Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Found 296 products of "Opioid Receptor"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
ORL1 antagonist 1
CAS:<p>ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).</p>Formula:C20H22ClN5Purity:98.92%Color and Shape:SolidMolecular weight:367.88ICI 154,129
CAS:<p>Selective δ opioid antagonist</p>Formula:C34H46N4O6SPurity:98%Color and Shape:SolidMolecular weight:638.82JTC-801 free base
CAS:<p>JTC-801 is a selective antagonist of the opioid receptor-like1 receptor (Ki: 8.2 nM).</p>Formula:C26H25N3O2Purity:98%Color and Shape:SolidMolecular weight:411.5LY 164929
CAS:<p>LY 164929 is a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding site.</p>Formula:C28H41N5O4Color and Shape:SolidMolecular weight:511.66SR8993
CAS:<p>SR8993 is a highly selective, brain-penetrant agonist of the nociceptin receptor.</p>Formula:C25H37FN4Purity:98%Color and Shape:SolidMolecular weight:412.59BMS-986124
CAS:<p>BMS-986124 is an allosteric modulator of the μ-Opioid Receptor.</p>Formula:C16H15BrClNO3S2Color and Shape:SolidMolecular weight:448.78DDD028
CAS:<p>DDD-028 is a potential non-opioid and non-cannabinoid analgesic. It was used for treating neuropathic and inflammatory pain.</p>Formula:C20H20N2Purity:98%Color and Shape:SolidMolecular weight:288.39Viminol
CAS:<p>Viminol is an opioid analgesic. Viminol is based on the α-pyrryl-2-aminoethanol structure, unlike any other class of opioids.</p>Formula:C21H31ClN2OPurity:98%Color and Shape:SolidMolecular weight:362.94Ici 174865
CAS:<p>Ici 174865 is a delta opioid receptor antagonist agent.</p>Formula:C38H53N5O7Color and Shape:SolidMolecular weight:691.86Endomorphin 1 acetate
CAS:<p>Endomorphin 1 acetate is a μ-opioid receptor agonist with antinociceptive and analgesic effects and can be used to study neurological diseases.</p>Formula:C36H42N6O7Color and Shape:SolidMolecular weight:670.75Axomadol
CAS:<p>Axomadol (EN3324) is a centrally active analgesic compound. It has opioid agonistic properties and inhibitory effects on the reuptake of monoamines.</p>Formula:C16H25NO3Purity:98%Color and Shape:SolidMolecular weight:279.37LY 281217
CAS:<p>LY 281217, an organic opioid agonist, can produce analgesic effects in mice.</p>Formula:C32H42N4O6Purity:98%Color and Shape:SolidMolecular weight:578.7Diallyl G
CAS:<p>Diallyl G is a delta-opioid receptor antagonist agent.</p>Formula:C38H53N5O8Color and Shape:SolidMolecular weight:707.86Loperamide oxide
CAS:<p>Loperamide oxide (R 58425) is a secreted antidiarrheal agent that increases peristalsis and inhibits intestinal absorption of water and ions.</p>Formula:C29H33ClN2O3Color and Shape:SolidMolecular weight:493.04CR-665 Acetate
CAS:<p>CR-665, a kappa-opioid agonist, is used potentially for the treatment of postoperative pain.</p>Formula:C38H53N9O6Color and Shape:SolidMolecular weight:731.899AZD7268
CAS:<p>AZD7268 is a potent, selective, reversible, and orally bioavailable agonist of δ-opioid receptor with CNS penetration.</p>Formula:C29H30N4O2SColor and Shape:SolidMolecular weight:498.64AT-076
CAS:<p>AT-076: κ-opioid (Ki=1.14 nM) & nociceptin (Ki=1.75 nM) noncompetitive antagonist; μ-opioid (Ki=1.67 nM) & δ-opioid (Ki=19.6 nM) competitive antagonist.</p>Formula:C26H35N3O3Color and Shape:SolidMolecular weight:437.57GSK1521498
CAS:<p>GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).</p>Formula:C24H23F2N4O4PPurity:98%Color and Shape:SolidMolecular weight:500.43Dup 747
CAS:<p>Dup 747 is an analgesic that binds with high affinity and selectivity to the kappa-opioid receptor.</p>Formula:C24H28Cl2N2O2Purity:98%Color and Shape:SolidMolecular weight:447.4σ1 Receptor/μ Opioid receptor modulator 1
CAS:<p>σ 1 Receptor/ μ Opioid receiver modulator 1 (Compound 44) is an effective σ 1 receptor antagonist (Ki=1.86 nM) and μ Opioid receptor agonists (Ki=2.1 nM).</p>Formula:C24H31FN2O2Color and Shape:SolidMolecular weight:398.51Norbinaltorphimine
CAS:<p>nor-Binaltorphimine dihydrochloride is a long-acting potent and highly selective kappa opioid receptor antagonist.</p>Formula:C40H43N3O6Color and Shape:SolidMolecular weight:661.79GSK1521498 free base
CAS:<p>GSK1521498 free base is an effective and selective μ-opioid receptor antagonist with potential applications in obesity, alcoholism, and drug addiction.</p>Formula:C24H20F2N4Purity:99.85%Color and Shape:SolidMolecular weight:402.44ADL-5747
CAS:<p>ADL-5747 (ADL-5747 (free base)) (free base) is a delta opioid receptor agonist used in the treatment of neurological disorders, skin and musculoskeletal</p>Formula:C24H28N2O3Purity:98.94% - 99.74%Color and Shape:SolidMolecular weight:392.49GR 89696 fumarate
CAS:<p>GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.</p>Formula:C23H29Cl2N3O7Purity:99.84%Color and Shape:SolidMolecular weight:530.4NNC 63-0532
CAS:<p>NNC 63-0532 is a potentnociceptin receptor agonist, Ki=7.3 nM, EC50=305 nM.</p>Formula:C27H29N3O3Purity:99.53%Color and Shape:SolidMolecular weight:443.54SCH-486757
CAS:<p>SCH-486757 is an agonist of nociceptin-1 (NOP1) and orphanin FQ peptide receptors and is used in the study of cough.</p>Formula:C24H23Cl2N3OPurity:99.53% - >99.99%Color and Shape:SolidMolecular weight:440.37Trimebutine CTB salt
CAS:<p>Trimebutine CTB salt (GIC-1001) is an opioid receptor agonist used in the study of pain.</p>Formula:C29H36N2O8S2Purity:99.85% - >99.99%Color and Shape:SolidMolecular weight:604.74IPAG
CAS:<p>IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.</p>Formula:C17H22IN3Purity:99.65%Color and Shape:SolidMolecular weight:395.28ICI 199,441 hydrochloride
CAS:<p>ICI 199,441 hydrochloride is a potent, selective agonist of κ-opioid receptor.</p>Formula:C21H25Cl3N2OPurity:99.57%Color and Shape:SolidMolecular weight:427.8ICI 204,448
CAS:<p>ICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of neurological diseases.</p>Formula:C23H27Cl3N2O4Purity:>99.99%Color and Shape:SolidMolecular weight:501.83Bevenopran
CAS:<p>Bevenopran (CB-5945) is a peripheral antagonist of μ-opioid receptor and can be used in studies about the treatment of opioid-induced bowel dysfunction.</p>Formula:C20H26N4O4Purity:98.69% - 98.9%Color and Shape:SolidMolecular weight:386.44JNJ-20788560
CAS:<p>JNJ-20788560 is a delta opioid receptor (DOR) agonist with analgesic activity. It is more selective for DOR than for mu opioid receptors (MOR).</p>Formula:C25H28N2O2Purity:98.02%Color and Shape:SolidMolecular weight:388.5ML-335
CAS:<p>ML-335, a μ-δ targeted agonist and MOR/DOR ligand, may lead to isomer-biased drugs with pain-relief properties.</p>Formula:C25H32N2O3Purity:98.52%Color and Shape:SolidMolecular weight:408.53AT-121
CAS:<p>AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, respectively).</p>Formula:C24H38N4O3SPurity:98.49% - 99.73%Color and Shape:SolidMolecular weight:462.65SNC 162
CAS:<p>SNC 162 is a potent and selective delta-opioid receptor (δ-opioid) agonist with analgesic, antidepressant and antiarrhythmic effects.</p>Formula:C27H37N3OPurity:98%Color and Shape:SolidMolecular weight:419.6CYT-1010
CAS:<p>CYT-1010, a mu-opioid receptor agonist; EC50: β-arrestin, 13.1 nM; cAMP, 0.0053 nM. Extracted from patent WO2013173730A2.</p>Formula:C35H40N6O5Purity:98%Color and Shape:SolidMolecular weight:624.73Mu opioid receptor antagonist 7
CAS:<p>Compound 24, also known as Mu opioid receptor antagonist 7, is a potent, centrally-acting µ-opioid receptor (µOR) antagonist with an inhibitory concentration (</p>Formula:C22H27ClN2O2Purity:98%Color and Shape:SolidMolecular weight:386.91Naloxonazine
CAS:<p>Naloxonazine, a potent, selective opiate mu-1 (μ1) antagonist, also influences leishmania through the modulation of host coding function.</p>Formula:C38H42N4O6Color and Shape:SolidMolecular weight:650.76μ opioid receptor agonist 3
CAS:<p>Compound 20, identified as μ opioid receptor agonist 3, is a potent µOR agonist that exhibits an EC50 value of 0.87 nM.</p>Formula:C22H28N2O2Purity:98%Color and Shape:SolidMolecular weight:352.47R-84760 hydrochloride
CAS:<p>R-84760, a potent κ-opioid receptor agonist, relieves tonic pain via supraspinal/spinal pathways, activating noradrenergic descent.</p>Formula:C19H25Cl3N2OSColor and Shape:SolidMolecular weight:435.84DPI-3290
CAS:<p>DPI-3290 is a specific agonist of opioid receptors (Ki: 0.18 nM, 0.46 nM, and 0.62 nM for δ-, μ-, and κ-opioid receptors, respectively) with potent</p>Formula:C30H34FN3O2Purity:98%Color and Shape:SolidMolecular weight:487.61Deltakephalin
CAS:<p>Deltakephalin is a synthetic, potent specific opiate delta receptors agonist.</p>Formula:C34H48N6O10Purity:98%Color and Shape:SolidMolecular weight:700.78Frakefamide
CAS:<p>Frakefamide: potent analgesic, μ-selective agonist, non-CNS penetrating.</p>Formula:C30H34FN5O5Purity:98%Color and Shape:SolidMolecular weight:563.62Icalcaprant
CAS:<p>Icalcaprant is a kappa-opioid receptor antagonist [1].</p>Formula:C23H26N4O3Purity:98%Color and Shape:SolidMolecular weight:406.48μ opioid receptor agonist 1
CAS:<p>μ opioid receptor agonist 1 (Compound H-1a) is an optically pure oxyheterocyclic substituted pyrroloxypyrazole derivative and an MOR receptor agonist that can</p>Formula:C26H38N4OColor and Shape:SolidMolecular weight:422.61Naloxonazine dihydrochloride
CAS:<p>μ1 receptor antagonist</p>Formula:C38H43ClN4O6Purity:98%Color and Shape:SolidMolecular weight:687.22ICI 204448
CAS:<p>ICI 204448 is a potent and peripherally selective κ-opioid agonist.</p>Formula:C23H26Cl2N2O4Color and Shape:SolidMolecular weight:465.37N-Benzylnaltrindole hydrochloride
CAS:<p>δ2 opioid receptor antagonist</p>Formula:C33H33ClN2O3Purity:98%Color and Shape:SolidMolecular weight:541.08Trap-101 hydrochloride
CAS:<p>nociceptin/orphanin FQ (NOP) receptor antagonist</p>Formula:C24H36ClN3O2Purity:98%Color and Shape:SolidMolecular weight:434.02ADL-08-0011
CAS:<p>ADL-08-0011 is an metabolite of alvimopan.</p>Formula:C23H29NO3Color and Shape:SolidMolecular weight:367.49
