Opioid Receptor
Opioid receptors are a group of G protein-coupled receptors that mediate the effects of endogenous and exogenous opioids. These receptors play a central role in pain modulation, mood regulation, and addictive behaviors. Opioid receptor agonists and antagonists are extensively used in pain management and addiction treatment, as well as in research on neurological and psychiatric disorders. At CymitQuimica, we provide a comprehensive selection of high-quality opioid receptor modulators to support your research in neurobiology, pain management, and addiction therapy.
Found 327 products of "Opioid Receptor"
Sort by
Purity (%)
0
100
|
0
|
50
|
90
|
95
|
100
ADL-5859
CAS:ADL-5859 HCl is a selective δ-opioid receptor agonist ( Ki: 0.8 nM), selectivity against opioid receptor κ, μ, and little inhibition for theFormula:C24H28N2O3·HClPurity:98.78% - 99.11%Color and Shape:SolidMolecular weight:428.95Ref: TM-T6175
1mg49.00€2mg66.00€5mg90.00€10mg166.00€25mg319.00€50mg492.00€100mg710.00€500mg1,468.00€1mL*10mM (DMSO)108.00€Orphanin FQ(1-11) acetate(178249-41-7 free base)
Nociceptin peptide fragment (1-11 aa), potent ORL1/KOR-3 agonist (Ki=55 nM), non-opioid, analgesic in mice.Formula:C51H79N15O16Purity:95.54%Color and Shape:SolidMolecular weight:1158.26BMS-986122
CAS:BMS-986122 (BMS 986122) is a positive allosteric modulator of μ-opioid receptors that increases β-arrestin recruitment stimulated by endomorphin 1 in U2OS-OPRM1Formula:C16H15BrClNO3S2Purity:98.42%Color and Shape:SolidMolecular weight:448.78Ref: TM-T26869
1mg46.00€5mg90.00€10mg152.00€25mg295.00€50mg447.00€100mg623.00€200mg880.00€1mL*10mM (DMSO)90.00€Leuphasyl TFA
CAS:Leuphasyl TFA: a long-lasting, degradation-resistant peptide & δ-opioid receptor agonist for signaling research.Formula:C31H40F3N5O9Purity:98.79%Color and Shape:SolidMolecular weight:683.67Methylnaltrexone bromide
CAS:Methylnaltrexone bromide (MOA-728) is one of the newer agents of peripherally-acting μ-opioid antagonists, acts to reverse the side effects of opioid drugs.Formula:C21H26BrNO4Purity:99.02%Color and Shape:SolidMolecular weight:436.35GRT2932Q
CAS:GRT2932Q is a nonpeptidic agonist of the opioid receptor-like 1 (ORL1) [1].Formula:C25H26ClN3OColor and Shape:SolidMolecular weight:419.95Viminol
CAS:Viminol is an opioid analgesic. Viminol is based on the α-pyrryl-2-aminoethanol structure, unlike any other class of opioids.Formula:C21H31ClN2OPurity:98%Color and Shape:SolidMolecular weight:362.94CR-665 Acetate
CAS:CR-665, a kappa-opioid agonist, is used potentially for the treatment of postoperative pain.Formula:C38H53N9O6Color and Shape:SolidMolecular weight:731.899GSK1521498 free base
CAS:GSK1521498 free base is an effective and selective μ-opioid receptor antagonist with potential applications in obesity, alcoholism, and drug addiction.Formula:C24H20F2N4Purity:99.85%Color and Shape:SolidMolecular weight:402.44Ref: TM-T11478L
1mg118.00€5mg282.00€10mg516.00€25mg1,007.00€50mg1,583.00€100mg2,322.00€1mL*10mM (DMSO)310.00€GSK1521498
CAS:GSK1521498 is a selective antagonist of the μ-opioid receptor (MOR).Formula:C24H23F2N4O4PPurity:98%Color and Shape:SolidMolecular weight:500.43ADL-5859 HCl
CAS:ADL-5859 is a delta-opioid receptor agonist.Formula:C24H28N2O3Purity:98%Color and Shape:SolidMolecular weight:392.49AZD7268
CAS:AZD7268 is a potent, selective, reversible, and orally bioavailable agonist of δ-opioid receptor with CNS penetration.Formula:C29H30N4O2SColor and Shape:SolidMolecular weight:498.64AT-076
CAS:AT-076: κ-opioid (Ki=1.14 nM) & nociceptin (Ki=1.75 nM) noncompetitive antagonist; μ-opioid (Ki=1.67 nM) & δ-opioid (Ki=19.6 nM) competitive antagonist.Formula:C26H35N3O3Color and Shape:SolidMolecular weight:437.57ML 190
CAS:ML 190 is a potent and selective κ opioid receptor (KOR) antagonist (Ki=129 nM), exhibiting an IC50=150 nM in β-arrestin assays, drug addiction.Formula:C27H32N6O3Purity:99.88%Color and Shape:SolidMolecular weight:488.58Ref: TM-T22995
1mg63.00€5mg137.00€10mg205.00€25mg447.00€50mg715.00€100mg964.00€1mL*10mM (DMSO)147.00€LY2048978
CAS:LY2048978: orally-active kappa antagonist, shows promise for mood and addiction in animal studies.Formula:C19H24N2O2Purity:98%Color and Shape:SolidMolecular weight:312.41Dup 747
CAS:Dup 747 is an analgesic that binds with high affinity and selectivity to the kappa-opioid receptor.Formula:C24H28Cl2N2O2Purity:98%Color and Shape:SolidMolecular weight:447.4Opioid receptor modulator 1
CAS:Opioid receptor modulator 1 is a modulator of opioid receptor.Formula:C18H23NO2Purity:98%Color and Shape:SolidMolecular weight:285.38ORL1 antagonist 1
CAS:ORL1 antagonist 1 is an o antagonist of pioid receptor-like 1 (ORL1) (IC50 of 61 nM).Formula:C20H22ClN5Purity:98.92%Color and Shape:SolidMolecular weight:367.88Ref: TM-T12320
1mg50.00€5mg105.00€10mg155.00€25mg224.00€50mg315.00€100mg424.00€200mg560.00€1mL*10mM (DMSO)108.00€TIPP
CAS:TIPP is an agent of delta opioid antagonist.Formula:C37H38N4O6Purity:98%Color and Shape:SolidMolecular weight:634.72SCH 221510
CAS:SCH 221510: oral NOP agonist, EC50=12 nM, Ki=0.3 nM, anxiolytic, for neurological research.Formula:C28H31NOPurity:99.74%Color and Shape:SolidMolecular weight:397.55μ opioid receptor agonist 2
CAS:μ opioid receptor agonist 2 （Compound H-3）is a MOR receptor agonist. μ opioid receptor agonist 2 can be used for the research of pain and pain related diseases.Formula:C25H34N4OColor and Shape:SolidMolecular weight:406.56Enadoline (Free Base)
CAS:Enadoline is a K-opioid agonist with visual and dissociative effects, studied for pain but dropped due to dysphoria.Formula:C24H32N2O3Color and Shape:SolidMolecular weight:396.52Azoenkephalin
CAS:Azoenkephalin is the azo bridge between tyrosine & phenylalanine of enkephalin molecule.Formula:C28H35N7O7Color and Shape:SolidMolecular weight:581.62ML138
CAS:ML138 is a probe for MLPCN, an agonist of the κ opioid receptor.Formula:C19H14Cl2N4OSColor and Shape:SolidMolecular weight:417.31Norbinaltorphimine
CAS:nor-Binaltorphimine dihydrochloride is a long-acting potent and highly selective kappa opioid receptor antagonist.Formula:C40H43N3O6Color and Shape:SolidMolecular weight:661.79σ1 Receptor/μ Opioid receptor modulator 1
CAS:σ 1 Receptor/ μ Opioid receiver modulator 1 (Compound 44) is an effective σ 1 receptor antagonist (Ki=1.86 nM) and μ Opioid receptor agonists (Ki=2.1 nM).Formula:C24H31FN2O2Color and Shape:SolidMolecular weight:398.51LY 164929
CAS:LY 164929 is a highly selective ligand for the lower affinity [3H]D-Ala2-D-Leu-5-enkephalin binding site.Formula:C28H41N5O4Color and Shape:SolidMolecular weight:511.66SR8993
CAS:SR8993 is a highly selective, brain-penetrant agonist of the nociceptin receptor.Formula:C25H37FN4Purity:98%Color and Shape:SolidMolecular weight:412.59BMS-986124
CAS:BMS-986124 is an allosteric modulator of the μ-Opioid Receptor.Formula:C16H15BrClNO3S2Color and Shape:SolidMolecular weight:448.78DDD028
CAS:DDD-028 is a potential non-opioid and non-cannabinoid analgesic. It was used for treating neuropathic and inflammatory pain.Formula:C20H20N2Purity:98%Color and Shape:SolidMolecular weight:288.39CP-866087
CAS:CP-866087 is a novel, potent and selective mu-opioid receptor antagonist for the study of female sexual dysfunction.Formula:C24H28N2O2Purity:99.56% - >99.99%Color and Shape:SoildMolecular weight:376.49Anrikefon
CAS:Anrikefon (HSK21542) is a kappa opioid receptor agonist with analgesic effect .Formula:C39H57N7O5Molecular weight:703.91GSK1521498 free base (hydrochloride)
CAS:GSK1521498 free base (hydrochloride) is a selective antagonist of the μ-opioid receptor (MOR).Formula:C24H21ClF2N4Purity:98%Color and Shape:SolidMolecular weight:438.9Ici 174865
CAS:Ici 174865 is a delta opioid receptor antagonist agent.Formula:C38H53N5O7Color and Shape:SolidMolecular weight:691.86LY 281217
CAS:LY 281217, an organic opioid agonist, can produce analgesic effects in mice.Formula:C32H42N4O6Purity:98%Color and Shape:SolidMolecular weight:578.7BW 373U86
CAS:BW373U86 (SNC86), a δ-opioid receptor agonist, demonstrates potent activity with an IC50 value of 1.49 nM and has shown to exhibit antidepressant-like effects [Formula:C27H37N3O2Color and Shape:SolidMolecular weight:435.6DIPPA hydrochloride
CAS:κ receptor antagonistFormula:C22H24Cl3N3OSPurity:98%Color and Shape:SolidMolecular weight:484.87JTC-801 free base
CAS:JTC-801 is a selective antagonist of the opioid receptor-like1 receptor (Ki: 8.2 nM).Formula:C26H25N3O2Purity:98%Color and Shape:SolidMolecular weight:411.5ICI 154,129
CAS:Selective δ opioid antagonistFormula:C34H46N4O6SPurity:98%Color and Shape:SolidMolecular weight:638.82Endomorphin 1 acetate
CAS:Endomorphin 1 acetate is a μ-opioid receptor agonist with antinociceptive and analgesic effects and can be used to study neurological diseases.Formula:C36H42N6O7Purity:99.74%Color and Shape:SolidMolecular weight:670.75Axomadol
CAS:Axomadol (EN3324) is a centrally active analgesic compound. It has opioid agonistic properties and inhibitory effects on the reuptake of monoamines.Formula:C16H25NO3Purity:98%Color and Shape:SolidMolecular weight:279.37Diallyl G
CAS:Diallyl G is a delta-opioid receptor antagonist agent.Formula:C38H53N5O8Color and Shape:SolidMolecular weight:707.86PF-4455242 HCl
CAS:PF-4455242 HCl is a selective and orally available κ-opioid receptor antagonist that exhibiting antidepressant effects.Formula:C21H29ClN2O2SPurity:99.59%Color and Shape:SolidMolecular weight:408.99Loperamide oxide
CAS:Loperamide oxide (R 58425) is a secreted antidiarrheal agent that increases peristalsis and inhibits intestinal absorption of water and ions.Formula:C29H33ClN2O3Color and Shape:SolidMolecular weight:493.04LY2444296
CAS:LY2444296 (FP3FBZ) is an orally active and selective antagonist of kappa opioid receptor(Ki = 1 nM).Formula:C24H22F2N2O2Purity:99.18%Color and Shape:SolidMolecular weight:408.44AT-121
CAS:AT-121 is a dual μ-opioid and neuropeptide receptor partial agonist (Kis 16.49 and 3.67 nM, respectively).Formula:C24H38N4O3SPurity:98.49% - 99.97%Color and Shape:SolidMolecular weight:462.65Ref: TM-T37610
1mg333.00€5mg787.00€10mg1,074.00€25mg1,510.00€50mg1,882.00€100mg2,375.00€500mg4,655.00€IPAG
CAS:IPAG is a potent σ-receptor antagonist (pKi=4.3). IPAG can induce cell apoptosis.Formula:C17H22IN3Purity:99.65%Color and Shape:SolidMolecular weight:395.28ICI 204,448
CAS:ICI 204,448 is a potent κ-opioid agonist with potential analgesic activity for the study of neurological diseases.Formula:C23H27Cl3N2O4Purity:>99.99%Color and Shape:SolidMolecular weight:501.83GR 89696 fumarate
CAS:GR 89696 fumarate is a highly selective κ2 opioid receptor agonist (IC50 = 0.04nM) with anti-pruritchy, anti-injury and neuroprotective effects.Formula:C23H29Cl2N3O7Purity:99.84%Color and Shape:SolidMolecular weight:530.4NNC 63-0532
CAS:NNC 63-0532 is a potentnociceptin receptor agonist, Ki=7.3 nM, EC50=305 nM.Formula:C27H29N3O3Purity:99.53%Color and Shape:SolidMolecular weight:443.54
