermorphin Analog, a heptapeptide from amphibian skin, binds μ-opioid receptors selectively and strongly.Formula:C44H59N11O10Purity:98%Color and Shape:SolidMolecular weight:901.43LY255582
CAS:LY255582 is a selective centrally active opioid receptor antagonist with high affinity for mu, delta and kappa receptors with Ki of 0.4 nM, 5.2, 2.0 nM,Formula:C22H35NO2Purity:98%Color and Shape:SolidMolecular weight:345.52R-6890
CAS:R-6890 is an opioid compound with analgesic properties.Formula:C21H24ClN3OColor and Shape:SolidMolecular weight:369.89
![[Phe1Ψ(CH2-NH)Gly2]Nociceptin(1-13)NH2](/_next/image/?url=https%3A%2Fstatic.cymitquimica.com%2Fproducts%2FTM%2Fthumb-webp%2FTP1988.webp&w=3840&q=75)
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