Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Found 296 products of "Opioid Receptor"
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FK 33-824
CAS:<p>FK 33-824, a stable synthetic analog of methionine enkephalin, reversible with naloxone.</p>Formula:C29H41N5O7SPurity:98%Color and Shape:SolidMolecular weight:603.73J-113397
CAS:<p>J-113397 is a potent and selective NOP receptor antagonist (IC50 = 2.3 nM).</p>Formula:C24H37N3O2Purity:98%Color and Shape:SolidMolecular weight:399.57BNTX
CAS:<p>BNTX (7-Benzylidenenaltrexone) is a selective δ1-opioid receptor antagonist. It competitively counteracts the antisecretory effects of DPDPE, Deltorphin 2, and DAMGO. BNTX is applicable in research focused on antinociceptive effects.</p>Formula:C27H27NO4Color and Shape:SolidMolecular weight:429.508Mu opioid receptor antagonist 4
<p>Compound 31: Potent, selective MOR antagonist; crosses blood-brain barrier; Ki & EC50: 0.38 nM; useful for OUD research.</p>Formula:C25H28N2O4SColor and Shape:SolidMolecular weight:452.57SB-612111 hydrochloride
<p>SB-612111 is a potent ORL-1 antagonist, with high affinity (Ki: 0.33 nM) and µ-receptor activity (Ki: 57.6 nM), blocking Nociceptin-induced pain.</p>Formula:C24H30Cl3NOColor and Shape:SolidMolecular weight:454.86RX 809055AX
CAS:<p>RX 809055AX is a long lasting opioid antagonist at mu and delta receptors.</p>Formula:C29H29ClN2O4Color and Shape:SolidMolecular weight:505SC13
CAS:<p>SC13, a novel mitragynine analog, exhibits low-efficacy agonism at Mu opioid receptors and provides antinociception while minimizing adverse effects.</p>Formula:C26H30N2O5Color and Shape:SolidMolecular weight:450.53BU09059
CAS:<p>BU09059 is a potent, selective, short-acting antagonist of the κ-opioid receptor (KOR).</p>Formula:C28H37N3O5Purity:98%Color and Shape:SolidMolecular weight:495.61Mu opioid receptor antagonist 3
<p>Potent, selective MOR antagonist (compound 26); crosses blood-brain barrier. Ki: 0.24 nM, EC50: 0.54 nM; for studying OUD.</p>Formula:C25H28N2O4SColor and Shape:SolidMolecular weight:452.57Allyphenyline oxalate
CAS:<p>The pKi values of Allyphenyline oxalate (compound 9) for the α2-adrenergic receptor subtypes α2A, α2B, and α2C are 7.24, 6.47, and 7.07, respectively.</p>Formula:C16H20N2O5Color and Shape:SolidMolecular weight:320.34rel-SB-612111 hydrochloride
CAS:<p>NOP receptor antagonist</p>Formula:C24H30Cl3NOPurity:98%Color and Shape:SolidMolecular weight:454.86Naldemedine tosylate
CAS:<p>Naldemedine (S-297995) tosylate, a PAMORA, targets μ-, δ-, κ-opioid receptors, aiding OIC research, may bind to SARS-CoV2's 3CL pro.</p>Formula:C39H42N4O9SColor and Shape:SolidMolecular weight:742.84(S)-MCOPPB
CAS:<p>(S)-MCOPPB is the S-enantiomer of MCOPPB, an orally active selective agonist for the Nociceptin/Orphanin FQ-Receptor. It inhibits signal transduction in mouse brain NOP receptors and is utilized in anxiety disorder research.</p>Formula:C26H40N4Color and Shape:SolidMolecular weight:408.623Opioid receptor antagonist 1
CAS:<p>Opioid receptor antagonist 1 (Compound 10) is an Orvinol-based antagonist of opioid receptors. It exhibits activity as an antagonist against the analgesic properties of morphine.</p>Formula:C24H29ClF3NO4Color and Shape:SolidMolecular weight:487.94Naltrindole 5′-isothiocyanate
CAS:<p>Naltrindole 5′-isothiocyanate (5'-NTII) is an irreversible delta opioid receptor antagonist that counters the analgesic effects induced by DSLET without altering the effects caused by DPDPE.</p>Formula:C27H25N3O3SColor and Shape:SolidMolecular weight:471.571Bromadoline
CAS:<p>Bromadoline is an opioid compound that exhibits anti-nociceptive properties in rodents.</p>Formula:C15H21BrN2OColor and Shape:SolidMolecular weight:325.244KNT-127
CAS:<p>KNT-127 is an agonist of δ-Opioid receptor.</p>Formula:C24H24N2O2Purity:98%Color and Shape:SolidMolecular weight:372.46(±)-J 113397
CAS:<p>(±)-J-113397 is a potent and selective non-peptidyl ORL1 receptor antagonist (K(i): cloned human ORL1=1.8 nM).</p>Formula:C24H37N3O2Color and Shape:SolidMolecular weight:399.575′-Guanidinonaltrindole
CAS:<p>5′-Guanidinonaltrindole (GNTI) is a selective antagonist of the kappa opioid receptor.</p>Formula:C27H29N5O3Color and Shape:SolidMolecular weight:471.551GNTI dihydrochloride
CAS:<p>κ opioid receptor antagonist</p>Formula:C27H30ClN5O3Purity:98%Color and Shape:SolidMolecular weight:508.01Sunobinop
CAS:<p>Sunobinop (S 117957) is an opioid receptor-like orphan receptor (ORL1) modulator.</p>Formula:C26H33N3O3Color and Shape:SolidMolecular weight:435.56σ1 Receptor/μ Opioid receptor modulator 2
CAS:<p>Compound 4x, also known as σ1 Receptor/μOpioid receptormodulator 2, acts as a μOR agonist and a σ1R antagonist, exhibiting a potent μOR EC50 of 0.6 nM and strong σ1R inhibitory activity (Ki: 363.7 nM). It demonstrates significant analgesic effects in various pain models.</p>Formula:C23H31N3OMolecular weight:365.51Norbinaltorphimine dihydrochloride
CAS:<p>Norbinaltorphimine dihydrochloride is a selective and potent κ opioid receptor antagonist that induces itch-associated responses in mice.</p>Formula:C40H45Cl2N3O6Purity:98.17% - 99.88%Color and Shape:SolidMolecular weight:734.71BU72
CAS:<p>BU72 is a potent, long-lasting agonist for μ and κ opioid receptors, with partial agonistic activity at the δ opioid receptor (EC50 values of 0.054, 0.033, and 0.58 nM, respectively). It provides strong, enduring analgesic effects primarily mediated through μ opioid receptors. BU72 also exhibits a prolonged duration of activity and can partially reverse morphine-induced analgesia. It is applicable in studies of opioid dependence.</p>Formula:C28H32N2O2Color and Shape:SolidMolecular weight:428.57Riminkefon
CAS:<p>Riminkefon is a kappa opioid receptor agonist .</p>Formula:C38H57N7O6Color and Shape:SolidMolecular weight:707.9JDTic Dihydrochloride
CAS:<p>JDTic Dihydrochloride is a high-affinity and selective κ-opioid receptor (KOR) antagonist that blocks dynorphin-KOR signalling,antidepressant.</p>Formula:C28H41Cl2N3O3Purity:98%Color and Shape:SolidMolecular weight:538.55Mu opioid receptor antagonist 8
CAS:<p>Muopioid Receptor Antagonist 8 (368) serves as an antagonist to the μ-opioid receptor, significantly inhibiting the activation of Gi induced by met-enkephalin at the µOR.</p>Formula:C36H35N3O4SColor and Shape:SolidMolecular weight:605.756β-Naltrexol
CAS:<p>6β-Naltrexol is a peripherally selective opioid antagonist that reduces constipation from opioids while minimizing central nervous system effects.</p>Formula:C20H25NO4Purity:99.933%Color and Shape:SolidMolecular weight:343.42DS34942424
<p>DS34942424 is an orally potent analgesic which did not exhibit mu opioid receptor agonist activity.</p>Formula:C15H17FN2OColor and Shape:SolidMolecular weight:260.31Mu opioid receptor antagonist 5
<p>Compound NAP: MOR antagonist, crosses blood-brain barrier, EC50: 1.14 nM, Ki: 0.37 nM, useful for OUD research.</p>Formula:C26H29N3O4Color and Shape:SolidMolecular weight:447.53BW 443C
CAS:<p>BW 443C is a selective agonist of mu-opioid receptor.</p>Formula:C33H46N10O10Color and Shape:SolidMolecular weight:742.791Mu opioid receptor antagonist 2
<p>Compound 25: potent, selective MOR antagonist, crosses blood-brain barrier (Ki: 0.37 nM, EC50: 0.44 nM), for OUD research.</p>Formula:C25H28N2O4SColor and Shape:SolidMolecular weight:452.57SB-612111
CAS:<p>SB-612111: potent ORL-1 antagonist, Ki=0.33 nM; μ-, κ-, δ-receptor Ki=57.6, 160.5, 2109 nM; blocks nociceptin's pain effect.</p>Formula:C24H29Cl2NOColor and Shape:SolidMolecular weight:418.40Isotodesnitazene
CAS:<p>Isotodesnitazene is an opioid compound that primarily targets the μ-opioid receptor (MOR). It exhibits EC50 values of 34.8 nM and 142 nM for MOR-βarr2 and MOR-mini-Gi, respectively. Isotodesnitazene can be utilized for research in opioid drugs.</p>Formula:C23H31N3OColor and Shape:SolidMolecular weight:365.51Anilopam
CAS:<p>Anilopam is an opioid analgesic belonging to the benzazepine class and acts as an agonist at opioid receptors.</p>Formula:C20H26N2OColor and Shape:SolidMolecular weight:310.4322-Thiocyanatosalvinorin A
CAS:<p>22-Thiocyanatosalvinorin A (RB-64) is a potent selective agonist for the kappa-opioid receptor, exhibiting an EC50 value of 0.077 nM.</p>Formula:C24H27NO8SColor and Shape:SolidMolecular weight:489.54CCG258747
CAS:<p>CCG258747 is a novel, selective inhibitor of the GRK2 subfamily.</p>Formula:C28H27FN4O4Color and Shape:SolidMolecular weight:502.54BNTX maleate
CAS:<p>δ1 opioid receptor antagonist</p>Formula:C31H31NO8Purity:98%Color and Shape:SolidMolecular weight:545.58Daeatal
CAS:<p>Dynorphin A ethylamide (1-9), the opioid activities were examined in the bioassays.</p>Formula:C56H93N19O10Purity:98%Color and Shape:SolidMolecular weight:1192.46Nalmefene
CAS:<p>Nalmefene (ORF 11676) is a μ-opioid antagonist and partial κ agonist used in the study of opioid overdose and alcohol dependence.</p>Formula:C21H25NO3Purity:99.86%Color and Shape:SolidMolecular weight:339.43Propiram fumarate HCl
CAS:<p>Propiram fumarate HClis an orally available Opioid receptors agonist with analgesic activity for the study of musculoskeletal pain.</p>Formula:C16H25N3O·xClHPurity:99.25%Color and Shape:SoildSR17018
CAS:<p>SR17018 is an mu-opioid-receptor (MOR) agonist, binding with GTPγS, with an EC50 of 97 nM.</p>Formula:C19H18Cl3N3OPurity:99.89%Color and Shape:SolidMolecular weight:410.72Cebranopadol
CAS:<p>Cebranopadol (GRT6005) is an analgesic NOP and opioid receptor agonist with Kis of 0.9 nM, 0.7 nM, 2.6 nM, 18 nM for human NOP, μ-opioid (MOP), κ-opioid (KOP)</p>Formula:C24H27FN2OPurity:98.32% - 99.78%Color and Shape:SolidMolecular weight:378.48Bromadoline maleate
CAS:<p>Bromadoline is an opioid analgesic selective for the μ-opioid receptor.</p>Formula:C19H25BrN2O5Purity:98%Color and Shape:SolidMolecular weight:441.322SR14150
CAS:<p>SR14150 is a partial agonist of high-affinity NOP receptor.</p>Formula:C21H30N2OPurity:98%Color and Shape:SolidMolecular weight:326.48MOR agonist-1
CAS:<p>MOR Agonist-1 is a μ-opioid receptor (MOR) agonist noted for its potent analgesic properties and is utilized in research concerning pain and associated</p>Formula:C22H26ClFN2O2Purity:98%Color and Shape:SolidMolecular weight:404.91
